Hirai Go 平井剛

… Alternative Names

HIRAI Go 平井剛

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Researcher Number	50359551
Other IDs	https://orcid.org/0000-0003-3420-555X
External Links
Affiliation (Current)	2023: 九州大学, 薬学研究院, 教授
Affiliation (based on the past Project Information) *help	2016 – 2023: 九州大学, 薬学研究院, 教授 2015: 国立研究開発法人理化学研究所, 袖岡有機合成化学研究室, 専任研究員 2014: 独立行政法人理化学研究所, 専任研究員 2010 – 2014: 独立行政法人理化学研究所, 袖岡有機合成化学研究室, 専任研究員 2005 – 2009: 独立行政法人理化学研究所, 袖岡有機合成化学研究室, 研究員 … More 2007: The Institute of Physical and Chemical Research, 袖岡有機合成化学研究室, 研究員 2004 – 2005: 独立行政法人理化学研究所, 研究員 2004: RIKEN, Research Scientist, 理化学研究所, 研究員 2003 – 2004: 東北大学, 多元物質科学研究所, 助手 Less
Review Section/Research Field	Principal Investigator Science and Engineering / Living organism molecular science / Basic Section 37020:Chemistry and chemical methodology of biomolecules-related / ケミカルバイオロジー / Chemical biology / Medium-sized Section 37:Biomolecular chemistry and related fields / Transformative Research Areas, Section (II) Except Principal Investigator Basic Section 38020:Applied microbiology-related / Bioorganic chemistry / Science and Engineering … More / Applied microbiology / Chemical biology / Chemical biology / Structural biochemistry / Living organism molecular science / Broad Section H Less
Keywords	Principal Investigator 有機合成 / シアリダーゼ / シアル酸 / 生物活性 / 分子プローブ / 構造活性相関 / 分子設計 / 複合糖質 / 代謝 / 有機化学 … More / 糖鎖 / 生体分子 / 中分子 / C-グリコシド / カップリング / ラジカル / 阻害剤 / グリコシル化 / 酸化的カップリング / Isobenzofuranone / PKCα / C1ドメイン / ドメイン選択性 / isobenzofuranone / Stille coupling / 不斉ジヒドロキシル化 / プロテインホスファターゼ / 不可逆的阻害剤 / 蛍光ラベル体 / ホオズキ / ステロイド / NF-kB / physalin / ワンポット反応 / ドミノ反応 / 生理活性 / シグナル伝達 / 酸化ステロイド / NF-κB / Physalin / タンパク質SUMO化 / 天然物 / 植物酸化ステロイド / 鍵構造アナログ / 作用機序解析 / 酵素反応 / プローブ / コンホメーション / ラジカルカップリング / C-H挿入反応 / C-H活性化 / グルコサミノグリカン / 代謝耐性型アナログ / ヒアルロナン / 水素添加反応 / 光反応 / 触媒的合成 / 擬天然物 / 擬複合糖質 … More Except Principal Investigator 阻害剤 / プロテインキナーゼC / RK-682 / PKC / 細胞死 / 細胞間コミュニケーション / 分裂酵母 / オキシリピン / ウロテインキナーゼC / 酵素 / コンホマーション / 細胞増殖 / ネクローシス / プロテインキナーゼ / プロテインホスファターゼ / フッ素 / インドリルマレイミイド / フッ素化 / バイオイソスター / フルオロホスホン酸 / タンパク質アセチル化 / アセチローム / 代謝酵素 / 翻訳関連因子 / リジン脱アセチル化酵素 / リジンアセチル化酵素 / 枯草菌 / コリネバクテリウム菌 / コリネバクテリウム / グルタミン酸生産 / タンパク質(リジン)アセチル化 / 枯草菌(Bacillus subtilis) / 必須タンパク質 / リン酸化プロテオーム / 脱アセチル化酵素 / プロテオミクス / シャペロン / HDAC / 酵素阻害剤 / Isobenzofuranone誘導体 / ホスファチジルセリン / 構造活性相関 / 有機合成 / Phosphatidylserine / ホルボールエステル / SUMO / 抗がん剤 / 脱SUMO化酵素 / SUMOylation / がん / ケミカルバイオロジー / NMR / マルチドメインタンパク質 / sortase / プロテインライゲーション / 構造解析 / 活性制御 / 目的指向型ライブラリー / チロシンホスファターゼ / テトロン酸 / アスコルビン酸 / ヘパラナーゼ / ライブラリー / テロン酸 / focused library / protein tyrosine phosphatase / inhibitor / tetronic acid / Ascorbic acid / heparanase / protein kinase C / 窒素代謝 / 脂質 / タンパク質 / 機能解析 Less

Catalytic synthesis of pseudo-natural products utilizing photo-reactionPrincipal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2023 – 2027
- Research Category
  
  Grant-in-Aid for Transformative Research Areas (A)
- Review Section
  
  Transformative Research Areas, Section (II)
- Research Institution
  Kyushu University
Diversity of oxidized lipids and their functional understanding
- Principal Investigator
  
  山田健一
- Project Period (FY)
  2023 – 2027
- Research Category
  
  Grant-in-Aid for Scientific Research (S)
- Review Section
  
  Broad Section H
- Research Institution
  Kyushu University
分裂酵母の細胞間コミュニケーションを担うオキシリピンの生合成経路の解明
- Principal Investigator
  
  八代田陽子
- Project Period (FY)
  2022 – 2024
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Review Section
  
  Basic Section 38020:Applied microbiology-related
- Research Institution
  Institute of Physical and Chemical Research
Synthetic chemistry for the development of oligosaccharide-type sialidase inhibitorsPrincipal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2021 – 2023
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 37020:Chemistry and chemical methodology of biomolecules-related
- Research Institution
  Kyushu University
中分子グライコミメティクスの開拓Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2021 – 2023
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 37:Biomolecular chemistry and related fields
- Research Institution
  Kyushu University
代謝安定型糖鎖を基盤とする高次生物機能中分子複合糖質アナログ創製Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2018 – 2019
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Research Institution
  Kyushu University
Synthetic chemistry for the development of oligosaccharide-type sialidase inhibitorsPrincipal Investigator
- Principal Investigator
  
  Hirai Go
- Project Period (FY)
  2018 – 2021
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 37020:Chemistry and chemical methodology of biomolecules-related
- Research Institution
  Kyushu University
Nitrogen Signaling Factor (NSF)-mediated cell-to-cell communication in fission yeast
- Principal Investigator
  
  Yashiroda Yoko
- Project Period (FY)
  2018 – 2020
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 38020:Applied microbiology-related
- Research Institution
  Institute of Physical and Chemical Research
代謝安定型糖鎖を基盤とする高次生物機能複合糖質アナログの創製Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2016 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Review Section
  
  Science and Engineering
- Research Institution
  Kyushu University
Development of a novel type of carbohydrate probesPrincipal Investigator
- Principal Investigator
  
  Hirai Go
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Chemical biology
- Research Institution
  Kyushu University
  Institute of Physical and Chemical Research
酸化ステロイドの鍵構造アナログ創製と作用機序解析Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2014 – 2015
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Review Section
  
  Science and Engineering
- Research Institution
  Institute of Physical and Chemical Research
Structural study of reconstitued full length PKC
- Principal Investigator
  
  MISHIMA Masaki
- Project Period (FY)
  2013 – 2014
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Structural biochemistry
- Research Institution
  Tokyo Metropolitan University
タンパク質ＳＵＭＯ化を阻害する天然物リガンドの合成供給と構造活性相関Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2012 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Review Section
  
  Science and Engineering
- Research Institution
  The Institute of Physical and Chemical Research
Study on chemical biology for protein SUMOylation
- Principal Investigator
  
  ITO Akihiro
- Project Period (FY)
  2011 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical biology
- Research Institution
  The Institute of Physical and Chemical Research
Synthetic approaches toward the identification of target proteins of physalinsPrincipal Investigator
- Principal Investigator
  
  HIRAI Go
- Project Period (FY)
  2010 – 2012
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  ケミカルバイオロジー
- Research Institution
  The Institute of Physical and Chemical Research
Proteomic approach for identification of lysine acetylation in bacteria
- Principal Investigator
  
  KOSONO Saori
- Project Period (FY)
  2009 – 2011
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Applied microbiology
- Research Institution
  The Institute of Physical and Chemical Research
Clarification research for molecular mechanism of a novel type of protein kinase C inhibitor
- Principal Investigator
  
  SODEOKA Mikiko
- Project Period (FY)
  2009 – 2011
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical biology
- Research Institution
  The Institute of Physical and Chemical Research
Development of a novel type of irreversible inhibitors for comprehensive analysis of protein phosphatase in cellsPrincipal Investigator
- Principal Investigator
  
  HIRAI Go
- Project Period (FY)
  2007 – 2008
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Living organism molecular science
- Research Institution
  The Institute of Physical and Chemical Research
細胞の増殖と死を制御する分子の創製と機能解析
- Principal Investigator
  
  袖岡幹子
- Project Period (FY)
  2004 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Science and Engineering
- Research Institution
  The Institute of Physical and Chemical Research
  Tohoku University
プロテインキナーゼC活性化機構の解明と新規阻害剤の開発Principal Investigator
- Principal Investigator
  
  平井剛
- Project Period (FY)
  2004 – 2005
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Living organism molecular science
- Research Institution
  The Institute of Physical and Chemical Research
  Tohoku University
Construction of focused library and the development of protein tyrosine phosphatase inhibitor
- Principal Investigator
  
  SODEOKA Mikiko
- Project Period (FY)
  2003 – 2004
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Living organism molecular science
- Research Institution
  TOHOKU UNIVERSITY
酵素のコンホメーションを認識する分子:阻害剤開発への新しいアプローチ
- Principal Investigator
  
  SODEOKA Mikiko
- Project Period (FY)
  2002 – 2003
- Research Category
  
  Grant-in-Aid for Exploratory Research
- Research Field
  
  Bioorganic chemistry
- Research Institution
  Tohoku University

[Journal Article] Harringtonine Ester Derivatives with Enhanced Antiproliferative Activities against HL-60 and HeLa Cells2022
- Author(s)
  Ochi Akihiro、Yoritate Makoto、Miyamoto Tomofumi、Usui Kazuteru、Yusakul Gorawit、Putalun Waraporn、Tanaka Hiroyuki、Hirai Go、Morimoto Satoshi、Sakamoto Seiichi
- Journal Title
  
  Journal of Natural Products
  
  Volume: 85 Issue: 2 Pages: 345-351
- DOI
  10.1021/acs.jnatprod.1c00888
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K15957, KAKENHI-PROJECT-21H02070, KAKENHI-PROJECT-20K05467, KAKENHI-PROJECT-21K19053
[Journal Article] Effect of Alkynyl Group on Reactivity in Photoaffinity Labeling with 2‐Thienyl‐Substituted α‐Ketoamide2022
- Author(s)
  Moriyama Takahiro、Mizukami Daiki、Yoritate Makoto、Usui Kazuteru、Takahashi Daisuke、Ota Eisuke、Sodeoka Mikiko、Ueda Tadashi、Karasawa Satoru、Hirai Go
- Journal Title
  
  Chemistry A European Journal
  
  Volume: 28 Issue: 11 Pages: 1-5
- DOI
  10.1002/chem.202103925
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K07016, KAKENHI-PROJECT-20K15957, KAKENHI-PROJECT-21H02070, KAKENHI-PROJECT-20K05467, KAKENHI-PROJECT-21K19053, KAKENHI-PROJECT-20K15290
[Journal Article] β-Glycosyl Trifluoroborates as Precursors for Direct α-C-Glycosylation: Synthesis of 2-Deoxy-α-C-glycosides2021
- Author(s)
  Daiki Takeda, Makoto Yoritate, Hiroki Yasutomi, Suzuka Chiba, Takahiro Moriyama, Atsushi Yokoo, Kazuteru Usui, Go Hirai*
- Journal Title
  
  Organic Letters
  
  Volume: 23 Issue: 5 Pages: 1940-1944
- DOI
  10.1021/acs.orglett.1c00402
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K05467, KAKENHI-PROJECT-20K15957, KAKENHI-PROJECT-18H02097
[Journal Article] Preparation of Oxysterols by C?H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst2021
- Author(s)
  Fujii Yui、Yoritate Makoto、Makino Kana、Igawa Kazunobu、Takeda Daiki、Doiuchi Daiki、Tomooka Katsuhiko、Uchida Tatsuya、Hirai Go
- Journal Title
  
  Molecules
  
  Volume: 27 Issue: 1 Pages: 225-225
- DOI
  10.3390/molecules27010225
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-20K15957, KAKENHI-PROJECT-21H02070, KAKENHI-PROJECT-21J13680, KAKENHI-PROJECT-21K19053
[Journal Article] Design, synthesis, and functional evaluation of triazine-based bivalent agents that simultaneously target the active site and hot spot of phosphatase Cdc25B2021
- Author(s)
  Nagaoka Yosei、Parvatkar Prakash、Hirai Go、Ohkanda Junko
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 48 Pages: 128265-128265
- DOI
  10.1016/j.bmcl.2021.128265
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K21248, KAKENHI-PUBLICLY-20H04769, KAKENHI-PROJECT-21H02070, KAKENHI-PROJECT-21K19053
[Journal Article] Ganglioside GM3 Analogues Containing Monofluoromethylene-Linked Sialoside: Synthesis, Stereochemical Effects, Conformational Behavior, and Biological Activities2020
- Author(s)
  Hirai Go、Kato Marie、Koshino Hiroyuki、Nishizawa Eri、Oonuma Kana、Ota Eisuke、Watanabe Toru、Hashizume Daisuke、Tamura Yuki、Okada Mitsuaki、Miyagi Taeko、Sodeoka Mikiko
- Journal Title
  
  JACS Au
  
  Volume: 1 Issue: 2 Pages: 137-146
- DOI
  10.1021/jacsau.0c00058
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-20K15290, KAKENHI-PROJECT-18H02097
[Journal Article] Synthesis of DFGH-Ring Derivatives of Physalins via One-Pot Construction of GH-Ring and Evaluation of Their NF-κB-Inhibitory Activity2020
- Author(s)
  Yoritate Makoto、Morita Yuki、Gemander Manuel、Morita Masaki、Yamashita Tomohiro、Sodeoka Mikiko、Hirai Go
- Journal Title
  
  Organic Letters
  
  Volume: 22 Issue: 22 Pages: 8877-8881
- DOI
  10.1021/acs.orglett.0c03255
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K15957, KAKENHI-PROJECT-18H02097
[Journal Article] Identification of novel fish sialidase genes responsible for KDN-cleaving activity2020
- Author(s)
  Shiozaki Kazuhiro、Uezono Keiya、Hirai Go、Honda Akinobu、Minoda Masaya、Wakata Ryuta
- Journal Title
  
  Glycoconjugate Journal
  
  Volume: 37 Issue: 6 Pages: 745-753
- DOI
  10.1007/s10719-020-09948-6
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19K06223, KAKENHI-PROJECT-18H02097
[Journal Article] Synthesis of All Stereoisomers of Monomeric Spectomycin A1/A2 and Evaluation of Their Protein SUMOylation‐Inhibitory Activity2019
- Author(s)
  Nomura Yusaku、Thuaud Frederic、Sekine Daisuke、Ito Akihiro、Maeda Satoko、Koshino Hiroyuki、Hashizume Daisuke、Muranaka Atsuya、Cruchter Thomas、Uchiyama Masanobu、Ichikawa Satoshi、Matsuda Akira、Yoshida Minoru、Hirai Go、Sodeoka Mikiko
- Journal Title
  
  Chemistry A European Journal
  
  Volume: 25 Issue: 35 Pages: 8387-8392
- DOI
  10.1002/chem.201901093
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04417, KAKENHI-PLANNED-18H05503, KAKENHI-PROJECT-18H02097, KAKENHI-PROJECT-17H06173, KAKENHI-PROJECT-26221204
[Journal Article] Enhancement of saccharothriolide production and discovery of a new metabolite, saccharothriolide C2, by combined-culture of Saccharothrix sp. and Tsukamurella pulmonis2019
- Author(s)
  Yulu Jiang, Shan Lu, Go Hirai, Taira Kato, Hiroyasu Onaka, Hideaki Kakeya
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 60 Issue: 15 Pages: 1072-1074
- DOI
  10.1016/j.tetlet.2019.03.034
- Peer Reviewed
- Data Source
  KAKENHI-PLANNED-17H06401, KAKENHI-PROJECT-17K19233, KAKENHI-PUBLICLY-18H04417, KAKENHI-PROJECT-18H02097
[Journal Article] Synthesis of CH2-Linked α(1,6)-Disaccharide Analogues by α-Selective Radical Coupling C-Glycosylation2019
- Author(s)
  Kiya Noriaki、Hidaka Yu、Usui Kazuteru、Hirai Go
- Journal Title
  
  Organic Letters
  
  Volume: 21 Issue: 6 Pages: 1588-1592
- DOI
  10.1021/acs.orglett.9b00133
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04417, KAKENHI-PROJECT-18H02097
[Journal Article] Synthesis of All Stereoisomers of RK460 and Evaluation of Their Activity and Selectivity as Abscisic Acid Receptor Antagonists2019
- Author(s)
  Mikame Yu、Yoshida Kazuko、Hashizume Daisuke、Hirai Go、Nagasawa Kazuo、Osada Hiroyuki、Sodeoka Mikiko
- Journal Title
  
  Chemistry A European Journal
  
  Volume: 25 Issue: 14 Pages: 3496-3500
- DOI
  10.1002/chem.201806056
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04417, KAKENHI-PROJECT-18H02097, KAKENHI-PROJECT-16K13094, KAKENHI-PROJECT-18H03945, KAKENHI-PUBLICLY-18H04387, KAKENHI-PROJECT-16K18662
[Journal Article] Thienyl-Substituted α-Ketoamide: A Less Hydrophobic Reactive Group for Photo-Affinity Labeling2018
- Author(s)
  Ota Eisuke、Usui Kazuteru、Oonuma Kana、Koshino Hiroyuki、Nishiyama Shigeru、Hirai Go、Sodeoka Mikiko
- Journal Title
  
  ACS Chemical Biology
  
  Volume: 13 Issue: 4 Pages: 876-880
- DOI
  10.1021/acschembio.7b00988
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K12760, KAKENHI-PROJECT-16K18846
[Journal Article] Synthesis of polyunsaturated fatty acid-containing glucuronosyl-diacylglycerol through direct glycosylation2017
- Author(s)
  Wang Qianqian、Kuramoto Yuta、Okazaki Yozo、Ota Eisuke、Morita Masaki、Hirai Go、Saito Kazuki、Sodeoka Mikiko
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 58 Issue: 30 Pages: 2915-2918
- DOI
  10.1016/j.tetlet.2017.06.034
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17K13263, KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K12760
[Journal Article] Synthesis of the Right-Side Structure of Type B Physalins2017
- Author(s)
  Morita Masaki、Kojima Shuntaro、Ohkubo Megumi、Koshino Hiroyuki、Hashizume Daisuke、Hirai Go、Maruoka Keiji、Sodeoka Mikiko
- Journal Title
  
  Israel Journal of Chemistry
  
  Volume: 57 Issue: 3-4 Pages: 309-318
- DOI
  10.1002/ijch.201600110
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-17K13263, KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K12760
[Journal Article] Comparative Characterization of the Leaf Tissue of Physalis alkekengi and Physalis peruviana Using RNA-seq and Metabolite Profiling2016
- Author(s)
  Atsushi Fukushima, Michimi Nakamura, Hideyuki Suzuki, Mami Yamazaki, Eva Knoch, Tetsuya Mori, Naoyuki Umemoto, Masaki Morita, Go Hirai, Mikiko Sodeoka, and Kazuki Saito
- Journal Title
  
  Frontiers in Plant Science
  
  Volume: 7 Pages: 1883-1883
- DOI
  10.3389/fpls.2016.01883
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-26850024, KAKENHI-PROJECT-15K12760, KAKENHI-PROJECT-26350967
[Journal Article] Identification of novel secreted fatty acids that regulate nitrogen catabolite repression in fission yeast.2016
- Author(s)
  Sun X, Hirai G, Ueki M, Hirota H, Wang Q, Hongo Y, Nakamura T, Hitora Y, Takahashi H, Sodeoka M, Osada H, Hamamoto M, Yoshida M, Yashiroda Y.
- Journal Title
  
  Scientific Reports
  
  Volume: 6 Issue: 1 Pages: 20856-20856
- DOI
  10.1038/srep20856
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-15K07376, KAKENHI-PROJECT-24619011, KAKENHI-PROJECT-15K12760, KAKENHI-PUBLICLY-26102744, KAKENHI-PROJECT-15J09122, KAKENHI-PROJECT-25660085
[Journal Article] A new carbamidemethyl-linked lanthanide chelating tag for PCS NMR spectroscopy of proteins in living HeLa cells.2016
- Author(s)
  Yuya Hikone, Go Hirai, Masaki Mishima, Kohsuke Inomata, Teppei Ikeya, Souichiro Arai, Masahiro Shirakawa, Mikiko Sodeoka, and Yutaka Ito
- Journal Title
  
  Journal of Biomolecular NMR
  
  Volume: 66 Issue: 2 Pages: 99-110
- DOI
  10.1007/s10858-016-0059-4
- Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-15H01645, KAKENHI-PUBLICLY-16H00779, KAKENHI-PUBLICLY-16H00847, KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K06979, KAKENHI-PROJECT-15K12760, KAKENHI-PROJECT-15K14494, KAKENHI-PLANNED-25120003
[Journal Article] Photochemical and Additive-free Coupling Reaction of α-Cumyl α-Ketoesters via Intermolecular C-H Bond Activation2016
- Author(s)
  Eisuke Ota, Yu Mikame, Go Hirai, Shigeru Nishiyama, Mikiko Sodeoka
- Journal Title
  
  Synlett
  
  Volume: 27 Issue: 07 Pages: 1128-1132
- DOI
  10.1055/s-0035-1561098
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-14J06218, KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K12760
[Journal Article] Rational Design and Synthesis of [5]Helicene-Derived Phosphine Ligands and Their Application in Pd-Catalyzed Asymmetric Reactions2016
- Author(s)
  Kosuke Yamamoto, Takashi Shimizu, Kazunobu Igawa, Katsuhiko Tomooka, Go Hirai, Hiroshi Suemune, and Kazuteru Usui
- Journal Title
  
  Scientific Reports
  
  Volume: 6 Issue: 1 Pages: 36211-36211
- DOI
  10.1038/srep36211
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-15K12760, KAKENHI-PROJECT-16K18846
[Journal Article] Total synthesis of natural derivatives and artificial analogs of 13-oxyingenol and their biological evaluation2016
- Author(s)
  Takayuki Ohyoshi, Yuki Tamura, Ichiro Hayakawa, Go Hirai, Yamato Miyazawa, Shota Funakubo, Mikiko Sodeoka, and Hideo Kigoshi
- Journal Title
  
  Org. Biomol. Chem.
  
  Volume: 14 Issue: 48 Pages: 11426-11437
- DOI
  10.1039/c6ob02268e
- NAID
  120007135231
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-16H01167, KAKENHI-PROJECT-26242073, KAKENHI-PROJECT-15K12760
[Journal Article] Focused Library with a Core Structure Extracted from Natural Products and Modified: Application to Phosphatase Inhibitors and Several Biochemical Findings2015
- Author(s)
  Go Hirai and Mikiko Sodeoka
- Journal Title
  
  Acc. Chem. Res.
  
  Volume: 48 Issue: 5 Pages: 1464-1473
- DOI
  10.1021/acs.accounts.5b00048
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K12760, KAKENHI-PUBLICLY-26102744
[Journal Article] Photo-induced formation of cyclopropanols from α-ketoamides via γ-C-H bond activation2015
- Author(s)
  Eisuke Ota, Yu Mikame, Go Hirai, Hiroyuki Koshino, Shigeru Nishiyama, Mikiko Sodeoka
- Journal Title
  
  Tetrahedron Lett.
  
  Volume: 56 Issue: 44 Pages: 5991-5994
- DOI
  10.1016/j.tetlet.2015.09.038
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K12760, KAKENHI-PUBLICLY-26102744, KAKENHI-PROJECT-14J06218
[Journal Article] Reactions of Carbonyl Compounds with Phosphorus Ylide Generated from Tribromofluoromethane and Tris(dimethylamino)phosphine2015
- Author(s)
  Go Hirai, Eri Nishizawa, Daiki Kakumoto, Masaki Morita, Mitsuaki Okada, Daisuke Hashizume, Sayoko Nagashima, Mikiko Sodeoka
- Journal Title
  
  Chem. Lett.
  
  Volume: 44 Issue: 10 Pages: 1389-1391
- DOI
  10.1246/cl.150523
- NAID
  130005101456
- ISSN
  0366-7022, 1348-0715
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K12760, KAKENHI-PUBLICLY-26102744
[Journal Article] C-シアロシド結合を有するガングリオシドアナログの創製2014
- Author(s)
  平井　剛
- Journal Title
  
  ファインケミカル
  
  Volume: 43 (No.2) Pages: 45-52
- Data Source
  KAKENHI-PUBLICLY-24102534
[Journal Article] RE12 Derivatives Displaying Vaccinia H1-related Phosphatase (VHR) Inhibition in the Presence of Detergent and Their Anti-Proliferative Activity against HeLa Cells2014
- Author(s)
  Frederic Thuaud, Shuntaro Kojima, Go Hirai, Kana Oonuma, Ayako Tsuchiya, Takako Uchida, Teruhisa Tsuchitomo, Mikiko Sodeoka
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 9 Pages: 2771-2782
- DOI
  10.1016/j.bmc.2014.03.012
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PUBLICLY-26102744
[Journal Article] 天然物を基にした両特異性プロテインホスファターゼ阻害剤の開発2014
- Author(s)
  平井剛
- Journal Title
  
  化学工業
  
  Volume: 65 Pages: 304-310
- Data Source
  KAKENHI-PUBLICLY-26102744
[Journal Article] Unexpected Diels-Alder/Carbonylene Cascade toward the Biomimetic Synthesis of Chloropupukeananin2013
- Author(s)
  T. Suzuki, Y. Miyajima, K. Suzuki, K. Iwakiri, M. Koshimizu, G. Hirai, M. Sodeoka, S.Kobayashi
- Journal Title
  
  Organic Letters
  
  Volume: 15 Issue: 7 Pages: 1748-1751
- DOI
  10.1021/ol400549q
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22390004, KAKENHI-PUBLICLY-24102534
[Journal Article] Development of bis-unsaturated ester aldehydes as amino-glue probes: sequential double azaelectrocyclization as a promising strategy for bioconjugation.2013
- Author(s)
  Tanaka, K., Nakamoto, Y., Siwu, ER., Pradipta, AR., Morimoto, K., Fujiwara, T., Yoshida, S., Hosoya, T., Tamura, Y., Hirai, G., Sodeoka, M., Fukase, K.
- Journal Title
  
  Org Biomol Chem.,
  
  Volume: 11 Issue: 42 Pages: 7326-7333
- DOI
  10.1039/c3ob41507d
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23241074, KAKENHI-PROJECT-23681047, KAKENHI-PUBLICLY-24102512, KAKENHI-PUBLICLY-24102518, KAKENHI-PUBLICLY-24102534, KAKENHI-PROJECT-25560410
[Journal Article] Contribution of Cage-Shaped Structure of Physalins to Their Mode of Action in Inhibition of NF-kB Action2013
- Author(s)
  M. Ozawa, M. Morita, G. Hirai, S. Tamura, M. Kawai, A. Tsuchiya, K. Oonuma, K. Maruoka, M. Sodeoka
- Journal Title
  
  ACS Med. Chem. Lett.
  
  Volume: 4 Issue: 8 Pages: 730-735
- DOI
  10.1021/ml400144e
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24102534, KAKENHI-PROJECT-24790109
[Journal Article] High-resolution heteronuclear multidimensional NMR of proteins living insect cells using a baculovirus protein expression system ≪2013
- Author(s)
  Jumpei Hamatsu, Daniel O'Donovan, Takashi Tanaka, Takahiro Shirai, Yuichiro Hourai, Tsutomu Mikawa, Teppei Ikeya, Masaki Mishima, Wayne Boucher, Brian O. Smith, Ernest D. Laue, Masahiro Shirakawa, Yutaka Ito 4
- Journal Title
  
  Journal of the American Chemical Society
  
  Volume: 135 Issue: 5 Pages: 1688-1691
- DOI
  10.1021/ja310928u
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J05888, KAKENHI-PLANNED-21121006, KAKENHI-PROJECT-22570147, KAKENHI-PUBLICLY-24121722, KAKENHI-PROJECT-24770101, KAKENHI-PUBLICLY-25117723, KAKENHI-PROJECT-25650025, KAKENHI-PUBLICLY-24113720
[Journal Article]2013
- Author(s)
  Masaaki Ozawa, Masaki Morita, Go Hirai, Satoru Tamura, Masao Kawai, Ayako Tsuchiya, Kana Oonuma, Keiji Maruoka, and Mikiko Sodeoka
- Journal Title
  
  ACS. Med. Chem. Lett.
  
  Volume: (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22603014
[Journal Article] Development of Novel Types of Biologically Active Compounds Based on Natural Products and Biomolecules2012
- Author(s)
  平井剛
- Journal Title
  
  YAKUGAKU ZASSHI
  
  Volume: 132 Issue: 1 Pages: 117-124
- DOI
  10.1248/yakushi.132.117
- NAID
  130001871951
- ISSN
  0031-6903, 1347-5231
- Year and Date
  2012-01-01
- Language
  Japanese
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22603014
[Journal Article]2012
- Author(s)
  Masaki Morita, Go Hirai, Meguni Ohkubo Hiroyuki Koshino, Daisuke Hashizume, Keiji Maruoka, and Mikiko Sodeoka
- Journal Title
  
  Org. Latt.
  
  Volume: 14 Pages: 3434-3437
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22603014
[Journal Article] Design and synthesis of protein kinase Cαactivators based on .'out of pocket' interactions2011
- Author(s)
  Hirai, G., Ohkubo, M., Tamura, Y. and Sodeoka, M.
- Journal Title
  
  Bioorg. Med. Chem. Lett
  
  Volume: 21 Pages: 3587-3590
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-21603016
[Journal Article] Design and Synthesis of Protein Kinase Cα activators based on 'out of pocket' interaction2011
- Author(s)
  Go Hirai
- Journal Title
  
  Bioorg.Med.Chem.Lett.
  
  Volume: 21 Issue: 12 Pages: 3587-3590
- DOI
  10.1016/j.bmcl.2011.04.108
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-21603016
[Journal Article] Asymmetric synthesis of isobenzofuranone derivatives and their unique character as protein kinase Cα(PKCα)activators2009
- Author(s)
  Go Hirai
- Journal Title
  
  Tetrahedron Lett. 50
  
  Pages: 3609-3612
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-21603016
[Journal Article] Asymmetric synthesis of isobenzofuranone derivatives and their unique character as protein kinase Cα(PKCα) activators2009
- Author(s)
  Hirai, G., Ogoshi, Y., Ohkubo, M., Tamura, Y., Watanabe, T., Shimizu, T. and Sodeoka, M.
- Journal Title
  
  Tetrahedron Lett
  
  Volume: 50 Pages: 3609-3612
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-21603016
[Journal Article] Synthesis of CH_2-Linked・(2,3)Sialylgalactose Analogue : On the Stereoselectivity of the Key Ireland-Claisen Rearrangement2008
- Author(s)
  Toru Watanabe, Go Hirai, Marie Kato, Daisuke Hashizume, Taeko Miyagi, Mikiko Sodeoka
- Journal Title
  
  Org. Lett. 10
  
  Pages: 4167-4170
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] Limited Inhibitory Effects of Oseltamivir and Zanamivir on Human Sialidases2008
- Author(s)
  Keiko Hata, Koichi Koseki, Kazunori Yamaguchi, Setsuko Moriya, Yasuo Suzuki, Sangchai Yingsakmongkon, Go Hirai, Mikiko Sodeoka, Mark von Itzstein, Taeko Miyagi
- Journal Title
  
  Antimicrob. Agents Chemother 52
  
  Pages: 3484-3491
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] Stereocontrolled and Convergent Entry to CF_2-Sialosides: Synthesis of CF_2-Linked Ganglioside GM42007
- Author(s)
  Go Hirai
- Journal Title
  
  Journal of the American Chemical Society 129
  
  Pages: 15420-15421
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] Importance of interaction between C1 domain and lipids in protein kinase Cα activation: Hydrophobic side chain direction isobenzofuranone ligands controls enzyme activation level2007
- Author(s)
  Go Hirai
- Journal Title
  
  ChemMedChem 2
  
  Pages: 1006-1009
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16073203
[Journal Article] Stereo-controlled and Convergent Entry to CF_2-Sialosides : Synthesis of CF_2-linked Ganglioside GM42007
- Author(s)
  Go Hirai
- Journal Title
  
  J. Am. Chem. Soc. 129
  
  Pages: 15420-15421
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16073203
[Journal Article] Stereocontrolled and Convergent Entry to CF_2-Sialosides : Synthesis of CF_2-Linked Ganglioside GM42007
- Author(s)
  Go Hirai, Toru Watanabe, Kazunori Yamaguchi, Taeko Miyagi, Mikiko Sodeoka
- Journal Title
  
  J. Am. Chem. Soc. 129
  
  Pages: 15420-15421
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] Importance of interaction between C1 domain and lipids in protein kinase Ca activation : Hydrophobic side chain direction in isobensofuranone ligands controls enzyme activation level2007
- Author(s)
  Go Hirai, Tadashi Shimizu, Toru Watanabe, Yosuke Ogoshi, Megumi Ohkubo, Mikiko Sodeoka
- Journal Title
  
  ChemMedChem 2
  
  Pages: 1006-1009
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] Importance of interaction between C1 domain and lipids in protein kinase Cα activation: Hydrophobic side chain direction in isobenzofuranone ligands controls enzyme activation level.2007
- Author(s)
  Go Hirai
- Journal Title
  
  Chem Med Chem 2
  
  Pages: 1006-1009
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19710195
[Journal Article] プロテインキナーゼC(PKC)の構造と活性化機構の解明を目指した新規C1ドメインリガンドの創製2006
- Author(s)
  平井剛, 清水忠, 袖岡幹子
- Journal Title
  
  有機合成化学協会誌 64
  
  Pages: 515-527
- NAID
  10017486844
- Data Source
  KAKENHI-PROJECT-16073203
[Journal Article] 低分子阻害剤によるタンパク質リン酸化の制御 : 構造変化と選択性2005
- Author(s)
  平井剛
- Journal Title
  
  実験医学増刊 23, No.4
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-15310144
[Journal Article] Control of the protein phosphorylation by small molecule inhibitors : protein structure and selectivity2005
- Author(s)
  Go Hirai
- Journal Title
  
  Experimental Medicine vol.23-No.4
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-15310144
[Journal Article] 低分子阻害剤によるタンパク質リン酸化の制御:構造変化と選択性2005
- Author(s)
  平井剛
- Journal Title
  
  実験医学増刊 Vol.23,No.4
  
  Pages: 199-204
- Data Source
  KAKENHI-PROJECT-16073203
[Journal Article] 低分子阻害剤によるタンパク質リン酸化の制御:構造変化と選択性2005
- Author(s)
  平井剛
- Journal Title
  
  実験医学増刊 Vol.23,No.4
  
  Pages: 199-204
- Data Source
  KAKENHI-PROJECT-15310144
[Journal Article] 低分子阻害剤によるタンパク質リン酸化の制御:構造変化と選択性2005
- Author(s)
  平井剛
- Journal Title
  
  実験医学増刊:ここまで進んだゲノム医科学と疾患研究 23・4
  
  Pages: 651-656
- Data Source
  KAKENHI-PROJECT-16710152
[Patent] 新規化合物、並びにかかる新規化合物を含む酵素阻害剤及びＡＢＰ2020
- Inventor(s)
  平井剛、森田昌樹、木室佑亮、土井一毅
- Industrial Property Rights Holder
  九州大学
- Industrial Property Rights Type
  特許
- Filing Date
  2020
- Overseas
- Data Source
  KAKENHI-PROJECT-18H02097
[Patent] 新規化合物、並びにかかる新規化合物を含む酵素阻害剤及びＡＢＰ2020
- Inventor(s)
  平井剛、森田昌樹、木室佑亮、土井一毅
- Industrial Property Rights Holder
  九州大学
- Industrial Property Rights Type
  特許
- Filing Date
  2020
- Overseas
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Patent] 新規化合物、並びにかかる新規化合物を含む酵素阻害剤及びＡＢＰ2019
- Inventor(s)
  平井剛、森田昌樹、木室佑亮
- Industrial Property Rights Holder
  平井剛、森田昌樹、木室佑亮
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2019-052106
- Filing Date
  2019
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Patent] シアル酸誘導体2016
- Inventor(s)
  平井剛、深澤亮、袖岡幹子
- Industrial Property Rights Holder
  平井剛、深澤亮、袖岡幹子
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2016-147705
- Filing Date
  2016-07-27
- Data Source
  KAKENHI-PROJECT-15K12760
[Patent] シアル酸誘導体2016
- Inventor(s)
  平井剛、深澤亮、袖岡幹子
- Industrial Property Rights Holder
  平井剛、深澤亮、袖岡幹子
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2016-147705
- Filing Date
  2016-07-27
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Efficient Synthetic Strategy for C-linked α-Galactosylceramide Analogues2022
- Author(s)
  Go Hirai
- Organizer
  7th International Symposium on Middle Molecular Strategy (ISMMS-7)/ 16th Meeting of the International Endotoxin and Innate Immunit Society (IEIIS-16)
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 代謝耐性型複合糖質のポテンシャル：アジュバントへの展開は可能か？2022
- Author(s)
  平井剛
- Organizer
  第15回次世代アジュバント研究会
- Invited
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] 直接C-グリコシル化反応を活用した糖鎖アナログの効率的合成法の開発2022
- Author(s)
  森山貴博、小野俊介、寄立麻琴、千馬鈴華、田邉理子、平井剛
- Organizer
  日本薬学会第142回年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 代謝耐性型複合糖質のポテンシャル：アジュバントへの展開は可能か？2022
- Author(s)
  平井剛
- Organizer
  第15回次世代アジュバント研究会
- Invited
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 代謝耐性型ヒアルロナンオリゴマーの合成研究2022
- Author(s)
  木谷憲昭、寄立麻琴、平井剛
- Organizer
  日本化学会第102春季年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 2-エキソメチレン型グルコシドの立体選択的合成と活性評価2022
- Author(s)
  伊ヶ崎孝洋、木室佑亮、寄立麻琴、平井剛
- Organizer
  日本薬学会第142回年会
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] グリコシルラジカルを基盤とした炭素連結型β-グルコシルセラミドの合成2022
- Author(s)
  千馬鈴華、森山貴博、小野俊介、寄立麻琴、平井
- Organizer
  日本化学会第102春季年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 2位にジフルオロメチレン基を有するグルコース誘導体の合成研究2022
- Author(s)
  古城真夏、寄立麻琴、平井剛
- Organizer
  日本化学会第102春季年会
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] Physalin類が有するDFGH環の新規合成法の開発2021
- Author(s)
  寄立麻琴、森田友己、森田昌樹、山下智大、袖岡幹子、平井剛
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 還元的光クロスカップリング反応を用いたKRN7000アナログの合成2021
- Author(s)
  小野俊介、寄立麻琴、森山貴博、長門石正孝、臼井一晃、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] グリコシルラジカルを基盤としたβ選択的なC-グリコシル化反応の開発2021
- Author(s)
  千馬鈴華、寄立麻琴、平井剛
- Organizer
  第58回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 2-エキソメチレン型β-グルコシドの立体選択的合成法の開発2021
- Author(s)
  古城真夏、寄立麻琴、平井剛
- Organizer
  第58回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] β-グリコシルボロン酸を用いたC-グリコシド合成法の開発2021
- Author(s)
  安冨弘樹、竹田大樹、千馬鈴華、寄立麻琴、平井剛
- Organizer
  第118回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] β-グリコシルボロン酸を用いた立体保持型C-グリコシル化の検討2021
- Author(s)
  安冨弘樹、竹田大樹、千葉鈴華、寄立麻琴、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 糸状菌 A. nidulans のアミラーゼ産生に対する代謝耐性型イソマルトースの効果2021
- Author(s)
  森山貴博, 木谷憲昭, 寄立麻琴, 加藤直樹, 沼本穂, 高橋俊二, 平井剛
- Organizer
  ケミカルバイオロジー学会第15回年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 立体選択的な2’-エキソメチレン型グルコシドの合成法開発2021
- Author(s)
  伊ヶ崎孝洋、寄立麻琴、平井剛
- Organizer
  第58回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] 基質－遷移状態ハイブリッドアナログ型α-glucosidase阻害剤の開発2021
- Author(s)
  土井一毅、木室佑亮、寄立麻琴、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Substrate-type Sialidase Inhibitors Involving Unique Mechanism-based Inhibition Machinery2021
- Author(s)
  Go Hirai, Ryo Fukazawa, Keiya Uezono, Kenta Mizui, Makoto Yoritate, Mikiko Sodeoka
- Organizer
  Pacifichem 2021: Recent advances in carbohydrate chemistry and chemical glycobiology (#111)
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] 2-エキソメチレン型β-グルコシドの立体選択的合成法の開発2021
- Author(s)
  古城真夏、寄立麻琴、平井剛
- Organizer
  創薬懇話会2021 in 京都
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] Synthesis and biological activity of C-linked glycan and glycolipid analogues2021
- Author(s)
  Go Hirai, Shunsuke Ono, Takahiro Moriyama, Makoto Yoritate
- Organizer
  Pacifichem 2021: Middle molecular strategy for regulation of protein-protein & protein-biomolecule interactions (#370)
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] グリコシルラジカルを基盤としたβ選択的なC-グリコシル化反応の開発2021
- Author(s)
  千馬鈴華、小野俊介、寄立麻琴、平井剛
- Organizer
  創薬懇話会2021 in 京都
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] Development of New Synthetic Method of the DFGH-ring of Physalin-Type Natural Products and SAR Study of the Pseudo- Natural Products2021
- Author(s)
  Yoritate, M.; Morita, Y.; Morita, M; Yamashita, T.; Sodeoka, M.; Hirai, G.
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 分裂酵母のオキシリピンを介した窒素代謝に関わる細胞間コミュニケーションの解明2021
- Author(s)
  橋本莉央、八代田陽子、大澤晋、平井剛、森山裕充、吉田稔
- Organizer
  日本農芸化学会2021年度大会
- Data Source
  KAKENHI-PROJECT-18H02131
[Presentation] グリコシルボロン酸を用いた2-デオキシ-C-グリコシド誘導体のα-選択的合成法の開発2021
- Author(s)
  竹田大樹、安冨弘樹、千馬鈴華、寄立麻琴、平井剛
- Organizer
  第40回日本糖質学会年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] コンフォメーション制御を志向したC-グリコシドアナログの開発2021
- Author(s)
  森山貴博、木谷憲昭、小野俊介、寄立誠、加藤直樹、高橋俊二、平井剛
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Efficient Synthetic Strategy for C-linked α-Galactosylceramide Analogues2021
- Author(s)
  Go Hirai
- Organizer
  7th International Symposium on Middle Molecular Strategy (ISMMS-7)/ 16th Meeting of the International Endotoxin and Innate Immunit Society (IEIIS-16)
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] 直接C-グリコシル化による代謝耐性型複合糖質アナログ合成2021
- Author(s)
  平井剛、森山貴博、小野俊介、千馬鈴華、木谷憲昭、寄立麻琴、加藤直樹、高橋俊二
- Organizer
  第40回日本糖質学会年会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] β-グリコシルボロン酸を用いた炭素連結型糖鎖の合成2021
- Author(s)
  竹田大樹、安冨弘樹、千葉鈴華、寄立麻琴、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Unique Activity of C-isomaltose analogues in A. nidulans2021
- Author(s)
  Takahiro Moriyama, Naoki Kato, Noriaki Kiya, Riko Tanabe, Makoto Yoritate, Minori Numamoto, Shunji Takahashi, Go Hirai
- Organizer
  AIMECS2121
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] C-グリコシドを基盤とした新規二糖アナログの合成と活性研究2021
- Author(s)
  木谷憲昭、寄立麻琴、平井剛
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 代謝耐性型中分子ヒアルロナンアナログの合成研究2021
- Author(s)
  木谷憲昭、森山貴博、寄立麻琴、平井剛
- Organizer
  第63回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] グリコシルボロン酸誘導体の合成とα-選択的な直接的2-デオキシ-C-グリコシド誘導体の新規合成法開発2021
- Author(s)
  竹田大樹、安冨弘樹、千馬鈴華、寄立麻琴、平井剛
- Organizer
  第31回万有福岡シンポジウム
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] ユニークな3次元構造をもつ糖―アミノ酸ハイブリッド骨格の構築2021
- Author(s)
  織田旺紀、寄立麻琴、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] グリコシルラジカルを基盤としたβ選択的C-グリコシル化反応の開発2021
- Author(s)
  千馬鈴華, 森山貴博, 小野俊介, 寄立麻琴, 平井剛
- Organizer
  第38回日本薬学会九州山口支部大会
- Data Source
  KAKENHI-PROJECT-21K19053
[Presentation] 2-エキソメチレン型UDP-グルコースの合成研究2021
- Author(s)
  山口昂太、木室佑亮、寄立麻琴、平井剛
- Organizer
  日本化学会第101春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 糖ヌクレオチドを模倣した糖転移酵素に対するABPの開発2021
- Author(s)
  山口昂太、木室佑亮、寄立麻琴、平井剛
- Organizer
  第33回若手研究者のためのセミナー
- Data Source
  KAKENHI-PROJECT-21H02070
[Presentation] 新規シアリダーゼ阻害剤の効率的合成を志向したシアル酸３位修飾法の開発2020
- Author(s)
  上薗慶也、寄立麻琴、平井剛
- Organizer
  第117回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 糖鎖分解の基質特性追跡：α-グルコシダーゼに対する概念実証2020
- Author(s)
  木室佑亮、土井一毅、寄立麻琴、平井剛
- Organizer
  第62回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] グリコシルボロン酸を用いた炭素連結型糖鎖の新規合成法の開発2020
- Author(s)
  竹田大樹、安冨弘樹、千葉鈴華、横尾淳、臼井一晃、寄立麻琴、平井剛
- Organizer
  反応と合成の進歩2020特別企画シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 還元的光クロスカップリング反応を用いたC-グリコシド誘導体の合成研究2020
- Author(s)
  小野俊介、長門石正孝、森山貴博、臼井一晃、寄立麻琴、平井剛
- Organizer
  第117回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] B-グリコシドの合成とカップリング反応によるC-グリコシドの合成2020
- Author(s)
  竹田大樹、安冨弘樹、千葉鈴華、横尾淳、臼井一晃、寄立麻琴、平井剛
- Organizer
  第117回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Metabolically Stable Analogues and Photo-Reactive Probe for Understanding Glycolipid Functions2020
- Author(s)
  Go Hirai
- Organizer
  The 93rd Annual Meeting of the Japanese Biochemical Society: Toward understanding and control of sugar-containing lipids by biology and chemistry
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 分裂酵母の窒素シグナリング因子を介した細胞間コミュニケーションにおける受容機構の解明2020
- Author(s)
  橋本莉央、八代田陽子、大澤晋、平井剛、森山裕充、吉田稔
- Organizer
  日本農芸化学会2020年度大会
- Data Source
  KAKENHI-PROJECT-18H02131
[Presentation] 新規炭素連結型イソマルトースアナログの合成研究2020
- Author(s)
  森山貴博、木谷憲昭、小野俊介、寄立誠、加藤直樹、高橋俊二、平井剛
- Organizer
  第117回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 代謝安定型Glc-CerおよびGal-Cerアナログの合成研究2020
- Author(s)
  寄立麻琴、日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  第30回万有福岡シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] α-グルコシダーゼに対する基質特異的代謝追跡プローブの開発2019
- Author(s)
  木室佑亮、土井一毅、森田昌樹、平井剛
- Organizer
  第21回薬学研究院若手セミナー
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] C-H挿入反応を用いたシアル酸3位の選択的修飾法の開発2019
- Author(s)
  上薗慶也、森田昌樹、平井剛
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 新規シアリダーゼ阻害剤の効率的な合成法の開発2019
- Author(s)
  上薗慶也、寄立麻琴、平井剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Synthetic studies of 1,6-C-linked disaccharide analogues based on direct radical coupling2019
- Author(s)
  Noriaki kiya, Yu Hidaka, Makoto Yoritate, Kazuteru Usui, Go Hirai
- Organizer
  European Carbohydrate Symposium (EurocarboXX)
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] α-グルコシダーゼに対する基質特異的代謝追跡プローブの開発2019
- Author(s)
  木室佑亮、土井一毅、森田昌樹、平井剛
- Organizer
  第31回若手研究者のためのセミナー
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Glycan probes: C-glycosides and photo-affinity probes2019
- Author(s)
  Go Hirai
- Organizer
  ACGG11
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] B-グリコシドの合成とC-グリコシド合成への応用2019
- Author(s)
  竹田大樹、安冨弘樹、横尾淳、臼井一晃、寄立麻琴、平井剛
- Organizer
  日本化学会第100春季年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] α-グルコシダーゼに対するSubstrate-specific Metabolism Monitoring Probe (SMMP)の開発2019
- Author(s)
  木室佑亮、土井一毅、森田昌樹、平井剛
- Organizer
  日本ケミカルバイオロジー学会　第14回年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 不安定なジエノフィルを用いるDiels-Alder反応を基盤とした天然物模倣型分子の合成研究2019
- Author(s)
  織田旺紀、森田昌樹、平井剛
- Organizer
  第56回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 新規複合糖質研究ツール：基質特異的分解追跡を可能にする分子プローブ2019
- Author(s)
  平井剛、木室佑亮、土井一毅、深澤亮、大沼可奈、袖岡幹子
- Organizer
  第38回日本糖質学会年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 2位エキソメチレン基を有するα-ガラクトシドの開発と活性評価2019
- Author(s)
  丸野瑛裕、木室佑亮、森田昌樹、寄立麻琴、平井剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 直接的α-C-グリコシル化を基盤とした1,6-炭素連結型二糖アナログの合成研究2019
- Author(s)
  木谷憲昭、日高悠、臼井一晃、加藤直樹、高橋俊二、平井剛
- Organizer
  第31回若手研究者のためのセミナー
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 代謝耐性型糖鎖を基盤とする炭素連結型メリビオサミンの合成研究2019
- Author(s)
  木谷憲昭、臼井一晃、寄立麻琴、平井剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Development of Substrate-specific Metabolism Monitoring probe for α-glucosidase2019
- Author(s)
  Yusuke Kimuro, Kazuki Doi, Masaki Morita, Makoto Yoritate, Go Hirai
- Organizer
  日本化学会第100春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 直接的ラジカルカップリング反応を基盤とする炭素連結型イソマルトース誘導体の合成研究2019
- Author(s)
  木谷憲昭、日高悠、臼井一晃、平井剛
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 直接的C-グリコシル化を基盤とした炭素連結型糖脂質アナログの合成研究2019
- Author(s)
  日高悠、木谷憲昭、寄立麻琴、臼井一晃、平井剛
- Organizer
  第116回有機合成シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 基質構造を基盤とした新規α-グルコシダーゼ阻害剤の開発2019
- Author(s)
  土井一毅、木室佑亮、寄立麻琴、平井剛
- Organizer
  日本化学会第100春季年会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 直接的α-C-グリコシル化を基盤とした1,6-炭素連結型二糖アナログの合成研究2019
- Author(s)
  木谷憲昭、日高悠、臼井一晃、加藤直樹、高橋俊二、平井剛
- Organizer
  第29回万有福岡シンポジウム
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 標識部位を導入したグリコシダーゼに対する新規mechanism-based inhibitorの開発2019
- Author(s)
  土井一毅、木室佑亮、平井剛
- Organizer
  第56回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Thienyl‐substituted α‐ketoamide: a less hydrophobic photoreactive group useful for analysis of carbohydrate‐protein interaction2019
- Author(s)
  Go Hirai
- Organizer
  European Carbohydrate Symposium (EurocarboXX)
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 炭素連結型イソマルトースアナログの構造活性相関研究2019
- Author(s)
  森山貴博、木谷憲昭、寄立麻琴、加藤直樹、高橋俊二、平井剛
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 炭素連結型糖脂質アナログの合成研究2019
- Author(s)
  日高悠、木谷憲昭、寄立麻琴、臼井一晃、○平井剛
- Organizer
  第37回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Synthesis of Biologically Active Molecules Based on Unique Right-Side Structure of Physalins2019
- Author(s)
  Yuki Morita, Manuel Gemander, Masaki Morita, Mikiko Sodeoka, Go Hirai
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 擬天然物を標的とする有機合成2019
- Author(s)
  平井剛
- Organizer
  第56回化学関連支部合同九州大会
- Invited
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] アトムトランスファー型ラジカルカップリング反応を利用した炭素連結型糖脂質の合成研究2019
- Author(s)
  寄立麻琴、日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  日本化学会第100春季年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] ホウ素グリコシド結合をもつ糖誘導体の合成とその利用2019
- Author(s)
  竹田大樹、横尾淳、安冨弘樹、臼井一晃、平井剛
- Organizer
  第56回化学関連支部合同九州大会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 2-エキソメチレン基を有するα-ガラクトシドの合成と機能評価2019
- Author(s)
  丸野瑛裕、木室佑亮、森田昌樹、寄立麻琴、平井剛
- Organizer
  第36回日本薬学会九州支部大会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 有機合成で新しいケミカルバイオロジーツールを創る2019
- Author(s)
  平井剛
- Organizer
  2019年度前期（春季）有機合成化学講習会　「新時代に飛躍する有機合成化学―機能性分子、材料から創薬まで―」
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 還元的クロスカップリング反応によるC-グリコシド誘導体の合成研究2019
- Author(s)
  小野俊介、長門石正孝、臼井一晃、寄立麻琴、平井剛
- Organizer
  第38回日本糖質学会年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 還元的光クロスカップリング反応によるC-グリコシド誘導体の合成研究2019
- Author(s)
  小野俊介、長門石正孝、臼井一晃、寄立麻琴、平井剛
- Organizer
  日本化学会第100春季年会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Synthesis and biological potential of carbohydrate analogues2019
- Author(s)
  Go Hirai
- Organizer
  19th Tateshina Conference
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 分子間カップリングを基盤とする炭素連結型2糖及び糖脂質アナログの合成研究2018
- Author(s)
  日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  第55回化学関連支部合同九州大会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 合成化学が拓く生物活性物質創製研究2018
- Author(s)
  平井剛
- Organizer
  生体機能関連化学部会若手の会　第30回サマースクール
- Invited
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] Synthetic studies of 1,6-C-linked disaccharide analogues based on radical coupling2018
- Author(s)
  Noriaki kiya, Yu Hidaka, Kazuteru Usui, Go Hirai
- Organizer
  IKCOC-14
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Synthetic studies of C-linked disaccharide analogues based on radical coupling2018
- Author(s)
  Yu Hidaka, Noriaki Kiya, Kazuteru Usui, Go Hirai
- Organizer
  IRCCS-CREST Joint Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 有機化学で複合糖質研究に挑む2018
- Author(s)
  平井剛
- Organizer
  第29回万有仙台シンポジウム　未来を指向した有機合成化学
- Invited
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] ラジカルカップリング反応を基盤とする炭素連結型2糖アナログの合成研究2018
- Author(s)
  木谷憲昭、日高悠、臼井一晃、平井剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 還元的クロスカップリング反応によるアリール C-グリコシドの合成研究2018
- Author(s)
  臼井一晃、長門石昌孝、郭義天、平井剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] ラジカルカップリングを基盤とする1,6-炭素連結型二糖アナログの合成研究2018
- Author(s)
  木谷憲昭、日高悠、臼井一晃、平井剛
- Organizer
  「有機合成化学を起点とするものづくり戦略」最終研究成果発表シンポジウム
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 分子間カップリングを基盤とする炭素連結型糖脂質アナログの合成研究2018
- Author(s)
  日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  創薬懇話会2018 in 志賀島
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 糖鎖に細工をする有機化学2018
- Author(s)
  平井剛
- Organizer
  有機合成化学協会東海支部主催　平成30年度有機合成セミナー
- Invited
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] フィサリン類の特異な右側構造の合成研究2018
- Author(s)
  森田昌樹、平井剛、袖岡幹子
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 有機化学で複合糖質研究に挑む2018
- Author(s)
  平井剛
- Organizer
  第29回万有仙台シンポジウム　未来を指向した有機合成化学
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 合成化学が拓く生物活性物質創製研究2018
- Author(s)
  平井剛
- Organizer
  生体機能関連化学部会若手の会　第30回サマースクール
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Focused Libraryのススメ2018
- Author(s)
  平井剛
- Organizer
  Asian Chemical Probe Research Hub Symposium：天然物有機化学・天然物合成とケミカルバイオロジー
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] C-H挿入反応を用いたシアル酸3位の選択的修飾法の開発2018
- Author(s)
  上薗慶也、臼井一晃、森田昌樹、平井剛
- Organizer
  第55回化学関連支部合同九州大会
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 光反応基官能基を導入した分裂酵母のシグナル分子の合成研究2018
- Author(s)
  水野雄太、森田昌樹、麻生真理子、平井剛
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 分子間カップリングを基盤とする炭素連結型糖脂質アナログの合成研究2018
- Author(s)
  日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  第30回若手研究者のためのセミナー
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 複合糖質を高機能化する有機化学2018
- Author(s)
  平井剛
- Organizer
  大塚創薬化学シンポジウム2018
- Invited
- Data Source
  KAKENHI-PROJECT-18H02097
[Presentation] 分子間カップリングを基盤とする炭素連結型糖脂質アナログの合成研究2018
- Author(s)
  日高悠、木谷憲昭、臼井一晃、平井剛
- Organizer
  第35回日本薬学会九州支部大会
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 複合糖質を高機能化する有機化学2018
- Author(s)
  平井剛
- Organizer
  大塚創薬化学シンポジウム2018
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] Synthesis of Unique Right-Side Structure of Physalins2018
- Author(s)
  Yuki Morita, Manuel Gemander, Masaki Morita, Mikiko Sodeoka, Go Hirai
- Organizer
  IRCCS-CREST Joint Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 天然物を高機能化する有機合成2018
- Author(s)
  平井剛
- Organizer
  日本化学会第98春季年会(2018)：天然有機化合物の全合成：効率的分子構築のための新しい反応と戦略（CSJカレントレビュー企画）
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 糖鎖に細工をする有機化学2018
- Author(s)
  平井剛
- Organizer
  有機合成化学協会東海支部主催　平成30年度有機合成セミナー
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04417
[Presentation] 非天然型複合糖質を創る2017
- Author(s)
  平井剛
- Organizer
  糸状菌分子生物学研究会　第5回若手の会 WS in SAGA
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Photoredox触媒を用いたクロスカップリングによるアリール C-グリコシドの合成研究2017
- Author(s)
  長門石昌孝、臼井一晃、郭義天、平井剛
- Organizer
  第34回日本薬学会九州支部大会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Synthesis of all the possible isomers of RK460 and its activity evaluation2017
- Author(s)
  三瓶悠、由田和津子、平井剛、長澤和夫、長田裕之、袖岡幹子
- Organizer
  日本化学会第97春季年会
- Place of Presentation
  慶應義塾大学日吉キャンパス
- Year and Date
  2017-03-15
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Click 反応によって連結可能なIn-cell NMR用常磁性金属イオンタグの開発2017
- Author(s)
  名取文彦、彦根佑哉、平井剛、三島正規、伊藤隆、袖岡幹子
- Organizer
  日本化学会第97春季年会
- Place of Presentation
  慶應義塾大学日吉キャンパス
- Year and Date
  2017-03-15
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 光反応基官能基を導入した分裂酵母のシグナル分子の合成研究2017
- Author(s)
  水野雄太、麻生真理子、平井剛
- Organizer
  第５４回化学関連支部合同九州大会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Synthetic Strategy Towards Unique Right-Side Structures of Physalins2017
- Author(s)
  Masaki Morita, Go Hirai, Mikiko Sodeoka
- Organizer
  ISONIS-11 & ISMMS-3
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] ラジカルカップリング反応を基盤とする炭素連結型２糖アナログの合成研究2017
- Author(s)
  木谷憲昭、臼井一晃、平井剛
- Organizer
  第５４回化学関連支部合同九州大会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 非天然型複合糖質を創る2017
- Author(s)
  平井剛
- Organizer
  糸状菌分子生物学研究会　第5回若手の会 WS in SAGA
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] 光親和性標識を目指した一置換α-ケトアミドの光反応性に関する理論的研究2017
- Author(s)
  三宅由希子、臼井一晃、太田英介、袖岡幹子、平井剛
- Organizer
  第29回若手研究者のためのセミナー
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 代謝に着目した中分子糖鎖分子の設計と機能2017
- Author(s)
  平井　剛
- Organizer
  日本薬学会第137年会一般シンポジウム「中分子創薬研究のフロンティア－反応集積化が導く中分子戦略：高次生物機能分子の創製－
- Place of Presentation
  仙台国際センター
- Year and Date
  2017-03-27
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 人工糖鎖を備えて未来の疾患と戦う2017
- Author(s)
  平井剛
- Organizer
  第7回CSJ化学フェスタ2017「10年後にはどんな分子ができる？有機合成化学者の「革命分子」への挑戦」 (2017.10.18)
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] 光親和性標識を志向した一置換α-ケトアミドの光反応性に関する理論的研究2017
- Author(s)
  三宅由希子、臼井一晃、太田英介、袖岡幹子、平井剛
- Organizer
  第５４回化学関連支部合同九州大会
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Synthesis of Natural Product Compartments for Finding Their Functions2017
- Author(s)
  平井剛
- Organizer
  The 3rd HU-TMU-KU Joint Symposium for Pharmaceutical Sciences
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Development of the Disaccharide-Type Activity-Based Probe for Sialidase2017
- Author(s)
  深澤亮、大沼可奈、加藤麻理依、平井剛、袖岡幹子
- Organizer
  日本化学会第97春季年会
- Place of Presentation
  慶應義塾大学日吉キャンパス
- Year and Date
  2017-03-17
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] Development of the Disaccharide-Type Activity-Based Probe for Sialidase2017
- Author(s)
  深澤亮、大沼可奈、加藤麻理依、平井剛、袖岡幹子
- Organizer
  日本化学会第97春季年会
- Place of Presentation
  慶應義塾大学日吉キャンパス
- Year and Date
  2017-03-15
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Synthesis of Monomers for Spectomycin B1, A Middle Size SUMOylation Inhibitor Molecule2017
- Author(s)
  Go Hirai
- Organizer
  7th CCS/CSJ Young Chemist Forum（第7回日中若手化学者フォーラム）
- Place of Presentation
  Keio University
- Year and Date
  2017-03-18
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] シアリダーゼに対する新規activity-based probeの開発2017
- Author(s)
  平井剛、深澤亮、大沼可奈、森田昌樹、加藤麻理依、袖岡幹子
- Organizer
  第35回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] 人工糖鎖を備えて未来の疾患と戦う2017
- Author(s)
  平井剛
- Organizer
  第7回CSJ化学フェスタ2017「10年後にはどんな分子ができる？有機合成化学者の「革命分子」への挑戦」 (2017.10.18)
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 代謝に着目した中分子糖鎖分子の設計と機能2017
- Author(s)
  平井剛
- Organizer
  日本薬学会第137年会一般シンポジウム「中分子創薬研究のフロンティア－反応集積化が導く中分子戦略：高次生物機能分子の創製－
- Place of Presentation
  仙台国際センター
- Year and Date
  2017-03-27
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] 有機化学を起点とするケミカルバイオロジー研究2017
- Author(s)
  平井剛
- Organizer
  徳島大学大学院「創薬先端合成化学特論」講演会
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] ラジカルカップリング反応を基盤とする炭素連結型2糖アナログの合成研究2017
- Author(s)
  木谷憲昭、日高悠、臼井一晃、平井剛
- Organizer
  第29回若手研究者のためのセミナー
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] α-ケトアミドを基盤とする新しい光親和性標識実験用プローブの開発2017
- Author(s)
  平井剛、太田英介、臼井一晃、大沼可奈、袖岡幹子
- Organizer
  日本ケミカルバイオロジー学会　第12回年会
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] 有機合成化学を起点とするケミカルバイオロジー研究2017
- Author(s)
  平井剛
- Organizer
  平成29年度有機合成化学講演会　－合成有機化学のフロンティア－
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Click反応によって連結可能なIn-cell NMR用常磁性金属イオンタグの開発2016
- Author(s)
  名取文彦、彦根佑哉、平井剛、三島正規、伊藤隆、袖岡幹子
- Organizer
  第6回CSJ化学フェスタ2016
- Place of Presentation
  タワーホール船堀
- Year and Date
  2016-11-14
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 単量体型スペクトマイシンの全立体異性体全合成とSUMO化阻害活性2016
- Author(s)
  野村勇作、Frederic Thuaud、関根大介、平井剛、前田里子、伊藤昭博、吉田稔、市川聡、松田彰、袖岡幹子
- Organizer
  日本化学会第96回春季年会
- Place of Presentation
  同志社大学京田辺キャンパス（京都府京田辺市）
- Year and Date
  2016-03-24
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 生物活性分子創製研究と有機合成研究の融合2016
- Author(s)
  平井剛
- Organizer
  熊本大学理学部化学特別講義C講演会
- Place of Presentation
  熊本大学理学部
- Year and Date
  2016-05-24
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] ケミカルバイオロジーに役立つものづくりを目指して2016
- Author(s)
  平井剛
- Organizer
  特別企画: 有機合成化学を起点とするものづくり戦略 (日本化学会第96回春季年会)
- Place of Presentation
  同志社大学京田辺キャンパス（京都府京田辺市）
- Year and Date
  2016-03-24
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] ABA受容体アンタゴニストRK460の全立体異性体合成と活性評価2016
- Author(s)
  三瓶悠、由田和津子、平井剛、長澤和夫、長田裕之、袖岡幹子
- Organizer
  第6回CSJ化学フェスタ2016
- Place of Presentation
  タワーホール船堀
- Year and Date
  2016-11-14
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] シアリダーゼの機能解析を志向した3位修飾型シアル酸誘導体の合成と活性評価2016
- Author(s)
  深澤亮、平井剛、加藤麻理依、大沼可奈、越野広雪、袖岡幹子
- Organizer
  第58回天然有機化合物討論会
- Place of Presentation
  東北大学萩ホール
- Year and Date
  2016-09-14
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] Norrish-typeⅡ反応を起こさないα-ケトアミドおよびα-ケトエステルの光反応2016
- Author(s)
  太田英介、三瓶悠、平井剛、越野広雪、長澤和夫、西山繁、袖岡幹子
- Organizer
  第109回有機合成シンポジウム2016年【春】
- Place of Presentation
  東京工業大学
- Year and Date
  2016-06-08
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] フィサリンの全合成研究: エンインメタセシスを基盤としたABC環部構築法の開拓2016
- Author(s)
  森田昌樹、平井剛、袖岡幹子
- Organizer
  日本化学会第96回春季年会
- Place of Presentation
  同志社大学京田辺キャンパス（京都府京田辺市）
- Year and Date
  2016-03-24
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 生物活性分子創製研究と有機合成研究の融合2016
- Author(s)
  平井　剛
- Organizer
  熊本大学理学部化学特別講義C講演会
- Place of Presentation
  熊本大学理学部
- Year and Date
  2016-05-24
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 高機能性複合糖質の創製2016
- Author(s)
  平井剛
- Organizer
  日本化学会中国四国支部地区化学講演会「「有機化学者による生命科学へのアプローチ」
- Place of Presentation
  岡山大学理学部
- Year and Date
  2016-12-10
- Invited
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] がん細胞選択的な細胞死誘導活性を有するγ-リノレン酸の機能性誘導体の創製2016
- Author(s)
  福島翔・平井剛・佐藤綾人・田村結城・どど孝介・袖岡幹子
- Organizer
  第6回CSJ化学フェスタ2016
- Place of Presentation
  タワーホール船堀
- Year and Date
  2016-11-14
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] 高機能性複合糖質の創製2016
- Author(s)
  平井　剛
- Organizer
  日本化学会中国四国支部地区化学講演会「有機化学者による生命科学へのアプローチ」
- Place of Presentation
  岡山大学理学部
- Year and Date
  2016-12-10
- Invited
- Data Source
  KAKENHI-PUBLICLY-16H01167
[Presentation] シアリダーゼの機能解析を志向した3位修飾型シアル酸誘導体の合成と活性評価2016
- Author(s)
  深澤亮、平井剛、加藤麻理依、大沼可奈、越野広雪、袖岡幹子
- Organizer
  第58回天然有機化合物討論会
- Place of Presentation
  東北大萩ホール
- Year and Date
  2016-09-15
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] Spectomycin A1全異性体の合成とSUMO化阻害活性2015
- Author(s)
  平井剛、野村勇作、Frederic Thuaud、前田里子、伊藤昭博、吉田稔、市川聡、松田彰、袖岡幹子
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学川内萩ホール（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] Synthetic strategy toward unique complex right-side structures of physalins2015
- Author(s)
  Masaki Morita, Shuntaro Kojima, Go Hirai, Mikiko Sodeoka
- Organizer
  Molecular Function of Natural Products: Advances towards Chemical Biology, PacifiChem 2015
- Place of Presentation
  Honolulu (USA)
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] Spectomycin A1全異性体の合成とSUMO化阻害活性2015
- Author(s)
  平井剛、野村勇作、Frederic Thuaud、前田里子、伊藤昭博、吉田稔、市川聡、松田彰、袖岡幹子
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学川内萩ホール（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] Spectomycin A1 全立体異性体の合成とSUMO化阻害活性2015
- Author(s)
  野村勇作、 Frederic Thuaud、関根大介、平井剛、前田里子、伊藤昭博、市川聡、松田彰、吉田稔、袖岡幹子
- Organizer
  第57回天然有機化合物討論会
- Place of Presentation
  神奈川県民ホール（神奈川県横浜市）
- Year and Date
  2015-09-09
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] Fluorine containing C-linked gangliosides GM3 analogs: Synthesis, conformational analysis, and biological activities2015
- Author(s)
  Go Hirai, Marie Kato, Kana Oonuma, Eri Nishizawa, Hiroyuki Koshino, Mikiko Sodeoka
- Organizer
  Molecular Function of Natural Products: Advances towards Chemical Biology, PacifiChem 2015
- Place of Presentation
  Honolulu (USA)
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] Fluorine containing C-linked gangliosides GM3 analogs: Synthesis, conformational analysis, and biological activities2015
- Author(s)
  Go Hirai, Marie Kato, Kana Oonuma, Eri Nishizawa, Hiroyuki Koshino, Mikiko Sodeoka
- Organizer
  Molecular Function of Natural Products: Advances towards Chemical Biology, PacifiChem 2015
- Place of Presentation
  Honolulu (USA)
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K12760
[Presentation] Fluorine Containing C-linked Gangliosides GM3 Analogues2014
- Author(s)
  Go Hirai
- Organizer
  Shibasaki Seminar
- Place of Presentation
  Bikaken, Gotanda, Tokyo
- Year and Date
  2014-11-14
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 糖脂質のケミカルバイオロジーを志向した有機化学2014
- Author(s)
  平井剛
- Organizer
  有機合成化学協会関東支部主催「若手研究者のためのセミナー」
- Place of Presentation
  東京大学、本郷キャンパス、東京
- Year and Date
  2014-11-15
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] シアリダーゼ耐性型ガングリオシドの創製2014
- Author(s)
  平井剛
- Organizer
  GlycoTOKYO2014シンポジウム
- Place of Presentation
  千葉大、松戸、千葉
- Year and Date
  2014-11-08
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 生物活性分子を創る：機能と構造に着目した合成化学的アプローチ2014
- Author(s)
  平井剛
- Organizer
  2014年度上智大学物質生命理工学部コロキウム
- Place of Presentation
  上智大学、四谷、東京
- Year and Date
  2014-07-08
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 天然物を基盤とする生物活性分子創製2014
- Author(s)
  平井剛
- Organizer
  理研シンポジウム「有機合成化学を起点とするものづくり戦略」
- Place of Presentation
  理化学研究所、和光市、埼玉
- Year and Date
  2014-06-09
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] Synthetic Study Aiming at SAR Investigations of Spectomycins2013
- Author(s)
  Yusaku Nomura, Frederic Thuaud, Go Hirai, Akihiro Ito, Minoru Yoshida, Mikiko Sodeoka
- Organizer
  3rd ACP Junior Symposium
- Place of Presentation
  Chiba, Japan
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Creation of Novel Biologically Active Molecules Designed Based on Natural Products2013
- Author(s)
  Go Hirai
- Organizer
  ACP lectureship Tour
- Place of Presentation
  Chulabhorn Research Institute, Mehidol University, Kasetsart University, Chulalongkorn University、Thailand
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Design and Development of Fluorine Containing Gangliosides: Establishing the Concept of Conformational Control2013
- Author(s)
  Go Hirai
- Organizer
  日本化学会第93春季年会アジア国際シンポジウム
- Place of Presentation
  立命館大学、滋賀県
- Year and Date
  2013-03-24
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Synthetic studies of spectomycins, protein SUMOylation inhibitors2013
- Author(s)
  Go Hirai
- Organizer
  The 2nd International Symposium on Chemical Biology of Natural Products: Target ID and Regulation of Bioactivity
- Place of Presentation
  Yokohama,Japan
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] 天然物を元に設計した新しい分子によるタンパク質リン酸化制御2012
- Author(s)
  平井　剛
- Organizer
  新学術領域研究「天然物ケミカルバイオロジー」第2回若手研究者ワークショップ
- Place of Presentation
  大阪大学、大阪
- Year and Date
  2012-10-30
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Isobenzofuranone誘導体を基盤としたProtein Kinase C阻害剤の開発2012
- Author(s)
  酒井基成、田村結城、平井剛、袖岡幹子
- Organizer
  日本薬学会第132年会
- Place of Presentation
  札幌
- Year and Date
  2012-03-31
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] 代謝安定性の獲得とコンホメーション制御を可能にする含フッ素ガングリオシド2012
- Author(s)
  平井　剛
- Organizer
  「有機合成化学を起点とするものづくり戦略」第2回ミニシンポジウム
- Place of Presentation
  北海道大学、北海道
- Year and Date
  2012-09-28
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Synthesis of Natural Product Derivatives Which Control the Post-translational Modifications of Proteins2012
- Author(s)
  Go Hirai
- Organizer
  The 1st International Symposium on Chemical Biology of Natural Products: Yarget ID and Regulation of Bioactivity
- Place of Presentation
  京都
- Year and Date
  2012-10-31
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 天然物を基に設計した新しい生理活性分子の合成と機能2012
- Author(s)
  平井剛
- Organizer
  工学院大学大学院講義「化学応用学特論A」
- Place of Presentation
  京都
- Year and Date
  2012-11-05
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 天然物を元に設計した新しい分子によるタンパク質リン酸化制御2012
- Author(s)
  平井剛
- Organizer
  新学術領域研究「天然物ケミカルバイオロジー」第2回若手研究者ワークショップ
- Place of Presentation
  大阪大学
- Year and Date
  2012-10-30
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 天然物を基に設計した新しい生理活性分子の合成と機能2012
- Author(s)
  平井　剛
- Organizer
  工学院大学大学院講義「化学応用学特論Ａ」
- Place of Presentation
  工学院大学、東京
- Year and Date
  2012-11-05
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] シアリダーゼ耐性型ガングリオシドGM3アナログの有機合成化学と生物活性2011
- Author(s)
  平井剛
- Organizer
  東北大学グローバルCOEプログラム「分子系高次構造体化学国際教育研究拠点」シンポジウム
- Place of Presentation
  仙台
- Year and Date
  2011-11-19
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Novel isobenzofuranone derivatives having Protein Kinase Cinhibitory activity2010
- Author(s)
  Yuki Tamura, Go Hirai, Megumi Ohkubo, Mikiko Sodeoka
- Organizer
  EMBO Conference Series, Chemical Biology 2010
- Place of Presentation
  Heidelberg, Germany
- Year and Date
  2010-09-24
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] Synthesis and biological evaluation of DEFGH-ring system of physalins2010
- Author(s)
  Go Hirai
- Organizer
  2010 RIKEN Chemical Biology International Symposium
- Place of Presentation
  理化学研究所、埼玉県和光市
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Design, synthesis, and biological evaluation of physalins analogues2010
- Author(s)
  Go Hirai
- Organizer
  Pacifichem 2010
- Place of Presentation
  Hawaii, USA
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 天然物や生体分子を基盤とした生理活性分子の創製2010
- Author(s)
  平井剛
- Organizer
  第54回日本薬学会関東支部大会
- Place of Presentation
  東京
- Year and Date
  2010-10-02
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] Synthesis and Biological Evaluation of DEFGH-ring System of Physalins、The 5th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-5)2010
- Author(s)
  Go Hirai
- Organizer
  The 1st New phase International Conference on Cutting-Edge Organic Chemistry in Asia (NICCEOCA-1)
- Place of Presentation
  Hsinchu, Taiwan
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 新規イソベンゾフラノン誘導体のPKC阻害機構の解析2010
- Author(s)
  田村結城、平井剛、袖岡幹子
- Organizer
  日本がん分子標的治療学会第14回学術集会
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] Synthesis and Biological Evaluation of DEFGH-ring System of Physalins2010
- Author(s)
  Go Hirai
- Organizer
  The 5th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-5), The 1st New phase International Conference on Cutting-Edge Organic Chemistry in Asia (NICCEOCA-1)
- Place of Presentation
  Hsinchu, Taiwan
- Year and Date
  2010-11-08
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 天然物や生体分子を基盤とした生理活性分子の創製2010
- Author(s)
  平井剛
- Organizer
  第54回日本薬学会関東支部大会
- Place of Presentation
  東京
- Year and Date
  2010-10-02
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Study on PKC inhibition by novel isobenzofuranone derivatives and their mechanism of action2009
- Author(s)
  Yuki Tamura, Go Hirai, Megumi Ohkubo, Mikiko Sodeoka
- Organizer
  The 25^<th> NAITO Conference on Chemical Biology[II]
- Place of Presentation
  Sapporo
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] 新規Isobenzofuranone誘導体のPKC阻害活性と作用機序に関する研究2009
- Author(s)
  田村結城、平井剛、大窪恵、袖岡幹子
- Organizer
  日本ケミカルバイオロジー学会第4回年会
- Place of Presentation
  神戸
- Data Source
  KAKENHI-PROJECT-21603016
[Presentation] Development of RK-682 enamide derivatives and attempts at comprehensive analysis of their target proteins in cells2008
- Author(s)
  Go Hirai
- Organizer
  THE 22nd NAITO CONFERENCE ON Chemical Biology[I]
- Place of Presentation
  Sapporo
- Year and Date
  2008-09-11
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] RK-682エナミド誘導体標的酵素の網羅的解析法の開発2008
- Author(s)
  平井剛
- Organizer
  日本化学会第88春季年会
- Place of Presentation
  立教大学
- Year and Date
  2008-03-29
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] RK-682エナミド誘導体標的酵素の網羅的解析法の開発2008
- Author(s)
  平井剛
- Organizer
  日本化学会第88春季年会
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] RK-682エナミド誘導体標的酵素の網羅的解析法の開発2008
- Author(s)
  平井剛
- Organizer
  日本化学会第88春季年会
- Place of Presentation
  立教大学
- Data Source
  KAKENHI-PROJECT-16073203
[Presentation] Development of RK-682 enamide derivatives and attempts at comprehensive analysis of their target proteins in cells2008
- Author(s)
  Go Hirai
- Organizer
  THE 22nd NAITO CONFERENCE ON Chemical Biology [I]
- Place of Presentation
  札幌
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] Development of Dual-specificity Protein Phosphatase Inhibitor2008
- Author(s)
  Go Hirai
- Organizer
  The First RIKEN Chemical Biolgy Deprtmnt Internatioal Symposium
- Place of Presentation
  熱海
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] RK-682エナミド誘導体標的酵素の網羅的解析法の開発2008
- Author(s)
  平井剛
- Organizer
  日本ケミカルバイオロジー研究会第三回年会
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] Synthesis of RK-682 enamide derivatives as novel dual-specificity protein phosphatase inhibitors2007
- Author(s)
  Go Hirai
- Organizer
  RIKEN International Symposium on Chemical Biology 2007
- Place of Presentation
  箱根・山のホテル
- Year and Date
  2007-11-12
- Data Source
  KAKENHI-PROJECT-16073203
[Presentation] 細胞内ホスファターゼ解析を志向した不可逆的阻害剤の開発2007
- Author(s)
  平井剛
- Organizer
  平成19年度「若手研究者のためのセミナー」
- Place of Presentation
  慶応大学
- Year and Date
  2007-10-27
- Data Source
  KAKENHI-PROJECT-19710195
[Presentation] Fluorine Containing C-linked Gangliosides Analogues
- Author(s)
  Go Hirai
- Organizer
  The First Asian Conference for "MONODUKURI" Strategy by Synthetic Organic Chemistry (ACMS)
- Place of Presentation
  Okinawa, Japan
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] 有機合成化学を活かした天然物基盤のケミカルバイオロジー研究
- Author(s)
  平井　剛
- Organizer
  早稲田大学講演会
- Place of Presentation
  早稲田大学
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] 生物活性物質を創る有機合成化学研究
- Author(s)
  平井　剛
- Organizer
  第1回慶應有機化学若手シンポジウム
- Place of Presentation
  慶應義塾大学
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] 分子設計と有機合成による高機能型生物活性分子の創製
- Author(s)
  平井剛
- Organizer
  第31回有機合成化学セミナー
- Place of Presentation
  志賀島、福岡
- Year and Date
  2014-09-17 – 2014-09-19
- Invited
- Data Source
  KAKENHI-PUBLICLY-26102744
[Presentation] 天然物を基に設計した新しい生理活性分子の合成と機能
- Author(s)
  平井剛
- Organizer
  工学院大学大学院講義「化学応用学特論Ａ」
- Place of Presentation
  工学院大学、東京都
- Invited
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] 酵素に分解されない糖脂質の開発
- Author(s)
  平井　剛
- Organizer
  東京大学工学部　化学生命工学科講演会「化学と生命のかけはし」
- Place of Presentation
  東京大学
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] 天然物を基にした分子設計を足がかりとするものづくり
- Author(s)
  平井　剛
- Organizer
  第3回CSJ化学フェスタ2013ナノ機能への挑戦－材料、素子、バイオ、そして未来－
- Place of Presentation
  船堀
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Creation of Novel Biologically Active Molecules Designed Based on Natural Products
- Author(s)
  Go Hirai
- Organizer
  ACP lectureship Tour at Chulabhorn Research Institute
- Place of Presentation
  Chulabhorn Research Institute, Thailand
- Invited
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] CHF連結型シアリルガラクトースの合成とコンホメーション
- Author(s)
  平井　剛
- Organizer
  理研シンポジウム：第14回分析・解析技術と化学の最先端
- Place of Presentation
  理化学研究所
- Invited
- Data Source
  KAKENHI-PUBLICLY-24102534
[Presentation] Creation of Novel Biologically Active Molecules Designed Based on Natural Products
- Author(s)
  Go Hirai
- Organizer
  ACP lectureship Tour at Mehidol University
- Place of Presentation
  Mehidol University, Thailand
- Invited
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Creation of Novel Biologically Active Molecules Designed Based on Natural Products
- Author(s)
  Go Hirai
- Organizer
  ACP lectureship Tour at Chulabhorn Research Institute
- Place of Presentation
  Kasetsart University, Thailand
- Invited
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] Creation of Novel Biologically Active Molecules Designed Based on Natural Products
- Author(s)
  Go Hirai
- Organizer
  ACP lectureship Tour at Chulabhorn Research Institute
- Place of Presentation
  Chulalongkorn University, Thailand
- Invited
- Data Source
  KAKENHI-PROJECT-22603014
[Presentation] In-cell NMRを志向したDOTA-M8リガンドの合成研究
- Author(s)
  彦根　佑哉，平井　剛，袖岡　幹子，三島　正規，伊藤　隆
- Organizer
  第５３回NMR討論会
- Place of Presentation
  吹田
- Year and Date
  2014-11-14 – 2014-11-16
- Data Source
  KAKENHI-PROJECT-25650025

1. SODEOKA Mikiko (60192142)

# of Collaborated Projects: 5 results

# of Collaborated Products: 9 results
2. HAMASHIMA Yoshitaka (40333900)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
3. Yashiroda Yoko (60360658)

# of Collaborated Projects: 2 results

# of Collaborated Products: 3 results
4. KOSONO Saori (90321760)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
5. SUZUKI Takehiro (60415198)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
6. TAMURA Yuki (50442984)

# of Collaborated Projects: 1 results

# of Collaborated Products: 7 results
7. TSUCHIYA Ayako (80442987)

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
8. OZAWA Masaaki (30617262)

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
9. ITO Akihiro (40391859)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
10. MISHIMA Masaki (70346310)

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
11. ITO Yutaka (80261147)

# of Collaborated Projects: 1 results

# of Collaborated Products: 2 results
12. 上村春樹 (60184975)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
13. 山田健一 (60346806)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
14. 柴田貴広 (80447838)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
15. 今井浩孝 (50255361)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
16. 小林進

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
17. 鈴木孝洋

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
18. 太田英介

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
19. 植木雅志

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
20. 田中克典

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
21. 深瀬浩一

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
22. 掛谷秀昭

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
23. 寄立麻琴

# of Collaborated Projects: 0 results

# of Collaborated Products: 3 results
24. 臼井一晃

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
25. 大神田淳子

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
26. 唐沢悟

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
27. 塩崎一弘

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

Hirai Go 平井 剛

HIRAI Go 平井 剛

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Catalytic synthesis of pseudo-natural products utilizing photo-reactionPrincipal Investigator

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Synthetic chemistry for the development of oligosaccharide-type sialidase inhibitorsPrincipal Investigator

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中分子グライコミメティクスの開拓Principal Investigator

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代謝安定型糖鎖を基盤とする高次生物機能中分子複合糖質アナログ創製Principal Investigator

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Synthetic chemistry for the development of oligosaccharide-type sialidase inhibitorsPrincipal Investigator

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代謝安定型糖鎖を基盤とする高次生物機能複合糖質アナログの創製Principal Investigator

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Development of a novel type of carbohydrate probesPrincipal Investigator

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酸化ステロイドの鍵構造アナログ創製と作用機序解析Principal Investigator

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タンパク質ＳＵＭＯ化を阻害する天然物リガンドの合成供給と構造活性相関Principal Investigator

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Hirai Go 平井剛

HIRAI Go 平井剛