SUMIYOSHI TAKAAKI 住吉孝明

… Alternative Names

住吉孝明スミヨシタカアキ

Sumiyoshi Takaaki 住吉孝明

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Researcher Number	50738911
Other IDs
Affiliation (Current)	2025: 関西大学, 化学生命工学部, 教授
Affiliation (based on the past Project Information) *help	2023: 関西大学, 化学生命工学部, 教授 2020 – 2021: 関西大学, 化学生命工学部, 教授 2019: 関西大学, 化学生命工学部, 准教授 2015 – 2016: 関西大学, 化学生命工学部, 准教授
Review Section/Research Field	Principal Investigator Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Drug development chemistry
Keywords	Principal Investigator 構造活性相関 / 創薬化学 / HDAC6 / タンパク分解誘導剤 / 細胞膜透過性 / HDAC / PROTAC / 血液脳関門 / ヒストン脱アセチル化酵素阻害剤 / 代謝安定性 … More / HDAC阻害剤 / 中枢移行性 / 抗うつ薬 / 脳移行性 / HDAC6阻害剤 / 中枢神経作用薬 / 有機合成化学 / Gタンパク結合型受容体 / 光学活性体 / 部分作動薬 / ムスカリン受容体作動薬 Less

Discovery of cell membrane permeable HDAC6 PROTACsPrincipal Investigator
- Principal Investigator
  
  住吉孝明
- Project Period (FY)
  2023 – 2025
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Kansai University
Drug discovery of CNS-penetrant histonedeacetylase inhibitorsPrincipal Investigator
- Principal Investigator
  
  Sumiyoshi Takaaki
- Project Period (FY)
  2019 – 2021
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Kansai University
Discovery of muscarinic acetylcholine receptor partial agonistsPrincipal Investigator
- Principal Investigator
  
  Sumiyoshi Takaaki
- Project Period (FY)
  2015 – 2016
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kansai University

All 2024 2023 2022 2021 2020 2019 2017 2016 2015

All Journal Article Presentation

[Journal Article] Acquired curved hair is caused by fusion of multiple hair matrix cells.2024
- Author(s)
  Horibe, I.; Izumi, S.; Ke, Y.; Tanahashi, N.; Takagi, Y.; Ishihara, R.; Nakano, T.; Sumiyoshi, T.; Nagaoka, Y.
- Journal Title
  
  J. Dermatol. Sci.
  
  Volume: 113 Issue: 3 Pages: 130-137
- DOI
  10.1016/j.jdermsci.2024.02.002
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K06061
[Journal Article] Cloning of two gene clusters involved in the catabolism of 2,4-dinitrophenol by Paraburkholderia sp. strain KU-46 and characterization of the initial DnpAB enzymes and a two-component monooxygenases DnpC1C2.2023
- Author(s)
  Liu, Y.; Yamamoto, T.; Kohaya, N.; Yamamoto, K.; Okano, K.; Sumiyoshi, T.; Hasegawa, Y.; Lau, P. C. K.; Iwaki, H.
- Journal Title
  
  J. Biosci. Bioeng.
  
  Volume: 136 Issue: 3 Pages: 223-231
- DOI
  10.1016/j.jbiosc.2023.05.013
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K06061
[Journal Article] Identification and Quantification of Short-Chain Aldehydes Generated from Hair by Ultraviolet Ray Irradiation2020
- Author(s)
  Horibe Ippei、Kitayama Shintaro、Nagai Mizuki、Kokuwano Yuri、Nakai Ayaka、Sumiyoshi Takaaki、Nagaoka Yasuo
- Journal Title
  
  Journal of Society of Cosmetic Chemists of Japan
  
  Volume: 54 Issue: 2 Pages: 169-176
- DOI
  10.5107/sccj.54.169
- NAID
  130007863959
- ISSN
  0387-5253, 1884-4146
- Year and Date
  2020-06-20
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07008
[Journal Article] A novel piperidine degradation mechanism in a newly isolated piperidine degrader <i>Pseudomonas</i> sp. strain KU43P2020
- Author(s)
  Yamamoto Taisei、Liu Yaxuan、Sumiyoshi Takaaki、Hasegawa Yoshie、Iwaki Hiroaki
- Journal Title
  
  J. Gen. Appl. Microbiol.
  
  Volume: 66 Issue: 5 Pages: 265-272
- DOI
  10.2323/jgam.2019.11.006
- NAID
  130007947210
- ISSN
  0022-1260, 1349-8037
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07008
[Journal Article] Design, Synthesis and Structure-Activity Relationship Study of Pyrilamine Derivatives as Histone Deacetylase Inhibitors2020
- Author(s)
  Hiranaka Seiya、Arata Mayumi、Nakata Akiko、Tanaka Akiko、Hashizume Yoshinobu、Kudo Norio、Ito Akihiro、Yoshida Minoru、Uesato Shinichi、Nagaoka Yasuo、Sumiyoshi Takaaki
- Journal Title
  
  HETEROCYCLES
  
  Volume: 101 Issue: 2 Pages: 726-726
- DOI
  10.3987/com-19-s(f)52
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07008
[Journal Article] GPR91 antagonist and TGF-β inhibitor suppressed collagen production of high glucose and succinate induced HSC activation2020
- Author(s)
  Sakai Mutsuko、Sumiyoshi Takaaki、Aoyama Takuma、Urayama Kenji、Yoshimura Ryoichi
- Journal Title
  
  Biochemical and Biophysical Research Communications
  
  Volume: 530 Issue: 2 Pages: 362-366
- DOI
  10.1016/j.bbrc.2020.07.141
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07008
[Journal Article] Discovery of new low-molecular-weight p53-Mdmx disruptors and their anti-cancer activities2016
- Author(s)
  Uesato, S.; Matsuura, Y.; Matsue, S.; Sumiyoshi, T.; Hirata, Y.; Takemoto, S.; Kawaratani, Y.; Yamai, Y.; Ishida, K.; Sasaki, T.; Enari, M.
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 24 Issue: 8 Pages: 1919-1926
- DOI
  10.1016/j.bmc.2016.03.021
- Peer Reviewed / Acknowledgement Compliant / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K18903, KAKENHI-PROJECT-24390222, KAKENHI-PROJECT-16K15317
[Journal Article] A Short Synthesis of (+)-β-Lycorane by Asymmetric Conjugate Addition Cascade.2015
- Author(s)
  Ｋｉｙｏｓｈｉ　Ｔｏｍｉｏｋａ
- Journal Title
  
  Ｔｅｔｒａｈｅｄｒｏｎ
  
  Volume: 71 Issue: 39 Pages: 7222-7226
- DOI
  10.1016/j.tet.2015.03.014
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24590035, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-26460005, KAKENHI-PROJECT-26460021, KAKENHI-PROJECT-15K18903
[Journal Article] Cyclic Model for the Asymmetric Conjugate Addition of Organolithiums with Enoates2015
- Author(s)
  Yasutomo Yamamoto
- Journal Title
  
  Synthesis
  
  Volume: 47 Issue: 15 Pages: 2256-2264
- DOI
  10.1055/s-0034-1380702
- NAID
  120005674638
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460021, KAKENHI-PROJECT-15K18903, KAKENHI-PROJECT-24590035
[Journal Article] Discovery of dihydroquinazolinone derivatives as potent, selective, and CNS-penetrant M1 and M4 muscrinic acetylcholine receptors agonists2015
- Author(s)
  Uruno, Y.; Konishi, Y.; Suwa, A.; Takai, K.; Tojo, K.; Nakako, T.; Sakai, M.; Enomoto, T.; Matsuda, H.; Kitamura, A.; Sumiyoshi, T.
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 25 Issue: 22 Pages: 5357-5361
- DOI
  10.1016/j.bmcl.2015.09.032
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] ホスホフルクトキナーゼ-1阻害剤トリプトリナミドの高活性異性体の絶対配置同定2023
- Author(s)
  懸樋涼、小林大貴、西村はる奈、矢島辰雄、吉田稔、長岡康夫、住吉孝明
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K06061
[Presentation] 氷再結晶化抑制活性を有するグルコバニリンとその誘導体の酵素合成およびそれらの細胞凍結保存への応用2023
- Author(s)
  林さくら、譚斌駿、河原秀久、住吉孝明、長岡康夫
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K06061
[Presentation] ツルムラサキ抽出エキスの成分が繊維芽細胞コラーゲン産生に及ぼす影響2023
- Author(s)
  棚橋七海、石川美月、住吉孝明、長岡康夫
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K06061
[Presentation] Streptomyces属菌由来ε-Poly-L-Lysine とその遺伝子複合体の細胞内分布と動態2023
- Author(s)
  佐野量子、白谷康太、住吉孝明、長岡康夫
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K06061
[Presentation] 細胞膜透過性向上を志向したヒドロキサム酸構造を有するpyrilamine型HDAC6阻害剤の探索合成2023
- Author(s)
  天野日菜子、平中誠弥、式田亮文、中田明子、新真由美、伊藤孝、伊藤昭博、吉田稔、布村一人、井手聡一郎、長岡康夫、住吉孝明
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K06061
[Presentation] Sirtuin2選択的阻害活性を有する長鎖脂肪酸アミド誘導体の合成2022
- Author(s)
  相原敬太、宮坂大成、中田明子、伊藤孝、工藤紀雄、伊藤昭博、吉田稔、長岡康夫、住吉孝明
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ホルホフルクトキナーゼ-1阻害剤トリプトリナミドの立体異性体の合成と構造活性相関2022
- Author(s)
  懸樋涼、小林大貴、西村はる菜、吉田稔、長岡康夫、住吉孝明
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ボロン酸構造を有するアセトアミノフェンプロドラッグの合成と評価2022
- Author(s)
  桝屋圭吾、夏谷格、加藤隆児、井尻好雄、長岡康夫、住吉孝明
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ヒト外毛根鞘細胞のコラーゲン産生と毛髪形状との相関性2022
- Author(s)
  柯兪如、堀部一平、叶妃美香、森田樹里、泉沙良、山崎鈴葉、住吉孝明、長岡康夫
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ε-ポリ-L-リシンとそのPEG化体を基盤とする核酸導入剤2022
- Author(s)
  蘇杭、長岡康夫、住吉孝明、石川雄也、藤井美沙、白谷康太
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] 中枢移行性を有するHDAC6選択的阻害剤の開発2022
- Author(s)
  橋本公佑、井手聡一郎、新真由美、中田明子、伊藤昭博、伊藤孝、工藤紀雄、吉田稔、長岡康夫、住吉孝明
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] グルコバニリンの氷再結晶化抑制活性2022
- Author(s)
  譚斌駿、藤井ちひろ、冨士剛弘、河原秀久、住吉孝明、長岡康夫
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] 水晶振動子マイクロバランス法を用いたGP96のタンパク-タンパク相互作用評価系の構築2022
- Author(s)
  宮地貴雅、住友倫子、伊藤健、長岡康夫、住吉孝明
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Synthesis and biological evaluation or stereoisomers of tryptolinamide as phosphofructokinase-1 inhibitor2021
- Author(s)
  Ryo KAKEHI, Hiroki KOBAYASHI, Haruna NISHIMURA, Minoru YOSHIDA, Yasuo NAGAOKA, Takaki SUMIYOSHI
- Organizer
  The 15th International Symposium in Science and Technology 2021
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Synthesis and biological evaluation of long-chain fatty acids amides as selective sirtuin2 inhibitors2021
- Author(s)
  Keita AIHARA, Taisei MIYASAKA, Akiko NAKATA, Akihiro ITO, Minoru YOSHIDA, Yasuo NAGAOKA, Takaaki SUMIYOSHI
- Organizer
  The 15th International Symposium in Science and Technology 2021
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Synthesis and evaluation of dioxazaborocane derivatives as acetaminophen prodrugs2021
- Author(s)
  Keigo MASUYA, Itaru NATSUTANI, Ryuji KATO, Yoshio IJIRI, Yasuo NAGAOKA, Takaaki SUMIYOSHI
- Organizer
  The 15th International Symposium in Science and Technology 2021
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Evaluation of protein-protein interaction between GP96 and oligopeptide permease using quartz crystal microbalance methodology2021
- Author(s)
  Takamasa MIYAJI, Tomoko SUMITOMO, Takeshi ITO, Yasuo NAGAOKA, Takaaki SUMIYOSHI
- Organizer
  The 15th International Symposium in Science and Technology 2021
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] マウスにおけるムスカリンM4受容体作動薬の抗精神病作用の評価2020
- Author(s)
  豊嶋友未香，中村元紀，吉田絵美，大橋千冬，廣瀬光之輔，石﨑悠斗，中村義弘，日垣愛生，清水佐紀，住吉孝明，大野行弘
- Organizer
  第94回日本薬理学会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Concese synthesis of M4 muscarinic acetylcholine receptor agonist2019
- Author(s)
  Yumika Toyoshima, Hirokazu Oho, Yasuo Nagaoka, Takaaki Sumiyoshi
- Organizer
  The 14th International Symposium in Science and Technology (ISST 2019)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Design and Synthesis of Propargyl Ester Containing Histone Deacetylase Inhibitors2019
- Author(s)
  Daisuke Sasaki, Seiya Hiranaka, Yasuo Nagaoka, and Takaaki Sumiyoshi
- Organizer
  The 14th International Symposium in Science and Technology (ISST 2019)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ヒトｉPS細胞由来心筋細胞からなる三次元心筋組織（LbL-3D Heart）を用いたCa2+イメージングによる薬理評価2019
- Author(s)
  恒川晴子, 塚本佳也, 住吉孝明, 赤木隆美, 長岡康夫, 明石満
- Organizer
  第19回日本再生医療学会総会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Design and Synthesis of Hybrid Compound of Pyrilamine and Histone Deacetylase 2 Inhibitor2019
- Author(s)
  Akifumi Shikida, Seiya Hiranaka, Norio Kudo, Minoru Yoshida, Yasuo Nagaoka, Takaaki Sumiyoshi
- Organizer
  The 14th International Symposium in Science and Technology (ISST 2019)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] Design, synthesis and evaluation of novel indoline derivatives as selective M1/M4 muscarinic acetylcholine receptors agonist2019
- Author(s)
  Yuka Ouchi, Hirokazu Oho, Yasuo NAGAOKA, and Takaaki SUMIYOSHI
- Organizer
  The 14th International Symposium in Science and Technology (ISST 2019)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ヒトｉPS細胞由来心筋細胞からなる三次元心筋組織体を用いたハイスループット心毒性評価システムの構築2019
- Author(s)
  恒川晴子, 塚本佳也, 住吉孝明, 赤木隆美, 長岡康夫, 明石満
- Organizer
  三大学医工薬連環科学教育研究機構研究発表会
- Data Source
  KAKENHI-PROJECT-19K07008
[Presentation] ヒストン脱アセチル化酵素（HDAC）阻害剤亜鉛結合部位の構造活性相関によるHDAC6選択的阻害剤の創製2017
- Author(s)
  平中誠弥、上里新一、長岡康夫、伊藤昭博、吉田稔、住吉孝明
- Organizer
  第21回関西大学先端科学技術シンポジウム
- Place of Presentation
  関西大学
- Year and Date
  2017-01-19
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] HDAC6選択的阻害活性を有するベンズアミド誘導体の探索研究2017
- Author(s)
  平中誠弥、上里新一、伊藤昭博、吉田稔、長岡康夫、住吉孝明
- Organizer
  日本薬学会第137年会
- Place of Presentation
  仙台国際センター・東北大学
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Efficient synthesis of (±)-coerulescine.2016
- Author(s)
  K. Takeuchi, K. Ishida, Y. Yamai, Y. Nagaoka, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] 脳移行性を有するヒストン脱アセチル化酵素（HDAC）阻害剤の探索研究2016
- Author(s)
  平中誠弥、上里新一、長岡康夫、伊藤昭博、吉田稔、平田佳之、住吉孝明
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学
- Year and Date
  2016-10-15
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Asymmetric synthesis of 3,3-disubstituted oxindoles using chiral acids.2016
- Author(s)
  M. Shimizu, Y. Yamai, K. Ishida, Y. Nagaoka, T. Sumiyoshi.
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Synthesis and biological evaluation of catechin derivatives.2016
- Author(s)
  K. Kawaguchi, S. Uesato, Y. Nagaoka, S. Yamasaki, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Synthesis and biological evaluation of benzamide derivatives as anti-cancer prodrugs.2016
- Author(s)
  R. Inoue, S. Takemoto, Y. Nakatsuji, Y. Nagaoka, S. Uesato, S. Oishi, M. Enari, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] p53活性化作用を有する2-aminobenzenethiol誘導体の探索研究2016
- Author(s)
  竹本涼穂，松浦佳宏，井上涼佑，江成政人，大石真也，藤井信孝，長岡康夫，上里新一，住吉孝明
- Organizer
  日本薬学会第136年会
- Place of Presentation
  パシフィコ横浜（神奈川）
- Year and Date
  2016-03-27
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Concise synthesis of spiro-fused oxindole derivatives.2016
- Author(s)
  I. Natsutani, R. Iwata, Y. Yamai, K. Ishida, Y. Nagaoka, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] ジケトピペラジン構造を有するヒストン脱アセチル化酵素阻害剤の探索研究2016
- Author(s)
  布袋彩菜，平田佳之，上里新一，長岡康夫，住吉孝明
- Organizer
  日本薬学会第136年会
- Place of Presentation
  パシフィコ横浜（神奈川）
- Year and Date
  2016-03-27
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Intramolecular macrocyclic cyclization by photo-affinity reaction.2016
- Author(s)
  R. Iiji, Y. Nagaoka, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Synthesis and biological evaluation of CNS-penetrant histone deacetylase inhibitor.2016
- Author(s)
  S. Hiranaka, Y. Nagaoka, S. Uesato, A. Ito, M. Yoshida, T. Sumiyoshi
- Organizer
  The 11th International Symposium in Science and Technology at Kansai University 2016
- Place of Presentation
  Kansai University
- Year and Date
  2016-07-26
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] 不斉非対称化反応を用いた光学活性3,3-ジ置換オキシインドールの合成研究2016
- Author(s)
  石田恭次、山井悠介、上里新一、長岡康夫、住吉孝明
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学
- Year and Date
  2016-10-15
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Synthesis and biological evaluation of benzamide derivatives as p53-Mdmx interaction inhibitors2015
- Author(s)
  Inoue, R.; Takemoto, S.; Oishi, S.; Enari, M.; Uesato, S.; Nagaoka, Y.; Sumiyoshi, T.
- Organizer
  The 10th International Symposium in Science and Technology 2015
- Place of Presentation
  Chulalongkorn University, Bangkok, Thailand
- Year and Date
  2015-08-31
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Intramolecular macrocyclic cyclization by photo-affinity reaction of benzophenone with alcohol2015
- Author(s)
  Iiji, R.; Ishida, K.; Nagaoka, Y.; Sumiyoshi, T.
- Organizer
  The 10th International Symposium in Science and Technology 2015
- Place of Presentation
  Chulalongkorn University, Bangkok, Thailand
- Year and Date
  2015-08-31
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Synthesis and biological evaluation of hybrid compounds of histone deacetylase inhibitor and histamine receptor blocker2015
- Author(s)
  Hiranaka, S.; Hotei, A.; Nagaoka, Y.; Sumiyoshi, T.
- Organizer
  The 10th International Symposium in Science and Technology 2015
- Place of Presentation
  Chulalongkorn University, Bangkok, Thailand
- Year and Date
  2015-08-31
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] Selective synthesis of 3,3-disubstituted oxindole and N-hydroxy oxindole via activation of carbonyl group by acid2015
- Author(s)
  Sumiyoshi, T.; Yamai, Y.; Ishida, K.; Shimizu, M.; Zhu, L.; Takeuchi, K.; Uesato, S.; Nagaoka, Y.
- Organizer
  The 10th International Symposium in Science and Technology 2015
- Place of Presentation
  Chulalongkorn University, Bangkok, Thailand
- Year and Date
  2015-08-31
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] 不斉非対称化反応を基盤とする3,3-disubstituted oxindole の合成研究2015
- Author(s)
  石田恭次，山井悠介，上里新一，長岡康夫，住吉孝明
- Organizer
  第65回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪大谷大学（大阪）
- Year and Date
  2015-10-17
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] オキシインドール環化反応の反応機構解明2015
- Author(s)
  山井悠介，石田恭次，竹内一喜，清水雅明，上里新一，長岡康夫，住吉孝明
- Organizer
  第65回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪大谷大学（大阪）
- Year and Date
  2015-10-17
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] 化学者からみた次世代創薬の動向と薬物動態研究者への期待2015
- Author(s)
  住吉孝明
- Organizer
  第 29回日本薬物動態学会ワークショップ
- Place of Presentation
  学術総合センター（東京）
- Year and Date
  2015-05-14
- Invited
- Data Source
  KAKENHI-PROJECT-15K18903
[Presentation] カルボニル基活性化を基盤とする置換oxindole化合物の簡便合成2015
- Author(s)
  山井悠介，石田恭次，周琳濤，竹内一喜，清水雅明，長岡康夫，住吉孝明
- Organizer
  第41回反応と合成の進歩シンポジウム
- Place of Presentation
  近畿大学（大阪）
- Year and Date
  2015-10-26
- Data Source
  KAKENHI-PROJECT-15K18903

1. NAKAMURA Arisa

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
2. NAMBARA Takuya

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
3. MURAKAMI Masato

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
4. YAMAMOTO Yasutomo

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

SUMIYOSHI TAKAAKI 住吉 孝明

住吉 孝明 スミヨシ タカアキ

Sumiyoshi Takaaki 住吉 孝明

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Discovery of cell membrane permeable HDAC6 PROTACsPrincipal Investigator

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Drug discovery of CNS-penetrant histonedeacetylase inhibitorsPrincipal Investigator

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Discovery of muscarinic acetylcholine receptor partial agonistsPrincipal Investigator

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[Journal Article] Acquired curved hair is caused by fusion of multiple hair matrix cells.2024

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[Journal Article] Cloning of two gene clusters involved in the catabolism of 2,4-dinitrophenol by Paraburkholderia sp. strain KU-46 and characterization of the initial DnpAB enzymes and a two-component monooxygenases DnpC1C2.2023

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[Journal Article] Identification and Quantification of Short-Chain Aldehydes Generated from Hair by Ultraviolet Ray Irradiation2020

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[Journal Article] A novel piperidine degradation mechanism in a newly isolated piperidine degrader <i>Pseudomonas</i> sp. strain KU43P2020

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[Journal Article] Design, Synthesis and Structure-Activity Relationship Study of Pyrilamine Derivatives as Histone Deacetylase Inhibitors2020

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[Journal Article] GPR91 antagonist and TGF-β inhibitor suppressed collagen production of high glucose and succinate induced HSC activation2020

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[Journal Article] Discovery of new low-molecular-weight p53-Mdmx disruptors and their anti-cancer activities2016

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[Journal Article] A Short Synthesis of (+)-β-Lycorane by Asymmetric Conjugate Addition Cascade.2015

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[Journal Article] Cyclic Model for the Asymmetric Conjugate Addition of Organolithiums with Enoates2015

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[Journal Article] Discovery of dihydroquinazolinone derivatives as potent, selective, and CNS-penetrant M1 and M4 muscrinic acetylcholine receptors agonists2015

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SUMIYOSHI TAKAAKI 住吉孝明

住吉孝明スミヨシタカアキ

Sumiyoshi Takaaki 住吉孝明