Yamaoka Yousuke 山岡庸介

… Alternative Names

YAMAOKA Yousuke 山岡庸介

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Researcher Number	60624723
Other IDs
Affiliation (Current)	2025: 兵庫医科大学, 薬学部, 講師
Affiliation (based on the past Project Information) *help	2022 – 2024: 兵庫医科大学, 薬学部, 講師 2016 – 2021: 京都大学, 薬学研究科, 助教 2015: 京都大学, 大学院薬学研究科, 助教 2014 – 2015: 京都大学, 薬学研究科(研究院), 助教 2013: 京都大学, ウイルス研究所, 助教
Review Section/Research Field	Principal Investigator Basic Section 33020:Synthetic organic chemistry-related / Chemical pharmacy / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related Except Principal Investigator Chemical pharmacy / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
Keywords	Principal Investigator 生物活性物質 / 複素環 / 中員環 / 酸 / 中員環合成 / イナミド / フロー合成 / 全合成 / 連続反応 / 天然物合成 … More / シクロブタン合成 / シクロブタン / 生理活性物質 / シクロブテン / イノラート / 含窒素複素環合成 / ルイス酸 / 薬学 / 有機化学 / インドリン / キノリン / 抗マラリア活性 / 有機合成 / 抗マラリア薬 / 複素環合成 … More Except Principal Investigator 小員環 / シクロブテン / 中員環 / 分子ひずみ / 面性不斉 / 不斉合成 / 反応開発 / シクロブタン / 刺激応答型分子 / 生理活性物質 / 炭素四員環 / イノラート / 多環芳香族化合物 / 酸化 / C-C結合開裂 / ひずみ化合物 / 刺激応答 / ADC / 精密有機合成 / ひずみ分子 / 生物活性分子 / 電子環状反応 / 新規反応 / ヘリセン / シクロブタノン / シクロプロパン / 生理活性天然物 / キラリティ / 有機材料 / 医薬候補化合物 / 小員環化合物 / 中員環化合物 / 触媒反応 / 合成化学 / 四員環炭化水素 / 生物活性天然物 / 機能性分子 / 天然物合成 / 有機合成 Less

Efficient Synthesis of Cyclobutanes by Multicomponent Reaction Using Ynolates and Its Application for Drug DiscoveryPrincipal Investigator
- Principal Investigator
  
  山岡庸介
- Project Period (FY)
  2024 – 2026
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Hyogo Medical University
formation of carbon four-membered rings using ynolate and its application for drug discoveryPrincipal Investigator
- Principal Investigator
  
  Yamaoka Yousuke
- Project Period (FY)
  2021 – 2023
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 33020:Synthetic organic chemistry-related
- Research Institution
  Hyogo Medical University
  Kyoto University
Design, Synthesis and Evaluation of Biologically Active Molecules Based on Ring Strain
- Principal Investigator
  
  Takasu Kiyosei
- Project Period (FY)
  2019 – 2021
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Kyoto University
Divergent Synthesis of Nitrogen-Containing Heterocycles by Sequential Reactions and Its Application to Drug DiscoveryPrincipal Investigator
- Principal Investigator
  
  Yamaoka Yousuke
- Project Period (FY)
  2018 – 2020
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 33020:Synthetic organic chemistry-related
- Research Institution
  Kyoto University
Efficient synthesis of nitrogen-containing compounds with yanamidesPrincipal Investigator
- Principal Investigator
  
  Yamaoka Yousuke
- Project Period (FY)
  2016 – 2017
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Stereocontrolled synthesis of poly-substituted medium-sized cyclic compounds by electrocyclic ring opening reaction and the synthesis of biologically active molecules
- Principal Investigator
  
  Takasu Kiyosei
- Project Period (FY)
  2016 – 2018
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Discovery of new reactions and utilities of 4-membered carbocyles based on their unique ring strains.
- Principal Investigator
  
  TAKASU KIYOSEI
- Project Period (FY)
  2013 – 2015
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Development of a Bronsted Acid-Promoted Ene-Ynamide CyclizationPrincipal Investigator
- Principal Investigator
  
  YAMAOKA Yousuke
- Project Period (FY)
  2013 – 2014
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University

All 2024 2023 2022 2021 2020 2019 2018 2017 2016 2015 2014 2013 Other

All Journal Article Presentation Book

[Book] Methods and Applications of Cycloaddition Reactions in Organic Syntheses2014
- Author(s)
  Yamaoka, Y. and Takasu, K.
- Total Pages
  20
- Publisher
  Wiley
- Data Source
  KAKENHI-PROJECT-25293002
[Journal Article] Entry into Lithium Ynolates from α,α,α-Tribromomethyl Ketones: Synthesis of Cyclobutenes via the [2 + 2] Cycloaddition with α,β-Unsaturated Carbonyls2024
- Author(s)
  Yamaoka Yousuke、Imahori Hidetaka、Namioka Motoki、Nishina Ryo、Kobori Yukiko、Ueda Motoki、Shindo Mitsuru、Takasu Kiyosei
- Journal Title
  
  Organic Letters
  
  Volume: 26 Issue: 9 Pages: 1896-1901
- DOI
  10.1021/acs.orglett.4c00202
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K17919, KAKENHI-PROJECT-23K18183, KAKENHI-PROJECT-21K05069, KAKENHI-PLANNED-21H05211, KAKENHI-PROJECT-23K24007
[Journal Article] Total Synthesis of Cryptopleurine and Its Analogues2022
- Author(s)
  Yamaoka Yousuke、Takasu Kiyosei、Yamakawa Takuro、Tateishi Kaito
- Journal Title
  
  Synthesis
  
  Volume: 54 Issue: 10 Pages: 2415-2422
- DOI
  10.1055/a-1730-8628
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19H03350, KAKENHI-ORGANIZER-21H05207
[Journal Article] Oxidative β-Cleavage of Fused Cyclobutanols Leading to Hydrofuran-Fused Polycyclic Aromatic Compounds2021
- Author(s)
  Kinouchi Hayate、Sugimoto Kazuma、Yamaoka Yousuke、Takikawa Hiroshi、Takasu Kiyosei
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 86 Issue: 18 Pages: 12615-12622
- DOI
  10.1021/acs.joc.1c01108
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19H03350, KAKENHI-PROJECT-21K18959, KAKENHI-PLANNED-21H05211
[Journal Article] Synthesis of Lactone-fused Cyclopropanes by Ring Contractive-Ketol Rearrangement of Ketal-Fused Cyclobutanones2021
- Author(s)
  Takasu, K.; Shigenaga, K.; Shimoda, K.; Takikawa, H.; Yamaoka
- Journal Title
  
  Heterocyles
  
  Volume: 103 Issue: 1 Pages: 177-177
- DOI
  10.3987/com-20-s(k)6
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19H03350
[Journal Article] Total Synthesis of (-)-Sigillin A: A Polychlorinated and Polyoxygenated Natural Product2020
- Author(s)
  Yamaoka Yousuke、Nakayama Takamori、Kawai Shota、Takasu Kiyosei
- Journal Title
  
  Organic Letters
  
  Volume: 22 Issue: 19 Pages: 7721-7724
- DOI
  10.1021/acs.orglett.0c02930
- NAID
  120006893993
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K05103, KAKENHI-PROJECT-19H03350
[Journal Article] Helical Nanographenes Embedded with Contiguous Azulene Units2020
- Author(s)
  Ogawa Naoki、Yamaoka Yousuke、Takikawa Hiroshi、Yamada Ken-ichi、Takasu Kiyosei
- Journal Title
  
  Journal of the American Chemical Society
  
  Volume: 142 Issue: 31 Pages: 13322-13327
- DOI
  10.1021/jacs.0c06156
- NAID
  120006888507
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19H03350, KAKENHI-PROJECT-19J14061, KAKENHI-PROJECT-18K06579, KAKENHI-PROJECT-19K22185
[Journal Article] Optical resolution via catalytic generation of chiral auxiliary2019
- Author(s)
  Kiyama Hiroki、Inokuma Tsubasa、Kuroda Yusuke、Yamaoka Yousuke、Takasu Kiyosei、Yamada Ken-ichi
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 60 Issue: 2 Pages: 175-177
- DOI
  10.1016/j.tetlet.2018.12.006
- NAID
  120006937697
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K06579, KAKENHI-PROJECT-18K14869, KAKENHI-PUBLICLY-18H04406, KAKENHI-PROJECT-16H05073
[Journal Article] Synthesis and Properties of Tribenzocarbazoles via an Acid-Promoted Retro (2+2)-Cycloaddition of Azapropellanes2018
- Author(s)
  Ogawa Naoki、Yamaoka Yousuke、Takikawa Hiroshi、Tsubaki Kazunori、Takasu Kiyosei
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 83 Issue: 15 Pages: 7994-8002
- DOI
  10.1021/acs.joc.8b00870
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K06548, KAKENHI-PUBLICLY-18H04406, KAKENHI-PROJECT-16H05073
[Journal Article] Silyl enol etherification by a Tf2NH/amine co-catalytic system for minimizing hazardous waste generation2018
- Author(s)
  Kurahashi Kei、Yamaoka Yousuke、Takemoto Yoshiji、Takasu Kiyosei
- Journal Title
  
  Reaction Chemistry & Engineering
  
  Volume: 3 Issue: 5 Pages: 626-630
- DOI
  10.1039/c8re00039e
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04406, KAKENHI-PROJECT-16H05073
[Journal Article] Synthesis of Multi-substituted Cyclobutenes: Cyclic Strategy for (2+2) Cycloaddition of Ketene Silyl Acetals with Propiolates2017
- Author(s)
  Y. Yamaoka, M. Ueda, T. Yamashita, K. Shimoda, K. Yamada, K. Takasu
- Journal Title
  
  Tetrahedron Lett
  
  Volume: 58 Issue: 30 Pages: 2944-2947
- DOI
  10.1016/j.tetlet.2017.06.039
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-16H01147, KAKENHI-PROJECT-16H05073
[Journal Article] Synthesis of pai-Extended Fluoranthenes via a KHMDS-Promoted Anion and Radical Reaction Cascade2017
- Author(s)
  N. Ogawa, Y. Yamaoka, K. Yamada, K. Takasu
- Journal Title
  
  Org. Lett.
  
  Volume: 19 Issue: 12 Pages: 3327-3330
- DOI
  10.1021/acs.orglett.7b01538
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-16H01147, KAKENHI-PROJECT-16H05073
[Journal Article] Synthesis and biological evaluation of steroidal derivatives bearing a small ring as vitamin D receptor agonists2017
- Author(s)
  N. Arichi, S. Fujiwara, M. Ishizawa, M. Makishima, D. H. Hua, K. Yamada, Y. Yamaoka, K. Takasu
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 27 Issue: 15 Pages: 3408-3411
- DOI
  10.1016/j.bmcl.2017.05.089
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01147, KAKENHI-PROJECT-16H05073
[Journal Article] Site-selective Benzoin-type Cyclization of Unsymmetrical Dialdoses Catalyzed by N-Heterocyclic Carbenes for Divergent Cyclitol Synthesis.2017
- Author(s)
  Bubwoon Kang, Yinli Wang, Satoru Kuwano, Yousuke Yamaoka, Kiyosei Takasu, Ken-ichi Yamada
- Journal Title
  
  Chem. Commun.
  
  Volume: 印刷中 Issue: 32 Pages: 4469-4472
- DOI
  10.1039/c7cc01191a
- NAID
  120006650105
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-15K18841, KAKENHI-PROJECT-16H05073, KAKENHI-PUBLICLY-16H01147
[Journal Article] Desymmetrization of Acid Anhydride with Asymmetric Esterification Catalyzed by Chiral Phosphoric Acid.2016
- Author(s)
  K. Yamada
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 57 Issue: 36 Pages: 4098-4100
- DOI
  10.1016/j.tetlet.2016.07.093
- NAID
  120006650106
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460005, KAKENHI-PROJECT-16H05073
[Journal Article] Use of a Catalytic Chiral Leaving Group for Asymmetric Substitutions at sp3-Hybridized Carbon Atoms: Kinetic Resolution of β-Amino Alcohols by p-Methoxybenzylation.2016
- Author(s)
  K. Yamada
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 55 Issue: 42 Pages: 13137-13141
- DOI
  10.1002/anie.201607208
- NAID
  120006556299
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460005, KAKENHI-PUBLICLY-16H01147, KAKENHI-PROJECT-16H05073
[Journal Article] Oxa- and Azacycle-formation via Migrative Cyclization of Sulfonylalkynol and Sulfonylalkynamide with N-Heterocyclic Carbene.2016
- Author(s)
  K. Yamada
- Journal Title
  
  J. Org. Chem
  
  Volume: 81 Issue: 6 Pages: 2652-2664
- DOI
  10.1021/acs.joc.6b00182
- NAID
  120006881403
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460005, KAKENHI-PROJECT-15K18841, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-25293002
[Journal Article] Hydrostannylation-Cross-Coupling Strategy for Stereoselective Synthesis of Alkylidenemalonates and Related α,β-Unsaturated Esters2015
- Author(s)
  Fujiwara, S.; Cadou, R.; Yamaoka, Y.; Takasu, K.; Yamada, K.
- Journal Title
  
  Eur. J. Org. Chem.
  
  Volume: none Issue: 2 Pages: 1264-1272
- DOI
  10.1021/jo502467m
- NAID
  120005623273
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-25293002, KAKENHI-PROJECT-25860006, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-26460005
[Journal Article] Synthesis of Steroidal Derivatives Bearing a Small Ring Using a Catalytic [2+2] Cycloaddition and a Ring-Contraction Rearrangement2015
- Author(s)
  Norihito Arichi, Kenji Hata, Yoshiji Takemoto, Ken-ichi Yamada, Yousuke Yamaoka, Kiyosei Takasu
- Journal Title
  
  Tetrahedron
  
  Volume: 71 Issue: 2 Pages: 233244-233244
- DOI
  10.1016/j.tet.2014.11.065
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-14J07573, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-26460005, KAKENHI-PROJECT-25293002
[Journal Article] An Arylative Ring Expansion Cascade of Fused Cyclobutenes via Short-Lived Intermediates with Planar Chirality.2015
- Author(s)
  K. Yamada
- Journal Title
  
  J. Am. Chem. Soc.
  
  Volume: 137 Issue: 30 Pages: 9579-9582
- DOI
  10.1021/jacs.5b06576
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460005, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-14J07573, KAKENHI-PROJECT-25293002
[Journal Article] Asymmetric Total Synthesis of Tylophorine via a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane.2015
- Author(s)
  K. Yamada
- Journal Title
  
  Synthesis
  
  Volume: 47 Issue: 18 Pages: 2819-2825
- DOI
  10.1055/s-0034-1380430
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460005, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-25293002
[Journal Article] Contiguous radical pivaloyloxymethylation-directed C(sp3)-H iodination of N-tosyl cycloalkanecarbaldimine.2015
- Author(s)
  Ｋｉｙｏｓｈｉ　Ｔｏｍｉｏｋａ
- Journal Title
  
  Tetrahedron Lettｅｒｓ
  
  Volume: 56 Issue: 23 Pages: 3086-3089
- DOI
  10.1016/j.tetlet.2014.11.105
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24590035, KAKENHI-PROJECT-25293002, KAKENHI-PUBLICLY-26105732, KAKENHI-PROJECT-26460005
[Journal Article] Organocatalytic Activation of the Leaving Group in the Intramolecular Asymmetric SN2' Reaction2015
- Author(s)
  Kuroda, Y.; Harada, S.; Oonishi, A.; Yamaoka, Y.; Yamada, K.; Takasu, K.
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 54 Pages: 8263-8266
- NAID
  120005670851
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-25293002
[Journal Article] 1. Equilibration of the EtAlCl2-Catalyzed [2 + 2] Cycloaddition of Silyl Enol Ethers: Diastereoselectivity Switch in the Synthesis of Fused Cyclobutanes2014
- Author(s)
  Hata, K.; Arichi, N.; Yamaoka, Y.; Yamada, K.; Takemoto, Y.; Takasu, K.
- Journal Title
  
  Asian J. Org. Chem.
  
  Volume: 3 Issue: 6 Pages: 706-710
- DOI
  10.1002/ajoc.201402042
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-25293002
[Journal Article] 2. Synthesis of Functionalized Polycyclic Aromatic Compounds via a Formal [2+2]-cycloaddition2014
- Author(s)
  Nagamoto, Y.; Yamaoka, Y.; Fujimura, S.; Takemoto, Y.; Takasu, K
- Journal Title
  
  Org. Lett.
  
  Volume: 16 Issue: 3 Pages: 1008-1011
- DOI
  10.1021/ol403757e
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24106719, KAKENHI-PROJECT-24659003, KAKENHI-PROJECT-25293002
[Journal Article] 5. Synthesis of 2,3,4,5-Tetra-substituted Pyrroles via a Base-Promoted Double Michael Reaction of Oxime-enoates with Nitroolefins2013
- Author(s)
  Kuroda, Y.; Imaizumi, K.; Yamada, K.; Yamaoka, Y.; Takasu, K.
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 54 Issue: 31 Pages: 4073-4075
- DOI
  10.1016/j.tetlet.2013.05.100
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24106719, KAKENHI-PROJECT-24790011, KAKENHI-PROJECT-25293002
[Journal Article] Enhanced Rate and Selectivity by Carboxylate Salt as a Basic Co-catalyst in Chiral N-Heterocyclic Carbene-Catalyzed Asymmetric Acylation of Secondary Alcohols.2013
- Author(s)
  K. Yamada
- Journal Title
  
  J. Am. Chem. Soc.
  
  Volume: 135 Issue: 31 Pages: 11485-11488
- DOI
  10.1021/ja4055838
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24790011, KAKENHI-PROJECT-25293002
[Presentation] 高酸化ジテルペンprovidencinの右セグメント合成研究2023
- Author(s)
  山岡庸介，西名亮，高須清誠
- Organizer
  日本薬学会　第143年会
- Data Source
  KAKENHI-PROJECT-21K05069
[Presentation] イノラートを用いた(2+2)環化付加によるシクロブテンのフロー合成2023
- Author(s)
  山岡庸介，浪岡雅樹，永木愛一郎，高須清誠
- Organizer
  日本薬学会　第143年会
- Data Source
  KAKENHI-PROJECT-21K05069
[Presentation] リチウムイノラートとα，β-不飽和カルボニル化合物との（2+2）環化付加反応のフロー法への応用2022
- Author(s)
  山岡庸介，浪岡雅樹，永木愛一郎，高須清誠
- Organizer
  日本プロセス化学会２０２２サマーシンポジウム
- Data Source
  KAKENHI-PROJECT-21K05069
[Presentation] マイクロフロー法でのリチウムイノラートとα,β-不飽和カルボニル化合物との (2+2) 環化付加反応によるシクロブテン合成2022
- Author(s)
  山岡庸介，浪岡雅樹，永木愛一郎，高須清誠
- Organizer
  第72回　日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-21K05069
[Presentation] 抗腫瘍活性ジテルペンprovidencin右セグメントの合成研究2022
- Author(s)
  山岡庸介，西名亮，高須清誠
- Organizer
  第72回　日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-21K05069
[Presentation] イナミドへの連続付加を用いたスピロインドリン合成2020
- Author(s)
  山岡庸介、山﨑大資、梶原大悟、瀧川紘、高須清誠
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] イナミドへの連続付加を用いたスピロインドリン合成2020
- Author(s)
  山岡庸介、山﨑大資、梶原大悟、瀧川紘、高須清誠
- Organizer
  第71回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] カリウム塩基を用いる分子内エノラート－オレフィンメタセシス2020
- Author(s)
  杉本和馬、紀之内颯、藤村駿、宮川泰典、山田健一、瀧川紘、山岡庸介、高須清誠
- Organizer
  第18回次世代を担う有機化学シンポジウム
- Data Source
  KAKENHI-PROJECT-19H03350
[Presentation] イナミドへの連続付加を用いたスピロインドリン合成2020
- Author(s)
  山岡庸介、山﨑大資、梶原大悟、瀧川紘、高須清誠
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] Helical Graphene Nanoribbons Embedded Polyazulene Framework2020
- Author(s)
  Naoki Ogawa, Yousuke Yamaoka, Hiroshi Takikawa, Kiyosei Takasu
- Organizer
  6th International Symposium on Middle Molecular Strategy (ISMMS-6)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19H03350
[Presentation] エンイナミドの連続環化反応による多環性キノリンの合成研究2019
- Author(s)
  山﨑大資、瀧川紘、山岡庸介、高須清誠
- Organizer
  第８６回日本分析化学会有機微量分析研究懇談会、第１１０回計測自動制御学会力学量計測部会、第３６回合同シンポジウム
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] オキサプロペランを用いる多環式スピロ化合物の合成法開発2019
- Author(s)
  小川直希、山岡庸介、瀧川紘、高須清誠
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-19H03350
[Presentation] イナミドの連続環化反応を利用した多環性キノリンの合成2019
- Author(s)
  山崎大資、山岡庸介、瀧川紘、高須清誠
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] Synthesis and Properties of Tribenzocarbazoles via an Acid Promoted Retro (2+2)-Cycloaddition of Azapropellanes2018
- Author(s)
  Naoki Ogawa, Yousuke Yamaoka. Hiroshi Takikawa, Kiyosei Takasu
- Organizer
  International Symposium on Main Group Chemistry Directed towards Organic Synthesis (MACOS)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] 植物の成長を制御するプロトイルダン類の合成2018
- Author(s)
  下田和摩、山岡庸介、瀧川紘、山田健一、高須清誠
- Organizer
  第60回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] 電子環状反応を利用したtrans-シクロアルケンの新規合成法とその応用2018
- Author(s)
  伊藤智裕, 堤正貴, 瀧川紘, 山田健一, 山岡庸介, 高須清誠
- Organizer
  モレキュラーキラリティ2018
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] エン-イナミドを用いた含窒素複素環の合成法の開発と応用2018
- Author(s)
  山岡庸介、山崎大資、篠崎麻紀子、武内奈央、山田健一、瀧川紘、高須清誠
- Organizer
  第44回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] ブレンステッド酸によるイナミドの分子内スピロ環化反応の開発2018
- Author(s)
  山岡庸介、山﨑大資、篠﨑麻紀子、山田健一、瀧川紘、高須清誠
- Organizer
  第68回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] イナミドとの連続反応によるスピロインドリン骨格の構築2018
- Author(s)
  山岡庸介、山崎大資、篠崎麻紀子、山田健一、瀧川紘、高須清誠
- Organizer
  第38回有機合成若手セミナー
- Data Source
  KAKENHI-PROJECT-18K05103
[Presentation] Total Synthesis of Echinocidin D by Using Lewis Acid Catalyzed [2+2] Cycloaddition2017
- Author(s)
  Kazuma Shimoda, Yousuke Yamaoka, Hiroshi Takikawa, Ken-ichi Yamada, Kiyosei Takasu
- Organizer
  The Eleventh International Symposium on Integrated Synthesis（ISONIS-11）
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] イナミドを用いた新規スピロインドリン合成法の開発2017
- Author(s)
  山岡庸介、山崎大資、篠崎麻紀子、山田健一、瀧川紘、高須清誠
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-16K18842
[Presentation] An Arylative Ring Expansion Cascade of Fused Cyclobutenes2017
- Author(s)
  Norihito Arichi, Yousuke Yamaoka, Ken-ichi Yamada, Kiyosei Takasu
- Organizer
  26th ISHC Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] 植物成長活性を有するmelleolideの合成研究2017
- Author(s)
  下田和摩、山岡庸介、山田健一、高須清誠
- Organizer
  創薬懇話会2017
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] エン‐イナミドを用いた含窒素複素環の簡便合成法の開発と応用2017
- Author(s)
  山岡庸介，吉田琢紘，篠崎麻紀子，武内奈央，山田健一，高須清誠
- Organizer
  第42回反応と合成の進歩シンポジウム
- Place of Presentation
  静岡市清水文化会館マリナート
- Year and Date
  2017-11-07
- Data Source
  KAKENHI-PROJECT-16K18842
[Presentation] イナミドを用いた含窒素複素環合成2017
- Author(s)
  山岡庸介
- Organizer
  第3回近畿薬学シンポジウム：化学系の若い力
- Invited
- Data Source
  KAKENHI-PROJECT-16K18842
[Presentation] エン-イナミドを用いたスピロインドール合成法の開発2016
- Author(s)
  山岡庸介、篠崎麻紀子、山田健一、高須清誠
- Organizer
  第64回日本薬学会近畿支部総会
- Place of Presentation
  大阪薬科大学
- Data Source
  KAKENHI-PROJECT-16K18842
[Presentation] Synthesis of Medium-sized trans-Cycloalkenes by Domino 4p-Electrocyclization－Alkylation of Fused Cyclobutenes2016
- Author(s)
  Tomohiro Ito, Ken-ichi Yamada, Yousuke Yamaoka, Kiyosei Takasu
- Organizer
  The Tenth International Symposium on Integrated Synthesis（ISONIS-10）
- Place of Presentation
  Awaji Umebutai
- Year and Date
  2016-11-18
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] Asymmetric Synthesis of Medium-Sized Ring Compounds via Short-Lived Cycloalkadiene Intermediates Based on Memory of Chirality Strategy2016
- Author(s)
  Norihito Arichi, Tomohiro Ito, Ken-ichi Yamada, Yousuke Yamaoka, Kiyosei Takasu
- Organizer
  Molecular Chirality Asia 2016
- Place of Presentation
  Osaka
- Year and Date
  2016-04-20
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05073
[Presentation] Efficient Synthesis of Nitrogen-containing Medium Rings with Ynamides2015
- Author(s)
  Yousuke Yamaoka, Nao Takeuchi, Ken-ichi Yamada, Kiyosei Takasu
- Organizer
  The 25th ISHC Congress
- Place of Presentation
  Santa Barbara, USA
- Year and Date
  2015-08-23
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] 面性不斉短寿命中間体を経由する縮環シクロブテンの環拡大反応2015
- Author(s)
  有地法人、山田健一、山岡庸介、高須清誠
- Organizer
  Symposium on Molecular Chirality 2015
- Place of Presentation
  早稲田大学西早稲田キャンパス
- Year and Date
  2015-06-22
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] Total Synthesis and Structural Revision of Paesslerin A2015
- Author(s)
  Yuzo Mogi, Ken-ichi Yamada, Yousuke Yamaoka, Kiyosei Takasu
- Organizer
  International Symposium of the Phytochemical Society of Asia 2015 (ISPSA2015) TOKUSHIMA
- Place of Presentation
  Tokushima Bunri University
- Year and Date
  2015-08-30
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] Total Synthesis of Paesslerin A2015
- Author(s)
  Yuzo Mogi, Kazato Inanaga, Takayuki Ishii, Hidetoshi Tokuyama, Masataka Ihara, Yousuke Yamaoka, Ken-ichi Yamada, Kiyosei Takasu
- Organizer
  The 39th Naito Conference「The chemistry of organocatalysts　有機分子触媒の化学」
- Place of Presentation
  シャトレーゼ　ガトーキングダム　サッポロ
- Year and Date
  2015-07-06
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] イナミドを用いた効率的中員環合成法の開発2014
- Author(s)
  山岡庸介、武内菜央、山田健一、高須清誠
- Organizer
  日本薬学会年会
- Place of Presentation
  熊本
- Data Source
  KAKENHI-PROJECT-25860006
[Presentation] イナミドを用いた中員環の効率的合成法の開発2014
- Author(s)
  山岡庸介、武内菜央、山田健一、高須清誠
- Organizer
  第６４回日本薬学会近畿支部総会
- Place of Presentation
  京都
- Year and Date
  2014-10-11
- Data Source
  KAKENHI-PROJECT-25860006
[Presentation] パラジウム触媒を用いた縮環シクロブテンのアリール化を伴う環拡大反応2014
- Author(s)
  有地法人、山田健一、山岡庸介、高須清誠
- Organizer
  第34回有機合成若手セミナー
- Place of Presentation
  大阪大学豊中キャンパス
- Year and Date
  2014-08-05
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] Marinoquinoline 類および aplidiopsamine A の全合成2013
- Author(s)
  山岡庸介、吉田琢紘、山田健一、高須清誠
- Organizer
  日本薬学会近畿支部大会
- Place of Presentation
  同志社女子大学
- Data Source
  KAKENHI-PROJECT-25860006
[Presentation] 多成分連続反応を利用する抗腫瘍活性テルペンPaesslerin Aの全合成
- Author(s)
  茂木雄三、稲永風人、石井崇之、徳山英利、井原正隆、山岡庸介、山田健一、高須清誠
- Organizer
  第56回天然有機化合物討論会
- Place of Presentation
  高知県立県民文化ホール・三翠園
- Year and Date
  2014-10-15 – 2014-10-17
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] 縮環シクロブタノールの環縮小転位を利用したtylophorine類の合成
- Author(s)
  谷口麻里枝、山岡庸介、山田健一、高須清誠
- Organizer
  第44回複素環化学討論会
- Place of Presentation
  札幌市民ホール（北海道）
- Year and Date
  2014-09-10 – 2014-09-12
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] Synthesis of Steroid Derivatives Bearing a Small Ring for the Conformational Fixation of D-Ring Side Chain
- Author(s)
  Norihito Arichi, Kenji Hata, Yamada Ken-ichi, Yosuke Yamaoka, Kiyosei Takasu
- Organizer
  20th International Conference on Organic Synthesis
- Place of Presentation
  Budapest, Hungary
- Year and Date
  2014-06-29 – 2014-07-04
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] Synthesis of 2,3,4,5-tetra-substituted pyrroles via a base-promoted double Michael reaction of oxime-enoates
- Author(s)
  Yusuke Kuroda, Kazuto IMaizumi, Ken-ichi Yamada, Yousuke Yamaoka, Kiyosei Takasu
- Organizer
  20th International Conference on Organic Synthesis
- Place of Presentation
  Budapest, Hungary
- Year and Date
  2014-06-29 – 2014-07-04
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] TOTAL SYNTHESIS OF PAESSLERIN A
- Author(s)
  Yuzo Mogi, Kazato Inanaga, Takayuki Ishii, Hidetoshi Tokuyama, Masataka Ihara, Yousuke Yamaoka, Ken-ichi Yamada, Kiyosei Takasu
- Organizer
  8th Singapore International Chemistry Conference (SICC-8)
- Place of Presentation
  the University Town campus of NUS, Singapore
- Year and Date
  2014-12-14 – 2014-12-17
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] イナミドを用いたキノリン骨格の効率的合成法の開発と Aplidiopsamine A の全合成
- Author(s)
  山岡庸介、篠崎麻紀子、吉田琢紘、山田健一、高須清誠
- Organizer
  日本薬学会第１３５年会
- Place of Presentation
  神戸
- Year and Date
  2015-03-25 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-25860006
[Presentation] 縮環シクロブタノールを経る多環芳香族化合物の合成と反応機構
- Author(s)
  山岡庸介、藤村駿、永本祐樹、山田健一、高須清誠
- Organizer
  第25回基礎有機化学討論会
- Place of Presentation
  東北大学川内北キャンパス・萩ホール
- Year and Date
  2014-09-07 – 2014-09-09
- Data Source
  KAKENHI-PROJECT-25293002
[Presentation] 効率的縮環シクロブタノール合成と多環芳香族炭化水素への応用
- Author(s)
  山岡庸介、藤村駿、永本祐樹、岸田明日美、山田健一、竹本佳司、高須清誠
- Organizer
  第12回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール（東京）
- Year and Date
  2014-05-23 – 2014-05-24
- Data Source
  KAKENHI-PROJECT-25293002

1. TAKASU KIYOSEI (10302168)

# of Collaborated Projects: 3 results

# of Collaborated Products: 37 results
2. HATTORI Akira (50300893)

# of Collaborated Projects: 3 results

# of Collaborated Products: 0 results
3. Shimoda Kazuma

# of Collaborated Projects: 1 results

# of Collaborated Products: 3 results
4. Ito Tomohiro

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
5. Ogawa Naoki

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
6. Tsutsumi Masaki

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
7. TAKIKAWA Hiroshi

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
8. 山田健一

# of Collaborated Projects: 0 results

# of Collaborated Products: 7 results
9. 新藤充

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
10. 鍬野哲

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

Yamaoka Yousuke 山岡 庸介

YAMAOKA Yousuke 山岡 庸介

Research Projects

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Co-Researchers

Efficient Synthesis of Cyclobutanes by Multicomponent Reaction Using Ynolates and Its Application for Drug DiscoveryPrincipal Investigator

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formation of carbon four-membered rings using ynolate and its application for drug discoveryPrincipal Investigator

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Design, Synthesis and Evaluation of Biologically Active Molecules Based on Ring Strain

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Divergent Synthesis of Nitrogen-Containing Heterocycles by Sequential Reactions and Its Application to Drug DiscoveryPrincipal Investigator

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Efficient synthesis of nitrogen-containing compounds with yanamidesPrincipal Investigator

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Stereocontrolled synthesis of poly-substituted medium-sized cyclic compounds by electrocyclic ring opening reaction and the synthesis of biologically active molecules

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Discovery of new reactions and utilities of 4-membered carbocyles based on their unique ring strains.

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Development of a Bronsted Acid-Promoted Ene-Ynamide CyclizationPrincipal Investigator

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[Book] Methods and Applications of Cycloaddition Reactions in Organic Syntheses2014

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[Journal Article] Entry into Lithium Ynolates from α,α,α-Tribromomethyl Ketones: Synthesis of Cyclobutenes via the [2 + 2] Cycloaddition with α,β-Unsaturated Carbonyls2024

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[Journal Article] Total Synthesis of Cryptopleurine and Its Analogues2022

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[Journal Article] Oxidative β-Cleavage of Fused Cyclobutanols Leading to Hydrofuran-Fused Polycyclic Aromatic Compounds2021

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[Journal Article] Synthesis of Lactone-fused Cyclopropanes by Ring Contractive-Ketol Rearrangement of Ketal-Fused Cyclobutanones2021

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[Journal Article] Total Synthesis of (-)-Sigillin A: A Polychlorinated and Polyoxygenated Natural Product2020

Author(s)

Yamaoka Yousuke 山岡庸介

YAMAOKA Yousuke 山岡庸介