yagi yusuke 屋木祐亮

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Yagi Yusuke 屋木祐亮

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Researcher Number	90802207
Other IDs
Affiliation (Current)	2025: 京都医療科学大学, 医療科学部, 講師 2025: 京都薬科大学, 薬学部, 研究員
Affiliation (based on the past Project Information) *help	2025: 京都医療科学大学, 医療科学部, 講師 2023: 京都医療科学大学, 医療科学部, 講師 2020 – 2022: 京都医療科学大学, 医療科学部, 助教 2019: 京都薬科大学, 薬学部, 研究員 2018: 京都薬科大学, 薬学部, ポストドクター
Review Section/Research Field	Principal Investigator Basic Section 52040:Radiological sciences-related
Keywords	Principal Investigator ラジオセラノスティクス / SPECT / PET / マイクロ波反応 / モレキュラーコンバーチブルプローブ / PET・SPECT / F-18標識反応 / モレキュラーコンバーチブル / GRP78 / 放射性医薬品 … More / がん治療 / 分子イメージング / 放射線科学 / マイクロ波 / ユニットカップリング型プローブ / ウレア誘導体 / 前立腺がん / 迅速合成 / 標識合成 / マイクロ波合成 / PSMA / 前立腺特異的膜抗原 Less

治療困難ながんの診断・治療を目的としたラジオセラノスティクスプローブの開発Principal Investigator
- Principal Investigator
  
  屋木祐亮
- Project Period (FY)
  2025 – 2027
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 52040:Radiological sciences-related
- Research Institution
  Kyoto University of Medical Science
Development of the Molecular convertible probe for Lung cancerPrincipal Investigator
- Principal Investigator
  
  屋木祐亮
- Project Period (FY)
  2022 – 2024
- Research Category
  
  Grant-in-Aid for Early-Career Scientists
- Review Section
  
  Basic Section 52040:Radiological sciences-related
- Research Institution
  Kyoto College of Medical Science
Development of Radio-Theranostics molecular probes for prostate cancerPrincipal Investigator
- Principal Investigator
  
  Yagi Yusuke
- Project Period (FY)
  2018 – 2021
- Research Category
  
  Grant-in-Aid for Early-Career Scientists
- Review Section
  
  Basic Section 52040:Radiological sciences-related
- Research Institution
  Kyoto College of Medical Science
  Kyoto Pharmaceutical University

All 2024 2023 2022 2021 2020 2019 2018

All Journal Article Presentation

[Journal Article] Novel [ 111 In]In-BnDTPA-EphA2-230-1 Antibody for Single-Photon Emission Computed Tomography Imaging Tracer Targeting of EphA22023
- Author(s)
  T. Furukawa, H. Kimura, M. Sasaki, T. Yamada, T. Iwasawa, Y. Yagi, K. Kato, H. Yasui
- Journal Title
  
  ACS Omega
  
  Volume: 8 Issue: 7 Pages: 7030-7035
- DOI
  10.1021/acsomega.2c07849
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-23K24189, KAKENHI-PROJECT-22K15852
[Journal Article] Effect of Water on Direct Radioiodination of Small Molecules/Peptides Using Copper-Mediated Iododeboronation in Water?Alcohol Solvent2023
- Author(s)
  Kondo Yuto、Kimura Hiroyuki、Sasaki Minon、Koike Sumina、Yagi Yusuke、Hattori Yasunao、Kawashima Hidekazu、Yasui Hiroyuki
- Journal Title
  
  ACS Omega
  
  Volume: 8 Issue: 27 Pages: 24418-24425
- DOI
  10.1021/acsomega.3c01974
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-22K15852, KAKENHI-PROJECT-21K06502
[Journal Article] Novel synthesis of an [18F]aryl boronic acid ester as a reagent for 18F-labeling via Suzuki coupling2022
- Author(s)
  Yagi Yusuke、Kimura Hiroyuki、Kondo Yuto、Higuchi Takahiro
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 104 Pages: 154010-154010
- DOI
  10.1016/j.tetlet.2022.154010
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-22K15852
[Journal Article] Copper-mediated radioiodination and radiobromination via aryl boronic precursor and its application to 125I/77Br?labeled prostate-specific membrane antigen imaging probes2022
- Author(s)
  Kondo Yuto、Kimura Hiroyuki、Sasaki Ichiro、Watanabe Shigeki、Ohshima Yasuhiro、Yagi Yusuke、Hattori Yasunao、Koda Manami、Kawashima Hidekazu、Yasui Hiroyuki、Ishioka Noriko S.
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 69 Pages: 116915-116915
- DOI
  10.1016/j.bmc.2022.116915
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K15852, KAKENHI-PROJECT-20K07056
[Journal Article] Copper-mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide2021
- Author(s)
  Yuto Kondo, Hiroyuki Kimura, Chiaki Fukumoto, Yusuke Yagi, Yasunao Hattori, Hidekazu Kawashima, Hiroyuki Yasui
- Journal Title
  
  Journal of Labelled Compounds and Radiopharmaceuticals
  
  Volume: - Issue: 8 Pages: 336-345
- DOI
  10.1002/jlcr.3925
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K08061, KAKENHI-PROJECT-19K08826, KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-20K07056, KAKENHI-PROJECT-21K06502
[Journal Article] A Putative Single-Photon Emission CT Imaging Tracer for Erythropoietin-Producing Hepatocellular A2 Receptor2021
- Author(s)
  Furukawa Takenori、Kimura Hiroyuki、Torimoto Hanae、Yagi Yusuke、Kawashima Hidekazu、Arimitsu Kenji、Yasui Hiroyuki
- Journal Title
  
  ACS Medicinal Chemistry Letters
  
  Volume: 12 Issue: 8 Pages: 1238-1244
- DOI
  10.1021/acsmedchemlett.1c00030
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-19K08826, KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-20K07056
[Journal Article] Aicardi-Goutieres syndrome-like encephalitis in mutant mice with constitutively active MDA52020
- Author(s)
  Onizawa Hideo、Kato Hiroki、Kimura Hiroyuki、Kudo Tomoo、Soda Nobumasa、Shimizu Shota、Funabiki Masahide、Yagi Yusuke、Nakamoto Yuji、Priller Josef、Nishikomori Ryuta、Heike Toshio、Yan Nan、Tsujimura Tohru、Mimori Tsuneyo、Fujita Takashi
- Journal Title
  
  International Immunology
  
  Volume: 33 Issue: 4 Pages: 225-240
- DOI
  10.1093/intimm/dxaa073
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-19K08299
[Journal Article] Synthesis of 18F-labeled streptozotocin derivatives and an in-vivo kinetics study using positron emission tomography2020
- Author(s)
  Arimitsu Kenji、Yagi Yusuke、Koshino Kazuhiro、Nishito Yukina、Higuchi Takahiro、Yasui Hiroyuki、Kimura Hiroyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 30 Issue: 17 Pages: 127400-127400
- DOI
  10.1016/j.bmcl.2020.127400
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-20K07056, KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-19J01778, KAKENHI-PROJECT-18K15608, KAKENHI-PROJECT-20K08061
[Journal Article] Efficient gallium-68 radiolabeling reaction of DOTA derivatives using a resonant-type microwave reactor2019
- Author(s)
  Yagi Yusuke、Shimizu Yoichi、Arimitsu Kenji、Nakamoto Yuji、Higuchi Takahiro、Togashi Kaori、Kimura Hiroyuki
- Journal Title
  
  Journal of Labelled Compounds and Radiopharmaceuticals
  
  Volume: 62 (3) Issue: 3 Pages: 132-138
- DOI
  10.1002/jlcr.3704
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-17K10377
[Journal Article] Structure?activity relationships of succinimidyl-Cys-C(O)-Glu derivatives with different near-infrared fluorophores as optical imaging probes for prostate-specific membrane antigen2018
- Author(s)
  Matsuoka Daiko、Watanabe Hiroyuki、Shimizu Yoichi、Kimura Hiroyuki、Yagi Yusuke、Kawai Ryoko、Ono Masahiro、Saji Hideo
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 26 Issue: 9 Pages: 2291-2301
- DOI
  10.1016/j.bmc.2018.03.015
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K15566, KAKENHI-PROJECT-17K19670
[Presentation] F-18間接標識用試薬ボロン酸誘導体3-[18F]TDBFB及び 4-[18F]TDBFBの最適化検討2024
- Author(s)
  屋木祐亮、木村寛之、樋口隆弘
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-22K15852
[Presentation] 鈴木カップリング反応を用いたF-18間接標識用試薬ボロン酸誘導体[18F]TDBFBの合成検討2023
- Author(s)
  屋木祐亮、木村寛之、樋口隆弘
- Organizer
  日本薬学会143年会
- Data Source
  KAKENHI-PROJECT-22K15852
[Presentation] Expanding the Versatility of F-18 Indirect Labeling: Optimizing the Synthesis of TDBFB Boronic Acid Derivatives for Indirect Labeling via Suzuki Coupling2023
- Author(s)
  Yusuke Yagi, Hiroyuki Kimura, Miu Ando, Kaho Kawaguchi, Ayano Sato, Airi Shimizu, Mihoko Fujimura, Takahiro Higuchi
- Organizer
  EANM’23 WORLD LEADING MEETING
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-22K15852
[Presentation] F-18標識ボロン酸誘導体との鈴木カップリング反応を用いた新規F-18標識法の開発2021
- Author(s)
  屋木祐亮、近藤悠斗、樋口隆弘、木村寛之
- Organizer
  日本薬学会第142年会
- Data Source
  KAKENHI-PROJECT-18K15566
[Presentation] In vitro characterization of metabolic trapping of a novel PET tracer for fatty acid oxidation, 18F-AS3504073-002020
- Author(s)
  Yasuhiro OHSHIMA, Yusuke YAGI, Hiroshi FUSHIKI, Christoph MAACK, Takahiro HIGUCHI
- Organizer
  EANM'20 virtual edition
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18K15566
[Presentation] 共振空洞型マイクロ波反応装置を用いた68Ga錯体形成反応の基礎評価2018
- Author(s)
  屋木祐亮, 木村寛之, 志水陽一, 有光健治, 中本裕士, 富樫かおり, 安井裕之
- Organizer
  第１３８回日本薬学会年会
- Data Source
  KAKENHI-PROJECT-18K15566

1. KIMURA Hiroyuki

# of Collaborated Projects: 0 results

# of Collaborated Products: 2 results
2. 岩澤卓弥

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
3. 加藤和則

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
4. 安井裕之

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
5. 河嶋秀和

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

yagi yusuke 屋木 祐亮

Yagi Yusuke 屋木 祐亮

Research Projects

Research Products

Co-Researchers

治療困難ながんの診断・治療を目的としたラジオセラノスティクスプローブの開発Principal Investigator

Principal Investigator

Project Period (FY)

Research Category

Review Section

Research Institution

Development of the Molecular convertible probe for Lung cancerPrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Review Section

Research Institution

Development of Radio-Theranostics molecular probes for prostate cancerPrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Review Section

Research Institution

[Journal Article] Novel [ 111 In]In-BnDTPA-EphA2-230-1 Antibody for Single-Photon Emission Computed Tomography Imaging Tracer Targeting of EphA22023

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Effect of Water on Direct Radioiodination of Small Molecules/Peptides Using Copper-Mediated Iododeboronation in Water?Alcohol Solvent2023

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Novel synthesis of an [18F]aryl boronic acid ester as a reagent for 18F-labeling via Suzuki coupling2022

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Copper-mediated radioiodination and radiobromination via aryl boronic precursor and its application to 125I/77Br?labeled prostate-specific membrane antigen imaging probes2022

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Copper-mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide2021

Author(s)

Journal Title

DOI

Data Source

[Journal Article] A Putative Single-Photon Emission CT Imaging Tracer for Erythropoietin-Producing Hepatocellular A2 Receptor2021

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Aicardi-Goutieres syndrome-like encephalitis in mutant mice with constitutively active MDA52020

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Synthesis of 18F-labeled streptozotocin derivatives and an in-vivo kinetics study using positron emission tomography2020

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Efficient gallium-68 radiolabeling reaction of DOTA derivatives using a resonant-type microwave reactor2019

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Structure?activity relationships of succinimidyl-Cys-C(O)-Glu derivatives with different near-infrared fluorophores as optical imaging probes for prostate-specific membrane antigen2018

Author(s)

Journal Title

DOI

Data Source

[Presentation] F-18間接標識用試薬ボロン酸誘導体3-[18F]TDBFB及び 4-[18F]TDBFBの最適化検討2024

Author(s)

Organizer

Data Source

[Presentation] 鈴木カップリング反応を用いたF-18間接標識用試薬ボロン酸誘導体[18F]TDBFBの合成検討2023

Author(s)

Organizer

yagi yusuke 屋木祐亮

Yagi Yusuke 屋木祐亮