Hirashima Shinichi 平島真一

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Hirashima Shin-ichi 平島真一

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Researcher Number	80642264
Other IDs
Affiliation (Current)	2025: 東京薬科大学, 薬学部, 准教授
Affiliation (based on the past Project Information) *help	2021 – 2023: 東京薬科大学, 薬学部, 准教授 2018 – 2020: 東京薬科大学, 薬学部, 講師 2016 – 2017: 東京薬科大学, 薬学部, 助教
Review Section/Research Field	Principal Investigator Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related Except Principal Investigator Chemical pharmacy
Keywords	Principal Investigator ヒドロホスフィニル化反応 / リンカルコゲニド化合物 / 不斉プロトン化反応 / ビシナルビスホスフィン誘導体 / リンカルコゲニド類 / 第二級ホスフィンカルコゲニド / ヒドロホスホニル化反応 / β-アミノホスフィン誘導体 / 第二級ホスフィンスルフィド / 不斉ヒドロホスフィニル化反応 / 光学活性有機リン化合物 … More Except Principal Investigator … More 薬学 / 触媒・化学プロセス / 有機化学 / 不斉反応 / 有機触媒 Less

求核部位選択性を鍵とする多彩なリンカルコゲニド類の合成展開Principal Investigator
- Principal Investigator
  
  平島真一
- Project Period (FY)
  2022 – 2024
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Tokyo University of Pharmacy and Life Science
Synthesis of chiral phosphorous compounds utilizing sulfurPrincipal Investigator
- Principal Investigator
  
  Hirashima Shin-ichi
- Project Period (FY)
  2019 – 2021
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Tokyo University of Pharmacy and Life Science
Development of novel push-pull ethylene organocatalysts and their application to synthesis of medicines
- Principal Investigator
  
  Miura Tsuyoshi
- Project Period (FY)
  2016 – 2018
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Tokyo University of Pharmacy and Life Science

All 2024 2023 2022 2021 2020 2019 2018 2017 2016

All Journal Article Presentation

[Journal Article] Regioselective One-Pot Synthesis of Vicinal Bisphosphine Derivatives from Nitroalkenes by Hydrophosphinylation/Elimination/Hydrophosphinylation2024
- Author(s)
  Hirota Eiki、Hirashima Shin-ichi、Morita Ryuki、Takase Junya、Matsushima Yasuyuki、Nakashima Kosuke、Akutsu Hiroshi、Miura Tsuyoshi
- Journal Title
  
  Organic Letters
  
  Volume: 26 Issue: 9 Pages: 1797-1802
- DOI
  10.1021/acs.orglett.3c04297
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510
[Journal Article] Synthesis of 2-Substituted Indoles via Migration Reaction of 3-Substituted Indoles with Triflic Acid2024
- Author(s)
 Nakashima Kosuke、Kudo Yuka、Matsushima Yasuyuki、Hirashima Shin-ichi、Miura Tsuyoshi
- Journal Title
 
 Chemical and Pharmaceutical Bulletin
 
 Volume: 72 Issue: 3 Pages: 336-339
- DOI
 10.1248/cpb.c23-00792
- ISSN
 0009-2363, 1347-5223
- Year and Date
 2024-03-25
- Language
 English
- Peer Reviewed
- Data Source
 KAKENHI-PROJECT-22K06510
[Journal Article] Fluorescent Rotary Switches: Four- vs Three-Substituted Phthalimide Boron Difluoride Schiff Base Complexes2023
- Author(s)
  Yordanov Dancho、Smolka Rastislav、Nakashima Kosuke、Hirashima Shin-ichi、Matsushima Yasuyuki、Vala Martin、Kraj?ovi? Jozef、Weiter Martin、Miura Tsuyoshi、Georgiev Anton
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 88 Issue: 24 Pages: 17206-17214
- DOI
  10.1021/acs.joc.3c02056
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-22K06510
[Journal Article] Vicinal All‐Carbon Quaternary Stereocenter Construction with Trifluoromethyl Groups via Organocatalytic Asymmetric Cascade Michael/Michael Reaction2023
- Author(s)
  Tsuyusaki Ryo、Nakashima Kosuke、Matsushima Yasuyuki、Hirashima Shin‐ichi、Miura Tsuyoshi
- Journal Title
  
  Chemistry ? An Asian Journal
  
  Volume: 19 Issue: 1
- DOI
  10.1002/asia.202300931
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510
[Journal Article] Highly efficient, asymmetric, and organocatalyst-based Henry reactions between α,β-unsaturated trifluoromethyl ketone and nitromethane2023
- Author(s)
  Tsuyusaki Ryo、Nakashima Kosuke、Shimomura Miki、Kawada Masahiro、Matsushima Yasuyuki、Hirashima Shin-ichi、Miura Tsuyoshi
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 117 Pages: 154375-154375
- DOI
  10.1016/j.tetlet.2023.154375
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510, KAKENHI-PROJECT-20K06948
[Journal Article] Catalytic Synthesis of Phthalide Derivatives via Asymmetric Bromolactonization of Stilbene‐type Carboxylic Acids usingN,N‐Dibenzyl Diaminomethylenemalononitrile as Organocatalyst2023
- Author(s)
 Matsushima Yasuyuki、Fukuda Shunsuke、Kobayashi Yusuke、Nezu Hiroyasu、Nakashima Kosuke、Hirashima Shin‐ichi、Miura Tsuyoshi
- Journal Title
 
 Asian Journal of Organic Chemistry
 
 Volume: 12 Issue: 7
- DOI
 10.1002/ajoc.202300254
- Peer Reviewed
- Data Source
 KAKENHI-PROJECT-22K06510
[Journal Article] Asymmetric Direct Vinylogous Conjugate Addition of α,β‐Unsaturated γ‐Butyrolactam to Acyl Acrylonitriles using Organocatalysts2023
- Author(s)
  Ishii Daiki、Hirashima Shin‐ichi、Nakashima Kosuke、Matsushima Yasuyuki、Sakai Takaaki、Akutsu Hiroshi、Miura Tsuyoshi
- Journal Title
  
  Asian Journal of Organic Chemistry
  
  Volume: － Issue: 5
- DOI
  10.1002/ajoc.202300082
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510, KAKENHI-PROJECT-20K06948
[Journal Article] Organocatalyzed Synthesis of Bicyclic γ‐Lactam Derivatives via Asymmetric Conjugate Addition of Cyclic β‐Keto Esters to Benzoyl Acrylonitriles2023
- Author(s)
  Matsushima Yasuyuki、Kubokawa Satsuki、Watanabe Mia、Nakashima Kosuke、Hirashima Shin‐ichi、Miura Tsuyoshi
- Journal Title
  
  Asian Journal of Organic Chemistry
  
  Volume: 13 Issue: 2
- DOI
  10.1002/ajoc.202300620
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510
[Journal Article] Asymmetric Friedel?Crafts Alkylation of Indoles with α,β‐unsaturated Trifluoromethyl Ketones Using a Squaramide Organocatalyst2022
- Author(s)
  Nakashima Kosuke、Hanamura Sumire、Imamura Aoi、Matsushima Yasuyuki、Hirashima Shin‐ichi、Miura Tsuyoshi
- Journal Title
  
  Asian Journal of Organic Chemistry
  
  Volume: 11 Issue: 10
- DOI
  10.1002/ajoc.202200403
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510, KAKENHI-PROJECT-20K06948
[Journal Article] Solvent-Triggered Long-Range Proton Transport in 7-Hydroxyquinoline Using a Sulfonamide Transporter Group2022
- Author(s)
  Nakashima Kosuke、Georgiev Anton、Yordanov Dancho、Matsushima Yasuyuki、Hirashima Shin-ichi、Miura Tsuyoshi、Antonov Liudmil
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 87 Issue: 10 Pages: 6794-6806
- DOI
  10.1021/acs.joc.2c00494
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510
[Journal Article] Asymmetric Direct Vinylogous Conjugate Addition of Substituted Furanone Derivatives to ( E )‐ and ( Z) ‐Benzoyl Acrylonitriles Using Organocatalysts2022
- Author(s)
 Ishii Daiki、Hirashima Shin‐ichi、Akutsu Hiroshi、Nakashima Kosuke、Matsushima Yasuyuki、Sakai Takaaki、Miura Tsuyoshi
- Journal Title
 
 Asian Journal of Organic Chemistry
 
 Volume: - Issue: 5
- DOI
 10.1002/ajoc.202200048
- Peer Reviewed
- Data Source
 KAKENHI-PROJECT-19K07002, KAKENHI-PROJECT-20K06948
[Journal Article] Synthesis of Chiral α‐Substituted β‐Aminophosphine Derivatives through Asymmetric Hydrophosphinylation Utilizing Secondary Phosphine Sulfides2022
- Author(s)
  Hirashima Shin‐ichi、Hirota Eiki、Matsushima Yasuyuki、Noda Naoki、Nishimura Yuya、Narushima Takefumi、Nakashima Kosuke、Miura Tsuyoshi
- Journal Title
  
  Chemistry ? An Asian Journal
  
  Volume: 17 Issue: 24
- DOI
  10.1002/asia.202200989
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510, KAKENHI-PROJECT-20K06948
[Journal Article] Asymmetric conjugate addition?cyclization of cyclohexane-1,2-dione with alkylidenemalononitriles using diaminomethylenemalononitrile organocatalyst2022
- Author(s)
  Matsushima Yasuyuki、Iino Yuta、Tsuruta Yuka、Nakashima Kosuke、Hirashima Shin-ichi、Miura Tsuyoshi
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 97 Pages: 153773-153773
- DOI
  10.1016/j.tetlet.2022.153773
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K06510, KAKENHI-PROJECT-20K06948
[Journal Article] Organocatalytic one-pot asymmetric synthesis of 6-trifluoromethyl-substituted 7,8-dihydrochromen-6-ol2022
- Author(s)
  K. Nakashima, A. Minai, Y. Okuaki, Y. Matsushima, S. Hirashima, T. Miura
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 95 Pages: 153733-153733
- DOI
  10.1016/j.tetlet.2022.153733
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K06948, KAKENHI-PROJECT-22K06510
[Journal Article] Asymmetric Henry Reaction of Trifluoromethyl Enones with Nitromethane Using a N,N ‐Dibenzyl Diaminomethylenemalononitrile Organocatalyst2022
- Author(s)
 Kawada Masahiro、Tsuyusaki Ryo、Nakashima Kosuke、Yamada Misaki、Kozakai Akihiro、Matsushima Yasuyuki、Hirashima Shin‐ichi、Miura Tsuyoshi
- Journal Title
 
 Chemistry - An Asian Journal
 
 Volume: 17 Issue: 4
- DOI
 10.1002/asia.202101299
- Peer Reviewed
- Data Source
 KAKENHI-PROJECT-19K07002, KAKENHI-PROJECT-20K06948
[Journal Article] Diaminomethylenemalononitrile as a Chiral Single Hydrogen Bond Catalyst: Application to Enantioselective Conjugate Addition of α‐Branched Aldehydes2021
- Author(s)
  Kawada Masahiro、Tsuyusaki Ryo、Nakashima Kosuke、Akutsu Hiroshi、Hirashima Shin‐ichi、Matsumoto Takashi、Yanai Hikaru、Miura Tsuyoshi
- Journal Title
  
  Chemistry- An Asian Journal
  
  Volume: 16 Issue: 16 Pages: 2272-2275
- DOI
  10.1002/asia.202100487
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07002, KAKENHI-PROJECT-20K06948
[Journal Article] Acylhydrazone Subunits as a Proton Cargo Delivery System in 7‐Hydroxyquinoline2021
- Author(s)
  Nakashima Kosuke、Petek Anton、Hori Yutaro、Georgiev Anton、Hirashima Shin‐ichi、Matsushima Yasuyuki、Yordanov Dancho、Miura Tsuyoshi、Antonov Liudmil
- Journal Title
  
  Chemistry - A European Journal
  
  Volume: 27 Issue: 45 Pages: 11559-11566
- DOI
  10.1002/chem.202101650
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-19K07002
[Journal Article] Asymmetric Conjugate Addition of Phosphonates to Enones Using Cinchona?Diaminomethylenemalononitrile Organocatalysts2020
- Author(s)
  Arai Ryoga、Hirashima Shin-ichi、Nakano Tatsuki、Kawada Masahiro、Akutsu Hiroshi、Nakashima Kosuke、Miura Tsuyoshi
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 85 Issue: 5 Pages: 3872-3878
- DOI
  10.1021/acs.joc.9b02553
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07002
[Journal Article] Asymmetric Direct Vinylogous Conjugate Addition of Substituted Furanone Derivatives to Benzoyl Acrylonitrile: Stereoselective Synthesis Toward Bicyclic γ-Lactams2020
- Author(s)
  Ishii Daiki、Hirashima Shin-ichi、Nakashima Kosuke、Akutsu Hiroshi、Sakai Takaaki、Matsushima Yasuyuki、Kawada Masahiro、Miura Tsuyoshi
- Journal Title
  
  Organic Letters
  
  Volume: 23 Issue: 2 Pages: 480-485
- DOI
  10.1021/acs.orglett.0c04004
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07002, KAKENHI-PROJECT-20K06948
[Journal Article] Asymmetric Conjugate Addition of α-Cyanoketones to Benzoyl Acrylonitrile Derivatives Using a Diaminomethylenemalononitrile Organocatalyst2020
- Author(s)
  Akutsu Hiroshi、Nakashima Kosuke、Kanetsuna Yuta、Kawada Masahiro、Hirashima Shin-ichi、Miura Tsuyoshi
- Journal Title
  
  Synthesis
  
  Volume: 52 Issue: 24 Pages: 3874-3880
- DOI
  10.1055/s-0040-1707285
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07002, KAKENHI-PROJECT-20K06948
[Journal Article] Highly efficient asymmetric conjugate addition of 5-benzylfurfurals to nitroalkenes using a thiourea organocatalyst2019
- Author(s)
  H. Akutsu, K. Nakashima, S. Hirashima, H. Matsumoto, Y. Koseki, T. Miura
- Journal Title
  
  Tetrahedron
  
  Volume: 75 Issue: 16 Pages: 2431-2435
- DOI
  10.1016/j.tet.2019.03.013
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Synthesis of chiral γ,γ-disubstituted γ-butenolides via direct vinylogous aldol reaction of substituted furanone derivatives with aldehydes2019
- Author(s)
  T. Sakai, S. Hirashima, Y. Matsushima, T. Nakano, D. Ishii, Y. Yamashita, K. Nakashima,
- Journal Title
  
  Org. Lett.
  
  Volume: 21 Issue: 8 Pages: 2606-2609
- DOI
  10.1021/acs.orglett.9b00574
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] 持続社会に応えうる高機能性水素結合供与型有機分子触媒の開発2018
- Author(s)
  平島真一，中島康介，三浦　剛
- Journal Title
  
  ファルマシア (Farumashia)
  
  Volume: 54 Pages: 938-942
- NAID
  130007494724
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Cinchona-iaminomethylenemalononitrile Organocatalyst for the Highly Enantioselective Hydrophosphonylation of Ketones and Enones2018
- Author(s)
  Arai Ryoga、Hirashima Shin-ichi、Kondo Junko、Nakashima Kosuke、Koseki Yuji、Miura Tsuyoshi
- Journal Title
  
  Organic Letters
  
  Volume: 20 Issue: 18 Pages: 5569-5572
- DOI
  10.1021/acs.orglett.8b02241
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Stereoselective conjugate addition of Ketones to Alkylidene Malonates using Thiourea-Sulfonamide organocatalyst2018
- Author(s)
  M. Kawada, K. Nakashima, S. Hirashima, T. Sakagami, Y. Koseki, T. Miura
- Journal Title
  
  Chirality
  
  Volume: 30 Issue: 11 Pages: 1515-1224
- DOI
  10.1002/chir.23015
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Asymmetric conjugate addition of α-cyanoketones to enones using diaminomethylenemalononitrile organocatalyst2018
- Author(s)
  K. Nakashima, Y. Noda, S. Hirashima, Y. Koseki, T. Miura
- Journal Title
  
  J. Org. Chem.
  
  Volume: 83 Issue: 4 Pages: 2402-2408
- DOI
  10.1021/acs.joc.7b02976
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Asymmetric Conjugate Addition of Nitroalkanes to Enones Using a Sulfonamide-thiourea Organocatalyst2017
- Author(s)
  M. Kawada, K. Nakashima, S. Hirashima, A. Yoshida, Y. Koseki, T. Miura
- Journal Title
  
  J. Org. Chem.
  
  Volume: 82 Issue: 13 Pages: 6986-6991
- DOI
  10.1021/acs.joc.7b00835
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Asymmetric conjugate addition of 5-benzylfurfurals to nitroalkenes using a diaminomethylenemalononitrile organocatalyst2017
- Author(s)
  H. Akutsu, K. Nakashima, S. Hirashima, M. Kitahara, Y. Koseki, T. Miura
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 58 Issue: 51 Pages: 4759-4762
- DOI
  10.1016/j.tetlet.2017.10.078
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Design of Novel Hydrogen-bonding Donor Organocatalysts and Their Application to Asymmetric Direct Aldol Reaction2017
- Author(s)
  H. Akutsu, K. Nakashima, H. Yanai, A. Kotani, S. Hirashima, T. Yamamoto, R. Takahashi, A. Yoshida, Y. Koseki, H. Hakamata, T. Matsumoto, T. Miura
- Journal Title
  
  Synlett
  
  Volume: 28 Issue: 11 Pages: 1363-1367
- DOI
  10.1055/s-0036-1558971
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178, KAKENHI-PROJECT-17K08224
[Journal Article] Squaramide-sulfonamide organocatalyst for asymmetric direct vinylogous aldol reactions2017
- Author(s)
  T. Sakai, S. Hirashima, Y. Yamashita, R. Arai, K. Nakashima, A. Yoshida, Y. Koseki, T. Miura,
- Journal Title
  
  J. Org. Chem
  
  Volume: 82 Issue: 9 Pages: 4661-4667
- DOI
  10.1021/acs.joc.7b00287
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K18838, KAKENHI-PROJECT-16K08178
[Journal Article] Asymmetric Conjugate Additions of Carbonyl Compounds to Nitroalkenes under Solvent-Free Conditions Using Fluorous Diaminomethylenemalononitrile Organocatalyst2017
- Author(s)
  S. Hirashima, T. Narushima, M. Kawada, K. Nakashima, K. Hanai, Y. Koseki, T. Miura
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 65 Issue: 12 Pages: 1185-1190
- DOI
  10.1248/cpb.c17-00596
- NAID
  130006235020
- ISSN
  0009-2363, 1347-5223
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Stereoselective conjugate addition of carbonyl compounds to maleimides using diaminomethyleneindenedione organocatalyst2016
- Author(s)
  Kosuke Nakashima, Masahiro Kawada, Shin-ichi Hirashima, Ayako Kosugi, Mana Kato,　Akihiro Yoshida, Yuji Koseki, Tsuyoshi Miura
- Journal Title
  
  Tetrahedron: Asymmetry
  
  Volume: 27 Issue: 17-18 Pages: 888-895
- DOI
  10.1016/j.tetasy.2016.07.002
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-16K08178
[Journal Article] Asymmetric Chlorination of β-Keto Esters Using Diaminomethylenemalononitrile Organocatalyst2016
- Author(s)
  Takaaki Sakai, Shin-ichi Hirashima, Kosuke Nakashima, Chie Maeda, Akihiro Yoshida, Yuji Koseki, Tsuyoshi Miura
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 64 Issue: 12 Pages: 1781-1784
- DOI
  10.1248/cpb.c16-00722
- NAID
  130005170646
- ISSN
  0009-2363, 1347-5223
- Language
  English
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] カルコゲンホスフィン酸を用いるアジリジンの不斉開環反応に関する研究2023
- Author(s)
  藤野亮, 平島真一, 壹岐朋佳, 馬場拓希, 野田直輝, 中島康介, 松島恭征, 三浦　剛
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 第二級ホスフィンスルフィドを用いた有機強塩基触媒による不斉プロトン化反応の開発2023
- Author(s)
  廣田瑛紀、平島真一、忠末千佳、鈴木杏奈、中島康介、松島恭征、三浦剛
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 有機分子触媒を用いた不斉ブロモラクトン化反応によるフタリド誘導体の合成2023
- Author(s)
  松島恭征、福田駿介、小林雄介、根津宏康、中島康介、平島真一、三浦剛
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 有機分子触媒を用いた高立体選択的トリフルオロメチル基含有スピロオキシインドールの合成2023
- Author(s)
  露崎龍、中島康介、松島恭征、平島真一、三浦剛
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] インドール環上におけるアルキル基転位反応に関する研究2023
- Author(s)
  中島康介、工藤夕加、松島恭征、平島真一、三浦剛
- Organizer
  第67回　日本薬学会　関東支部大会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 有機分子触媒を用いたトリフルオロメチルエノンへの高立体選択的なヘンリー反応の開発2023
- Author(s)
  露崎　龍、下村　実希、河田　雅宏、中島　康介、松島　恭征、平島　真一、三浦　剛
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 有機分子触媒を用いたフラン誘導体の位選択的不斉反応2023
- Author(s)
  阿久津裕士、玉井奎伍、敏蔭悠太郎、冨永涼太、中島康介、平島真一、吉田彰宏、三浦剛、山ノ井孝
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 第二級ホスフィンスルフィドをプロ求核剤とする不斉プロトン化反応の開発2023
- Author(s)
  廣田瑛紀、平島真一、忠末千佳、鈴木杏奈、中島康介、松島恭征、三浦剛
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 不斉共役付加反応を利用した2-アザビシクロ[3.3.0]オクタン誘導体の合成2023
- Author(s)
  松島恭征、窪川颯月、渡邉美亜、中島康介、平島真一、三浦剛
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 7-hydroxyquinolineにおけるacylhydrazoneによる分子内プロトン移動システム2022
- Author(s)
  中島康介、Petek Anton、堀祐太郎、Georgiev Anton、平島真一、松島恭征、Yordanov Dancho、三浦剛、Antonov Liudmil
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 有機分子触媒を用いた立体選択的スピロインドリン-3-オン誘導体の合成2022
- Author(s)
  中島康介、花村菫、今村碧、松島恭征、平島真一、三浦剛
- Organizer
  第66回　日本薬学会　関東支部大会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 第二級ホスフィンスルフィドを用いた光学活性有機リン化合物の効率的な合成法の開発2022
- Author(s)
  廣田瑛紀、平島真一、松島恭征、野田直輝、西村祐哉、成島岳史、中島康介、三浦剛
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 有機触媒を用いたトリフルオロメチルエノンへの高立体選択的ヘンリー反応2022
- Author(s)
  露崎龍、下村実希、河田雅宏、中島康介、松島恭征、平島真一、三浦剛
- Organizer
  医薬工三大学連携シンポジウム
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 酸化的スピロラクトン化によるキラルスピロオキシインドールの合成2022
- Author(s)
  奥秋祐壱、中島康介、松島恭征、平島真一、三浦剛
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] α,β-不飽和-γ-ブチロラクタムのβ-シアノエノンに対する不斉直截的ビニロガスマイケル付加反応2022
- Author(s)
  石井大暉、平島真一、坂井崇亮、中島康介、松島恭征、三浦剛
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 有機分子触媒を用いた不斉マイケル付加-環化反応による2-アミノ-4H-クロメン誘導体の合成2022
- Author(s)
  飯野雄太、松島恭征、鶴田悠夏、中島康介、平島真一、三浦剛
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] インドールとα,β-不飽和トリフルオロメチルケトンの不斉フリーデルクラフツアルキル化反応2022
- Author(s)
  今村碧、中島康介、花村菫、松島恭征、平島真一、三浦剛
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 新規ジアミノメチレンマロノニトリル触媒を用いたトリフルオロメチルエノンに対する不斉ヘンリー反応の開発2022
- Author(s)
  露崎龍、河田雅宏、中島康介、松島恭征、平島真一、三浦剛
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 持続可能社会の実現に向けた新規有機分子触媒の開発2022
- Author(s)
  平島真一
- Organizer
  CPhI/ICSE/P-MEC/bioLIVE/InnoPack/FDF/NEX Japan 2022
- Invited
- Data Source
  KAKENHI-PROJECT-22K06510
[Presentation] 新規キラル二環性γ-ラクタム誘導体の効率合成2021
- Author(s)
  石井大暉、平島真一、阿久津裕士、中島康介、松島恭征、坂井崇亮、三浦剛
- Organizer
  第47回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 不斉直接ビニロガス共役付加反応を利用した二環性γ-ラクタム誘導体の合成2021
- Author(s)
  石井大暉、平島真一、中島康介、阿久津裕士、坂井崇亮、松島恭征、河田雅宏、三浦剛
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] グリーンケミストリーを基盤とした有機分子触媒的不斉反応の開発2020
- Author(s)
  平島真一
- Organizer
  第64回日本薬学会関東支部大会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] ビシナルビスホスフィン誘導体の位置選択的ワンポット合成法の開発2020
- Author(s)
  廣田瑛紀、平島真一、森田龍輝、髙瀬純也、阿久津裕士、河田雅宏、中島康介、三浦　剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 不斉direct vinylogous Michael付加反応によるγ,γ-二置換 γ-ブテノリドの合成研究2020
- Author(s)
  石井大暉、平島真一、坂井崇亮、阿久津裕士、河田雅宏、中島康介、三浦　剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-19K07002
[Presentation] 有機分子触媒を用いたα-シアノケトンとβ-シアノエノンとの不斉共役付加反応2019
- Author(s)
  兼綱祐太、阿久津裕士、中島康介、栁沢紫苑、平島真一、古石裕治、三浦剛
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 第二級ホスフィンスルフィドを用いた不斉ホスファ‐マイケル付加反応の開発2019
- Author(s)
  藤野佑樹，平島真一，岡崎時夫，柴沼早希，中島康介，古石裕治，三浦剛
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 硫黄元素の特性を活かした不斉ヒドロホスフィニル化反応の開発2018
- Author(s)
  藤野佑樹，平島真一，柴沼早希，中島康介，古石裕治，三浦剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] フルオラス有機分子触媒を用いた不斉direct vinylogous aldol反応2018
- Author(s)
  松島恭征，坂井崇亮,　平島真一,　山下祥史,　中野　樹,　中島康介,　古石裕治,　三浦　剛
- Organizer
  フルオラス科学研究会第11回シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いたα,β-不飽和トリフルオロメチルケトンに対する不斉Henry反応の開発2018
- Author(s)
  河田雅宏, 中島康介, 山田美咲, 平島真一, 古石裕治，三浦剛
- Organizer
  第44回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 不斉 direct vinylogous aldol 反応によるγ,γ-二置換 γ-butenolideの合成研究2018
- Author(s)
  坂井崇亮,　平島真一,　山下祥史,　中野　樹,　中島康介,　古石裕治,　三浦　剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いたフラン誘導体の不斉ε位アルキル化反応2018
- Author(s)
  阿久津裕士，松本　光，中島康介，平島真一，古石裕治，三浦　剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] DMM型有機分子触媒を用いたフルフラール誘導体の不斉ε位アルキル化反応2018
- Author(s)
  阿久津裕士、中島康介、平島真一、古石裕治、三浦剛
- Organizer
  第44回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機触媒を用いた1,4-付加選択的不斉ヒドロホスホニル化反応の開発2018
- Author(s)
  新井　亮雅、平島　真一、中島　康介、古石　裕治、三浦　剛
- Organizer
  日本薬学会第62回関東支部大会シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いたα-シアノケトンのエノンへの不斉共役付加反応の開発2017
- Author(s)
  〇野田優太、中島康介、平島真一、古石裕治、三浦剛
- Organizer
  日本薬学会第137年会
- Place of Presentation
  東北大学
- Year and Date
  2017-03-25
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] スクアラミド-スルホンアミド有機触媒を用いた不斉direct vinylogous aldol 反応2017
- Author(s)
  坂井崇亮，平島真一，山下祥史，新井亮雅，中島康介，古石裕治，三浦剛
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いる不飽和ケトンに対する位置選択的不斉ヒドロホスホニル化反応の開発2017
- Author(s)
  新井　亮雅、平島　真一、中島　康介、古石　裕治、三浦　剛
- Organizer
  日本薬学会第61回関東支部大会シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] フルオラス有機分子触媒を用いた不斉ヒドロホスフィニル化反応2017
- Author(s)
  藤野　佑樹、平島　真一、成島　岳史、中島　康介、古石　裕治、三浦　剛
- Organizer
  フルオラス科学研究会第10回シンポジウム
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] ジアミノメチレンマロノニトリル型有機分子触媒を用いる不斉クロロ化反応の開発2017
- Author(s)
  〇坂井崇亮、平島真一、前田知恵、中島康介、吉田彰宏、古石裕治、三浦剛
- Organizer
  日本薬学会第137年会
- Place of Presentation
  東北大学
- Year and Date
  2017-03-25
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いた5-アルキルフルフラール誘導体の不斉ε位アルキル化反応2017
- Author(s)
  〇阿久津裕士、中島康介、平島真一、古石裕治、三浦剛
- Organizer
  日本薬学会第137年会
- Place of Presentation
  東北大学
- Year and Date
  2017-03-25
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] ケトン類に対する有機分子触媒的不斉ヒドロホスホニル化反応の開発2017
- Author(s)
  〇新井亮雅、平島真一、近藤純子、中島康介、古石裕治、三浦剛
- Organizer
  日本薬学会第137年会
- Place of Presentation
  東北大学
- Year and Date
  2017-03-25
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] スルホンアミドーチオウレア型有機分子触媒を用いた不斉反応2016
- Author(s)
  ◯河田雅宏、中島康介、平島真一、坂上徹、鈴木智博、野田優太、吉田彰宏、古石裕治、三浦剛
- Organizer
  第42回反応と合成の進歩シンポジウム
- Place of Presentation
  静岡市清水文化会館マリナート
- Year and Date
  2016-11-07
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] フルオラス有機分子触媒を用いたフラン誘導体の不斉アルキル化反応2016
- Author(s)
  ◯阿久津裕士、中島康介、平島真一、吉田彰宏、古石裕治、三浦剛
- Organizer
  フルオラス科学研究会第9回シンポジウム
- Place of Presentation
  名古屋大学
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 有機分子触媒を用いたカルボニル化合物のマレイミドへの不斉共役付加反応2016
- Author(s)
  ◯河田雅宏、中島康介、平島真一、小杉綾子、加藤真奈、吉田彰宏、古石裕治、三浦剛
- Organizer
  創薬懇話会2016
- Place of Presentation
  エクシブ蓼科
- Year and Date
  2016-06-30
- Data Source
  KAKENHI-PROJECT-16K08178
[Presentation] 新規有機分子触媒を用いた不斉Pudovik反応の開発2016
- Author(s)
  ○三浦剛、新井亮雅、平島真一、中島康介、古石裕治
- Organizer
  BIOtech 2016
- Place of Presentation
  東京ビッグサイト
- Year and Date
  2016-05-11
- Data Source
  KAKENHI-PROJECT-16K08178

1. Miura Tsuyoshi (40297023)

# of Collaborated Projects: 1 results

# of Collaborated Products: 30 results
2. 中島康介

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

Hirashima Shinichi 平島 真一

Hirashima Shin-ichi 平島 真一

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求核部位選択性を鍵とする多彩なリンカルコゲニド類の合成展開Principal Investigator

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Synthesis of chiral phosphorous compounds utilizing sulfurPrincipal Investigator

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Development of novel push-pull ethylene organocatalysts and their application to synthesis of medicines

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[Journal Article] Regioselective One-Pot Synthesis of Vicinal Bisphosphine Derivatives from Nitroalkenes by Hydrophosphinylation/Elimination/Hydrophosphinylation2024

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[Journal Article] Synthesis of 2-Substituted Indoles <i>via</i> Migration Reaction of 3-Substituted Indoles with Triflic Acid2024

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[Journal Article] Fluorescent Rotary Switches: Four- vs Three-Substituted Phthalimide Boron Difluoride Schiff Base Complexes2023

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[Journal Article] Vicinal All‐Carbon Quaternary Stereocenter Construction with Trifluoromethyl Groups via Organocatalytic Asymmetric Cascade Michael/Michael Reaction2023

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[Journal Article] Highly efficient, asymmetric, and organocatalyst-based Henry reactions between α,β-unsaturated trifluoromethyl ketone and nitromethane2023

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[Journal Article] Catalytic Synthesis of Phthalide Derivatives via Asymmetric Bromolactonization of Stilbene‐type Carboxylic Acids using<i>N,N</i>‐Dibenzyl Diaminomethylenemalononitrile as Organocatalyst2023

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[Journal Article] Asymmetric Direct Vinylogous Conjugate Addition of α,β‐Unsaturated γ‐Butyrolactam to Acyl Acrylonitriles using Organocatalysts2023

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[Journal Article] Organocatalyzed Synthesis of Bicyclic γ‐Lactam Derivatives via Asymmetric Conjugate Addition of Cyclic β‐Keto Esters to Benzoyl Acrylonitriles2023

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[Journal Article] Asymmetric Friedel?Crafts Alkylation of Indoles with α,β‐unsaturated Trifluoromethyl Ketones Using a Squaramide Organocatalyst2022

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[Journal Article] Solvent-Triggered Long-Range Proton Transport in 7-Hydroxyquinoline Using a Sulfonamide Transporter Group2022

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[Journal Article] Asymmetric Direct Vinylogous Conjugate Addition of Substituted Furanone Derivatives to ( <i>E</i> )‐ and ( <i>Z)</i> ‐Benzoyl Acrylonitriles Using Organocatalysts2022

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Hirashima Shinichi 平島真一

Hirashima Shin-ichi 平島真一