NISHIDE Kiyoharu 西出喜代治

… Alternative Names

西出喜代治

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Researcher Number	10237711
Other IDs
External Links
Affiliation (based on the past Project Information) *help	2013: 武庫川女子大学, 薬学部, 教授 2010: 武庫川女子大学, 薬学部, 教授 2004 – 2005: 広島国際大学, 薬学部, 教授 1997 – 2003: 京都薬科大学, 薬学部, 助教授 1995 – 1996: 京都薬科大学, 講師 1995: 京都薬科大学, 薬学部, 講師 1993 – 1994: 京都薬科大学, 薬学部, 助手
Review Section/Research Field	Principal Investigator Chemical pharmacy / Chemical pharmacy Except Principal Investigator Chemical pharmacy / Chemical pharmacy / Bioorganic chemistry / Biological Sciences
Keywords	Principal Investigator Nucleophile-Electrophile Interaction / retention of configuration / optically active alcohol / sulfoxide / thio ether / reductive desulfurization / hypophosphite / Raney nickel / Diels-Alder Reaction / Aliphatic Fluorocyanides … More / Stereoselective Protonation / Through Space n_F → π^* Interaction / X-Ray Crystallographic Analysis / Cyano group / Fluoro group / 立体配座固定 / Through space n_0→π^Interaction / van der Waals radii / 立体選択的アルキル化 / 立体選択的プロトン化 / Through Space n_0→σ^Interaction / Through Space n_0→π^Interaction / 脂肪族直鎖化合物 / Diels-Alder反応 / 脂肪族直鎖フルオロシアノ化合物 / 立体選択的プロトン化反応 / Through Space n_F→π^ Interaction / X-線構造解析 / シアノ基 / フッ素基 / alpha, beta-unsaturated ketone / α,β-unsaturated ketone / reductive desulfrization / α, β-unsaturated ketone / 無臭スルフィド / TMSBT / TMSBM / 脱アルキル化反応 / 1-ドデカンチオール / 無臭チオール / 無臭Swern酸化 / 無臭Corey-Kim酸化 / メチルモルホリノヘキシルスルホキシド(MMSO) / メチルモルホリノヘキシルスルフィド(MMS) / ドデシルメチルスルホキシド(Dod-S(O)-Me) / ドデシルメチルスルフィド(Dod-S-Me) / 無臭硫黄反応剤 / チオ糖 / 無臭1,3-プロパンジチオール / 無臭ベンゼンチオール / 無臭フェニルメタンチオール / ビス(4-トリメチルシリルフェニル)ジセレニド / 無臭有機セレン反応剤 / 無臭ボランスルフィド錯体 / グリーンケミストリー / 光学活性α-ヒドロキシアルデヒド / 光学活性モノチオアセタール / Raney Nickel-Combination System / 還元的脱硫反応 / キラルメルカプトアルコール / 光学活性二級アルコール / 高選択的不斉還元反応 / 不斉Tandem Michael-MPV反応 / (-)-Eptazocine / (-)-Aphanorphine / Quaternary Carbon / (+)-1,1′-Binaphthol / (+)-Blastmycinone / Alkhlation / (S)-2-Methoxymethylpyrrolidine / Tetronic Acid … More Except Principal Investigator pentafluorobenzoic acid / α,β-不飽和ケトン / mycestericin / FTY720 / FK506 / 2-alkyl-2-amino-1,3-propanediol / ISP-I / リサイクル / 複素環 / 有機合成 / odorless sulfide / odorless thiol / three contiguous chiral centers / dimethylchloroaluminum / MPV reduction / Michael addition / mercapto alcohol / 不斉MPV反応 / 不斉ミカエル付加 / カプトプリル / Raney-Nickel / 不斉プロトン化 / α, β-不飽和アミド / α, β-不飽和エステル / 3連続不斉炭素構築 / conjugate addition-protonation-MPV還元 / 3,4-ジヒドロ-2H-チオピラン / [4+2]cycloaddition-elimination / 1,3-オキサチアン / 光学活性メルカプトアルコール / γ-ブチロラクトン / Michael付加 / キラルアルコール / メルカプト基 / 無臭スルフィド / 無臭チオール / 3連続不斉炭素 / ジメチルクロロアルミニウム / MPV還元 / Michase付加 / メルカプトアルコール / Optically Active Alcohols / Asymmetric Bifunctional Group Exchange Reaction / Asymmetric Protonation / Dynamic Kinetic Resolution / Anymmetric 1,7-Hydride Shift / Asymmetric Tandem Michael-MPV Reaction / Chinal Mercapto Alcohols / α,β-Unsaturated Compounds / 1,7-水素転位 / 光学活性アリルアルコール / 不斉Michael付加反応 / 光学活性γ-メルカプトアルコール / 不斉TandemMichael-MPV反応 / 光学活性アルコール / 不斉官能基交換型反応 / 不斉プロトン化反応 / 動的速度論的分割 / 不斉1,7-水素転位 / 不斉Tandem Michael-MPV反応 / キラルメルカプトアルコール / α,β-不飽和カルボニル化合物 / cyclosporin / vegetable wasps plant worms / immunosuppresant / サクロスポリン / 2-alkyl-2-aminopropanediol / ツクツクボウシタケ / FK720 / サイクロスポリン / Mycestericin / 冬虫夏草 / 免疫抑制剤 / 高効率的 / 触媒的不斉水素移動型還元反応 / 有機合成反応 / 複素環化合物 / 環境調和型 / 不斉合成 / キラルリガンド / イオン化合物 / 触媒 / リガンド / イオン液体 / イオン性化合物 / 不斉還元 / NF-1147 / 選択的阻害 / II型トポイソメラーゼ / ヒト乳癌MDA-MB-231 / 環式アミノアルコール / シクロブタン骨格 / 新規ピリミジン系抗癌剤 / optically active sec-alcohol / intramoleculat MPV reduction / Lewis acid / chiral 3-mercaptoalcohol / dedithioacetalization / demonothioacetalization / silver salt-iodine Less

Development and application of the environmental friendly and highly efficient organic synthesis using characteristics of the heterocycle
- Principal Investigator
  
  KAWASAKI Ikuo
- Project Period (FY)
  2011 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Mukogawa Women's University
Development and application of the environmental friendly organic synthesis using characteristics of the heterocycle
- Principal Investigator
  
  KAWASAKI Ikuo
- Project Period (FY)
  2008 – 2010
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Mukogawa Women's University
無臭チオール・スルフィドの開発とその有機反応への応用Principal Investigator
- Principal Investigator
  
  西出喜代治
- Project Period (FY)
  2003 – 2005
- Research Category
  
  Grant-in-Aid for Exploratory Research
- Research Field
  
  Chemical pharmacy
- Research Institution
  Hiroshima International University
  Kyoto Pharmaceutical University
Studies on the construction of multi-contiguous asymmetric synthesis using mercapto alcohol as a chiral template
- Principal Investigator
  
  NODE Manabu
- Project Period (FY)
  2001 – 2003
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
新しい作用機序を有する新規ピリミジン系抗ガン剤の開発研究
- Principal Investigator
  
  野出學
- Project Period (FY)
  2000
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas (C)
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto Pharmaceutical University
Studies on the Through Space n_0 → π^* and n_0 → σ^* InteractionPrincipal Investigator
- Principal Investigator
  
  NISHIDE Kiyoharu
- Project Period (FY)
  1999 – 2000
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
Studies on the Development of Novel Asymmetric Multi-Functional MPV Reduction
- Principal Investigator
  
  NODE Manabu
- Project Period (FY)
  1997 – 1999
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
Exploitation of a New Method for the Reductive Desulfurization without Racemization of a Secondary AlcoholPrincipal Investigator
- Principal Investigator
  
  NISHIDA Kiyoharu
- Project Period (FY)
  1997 – 1998
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
官能基交換型新規不斉合成反応の開発研究Principal Investigator
- Principal Investigator
  
  西出喜代治
- Project Period (FY)
  1995
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
Design of Immunosuppressant Possessing Novel Mechanisms
- Principal Investigator
  
  FUJITA Tetsuro
- Project Period (FY)
  1995 – 1996
- Research Category
  
  Grant-in-Aid for Scientific Research (A)
- Research Field
  
  Bioorganic chemistry
- Research Institution
  Setsunan University, Faculty of Pharmaceutical Sciences
新しい脱モノチオアセタール化反応剤の開発とその不斉合成への応用
- Principal Investigator
  
  野出學
- Project Period (FY)
  1994
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University
beta位にヘテロ原子を有する不飽和エステル類のalpha及びgamma選択的不斉アルキル化反応の開発Principal Investigator
- Principal Investigator
  
  西出喜代治
- Project Period (FY)
  1993
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto Pharmaceutical University

All 2014 2013 2012 2011 2006 2005 2004 2003 2002

All Journal Article Presentation Book

[Book] 有機医薬品合成化学　ターゲット分子の合成2011
- Author(s)
  西出喜代治、前崎直容　編集、池田潔、川崎郁勇、鳥山正晴、春沢信哉、細井信造、本橋重康、山下正行
- Total Pages
  331
- Publisher
  廣川書店
- Data Source
  KAKENHI-PROJECT-23590031
[Journal Article] A novel one-step synthesis of benzo[b]furo[3,2-b]pyridines having an amino group at the 4-position from benzo[b]furo[3,2-d][1,3]oxazine2013
- Author(s)
  Yukako Tabuchi, Yusa Kakumoto, Hitomi Uchimoto, Ikuo Kawasaki, Yoshitaka Ohishi, and Kiyoharu Nishide
- Journal Title
  
  Heterocycles
  
  Volume: 87 Issue: 1 Pages: 177-191
- DOI
  10.3987/com-12-12615
- NAID
  40019530809
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23590031
[Journal Article] A novel one-step synthesis of benzo[b]furo- [3,2-b]pyridines having an amino group at the 4-position from benzo[b]furo[3,2-d][1,3]oxa-2013
- Author(s)
  Y. Tabuchi, Y. Kakumoto, H. Uchimoto, I. Kawasaki, Y. Ohishi, and K. Nishide
- Journal Title
  
  Heterocycles
  
  Volume: 87 (1) Pages: 177-191
- Data Source
  KAKENHI-PROJECT-23590031
[Journal Article] Preparation of Benzo[<i>b</i>]furans Having Five-Membered Heterocycles at the 2-Position and 2-(4-Alkylcarbamoylbuta-1,3-dienyl)benzo[<i>b</i>]furans, and Their Cysteinyl Leukotriene Receptor (cysLT1, cysLT2) Inhibitory Activity2012
- Author(s)
  Yukiko Akai, Yukako Tabuchi, Kumiko Ando, Azusa Ito, Yoko Sakata, Ikuo Kawasaki, Takahiro Ohishi, Masayuki Yamashita, Shunsaku Ohta, Kiyoharu Nishide, Yoshitaka Ohishi
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 60 Issue: 11 Pages: 1461-1467
- DOI
  10.1248/cpb.c12-00560
- NAID
  130001852386
- ISSN
  0009-2363, 1347-5223
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23590031
[Journal Article] Preparation of benzo[b]furans having five- membered heterocycles at the 2-position and 2-(4-alkylcarbamoylbuta-1,3-dienyl)benzo[b]f urans, and their cysteinyl leukotriene receptor (cysLT1, cysLT2) inhibitory activity2012
- Author(s)
  Yukiko Akai, Y. Tabuchi, K. Ando, A. Ito, Y. Sakata, I. Kawasaki, T. Ohishi, M. Yamashita, S. Ohta, Nishide, Y. Ohishi
- Journal Title
  
  Chem. Pharm. Bull
  
  Volume: 60 (11) Pages: 1461-1467
- NAID
  130001852386
- Data Source
  KAKENHI-PROJECT-23590031
[Journal Article] Preparation and Application of Odorless 1,3-Propanedithiol Reagents2006
- Author(s)
  Nishide, K., Node, M.et al.
- Journal Title
  
  Chem.Pharm.Bull. 54・1
  
  Pages: 141-146
- NAID
  110004820345
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] Odorless Diphenyl Diselenide and Diphenyl Disulfide : Syntheses and Applications2005
- Author(s)
  Nishide, K., Node, M.et al.
- Journal Title
  
  Synthesis ・3
  
  Pages: 447-457
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] The application of phenylmethanethiol and benzenethiol derivative as odorless organosulfur reagents in the synthesis of thiosugars and thioglycosides2005
- Author(s)
  Nishide, K., Node, M.et al.
- Journal Title
  
  Carbohydrate Research 340・15
  
  Pages: 2360-2368
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] 無臭有機硫黄反応剤の開発と応用2004
- Author(s)
  西出喜代治, 野出學
- Journal Title
  
  有機合成化学協会誌 62・9
  
  Pages: 895-910
- NAID
  10013510253
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] A practical improvement of odorless Corey-Kim and Swern oxidations2004
- Author(s)
  Nishide, K.et al.
- Journal Title
  
  Green Chem. 6・3
  
  Pages: 142-146
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] Development of Odorless Thiols and Sulfides and Their Applications to Organic Synthesis2004
- Author(s)
  Nishide, K.et al.
- Journal Title
  
  Monatshefte fur Chemie / Chemical Monthly 135・2
  
  Pages: 189-200
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] Dod-S-Me and Methyl 6-Morpholinohexyl Sulfide (MMS) as New Odorless Borane Carriers2004
- Author(s)
  Nishide, K., Node, M.et al.
- Journal Title
  
  Synthesis ・7
  
  Pages: 1003-1006
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] New odorless method for the Corey-Kim and Swern oxidations utilizing dodecyl methyl sulfide2003
- Author(s)
  Ohsugi, S., Nishide, K.et al.
- Journal Title
  
  Tetrahedron 59・42
  
  Pages: 8393-8398
- Data Source
  KAKENHI-PROJECT-15659005
[Journal Article] New odorless protocols for the Swern and Corey-Kim oxidations2002
- Author(s)
  Nishide, K.et al.
- Journal Title
  
  Tetrahedron Lett. 43・29
  
  Pages: 5177-5179
- Data Source
  KAKENHI-PROJECT-15659005
[Presentation] 77Se NMRを用いた1,2-Bis(arylseleno)-1-alkenesのanti脱離の機構2014
- Author(s)
  多羅尾あさみ、杉本　衣梨、松澤　香月、池田　未来、内本ひとみ、有光　健治、川崎　郁勇、西出　喜代治
- Organizer
  日本薬学会第134年会
- Place of Presentation
  熊本
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 1,2-Bis[4-(trimethylsilyl)phenylseleno]-1-alkenesの酸化により合成したselenoxideの77Se NMRを用いる脱離反応の検討2013
- Author(s)
  多羅尾あさみ、松澤香月、内本ひとみ、有光健治、川崎郁勇、西出喜代治
- Organizer
  33回有機合成若手セミナー明日の有機合成を担う人のために
- Place of Presentation
  神戸市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 1,2-Bis(arylseleno)-1-alkenesの酸化により合成したbisselenoxideの77Se NMRを用いた脱離反応の検討2013
- Author(s)
  多羅尾あさみ、南前奈美、太田千絢、内本ひとみ、有光健治、川崎郁勇、西出喜代治
- Organizer
  63回日本薬学会近畿支部大会
- Place of Presentation
  京田辺市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 幾つかのbenzo[b]furo[3,2-d][1,3]oxazine誘導体からの新規benzo[b]furo[3,2-b]pyridine誘導体の合成2013
- Author(s)
  田渕裕佳子、角本悠早、佐々木麻耶、伊藤由紀江、内本ひとみ、川崎郁勇、大石義孝、西出喜代治
- Organizer
  日本薬学会第133年会
- Place of Presentation
  横浜
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 1,2-Bis(arylseleno)alkenes の酸化-Selenoxideの脱離メカニズムの検討-2012
- Author(s)
  田渕裕佳子, 多羅尾あさみ, 杉本衣梨, 南前奈美, 石田久美, 太田千絢, 清水友香, 内本ひとみ, 川崎郁勇, 西出喜代治
- Organizer
  62回日本薬学会近畿支部大会
- Place of Presentation
  西宮市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 光学活性 4-hydroxy-2-pipecolic acid 誘導体の簡便な不斉合成2012
- Author(s)
  川崎郁勇、内本ひとみ、久留米愛、田渕裕佳子、太田俊作、山下正行、西出喜代治
- Organizer
  42回複素環化学討論会
- Place of Presentation
  京都市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 再利用可能な不斉水素移動型還元反応を利用した光学活性テルブタリンの合成研究2012
- Author(s)
  川崎郁勇, 窪弥生, 東美帆, 内本ひとみ, 田渕裕佳子, 山下正行, 太田俊作, 西出喜代治
- Organizer
  日本薬学会第132年会
- Place of Presentation
  札幌市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] 新規benzo[b]furo[3,2-b]pyridine誘導体合成法の開発2012
- Author(s)
  田渕　裕佳子・角本　悠早・内本　ひとみ・川崎　郁勇・大石　義孝・西出　喜代治
- Organizer
  42回複素環化学討論会
- Place of Presentation
  京都市
- Data Source
  KAKENHI-PROJECT-23590031
[Presentation] イオン液体中でのリサイクル可能な不斉水素移動型還元反応を利用する光学活性テルブタリンの合成に用いる基質の検討2011
- Author(s)
  川崎郁勇、内本ひとみ、窪弥生、田渕裕佳子、山下正行、太田俊作、西出喜代治
- Organizer
  31回有機合成若手セミナー
- Place of Presentation
  京都市
- Data Source
  KAKENHI-PROJECT-23590031

1. NODE Manabu (60027076)

# of Collaborated Projects: 8 results

# of Collaborated Products: 0 results
2. KAWASAKI Ikuo (00234055)

# of Collaborated Projects: 2 results

# of Collaborated Products: 13 results
3. YAMASHITA Yamashita (20239982)

# of Collaborated Projects: 2 results

# of Collaborated Products: 5 results
4. UCHIMOTO Hitomi (23590031)

# of Collaborated Projects: 1 results

# of Collaborated Products: 11 results
5. FUJITA Tetsuro (40027024)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
6. HAMAMAMICHI Norimitsu (60054011)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
7. 田渕裕佳子 (80509943)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
8. 久留米愛 (40454475)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
9. CHIBA Kenji

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
10. SASAKI Shigeo

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results

NISHIDE Kiyoharu 西出 喜代治

西出 喜代治

Research Projects

Research Products

Co-Researchers

Development and application of the environmental friendly and highly efficient organic synthesis using characteristics of the heterocycle

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Development and application of the environmental friendly organic synthesis using characteristics of the heterocycle

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

無臭チオール・スルフィドの開発とその有機反応への応用Principal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Studies on the construction of multi-contiguous asymmetric synthesis using mercapto alcohol as a chiral template

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

新しい作用機序を有する新規ピリミジン系抗ガン剤の開発研究

Principal Investigator

Project Period (FY)

Research Category

Review Section

Research Institution

Studies on the Through Space n_0 → π^* and n_0 → σ^* InteractionPrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Studies on the Development of Novel Asymmetric Multi-Functional MPV Reduction

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Exploitation of a New Method for the Reductive Desulfurization without Racemization of a Secondary AlcoholPrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

官能基交換型新規不斉合成反応の開発研究Principal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Design of Immunosuppressant Possessing Novel Mechanisms

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

新しい脱モノチオアセタール化反応剤の開発とその不斉合成への応用

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

beta位にヘテロ原子を有する不飽和エステル類のalpha及びgamma選択的不斉アルキル化反応の開発Principal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

[Book] 有機医薬品合成化学 ターゲット分子の合成2011

Author(s)

Total Pages

NISHIDE Kiyoharu 西出喜代治

西出喜代治

[Book] 有機医薬品合成化学　ターゲット分子の合成2011