Kitamura Yoshiaki 喜多村徳昭

… Alternative Names

喜多村徳昭キタムラヨシアキ

KITAMURA Yoshiaki 喜多村徳昭

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Researcher Number	10503659
Other IDs	https://orcid.org/0000-0002-5785-6892
Affiliation (Current)	2025: 岐阜大学, 工学部, 准教授
Affiliation (based on the past Project Information) *help	2022 – 2023: 岐阜大学, 工学部, 助教 2016 – 2017: 岐阜大学, 工学部, 助教 2010 – 2012: 岐阜大学, 工学部, 助教
Review Section/Research Field	Principal Investigator Drug development chemistry / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
Keywords	Principal Investigator 核酸医薬 / 簡便合成 / 多様性指向型合成 / 核酸オリゴマー / 生理活性 / 有機化学 / 薬学 / 効率的合成 / ポスト修飾 / CuAAC … More / 分解酵素耐性 / 環境応答 / 機能性短鎖RNA / オリゴ核酸修飾 / siRNA Less

核酸医薬開発の推進を目指した核酸オリゴマーの革新的合成法の開発Principal Investigator
- Principal Investigator
  
  喜多村徳昭
- Project Period (FY)
  2022 – 2024
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Gifu University
Development of sophisticated small RNAs utilizing the properties of functional groupsPrincipal Investigator
- Principal Investigator
  
  KITAMURA Yoshiaki
- Project Period (FY)
  2016 – 2017
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Gifu University
Novel modification method of oligonucleotides for siRNA medicinePrincipal Investigator
- Principal Investigator
  
  KITAMURA Yoshiaki
- Project Period (FY)
  2010 – 2012
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Gifu University

All 2024 2023 2018 2017 2016 2012 2011 Other

All Journal Article Presentation

[Journal Article] Nucleobase azide-ethynylribose click chemistry contributes to stabilizing oligonucleotide duplexes and stem-loop structures2017
- Author(s)
  Yoshiaki Kitamura, Ryo Asakura, Koki Terazawa, Aya Shibata, Masato Ikeda, Yukio Kitade
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 27 Issue: 12 Pages: 2655-2658
- DOI
  10.1016/j.bmcl.2017.04.023
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K18911
[Journal Article] Introduction of 2-O-benzyl abasic nucleosides to the 3'-overhang regions of siRNAs greatly improves nuclease resistance2017
- Author(s)
  Yuki Nagaya, Yoshiaki Kitamura, Aya Shibata, Masato Ikeda, Yukihiro Akao, Yukio Kitade
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 27 Issue: 24 Pages: 5454-5456
- DOI
  10.1016/j.bmcl.2017.10.070
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K18911
[Journal Article] Practical modification of peptides using ligand-free copper-catalyzed azide-alkyne cycloaddition2016
- Author(s)
  Yoshiaki Kitamura, Ryo Sakamoto, Takao Shiraishi, Haruka Oguri, Satoshi Ohno, Yukio Kitade
- Journal Title
  
  Tetrahedron
  
  Volume: 72 Issue: 27-28 Pages: 4016-4021
- DOI
  10.1016/j.tet.2016.05.029
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-16K18911
[Journal Article] Synthesis and biological properties of chemically modified siRNAs bearing 1-deoxy-D-ribofuranose in their 3'-overhang region2012
- Author(s)
  Kazumi Taniho, Remi Nakashima, Mahmoud Kandeel, Yoshiaki Kitamura, Yukio Kitade
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 22 Issue: 7 Pages: 2518-2521
- DOI
  10.1016/j.bmcl.2012.01.132
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22790107
[Journal Article] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofuranose as a versatile scaffold2012
- Author(s)
  Yoshiaki Kitamura, Kana Edayoshi, Yukio Kitade
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 53 Issue: 51 Pages: 6987-6989
- DOI
  10.1016/j.tetlet.2012.10.053
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22790107, KAKENHI-PROJECT-24390025
[Journal Article] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofura- nose as a versatile scaffold2012
- Author(s)
  Yoshiaki Kitamura、 Kana Edayoshi 、 Yukio Kitad
- Journal Title
  
  Tetrahedron Lett
  
  Volume: 53 Pages: 6987-6989
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22790107
[Journal Article] Synthesis and biological properties of chemically modified siRNAs bearing 1-deoxy-D-ribofuranose in their 3′-overhang region2012
- Author(s)
  Kazumi Taniho、Remi Nakashima、Mahmoud Kandeel、 Yoshiaki Kitamura、 Yukio Kitade
- Journal Title
  
  Bioorg. Med. Chem. Lett
  
  Volume: 22 Pages: 2518-2521
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] 核酸オリゴマーの新規合成法の開発を指向した5'位官能基化チミジンモノマーの合成とリン酸ジエステルとの反応2024
- Author(s)
  山口莉沙、喜多村徳昭
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-22K06501
[Presentation] 新規核酸オリゴマー構築法の開発を目指した5'位官能基化ヌクレオシド誘導体の合成2023
- Author(s)
  山口莉沙、天野夏妃、喜多村徳昭
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K06501
[Presentation] Preparation of nucleoside 3'-phosphate derivatives functionalized at 5'-position as monomer units for novel strategies to oligonucleotide synthesis2023
- Author(s)
  Yoshiaki Kitamura, Risa Yamaguchi, Natsuki Amano
- Organizer
  第50回国際核酸化学シンポジウム（ISNAC2023）
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-22K06501
[Presentation] 塩基部欠損ヌクレオシド類を 3’末端に有する siRNA の合成と性質評価2018
- Author(s)
  長屋優貴, 喜多村徳昭, 柴田綾, 池田将, 赤尾幸博, 北出幸夫
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] Nucleobase azide-ethynylribose click chemistry: stabilizing oligonucleotide duplexes and stem-loop structures2017
- Author(s)
  Yoshiaki Kitamura, Ryo Asakura, Koki Terazawa, Aya Shibata, Masato Ikeda, Yukio Kitade
- Organizer
  第44回国際核酸化学シンポジウム（ISNAC2017）・日本核酸化学会第1回年会
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] リボース誘導体を母核とする新規traceless型リンカーの開発2017
- Author(s)
  寺澤康輝, 喜多村徳昭, 長屋優貴, 柴田綾, 池田将, 北出幸夫
- Organizer
  日本病院薬剤師会東海ブロック・日本薬学会東海支部合同学術大会2017
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] Nucleobase azide-ethynylribose click chemistry contributes to stabilizing oligonucleotide duplexes and stem-loop　structures2017
- Author(s)
  Yoshiaki Kitamura, Ryo Asakura, Koki Terazawa, Aya Shibata, Masato Ikeda, Yukio Kitade
- Organizer
  第26回国際複素環化学会議（26th ISHC Congress）
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] Synthesis of chemically modified siRNAs bearing high affinity molecules for human Argonaute 2 PAZ domain and their biological properties2016
- Author(s)
  Yoshiaki Kitamura, Yuki Nagaya, Kazuhito Kondo, Ryo Asakura, Qin Ren, Mahmoud Kandeel, Aya Shibata, Masato Ikeda, Yukio Kitade
- Organizer
  第43回国際核酸化学シンポジウム（ISNAC2016）
- Place of Presentation
  熊本大学（熊本）
- Year and Date
  2016-09-27
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] トリアゾール環形成による二本鎖核酸の安定化2016
- Author(s)
  朝倉領、喜多村徳昭、柴田綾、池田将、北出幸夫
- Organizer
  日本病院薬剤師会東海ブロック・日本薬学会東海支部合同学術大会2016
- Place of Presentation
  長良川国際会議場（岐阜）
- Year and Date
  2016-10-30
- Data Source
  KAKENHI-PROJECT-16K18911
[Presentation] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofuranose and its applications2012
- Author(s)
  Kana Edayoshi 、 Yoshiaki Kitamura、Masato Ikeda 、 Yukio Kitade
- Organizer
  第39回国際核酸化学シンポジウム
- Place of Presentation
  名古屋
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] 1-Deoxy-1-ethynyl-β-D-ribofuranoseの立体選択的合成2012
- Author(s)
  枝吉佳奈、喜多村徳昭、北出幸夫
- Organizer
  平成 24 年度日本薬学会東海支部例会
- Place of Presentation
  静岡
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] Synthesis of 1-deoxy-D-ribofuranose and its application for RNAi studies2011
- Author(s)
  Kazumi Taniho, Yoshiaki Kitamura, Yukio Kitade
- Organizer
  第38回国際核酸化学シンポジウム(ISNAC2011)
- Place of Presentation
  北海道大学(札幌)
- Year and Date
  2011-11-09
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] 塩基部欠損型ヌクレオシドを導入した2-5Aアナログの合成とその生物活性2011
- Author(s)
  谷保和美、喜多村徳昭、北出幸夫
- Organizer
  平成23年度日本薬学会東海支部例会
- Place of Presentation
  金城学院大学(名古屋)
- Year and Date
  2011-07-09
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] Synthesis of 1-deoxy-D-ribo- furanose and its application for RNAi studies2011
- Author(s)
  Kazumi Taniho、Yoshiaki Kitamura、Yukio Kitade
- Organizer
  第38回国際核酸化学シンポジウム
- Place of Presentation
  札幌
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] 1-Deoxy-1-ethynyl-β-D-ribofuranoseの立体選択的合成
- Author(s)
  枝吉佳奈, 喜多村徳昭, 北出幸夫
- Organizer
  平成24年度日本薬学会東海支部例会
- Place of Presentation
  静岡県立大学（静岡）
- Data Source
  KAKENHI-PROJECT-22790107
[Presentation] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofuranose and its applications
- Author(s)
  Kana Edayoshi, Yoshiaki Kitamura, Masato Ikeda, Yukio Kitade
- Organizer
  第39回国際核酸化学シンポジウム（ISNAC2012）
- Place of Presentation
  名古屋大学（名古屋）
- Data Source
  KAKENHI-PROJECT-22790107

1. KITADE Yukio (20137061)

# of Collaborated Projects: 2 results

# of Collaborated Products: 19 results
2. IKEDA Masato (20432867)

# of Collaborated Projects: 2 results

# of Collaborated Products: 10 results
3. UENO Yoshihito (20250467)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
4. AYA SHIBATA (50462693)

# of Collaborated Projects: 1 results

# of Collaborated Products: 8 results

Kitamura Yoshiaki 喜多村 徳昭

喜多村 徳昭 キタムラ ヨシアキ

KITAMURA Yoshiaki 喜多村 徳昭

Research Projects

Research Products

Co-Researchers

核酸医薬開発の推進を目指した核酸オリゴマーの革新的合成法の開発Principal Investigator

Principal Investigator

Project Period (FY)

Research Category

Review Section

Research Institution

Development of sophisticated small RNAs utilizing the properties of functional groupsPrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

Novel modification method of oligonucleotides for siRNA medicinePrincipal Investigator

Principal Investigator

Project Period (FY)

Research Category

Research Field

Research Institution

[Journal Article] Nucleobase azide-ethynylribose click chemistry contributes to stabilizing oligonucleotide duplexes and stem-loop structures2017

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Introduction of 2-O-benzyl abasic nucleosides to the 3'-overhang regions of siRNAs greatly improves nuclease resistance2017

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Practical modification of peptides using ligand-free copper-catalyzed azide-alkyne cycloaddition2016

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Synthesis and biological properties of chemically modified siRNAs bearing 1-deoxy-D-ribofuranose in their 3'-overhang region2012

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofuranose as a versatile scaffold2012

Author(s)

Journal Title

DOI

Data Source

[Journal Article] Stereoselective synthesis of 1-deoxy-1-ethynyl-β-D-ribofura- nose as a versatile scaffold2012

Author(s)

Journal Title

Data Source

[Journal Article] Synthesis and biological properties of chemically modified siRNAs bearing 1-deoxy-D-ribofuranose in their 3′-overhang region2012

Author(s)

Journal Title

Data Source

[Presentation] 核酸オリゴマーの新規合成法の開発を指向した5'位官能基化チミジンモノマーの合成とリン酸ジエステルとの反応2024

Author(s)

Organizer

Data Source

[Presentation] 新規核酸オリゴマー構築法の開発を目指した5'位官能基化ヌクレオシド誘導体の合成2023

Author(s)

Organizer

Data Source

[Presentation] Preparation of nucleoside 3'-phosphate derivatives functionalized at 5'-position as monomer units for novel strategies to oligonucleotide synthesis2023

Author(s)

Organizer

Data Source

[Presentation] 塩基部欠損ヌクレオシド類を 3’末端に有する siRNA の合成と性質評価2018

Author(s)

Organizer

Data Source

[Presentation] Nucleobase azide-ethynylribose click chemistry: stabilizing oligonucleotide duplexes and stem-loop structures2017

Author(s)

Organizer

Data Source

[Presentation] リボース誘導体を母核とする新規traceless型リンカーの開発2017

Author(s)

Organizer

Kitamura Yoshiaki 喜多村徳昭

喜多村徳昭キタムラヨシアキ

KITAMURA Yoshiaki 喜多村徳昭

[Presentation] Nucleobase azide-ethynylribose click chemistry contributes to stabilizing oligonucleotide duplexes and stem-loop　structures2017