Ohno Hiroaki 大野浩章

… Alternative Names

OHNO Hiroaki 大野浩章

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Researcher Number	30322192
Other IDs
External Links
Affiliation (Current)	2025: 京都大学, 薬学研究科, 教授
Affiliation (based on the past Project Information) *help	2022 – 2024: 京都大学, 薬学研究科, 教授 2015 – 2020: 京都大学, 薬学研究科, 教授 2013 – 2016: 京都大学, 薬学研究科(研究院), 教授 2014: 京都大学, 大学院薬学研究科, 教授 2011 – 2013: 京都大学, 薬学研究科(研究院), 准教授 … More 2011: 京都大学, 大学院・薬学研究科, 准教授 2007 – 2011: Kyoto University, 薬学研究科, 准教授 2005 – 2006: 京都大学, 薬学研究科, 助教授 2004: 大阪大学, 薬学研究所, 助手 2000 – 2004: 大阪大学, 薬学研究科, 助手 Less
Review Section/Research Field	Principal Investigator Chemical pharmacy / Science and Engineering / Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related / Basic Section 47050:Environmental and natural pharmaceutical resources-related / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Medium-sized Section 33:Organic chemistry and related fields / Transition State Control / Chemical pharmacy Except Principal Investigator Drug development chemistry / Biological Sciences / Medium-sized Section 49:Pathology, infection/immunology, and related fields / Chemical pharmacy / Chemical pharmacy
Keywords	Principal Investigator 連続反応 / 金触媒 / アルカロイド / インドール / 反応集積化 / 有機化学 / アレン / パラジウム / 中分子 / 創薬 … More / スフィンゴ脂質 / カルバゾール / Ergotアルカロイド / 原子効率 / 多成分反応 / スルファミド / 複素環 / パラジウム触媒 / ケミカルスペース / ひずみ分子 / π共役分子 / ベンゾフルオランテン / ジベンゾフルオレン / フェナントレン / π共役系 / お椀型分子 / ビニルカチオン / 多環式芳香族化合物 / 天然物合成 / マクロ環化 / 骨格構築 / 多環式骨格 / 近接効果 / ストリクタミン / キノカルシン / 天然物 / 薬らしさ / 化合物ライブラリー / 全合成 / 多重結合 / キナーゼ阻害剤 / アセトゲニン / 遷移金属触媒 / 多環式芳香環 / 全合成研究 / 抗腫瘍活性 / テトラヒドロフラン / 構造活性相関研究 / ポリイン / インドールアルカロイド / アルケンイソスター / C-H活性化 / リゼルグ酸 / β-カルボリン / アミジン / イソキノリン / 金 / 銅 / ベンゾイソインドール / CH活性化 / 銅触媒 / ソクロブタン / 環化付加反応 / パラジウムカルベン / シクロプロパン / ヘテロ中員環 / タンデム反応 / 触媒反応 / 立体選択的合成 / 軸不斉 / ジエチル亜鉛 / 有機銅試薬 / アミノアレン … More Except Principal Investigator ケモカイン / CXCR4 / 癌 / 構造活性相関 / ペプチド / スクリーニング / 天然物 / 複素環 / キナーゼ / 創薬テンプレート / 薬剤耐性 / GPR54 / パラジウム触媒 / 抗ウイルス薬 / ヌクレオカプシド / エボラウイルス / BIRドメイン / カスパーゼ / SH2ドメイン / 医薬品探索 / キラル化合物 / 環状ペプチド / 合理的分子設計 / GPCR / π-Allyl Palladium / Amino Allenes / Diethylzinc / Palladium Catalyst / Sulfinyl Anion / Ketyl Radical / Spirocyclization / Samarium Iodide / アレン / HMPA / SmI2 / π-アリルパラジウム錯体 / アミノアレン / ジエチル亜鉛 / スルフィニルアニオン / ケチルラジカル / スピロ閉環反応 / ヨウ化サマリウム / 天然有機化合物 / 鏡像体 / 生物活性化合物 / アッセイ / 化合物ライブラリー / 複素環骨格構築反応 / ケモカイン受容体 / ドラッグライク / 分子設計 / キネシンモータータンパク / FC131 / jaspine B / スフィンゴシンキナーゼ / プロテインキナーゼCK2 / ホモロジーモデル / CXCR7ケモカイン受容体 / CXCR4ケモカイン受容体 / キネシン / KSP / CK2 / CXCR7 / 固相反応 / コンビナトリアル合成 / インドール / インドリン / キノリン / イソキノリン / 多成分反応 / ケミカルバイオロジー / ドラッグ指向性 / 化合物バンク / Kisspeptin / Eg5 / SDF-1 / ビニルスルホキシド / スルフェン酸亜鉛 / タンデム反応 / シクロプロパン / パラジウムカルベン Less

フィロウイルスの増殖機構の分子構造基盤の解明と制御法の開発
- Principal Investigator
  
  野田岳志
- Project Period (FY)
  2024 – 2026
- Research Category
  
  Grant-in-Aid for Scientific Research (A)
- Review Section
  
  Medium-sized Section 49:Pathology, infection/immunology, and related fields
- Research Institution
  Kyoto University
Natural product syntheses based on cascade cyclization and their applications to middle-molecule drug modalitiesPrincipal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2023 – 2026
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
  Basic Section 47050:Environmental and natural pharmaceutical resources-related
  Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related
- Research Institution
  Kyoto University
Synthesis of Novel Bowl-Shaped Highly pi-Conjugated Molecules Based on the Original Vinylcation FormationPrincipal Investigator
- Principal Investigator
  
  Ohno Hiroaki
- Project Period (FY)
  2022 – 2023
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 33:Organic chemistry and related fields
- Research Institution
  Kyoto University
Alkaloid Synthesis and Its Middle Molecular Strategy Based on Reaction IntegrationPrincipal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2018 – 2019
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Research Institution
  Kyoto University
Synthetic and medicinal studies on bioactive indole alkaloids based on direct construction of polycyclic ring systemsPrincipal Investigator
- Principal Investigator
  
  Hiroaki Ohno
- Project Period (FY)
  2017 – 2020
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Precise activation based on transition state control using neighboring effect and its medicinal applicationPrincipal Investigator
- Principal Investigator
  
  Ohno Hiroaki
- Project Period (FY)
  2015 – 2018
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Transition State Control
- Research Institution
  Kyoto University
Development of Novel Drug Discovery Technologies for Target Proteins with Elusive Molecular Basis
- Principal Investigator
  
  Fujii Nobutaka
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Develoment of a screening platform using mirror-image proteins and their application to drug discovery
- Principal Investigator
  
  Shinya Oishi
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
原子移動型反応の高度集積化による多環式芳香族化合物の合成と創薬展開Principal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2012 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Review Section
  
  Science and Engineering
- Research Institution
  Kyoto University
Development and application of a novel screening technolgy toward effective uses of chemical library
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2012 – 2014
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Innovative Molecular Transformations Based on Consecutive pai-Activation and Their Medicinal ApplicationsPrincipal Investigator
- Principal Investigator
  
  Hiroaki Ohno
- Project Period (FY)
  2012 – 2016
- Research Category
  
  Grant-in-Aid for Young Scientists (A)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Practical medicinal chemistry on the basis of protein chemistry, computational science and synthetic technologies for a variety of heterocycles
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2011 – 2014
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
触媒的多成分反応・高原子効率反応の高度集積化と創薬展開Principal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2010 – 2011
- Research Category
  
  Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
- Review Section
  
  Science and Engineering
- Research Institution
  Kyoto University
Divergent syntheses of biologically active compounds based on catalytic cascade cyclization reactionsPrincipal Investigator
- Principal Investigator
  
  OHNO Hiroaki
- Project Period (FY)
  2010 – 2011
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
多重標的創薬概念に基づくがん化学療法の新機軸
- Principal Investigator
  
  OISHI Shinya, 藤井信孝
- Project Period (FY)
  2008 – 2009
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
GPCR周辺の細胞外環境解明のためのケミカルプローブの創出と応用
- Principal Investigator
  
  大石真也, 藤井信孝
- Project Period (FY)
  2008 – 2009
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
Development of highly atom-economical synthetic methods based on catalytic cascade reactionsPrincipal Investigator
- Principal Investigator
  
  OHNO Hiroaki
- Project Period (FY)
  2007 – 2009
- Research Category
  
  Grant-in-Aid for Young Scientists (A)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
癌転移・骨髄依存薬物耐性の動的超分子機構解明のケミカルプローブ創出と創薬展開
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2006 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
ドラッグ指向性化合物バンクの構築と創薬展開
- Principal Investigator
  
  藤井信孝
- Project Period (FY)
  2006 – 2007
- Research Category
  
  Grant-in-Aid for Exploratory Research
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
複雑な構造を有する生物活性複素環の一挙合成法の開発と環境調和型連続反応への展開Principal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2005 – 2006
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
パラジウム触媒を用いた新規反応活性種の創出と合成反応への利用
- Principal Investigator
  
  TANAKA Tetsuaki
- Project Period (FY)
  2003 – 2004
- Research Category
  
  Grant-in-Aid for Exploratory Research
- Research Field
  
  Chemical pharmacy
- Research Institution
  Osaka University
生物活性を有する含窒素複素環の自在な合成を指向した新規環形成反応の開発研究Principal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2003 – 2004
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Osaka University
Synthesis of Biologically Active Compounds Using Potential Utility of Transition Metals
- Principal Investigator
  
  TANAKA Tetsuaki
- Project Period (FY)
  2001 – 2002
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Osaka University
高活性な降圧剤及びプロテアーゼ阻害剤の開発を指向したアミノアレンの合成研究Principal Investigator
- Principal Investigator
  
  大野浩章
- Project Period (FY)
  2000 – 2001
- Research Category
  
  Grant-in-Aid for Encouragement of Young Scientists (A)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Osaka University

[Book] Transition-Metal-Mediated Aromatic Ring Construction2013
- Author(s)
  Ohno, H.
- Total Pages
  797
- Publisher
  Wiley-VCH
- Data Source
  KAKENHI-PROJECT-24689001
[Book] Transition-Metal-Mediated Aromatic Ring Construction2013
- Author(s)
  Ohno, H.
- Total Pages
  797
- Publisher
  Wiely-VCH
- Data Source
  KAKENHI-PUBLICLY-24106720
[Book] Synthesis by substitution, linear allene, in science of synthesis.2007
- Author(s)
  Ohno H.
- Publisher
  Thieme
- Data Source
  KAKENHI-PROJECT-18015027
[Book] Aziridines and Epoxides in Organic Synthesis2005
- Author(s)
  Hiroaki Ohno
- Total Pages
  492
- Publisher
  Wiley-VCH : Weinheim
- Data Source
  KAKENHI-PROJECT-17790013
[Book] Modern Allene Chemistry (Vol.1)2004
- Author(s)
  Hiroaki Ohno
- Total Pages
  592
- Publisher
  Wiley-VCH : Weinheim
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Synthesis of labionin and avionin precursors via a nitrogen-centred-radical-triggered 1,5-HAT reaction of Tris derivatives2024
- Author(s)
  Yamaguchi Ayuta、Obiya Naoki、Arichi Norihito、Oishi Shinya、Ohno Hiroaki、Inuki Shinsuke
- Journal Title
  
  Organic & Biomolecular Chemistry
  
  Volume: 22 Issue: 10 Pages: 2049-2055
- DOI
  10.1039/d3ob02037a
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K17975, KAKENHI-PROJECT-23K27294
[Journal Article] Construction of a Bicyclo[2.2.2]octene Skeleton via a Visible-Light-Mediated Radical Cascade Reaction of Amino Acid Derivatives with <i>N</i>-(2-Phenyl)benzoyl Groups2023
- Author(s)
  Yoshida Yuki、Takeuchi Haruka、Nakagawa Kohei、Fujii Toshiki、Arichi Norihito、Oishi Shinya、Ohno Hiroaki、Inuki Shinsuke
- Journal Title
  
  Organic Letters
  
  Volume: 25 Issue: 26 Pages: 4846-4851
- DOI
  10.1021/acs.orglett.3c01586
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K27294
[Journal Article] Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I)2023
- Author(s)
  Tsuji Atsuhito、Masuya Takahiro、Arichi Norihito、Inuki Shinsuke、Murai Masatoshi、Miyoshi Hideto、Ohno Hiroaki
- Journal Title
  
  ACS Medicinal Chemistry Letters
  
  Volume: 14 Issue: 2 Pages: 211-216
- DOI
  10.1021/acsmedchemlett.2c00504
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K19028, KAKENHI-PROJECT-22K14837, KAKENHI-PROJECT-22KJ1917, KAKENHI-PROJECT-23K23540
[Journal Article] Gold(I)‐Catalyzed Bis‐Cyclization of Allenynes for the Synthesis of Strained and Planar Polycyclic Compounds2023
- Author(s)
  Tsuno Hitomi、Shen Jingfeng、Komatsu Hiroki、Arichi Norihito、Inuki Shinsuke、Ohno Hiroaki
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 62 Issue: 35
- DOI
  10.1002/anie.202307532
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K19028, KAKENHI-PROJECT-23K27294
[Journal Article] Alkoxymigration onto α‐Imino Gold Carbenes for Constructing Propellane‐Type Indolines2023
- Author(s)
  Greiner Luca C.、Arichi Norihito、Inuki Shinsuke、Ohno Hiroaki
- Journal Title
  
  Asian Journal of Organic Chemistry
  
  Volume: 12 Issue: 7
- DOI
  10.1002/ajoc.202300232
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K19028, KAKENHI-PROJECT-23K27294
[Journal Article] Archaeal glycerolipids are recognized by C-type lectin receptor Mincle.2023
- Author(s)
  Oka S, Watanabe M, Ito E, Takeyama A, Matsuoka T, Takahashi M, Izumi Y, Arichi N, Ohno H*, Yamasaki S*, Inuki S*.
- Journal Title
  
  Journal of the American Chemical Society
  
  Volume: 145(33) Issue: 33 Pages: 18538-18548
- DOI
  10.1021/jacs.3c05473
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K18924, KAKENHI-PROJECT-23K17975, KAKENHI-PLANNED-22H05183, KAKENHI-PLANNED-22H05185, KAKENHI-PROJECT-23H00403, KAKENHI-PROJECT-23K23151, KAKENHI-PROJECT-23K27294
[Journal Article] Gold(I)-Catalyzed Cascade Cyclization of Alkynyl Indoles for the Stereoselective Construction of the Quaternary Carbon Center of Akuammiline Alkaloids2023
- Author(s)
  Hashimoto Naoki、Taguchi Junichi、Arichi Norihito、Inuki Shinsuke、Ohno Hiroaki
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 88 Issue: 24 Pages: 17306-17321
- DOI
  10.1021/acs.joc.3c02142
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K19028, KAKENHI-PROJECT-23K27294
[Journal Article] Establishment of an MR1 Presentation Reporter Screening System and Identification of Phenylpropanoid Derivatives as MR1 Ligands2023
- Author(s)
  Matsuoka Takuro、Hattori Akira、Oishi Shinya、Araki Mitsugu、Ma Biao、Fujii Toshiki、Arichi Norihito、Okuno Yasushi、Kakeya Hideaki、Yamasaki Sho、Ohno Hiroaki、Inuki Shinsuke
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: 66 Issue: 17 Pages: 12520-12535
- DOI
  10.1021/acs.jmedchem.3c01122
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23K17975, KAKENHI-PROJECT-22K06677, KAKENHI-PROJECT-22KJ1866, KAKENHI-PLANNED-22H05183, KAKENHI-PLANNED-23H04882, KAKENHI-PROJECT-23H00403, KAKENHI-PROJECT-23K27294
[Journal Article] A Proximity‐Induced Fluorogenic Reaction Triggered by Antibody?Antigen Interactions with Adjacent Epitopes2023
- Author(s)
  Nishiyama Kentaro、Akiba Hiroki、Nagata Satoshi、Tsumoto Kouhei、Kamada Haruhiko、Ohno Hiroaki
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 62 Issue: 30
- DOI
  10.1002/anie.202306431
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-21K06453, KAKENHI-PROJECT-23K27294
[Journal Article] Gold(I)‐Catalyzed Benzylic C(sp3)-H Functionalizations: Divergent Synthesis of Indole[a]‐ and [b]‐Fused Polycycles2022
- Author(s)
  Greiner Luca C.、Arichi Norihito、Inuki Shinsuke、Ohno Hiroaki
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 62 Issue: 3
- DOI
  10.1002/anie.202213653
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22K19028
[Journal Article] Nonbiomimetic total synthesis of indole alkaloids using alkyne-based strategies2021
- Author(s)
  Ohno Hiroaki、Inuki Shinsuke
- Journal Title
  
  Organic & Biomolecular Chemistry
  
  Volume: 19 Issue: 16 Pages: 3551-3568
- DOI
  10.1039/d0ob02577a
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17H03971
[Journal Article] Total Synthesis of (+)-Polyoxamic Acid via Visible-Light-Mediated Photocatalytic β-Scission and 1,5-Hydrogen Atom Transfer of Glucose Derivative2020
- Author(s)
  Matsuoka Takuro、Inuki Shinsuke、Miyagawa Takashi、Oishi Shinya、Ohno Hiroaki
- Journal Title
  
  The Journal of Organic Chemistry
  
  Volume: 85 Issue: 12 Pages: 8271-8278
- DOI
  10.1021/acs.joc.0c00910
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K06938, KAKENHI-PUBLICLY-20H04773, KAKENHI-PROJECT-17H03971
[Journal Article] Total Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso ‐Cyclization2020
- Author(s)
  Takeuchi Haruka、Inuki Shinsuke、Nakagawa Kohei、Kawabe Takaaki、Ichimura Atsuhiko、Oishi Shinya、Ohno Hiroaki
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 59 Issue: 47 Pages: 21210-21215
- DOI
  10.1002/anie.202009399
- NAID
  120006898144
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K06938, KAKENHI-PUBLICLY-20H04773, KAKENHI-PROJECT-17H03971
[Journal Article] Gold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines2020
- Author(s)
  A. Yamaguchi, S. Inuki, Y. Tokimizu, S. Oishi, H. Ohno
- Journal Title
  
  J. Org. Chem.
  
  Volume: 85 Issue: 4 Pages: 2543-2559
- DOI
  10.1021/acs.joc.9b03256
- NAID
  120006817609
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408, KAKENHI-PUBLICLY-18H04615, KAKENHI-PROJECT-17H03971
[Journal Article] Total Synthesis of Dictyodendrins A－F by the Gold‐Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole2020
- Author(s)
  Matsuoka Junpei、Inuki Shinsuke、Matsuda Yuka、Miyamoto Yoichi、Otani Mayumi、Oka Masahiro、Oishi Shinya、Ohno Hiroaki
- Journal Title
  
  Chemistry － A European Journal
  
  Volume: 26 Issue: 49 Pages: 11150-11157
- DOI
  10.1002/chem.202001950
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20K06455, KAKENHI-PROJECT-17H03971
[Journal Article] Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes2019
- Author(s)
  T. Ikeuchi, S. Inuki, S. Oishi, H. Ohno
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 58 Issue: 23 Pages: 7792-7796
- DOI
  10.1002/anie.201903384
- NAID
  120006634622
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408, KAKENHI-PROJECT-17H03971
[Journal Article] Construction of Quaternary Carbon Stereocenter of α-Tertiary Amine through Remote C-H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin2019
- Author(s)
  Miyagawa Takashi、Inuki Shinsuke、Oishi Shinya、Ohno Hiroaki
- Journal Title
  
  Organic Letters
  
  Volume: 21 Issue: 14 Pages: 5485-5490
- DOI
  10.1021/acs.orglett.9b01778
- NAID
  120006719313
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04615, KAKENHI-PROJECT-17H03971
[Journal Article] Construction of the Pyrrolo[2,3-d]carbazole Core of Spiroindoline Alkaloids by Gold-Catalyzed Cascade Cyclization of Ynamide2019
- Author(s)
  J. Matsuoka, H. Kumagai, S. Inuki, S. Oishi, H. Ohno
- Journal Title
  
  J. Org. Chem.
  
  Volume: 84 Issue: 14 Pages: 9358-9363
- DOI
  10.1021/acs.joc.9b01149
- NAID
  120006708241
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408, KAKENHI-PROJECT-17H03971, KAKENHI-PROJECT-18J12107
[Journal Article] Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds2018
- Author(s)
  N. Hamada, A. Yamaguchi, S. Inuki, S. Oishi, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 20 Issue: 15 Pages: 4401-4405
- DOI
  10.1021/acs.orglett.8b01524
- NAID
  120006634623
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-17H03971
[Journal Article] Direct synthesis of aryl-annulated [c]carbazoles by gold(I)-catalysed cascade reaction of azide-diynes and arenes2018
- Author(s)
  Yuiki Kawada, Shunsuke Ohmura, Misaki Kobayashi, Wataru Nojo, Masaki Kondo, Yuka Matsuda, Junpei Matsuoka, Shinsuke Inuki, Shinya Oishi, Chao Wang, Tatsuo Saito, Masanobu Uchiyama, Takanori Suzuki, Hiroaki Ohno
- Journal Title
  
  Chem. Sci.
  
  Volume: 9 Issue: 44 Pages: 8416-8416
- DOI
  10.1039/c8sc03525c
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18K06544, KAKENHI-PROJECT-18K06571, KAKENHI-PUBLICLY-18H04376, KAKENHI-PROJECT-15H03790, KAKENHI-PROJECT-18J12107, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-16K13968
[Journal Article] Introduction of a Polar Functional Group to the Lipid Tail of 4-<i>epi</i>-Jaspine B Affects Sphingosine Kinase Isoform Selectivity2018
- Author(s)
  S. Inuki, T. Miyagawa, S. Oishi, H. Ohno
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 66 Issue: 9 Pages: 866-872
- DOI
  10.1248/cpb.c18-00366
- NAID
  130007479591
- ISSN
  0009-2363, 1347-5223
- Year and Date
  2018-09-01
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408, KAKENHI-PUBLICLY-18H04615, KAKENHI-PROJECT-17H03971
[Journal Article] Head-to-Tail Macrocyclization of Cysteine-Free Peptides Using an o-Aminoanilide Linker2018
- Author(s)
  T. Ohara, M. Kaneda, T. Saito, N. Fujii, H. Ohno, S. Oishi
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 28 Issue: 8 Pages: 1283-1286
- DOI
  10.1016/j.bmcl.2018.03.027
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-15J05499
[Journal Article] Direct Synthesis of Aryl-Annulated [c]Carbazoles by Gold(I)-Catalysed Cascade Reaction of Azide-Diynes and Arenes2018
- Author(s)
  Y. Kawada, S. Ohmura, M. Kobayashi, W. Nojo, M. Kondo, Y. Matsuda, J. Matsuoka, S. Inuki, S. Oishi, C. Wang, T. Saito, M. Uchiyama, T. Suzuki, H. Ohno
- Journal Title
  
  Chem. Sci.
  
  Volume: 9 Pages: 8416-8425
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17H03971
[Journal Article] Direct Synthesis of Aryl-Annulated [c]Carbazoles by Gold(I)-Catalysed Cascade Reaction of Azide-Diynes and Arenes2018
- Author(s)
  Y. Kawada, S. Ohmura, M. Kobayashi, W. Nojo, M. Kondo, Y. Matsuda, J. Matsuoka, S. Inuki, S. Oishi, C. Wang, T. Saito, M. Uchiyama, T. Suzuki, H. Ohno
- Journal Title
  
  Chem. Sci.
  
  Volume: 9 Pages: 8416-8425
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Journal Article] Synthesis of Jaspine B Regioisomers through Palladium-Catalyzed Stereoselective Tetrahydrofuran Formation: Insight into the Ligand Recognition of Sphingosine Kinases2018
- Author(s)
  Miyagawa, S. Inuki, M. Honda, S. Nakamura, I. Nakanishi, N. Fujii, S. Oishi, H. Ohno
- Journal Title
  
  Tetrahdron
  
  Volume: 74 Issue: 15 Pages: 1802-1809
- DOI
  10.1016/j.tet.2018.02.042
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PUBLICLY-18H04408, KAKENHI-PROJECT-17H03971
[Journal Article] Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3)2018
- Author(s)
  Sekiguchi Haruka、Kuroyanagi Tomoko、Rhainds David、Kobayashi Kazuya、Kobayashi Yuka、Ohno Hiroaki、Heveker Nikolaus、Akaji Kenichi、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: 61 Issue: 8 Pages: 3745-3751
- DOI
  10.1021/acs.jmedchem.8b00336
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-16H05104
[Journal Article] Identification of Selective Inhibitors of Sphingosine Kinases 1 and 2 through a Structure-Activity Relationship Study of 4-epi-Jaspine B2017
- Author(s)
  H. Ohno, M. Honda, N. Hamada, J. Miyagaki, A. Iwata, K. Otsuki, T. Maruyama, S. Nakamura, I. Nakanishi, S. Inuki, N. Fujii, S. Oishi
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 25 Issue: 12 Pages: 3046-3052
- DOI
  10.1016/j.bmc.2017.03.059
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-17H03971
[Journal Article] Synthesis of Grb2 SH2 domain proteins for mirror-image screening systems.2017
- Author(s)
  Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S.
- Journal Title
  
  Bioconjugate Chemistry
  
  Volume: 28 Issue: 2 Pages: 609-619
- DOI
  10.1021/acs.bioconjchem.6b00692
- Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-26350976, KAKENHI-PROJECT-15H04653
[Journal Article] Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold2017
- Author(s)
  N. Hamada, Y. Yoshida, S. Oishi, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 19 Pages: 3875-3878
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17H03971
[Journal Article] Synthesis of the Src SH2 domain and its application in bioassays for mirror-image screening2017
- Author(s)
  Shu Keitou、Noguchi Taro、Honda Kaori、Kondoh Yasumitsu、Osada Hiroyuki、Ohno Hiroaki、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  RSC Advances
  
  Volume: 7 Issue: 61 Pages: 38725-38732
- DOI
  10.1039/c7ra07445j
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-15H04653
[Journal Article] Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction.2017
- Author(s)
  Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S
- Journal Title
  
  Bioorg Med Chem Lett
  
  Volume: 印刷中 Issue: 11 Pages: 2571-2574
- DOI
  10.1016/j.bmcl.2017.03.082
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-26350976, KAKENHI-PROJECT-15H04653
[Journal Article] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles2017
- Author(s)
  J. Matsuoka, Y. Matsuda, Y. Kawada, S. Oishi, H. Ohno
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 56 Issue: 26 Pages: 7444-7448
- DOI
  10.1002/anie.201703279
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-17H03971
[Journal Article] Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold2017
- Author(s)
  N. Hamada, Y. Yoshida, S. Oishi, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 19 Pages: 3875-3878
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061
[Journal Article] Development of novel NK3 receptor antagonists with reduced environmental impact2016
- Author(s)
  Yamamoto Koki、Okazaki Shiho、Ohno Hiroaki、Matsuda Fuko、Ohkura Satoshi、Maeda Kei-ichiro、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 24 Issue: 16 Pages: 3494-3500
- DOI
  10.1016/j.bmc.2016.05.054
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15H04654
[Journal Article] Gold-Catalyzed Three-Component Spirocyclization: a One-Pot Approach to Functionalized Pyrazolidines2016
- Author(s)
  B. Wagner, W. Hiller, H. Ohno, N. Krause
- Journal Title
  
  Org. Biomol. Chem.
  
  Volume: 14 Issue: 5 Pages: 1579-1583
- DOI
  10.1039/c5ob02453f
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001
[Journal Article] Screening of a virtual mirror-image library of natural products2016
- Author(s)
  T. Noguchi, S. Oishi, K. Honda, Y. Kondoh, T. Saito, H. Ohno, H. Osada, N. Fujii
- Journal Title
  
  Chem. Comm.
  
  Volume: 52 Issue: 49 Pages: 7653-7656
- DOI
  10.1039/c6cc03114e
- Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-26350976
[Journal Article] Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne2016
- Author(s)
  S. Naoe, Y. Yoshida, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem.
  
  Volume: 81 Issue: 13 Pages: 5690-5698
- DOI
  10.1021/acs.joc.6b00720
- NAID
  120006634624
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654
[Journal Article] Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization2016
- Author(s)
  D. Nishiyama, A. Ohara, H. Chiba, H. Kumagai, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 18 Issue: 7 Pages: 1670-1673
- DOI
  10.1021/acs.orglett.6b00536
- NAID
  120006634625
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Structure-Activity Relationship Study of 4-(Thiazol-5-yl)benzoic Acid Derivatives as Potent Protein Kinase CK2 Inhibitors2016
- Author(s)
  H. Ohno, D. Minamiguchi, S. Nakamura, K. Shu, S. Okazaki, M. Honda, R. Misu, H. Moriwaki, S. Nakanishi, S. Oishi, T. Kinoshita, I. Nakanishi, N. Fujii
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 24 Issue: 5 Pages: 1136-1141
- DOI
  10.1016/j.bmc.2016.01.043
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor2016
- Author(s)
  D. Nishiyama, Y. Sakai, H. Sekiguchi, H. Chiba, R. Misu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 64 Issue: 7 Pages: 996-1003
- DOI
  10.1248/cpb.c16-00302
- NAID
  130005160050
- ISSN
  0009-2363, 1347-5223
- Language
  English
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654
[Journal Article] Convenient Synthesis of Spiroindole Derivatives via Palladium-Catalyzed Cyclization of Propargyl Chlorides2015
- Author(s)
  A. Iwata , S. Inuki, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Tetrahedron
  
  Volume: 71 Issue: 37 Pages: 6580-6585
- DOI
  10.1016/j.tet.2015.05.006
- NAID
  120005674646
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001
[Journal Article] Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation2015
- Author(s)
  Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H.
- Journal Title
  
  Chem. Eur. J.
  
  Volume: 21 Issue: 4 Pages: 1463-1467
- DOI
  10.1002/chem.201405903
- NAID
  120005613671
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24689001
[Journal Article] Direct Construction of Fused Indoles by Gold-Catalyzed Cascade Cyclization of Conjugated Diynes2015
- Author(s)
  Saori Naoe, Tatsuo Saito, Masanobu Uchiyama, Shinya Oishi, Nobutaka Fujii, and Hiroaki Ohno
- Journal Title
  
  Organic Letters
  
  Volume: 17 Issue: 7 Pages: 1774-1777
- DOI
  10.1021/acs.orglett.5b00550
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-13J07518, KAKENHI-PROJECT-24229001, KAKENHI-PROJECT-24689001
[Journal Article] Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines via the Rearrangement of a Propargyl Group2015
- Author(s)
  Y. Tokimizu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 54 Issue: 27 Pages: 7862-7866
- DOI
  10.1002/anie.201502256
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001
[Journal Article] Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists.2015
- Author(s)
  Misu R, Yamamoto K, Yamada A, Noguchi T, Ohno H, Yamamura T, Okamura H, Matsuda F, Ohkura S, Oishi S, Fujii N.
- Journal Title
  
  MedChemCommun
  
  Volume: 6 Issue: 3 Pages: 469-476
- DOI
  10.1039/c4md00514g
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-24380154
[Journal Article] Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group2015
- Author(s)
  M. Taguchi, Y. Tokimizu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 17 Issue: 24 Pages: 6250-6253
- DOI
  10.1021/acs.orglett.5b03254
- NAID
  120006634626
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides2015
- Author(s)
  Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi ASK, Ohno H.
- Journal Title
  
  Org. Lett.
  
  Volume: 17 Issue: 3 Pages: 604-607
- DOI
  10.1021/ol503623m
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24689001
[Journal Article] The Synthesis of Alkaloids Using a Transition-Metal-Catalyzed Intramolecular Amination Reaction2014
- Author(s)
  H. Ohno, et al.
- Journal Title
  
  Synlett
  
  Volume: 25 Issue: 02 Pages: 179-192
- DOI
  10.1055/s-0033-1340165
- NAID
  120005587794
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24106720, KAKENHI-PROJECT-24689001
[Journal Article] Dual Gold Catalysis : Synthesis of Polycyclic Compounds via C-H Insertion of Gold Vinylidenes2014
- Author(s)
  Yusuke Tokimizu
- Journal Title
  
  Chem. Eur. J.
  
  Volume: 20 Issue: 49 Pages: 16331-16336
- DOI
  10.1002/chem.201404987
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06069, KAKENHI-PROJECT-24689001
[Journal Article] Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation.2014
- Author(s)
  Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N.
- Journal Title
  
  J. Med. Chem.
  
  Volume: 57 Issue: 20 Pages: 8646-8651
- DOI
  10.1021/jm500771w
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-24380154
[Journal Article] Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of lndoloquinolines2014
- Author(s)
  Tokimizu Y, Oishi S Fujii N, Ohno H.
- Journal Title
  
  Org. Lett.
  
  Volume: 16 Issue: 11 Pages: 3138-3141
- DOI
  10.1021/ol5012604
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24689001
[Journal Article] Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors2014
- Author(s)
  Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 12 Pages: 3171-3179
- DOI
  10.1016/j.bmc.2014.04.008
- NAID
  120005466732
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23390025
[Journal Article] Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation2014
- Author(s)
  Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii and Hiroaki Ohno
- Journal Title
  
  Chemical Communications
  
  Volume: 50 Issue: 3 Pages: 298-300
- DOI
  10.1039/c3cc46511j
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J05601, KAKENHI-PROJECT-23390025, KAKENHI-PUBLICLY-24106720, KAKENHI-PROJECT-24689001
[Journal Article] Gold-Catalyzed Atom-Economical Cascade Reactions of Alkynes for Ring Formation2014
- Author(s)
  H. Ohno et al.
- Journal Title
  
  Journal of Synthetic Organic Chemistry, Japan
  
  Volume: 72 Issue: 11 Pages: 1218-1227
- DOI
  10.5059/yukigoseikyokaishi.72.1218
- NAID
  130004749120
- ISSN
  0037-9980, 1883-6526
- Language
  Japanese
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-24689001
[Journal Article] Synthesis of IB-01212 by multiple N-methylations of peptide bonds.2014
- Author(s)
  Nabika R, Oishi S, Misu R, Ohno H, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 21 Pages: 6156-6162
- DOI
  10.1016/j.bmc.2014.08.036
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07872, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659004
[Journal Article] Synthesis and Applications of Vinylaziridines and Ethynylaziridines2014
- Author(s)
  H. Ohno
- Journal Title
  
  Chem. Rev.
  
  Volume: 114 Issue: 16 Pages: 7784-7814
- DOI
  10.1021/cr400543u
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24689001
[Journal Article] Design and synthesis of fluorescent probes for GPR54.2014
- Author(s)
  Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 13 Pages: 3325-3330
- DOI
  10.1016/j.bmc.2014.04.052
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-26252046
[Journal Article] Synthesis and biological evaluation of the [D-MeAlall]-epimer of coibamide A.2014
- Author(s)
  Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 25 Issue: 2 Pages: 302-306
- DOI
  10.1016/j.bmcl.2014.11.044
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07872, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659004
[Journal Article] Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility2014
- Author(s)
  Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N.
- Journal Title
  
  ACS Med. Chem. Lett.
  
  Volume: 5 Issue: 5 Pages: 566-571
- DOI
  10.1021/ml500016j
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23390025
[Journal Article] Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes2013
- Author(s)
  Misu R, Oishi S, Setsuda S, Noguchi T, Kaneda M, Ohno H, Evans B, Navenot JM, Peiper SC, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 23 Issue: 9 Pages: 2628-2631
- DOI
  10.1016/j.bmcl.2013.02.098
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007
[Journal Article] Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 4041822013
- Author(s)
  Tsukasa Mizuhara, Shinya Oishi, Hiroaki Ohno, Kazuya Shimura, Masao Matsuoka, Nobutaka Fujii
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 21 Issue: 7 Pages: 2079-2087
- DOI
  10.1016/j.bmc.2013.01.016
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J01895, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24791021
[Journal Article] Convergent Synthesis of (-)-Quinocarcin Based on the Combination of Sonogashira Coupling and Gold (I)-Catalyzed 6-endo-dig Hydroamination2013
- Author(s)
  Hiroaki Chiba, Yuki Sakai, Ayako Ohara, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno
- Journal Title
  
  Chemistry A European Journal
  
  Volume: (in press) Issue: 27 Pages: 8875-8883
- DOI
  10.1002/chem.201300687
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J01905, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Recent Advances in the Construction of Polycyclic Compounds via Palladium-Catalyzed Atom-Economical Cascade Reactions2013
- Author(s)
  Ohno, H.
- Journal Title
  
  Asian J. Org. Chem.
  
  Volume: 2 Issue: 1 Pages: 18-28
- DOI
  10.1002/ajoc.201200128
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001
[Journal Article] Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors2013
- Author(s)
  Hou Z, Oishi S, Suzuki Y, Kure T, Nakanishi I., Hirasawa A, Tsujimoto G, Ohno H, Fujii N.
- Journal Title
  
  Org. Biomol. Chem.
  
  Volume: 11 Issue: 20 Pages: 3288-3296
- DOI
  10.1039/c3ob40223a
- NAID
  120005474525
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23659038, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents2013
- Author(s)
  Mizuhara T, Kato T, Hirai A, Kurihara H, Shimada Y, Taniguchi M, Maeta M, Togami H, Shimura K, Matsuoka M, Okazaki S, Takeuchi T, Ohno H, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 23 Issue: 16 Pages: 4557-4561
- DOI
  10.1016/j.bmcl.2013.06.026
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24791021
[Journal Article] Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors.2013
- Author(s)
  Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Kubo T, Kaneda M, Ohno H, Osada H, Fujii N
- Journal Title
  
  Bioorg Med Chem Lett
  
  Volume: 23 Issue: 13 Pages: 3802-3805
- DOI
  10.1016/j.bmcl.2013.04.094
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23510287, KAKENHI-PROJECT-24659046
[Journal Article] Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis2013
- Author(s)
  Yoshimitsu Y, Miyagaki J, Oishi S, Fujii N, Ohno H.
- Journal Title
  
  Tetrahedron
  
  Volume: 69 Issue: 21 Pages: 4211-4220
- DOI
  10.1016/j.tet.2013.03.091
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659046, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Palladium-Catalyzed Medium-Ring Formation for Construction of the Core Structure of Laurencia Oxacycles: Synthetic Study of Laurendecumallene B2013
- Author(s)
  Y. Yoshimitsu, H. Ohno, et al.
- Journal Title
  
  Org. Lett.
  
  Volume: 15 Issue: 12 Pages: 3046-3049
- DOI
  10.1021/ol401231y
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24106720, KAKENHI-PROJECT-24689001
[Journal Article] 5,10-Dihydrobenzo [a] indolo [2,3-c] carbazole : A Highly Fluorescent Disk-shaped Electron Donor Exhibiting Dual UVvisNIR and Fluorescence Spectral Changes upon Electrolysis2013
- Author(s)
  Yusuke Tokimizu
- Journal Title
  
  Chem. Lett.
  
  Volume: 42 Issue: 9 Pages: 1001-1003
- DOI
  10.1246/cl.130388
- NAID
  10031194320
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06069, KAKENHI-PUBLICLY-24106720, KAKENHI-PROJECT-24689001
[Journal Article] Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds2013
- Author(s)
  H. Ohno
- Journal Title
  
  Isr. J. Chem.
  
  Volume: 53 Issue: 11-12 Pages: 869-882
- DOI
  10.1002/ijch.201300054
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-24106720, KAKENHI-PROJECT-24689001
[Journal Article] Structure-Activity Relationship Study of a CXC Chemokine Receptor Type 4 Antagonist, FC131, Using a Series of Alkene Dipeptide Isosteres2012
- Author(s)
  Kobayashi K., et al
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: (in press) Issue: 6 Pages: 2746-2757
- DOI
  10.1021/jm2016914
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J02083, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23570192, KAKENHI-PROJECT-23689007
[Journal Article] Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists.2012
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot J, Peiper S, Fujii N.
- Journal Title
  
  Bioconjug. Chem.
  
  Volume: 23 Issue: 6 Pages: 1259-1265
- DOI
  10.1021/bc300084h
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23659038, KAKENHI-PROJECT-23689007
[Journal Article] Structure-based Design of Novel Potent CK2 Inhibitors with Phenyl-azole Scaffolds.2012
- Author(s)
  Z. Hou, I. Nakanishi, T. Kinoshita, Y. Takei, M. Yasue, R. Misu, Y. Suzuki, S. Nakamura, T. Kure, H. Ohno, K. Murata, K. Kitaura, A. Hirasawa, G. Tsujimoto, S. Oishi, N. Fujii.
- Journal Title
  
  J. Med. Chem.
  
  Volume: 55 Issue: 6 Pages: 2899-2903
- DOI
  10.1021/jm2015167
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590110, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23659038
[Journal Article] Double C-H Functionalization in Sequential Order : Direct Synthesis of Polycyclic Compounds by a Palladium-Catalyzed C-H Alkenylation-Arylation Cascade2012
- Author(s)
  Ohno, H., Tanaka, T., et al
- Journal Title
  
  Chem.Eur.J.
  
  Volume: 18(印刷中) Issue: 17 Pages: 5352-5360
- DOI
  10.1002/chem.201103819
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22390021, KAKENHI-PROJECT-22590005, KAKENHI-PROJECT-23790130, KAKENHI-PROJECT-24590008
[Journal Article] Efficient Synthesis of Aminomethylated Azaindoles and Corresponding Pyrrole-Fused Derivatives by Copper-Catalyzed Domino Multicomponent Coupling and Cyclization2012
- Author(s)
  Hou, Z., Ohno, H., et al
- Journal Title
  
  Tetrahedron
  
  Volume: 68 Issue: 6 Pages: 1695-1703
- DOI
  10.1016/j.tet.2011.12.059
- NAID
  120003874274
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22590005, KAKENHI-PROJECT-23390025
[Journal Article] Total Synthesis of (-)-Quinocarcin by Gold(I)-Catalyzed Regioselective Hydroamination2012
- Author(s)
  Hiroaki Chiba, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 51 Issue: 36 Pages: 9169-9172
- DOI
  10.1002/anie.201205106
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J01905, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Development and application of fluorescent SDF-1 derivatives2012
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N.
- Journal Title
  
  Future Med. Chem.
  
  Volume: 4 Issue: 7 Pages: 837-844
- DOI
  10.4155/fmc.12.31
- NAID
  120005285488
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23590636, KAKENHI-PROJECT-23659038, KAKENHI-PROJECT-23689007
[Journal Article] Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles.2012
- Author(s)
  Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Journal Title
  
  Org. Biomol. Chem.
  
  Volume: 10 Issue: 33 Pages: 6792-6802
- DOI
  10.1039/c2ob25904d
- NAID
  120005302103
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24791021
[Journal Article] Gold(I)-Catalyzed Regioselective Inter/Intramolecular Addition Cascade of Di- and Triynes for Direct Construction of Substituted Naphthalenes2012
- Author(s)
  Naoe, S. and Ohno, H. et al.
- Journal Title
  
  J. Org. Chem.
  
  Volume: 77 Issue: 11 Pages: 4907-4916
- DOI
  10.1021/jo300771f
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Structure-activity relationship study of pyrimido[1, 2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents.2012
- Author(s)
  Tsukasa Mizuhara, Shinya Oishi, Hiroaki Ohno, Kazuya Shimura, Masao Matsuoka, Nobutaka Fujii
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 20 Issue: 21 Pages: 6334-6441
- DOI
  10.1016/j.bmc.2012.08.030
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J01895, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24791021
[Journal Article] Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (-)-quinocarcinamide2012
- Author(s)
  Hiroaki Chiba, Yuki Sakai, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno
- Journal Title
  
  Tetrahedron Letters
  
  Volume: 53 Issue: 46 Pages: 6273-6276
- DOI
  10.1016/j.tetlet.2012.09.030
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J01905, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] Design and synthesis of novel class of CK2 inhibitors : application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles.2012
- Author(s)
  Suzuki Y, Oishi S, Takei Y, Yasue M, Misu R, Naoe S, Hou Z, Kure T, Nakanishi I, Ohno H, Hirasawa A, Tsujimoto G, Fujii N.
- Journal Title
  
  Org. Biomol. Chem.
  
  Volume: 10 Issue: 25 Pages: 4907-4915
- DOI
  10.1039/c2ob25298h
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23659038
[Journal Article] Gold-Catalyzed Three-Component Annulation : Efficient Synthesis of Highly Functionalized Dihydropyrazoles from Alkynes, Hydrazines, and Aldehydes or Ketones2012
- Author(s)
  Suzuki, Y., Ohno, H., et al
- Journal Title
  
  Org.Lett.
  
  Volume: 14 Issue: 1 Pages: 326-329
- DOI
  10.1021/ol203072u
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22590005, KAKENHI-PROJECT-23390025
[Journal Article] Pachastrissamine (Jaspine B) and Its Stereoisomers Inhibit Sphingosine Kinases and Atypical Protein Kinase C2011
- Author(s)
  Yoshimitsu Y.Oishi S.miyagaki J.Inuki S.Ohno H.Fujii N.
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 19 Issue: 18 Pages: 5402-5408
- DOI
  10.1016/j.bmc.2011.07.061
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-11J02576, KAKENHI-PROJECT-23390025
[Journal Article] Direct Synthesis of Fused-Indoles by Gold-Catalyzed Cascade Cyclization of Diynes2011
- Author(s)
  Hirano, K., Ohno H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Pages: 1212-1227
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Formal Total Synthesis of (+)-Lysergic Acid via Zinc (II)-Mediated Regioselective Ring-Opening Reduction of 2-Alkynyl-3-indolyloxirane2011
- Author(s)
  Iwata, A., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Issue: 13 Pages: 5506-5512
- DOI
  10.1021/jo2008324
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22590005
[Journal Article] Direct Synthesis of Highly Fused Perimidines by Copper (I)-Catalyzed Hydroamination of 2-Ethynylbenzaldehydes2011
- Author(s)
  Tokimizu, Y., Ohno, H., et al
- Journal Title
  
  Tetrahedron
  
  Volume: 67 Issue: 29 Pages: 5168-5175
- DOI
  10.1016/j.tet.2011.05.051
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22590005
[Journal Article] Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups2011
- Author(s)
  Inuki, S., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Pages: 2072-2084
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Gold (I)-Catalyzed Polycyclizations of Poly (enyne) anilines Based on Hydroamination and Consecutive Hydroarylation Cascade2011
- Author(s)
  Hirano, K., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Issue: 21 Pages: 9068-9080
- DOI
  10.1021/jo2018119
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PUBLICLY-22106522, KAKENHI-PROJECT-22590005, KAKENHI-PROJECT-22790009
[Journal Article] Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and(+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups2011
- Author(s)
  Inuki, S., Ohno H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Pages: 2072-2084
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Direct Synthesis of Fused-IndoIes by Gold-Catalyzed Cascade Cyclization of Diynes2011
- Author(s)
  Hirano, K., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 76 Pages: 1212-1227
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Palladium-Catalyzed Construction of Polycyclic Hetetocycles by an Alkyne Insertion and Direct Arylation Cascade2011
- Author(s)
  Ohno, H., Tanaka, T., et al
- Journal Title
  
  Synthesis
  
  Volume: 2011 Issue: 16 Pages: 2567-2578
- DOI
  10.1055/s-0030-1260098
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521, KAKENHI-PROJECT-22590005
[Journal Article] Enantioselective Total Synthesis of(+)-Lysergic Acid,(+)-Lysergol, and(+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups2011
- Author(s)
  S. Inuki, A. Iwata, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 76(7) Issue: 7 Pages: 2072-2084
- DOI
  10.1021/jo102388e
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Direct Synthesis of Fused-Indoles by Gold-Catalyzed Cascade Cyclization of Diynes2011
- Author(s)
  K. Hirano, Y. Inaba, N. Takahashi, M. Shimano, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 76(5) Issue: 5 Pages: 1212-1227
- DOI
  10.1021/jo102507c
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] "Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors"2011
- Author(s)
  Takeuchi T, Oishi S, Watanabe T, Ohno H, Sawada J, Matsuno K,Asai A, Asada N, Kitaura K, Fujii N.
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: 54巻 Issue: 13 Pages: 4839-4846
- DOI
  10.1021/jm200448n
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590067, KAKENHI-PROJECT-23390025
[Journal Article] Direct Synthesis of Quinazolines through Copper-Catalyzed Domino Alkynylation and Cyclization of Aniline-Derived Benzamidines2010
- Author(s)
  Ohta, Y., Ohno H., et al.
- Journal Title
  
  Org.Lett.
  
  Volume: 12 Pages: 3963-3965
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates.2010
- Author(s)
  S.Inuki, Y.Yoshimitsu, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 75(11)
  
  Pages: 3831-3842
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Synthesis of Fused and Linked Bicyclic Nitrogen Heterocycles by Palladium-Catalyzed Domino Cyclization of Propargyl Bromides2010
- Author(s)
  Okano, A., Ohno, H., et al
- Journal Title
  
  Chem.Eur.J.
  
  Volume: 16 Pages: 8410-8418
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Gold-Catalyzed Intramolecular Alkyne Cycloisomerization Cascade : Direct Synthesis of Aryl-Annulated[a]carbazoles from Aniline-Substituted Diethynylarenes2010
- Author(s)
  Hirano, K., Ohno, H., et al
- Journal Title
  
  Adv.Synth.Catal.
  
  Volume: 352 Pages: 368-372
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Direct Synthesis of Quinazolines through Copper-Catalyzed Reaction of Aniline-Derived Benzamidines2010
- Author(s)
  Y. Ohta, Y. Tokimizu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Org. Lett
  
  Volume: 12(17) Issue: 17 Pages: 3963-3965
- DOI
  10.1021/ol1016756
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates2010
- Author(s)
  Inuki, S., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3831-3842
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Construction of Linked Nitrogen Heterocycles by Palladium(0)-Catalyzed Intramolecular Domino Cyclization of 2-Alkynylaziridines Bearing a 2-Aminoethyl Group via Ring Expansion with Isocyanate2010
- Author(s)
  Okano, A., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3396-3400
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Synthesis of Fused and Linked Bicyclic Nitrogen Heterocycles by Palladium-Catalyzed Domino Cyclization of Propargyl Bromides2010
- Author(s)
  Okano, A., Ohno, H., et al.
- Journal Title
  
  Chem.Eur.J.
  
  Volume: 16 Pages: 8410-8418
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Construction of Linked Nitrogen Heterocycles by Palladium(0)-Catalyzed Intramolecular Domino Cyclization of 2-Alkynylaziridines Bearing a 2-Aminoethyl Group via Ring Expansion with Isocyanate2010
- Author(s)
  A. Okano, S. Oishi, T. Tanaka, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 75(10) Issue: 10 Pages: 3396-3400
- DOI
  10.1021/jo100462w
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Construction of Linked Nitrogen Heterocycles by Palladium(0)-Catalyzed Intramolecular Domino Cyclization of 2-Alkynylaziridines Bearing a 2-Aminoethyl Group via Ring Expansion with Isocyanate2010
- Author(s)
  Okano, A., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3396-3400
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B)2010
- Author(s)
  Yoshimitsu, Y., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3843-3846
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B).2010
- Author(s)
  Y.Yoshimitsu, S.Inuki, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 75(11)
  
  Pages: 3843-3846
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Direct Synthesis of Quinazolines through Copper-Catalyzed Domino Alkynylation and Cyclization of Aniline-Derived Benzamidines2010
- Author(s)
  Ohta, Y., Ohno, H., et al
- Journal Title
  
  Org.Lett.
  
  Volume: 12 Pages: 3963-3965
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine(Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates2010
- Author(s)
  S. Inuki, Y. Yoshimitsu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 75(11) Issue: 11 Pages: 3831-3842
- DOI
  10.1021/jo100544v
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Gold-Catalyzed Intramolecular Alkyne Cycloisomerization Cascade : Direct Synthesis of Aryl-Annulated[a]carbazoles from Aniline-Substituted Diethynylarenes2010
- Author(s)
  Hirano, K., Ohno, H., et al.
- Journal Title
  
  Adv.Synth.Catal.
  
  Volume: 352 Pages: 368-372
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Efficient Synthesis of Pyrimido[1,2-c][1,3]benzothiazin-6-imines and Related Tricyclic Heterocycles by S_NAr-Type C-S, C-N, or C-O Bond Formation with Heterocumulenes2010
- Author(s)
  Mizuhara, T., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 265-268
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Efficient Synthesis of Pyrimido[1,2-c][1,3]- benzothiazin-6-imines and Related Tricyclic Heterocycles by SNAr-Type C-S, C-N, or C-O Bond Formation with Heterocumulenes.2010
- Author(s)
  T.Mizuhara, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 75(1)
  
  Pages: 265-268
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine(Jaspine B)2010
- Author(s)
  Yoshimitsu, Y., Ohno H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3843-3846
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Gold-Catalyzed Intramolecular Alkyne Cycloisomerization Cascade: Direct Synthesis of Aryl-Annulated[ a]carbazoles from Aniline-Substituted Diethynylarenes.2010
- Author(s)
  K.Hirano, Y.Inaba, T.Watanabe, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Adv.Synth.Catal. 352(2)
  
  Pages: 368-372
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Construction of Linked Nitrogen Heterocycles by Palladium(0)-Catalyzed Intramolecular Domino Cyclization of 2-Alkynylaziridines Bearing a 2-Aminoethyl Group via Ring Expansion with Isocyanate2010
- Author(s)
  Okano, A., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3396-3400
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Construction of Linked Nitrogen Heterocycles by Palladium(0)-Catalyzed Intramolecular Domino Cyclization of 2-Alkynylaziridines Bearing a 2-Aminoethyl Group via Ring Expansion with Isocyanate2010
- Author(s)
  A.Okano, S.Oishi, T.Tanaka, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 75(10)
  
  Pages: 3396-3400
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine(Jaspine B)2010
- Author(s)
  Y. Yoshimitsu, S. Inuki, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 75(11) Issue: 11 Pages: 3843-3846
- DOI
  10.1021/jo1005284
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B)2010
- Author(s)
  Yoshimitsu, Y., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3843-3846
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Synthesis of Fused and Linked Bicyclic Nitrogen Heterocycles by Palladium-Catalyzed Domino Cyclization of Propargyl Bromide.2010
- Author(s)
  A.Okano, K.Tsukamoto, S.Kosaka, H.Maeda, S.Oishi, T.Tanaka, N.Fujii, H.Ohno.
- Journal Title
  
  Chem.Eur.J. 16(28)
  
  Pages: 8410-8418
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Efficient Synthesis of Pyrimido[1,2-c][1,3]benzothiazin-6-imines and Related Tricyclic Heterocycles by S_NAr-Type C-S, C-N, or C-O Bond Formation with Heterocumulenes2010
- Author(s)
  Mizuhara, T., Ohno H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 265-268
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates2010
- Author(s)
  Inuki, S., Ohno H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3831-3842
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Direct Synthesis of Quinazolines through Copper-Catalyzed Domino Alkynylation and Cyclization of Aniline-Derived Benzamidines2010
- Author(s)
  Ohta, Y., Ohno, H., et al.
- Journal Title
  
  Org.Lett.
  
  Volume: 12 Pages: 3963-3965
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Gold-Catalyzed Intramolecular Alkyne Cycloisomerization Cascade : Direct Synthesis of Aryl-Annulated[a] carbazoles from Aniline-Substituted Diethynylarenes2010
- Author(s)
  K. Hirano, Y. Inaba, T. Watanabe, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Adv. Synth. Catal
  
  Volume: 352(2) Issue: 2-3 Pages: 368-372
- DOI
  10.1002/adsc.200900880
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Synthesis of Fused and Linked Bicyclic Nitrogen Heterocycles by Palladium-Catalyzed Domino Cyclization of Propargyl Bromides2010
- Author(s)
  Okano, A., Ohno, H., et al.
- Journal Title
  
  Chem.Eur.J.
  
  Volume: 16 Pages: 8410-8418
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Gold-Catalyzed Intramolecular Alkyne Cycloisomerization Cascade : Direct Synthesis of Aryl-Annulated[α]carbazoles from Aniline-Substituted Diethynylarenes2010
- Author(s)
  Hirano, K, Ohno, H., et al.
- Journal Title
  
  Adv.Synth.Catal.
  
  Volume: 352 Pages: 368-372
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres2010
- Author(s)
  Narumi T, Ohno H, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 8 Pages: 616-621
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Synthesis of Fused and Linked Bicyclic Nitrogen Heterocycles by Palladium-Catalyzed Domino Cyclization of Propargyl Bromides2010
- Author(s)
  A. Okano, K. Tsukamoto, S. Kosaka, H. Maeda, S. Oishi, T. Tanaka, N. Fujii, H. Ohno
- Journal Title
  
  Chem. Eur. J
  
  Volume: 16(28) Issue: 28 Pages: 8410-8418
- DOI
  10.1002/chem.201000653
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates2010
- Author(s)
  Inuki, S., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 3831-3842
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres2010
- Author(s)
  Narumi T, Ohno H, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 8 Pages: 616-621
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Efficient Synthesis of Pyrimido[1, 2-c][1, 3] benzothiazin-6-imines and Related Tricyclic Heterocycles by SNAr-Type C-S, C-N, or C-O Bond Formation with Heterocumulenes2010
- Author(s)
  T. Mizuhara, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem
  
  Volume: 75(1) Issue: 1 Pages: 265-268
- DOI
  10.1021/jo902327n
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-22590005
[Journal Article] Efficient Synthesis of Pyrimido [1,2-c][1,3]benzothiazin-6-imines and Related Tricyclic Heterocycles by S_NAr-Type C-S, C-N, or C-O Bond Formation with Heterocumulenes2010
- Author(s)
  Mizuhara, T., Ohno, H., et al
- Journal Title
  
  J.Org.Chem.
  
  Volume: 75 Pages: 265-268
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22106521
[Journal Article] Direct Synthesis of Quinazolines through Copper-Catalyzed Reaction of Aniline-Derived Benzamidines.2010
- Author(s)
  Y.Ohta, Y.Tokimizu, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett 12(17)
  
  Pages: 3963-3965
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Construction of Nitrogen Heterocycles Bearing an Aminomethyl Group by Copper-Catalyzed Domino Three-Component Coupling-Cyclization2009
- Author(s)
  Y.Ohta, H.Chiba, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 74(18)
  
  Pages: 7052-7058
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Construction of Nitrogen Heterocycles Bearing an Aminomethyl Group by Copper-Catalyzed Domino Three-Component Coupling-Cyclization2009
- Author(s)
  Ohta, Y., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 7052-7058
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes.2009
- Author(s)
  S.Inuki, Y.Yoshimitsu, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett. 11(19)
  
  Pages: 4478-4481
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-ccopper-mediated SN2' alkylation2009
- Author(s)
  Kobayashi K, Oishi S, Ohno H, Fujii N, et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 4626-4629
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Rapid Access to 3-(Aminomethyl)isoquinoline-Fused Polycyclic Compounds by Copper-Catalyzed Four-Component Coupling, Cascade Cyclisation and Oxidation.2009
- Author(s)
  Y.Ohta, Y.Kubota, T.Watabe, H.Chiba, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 74(16)
  
  Pages: 6299-6302
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Rapid Access to 3-(Aminomethyl)isoquinoline-Fused Polycyclic Compounds by Copper-Catalyzed Four-Component Coupling, Cascade Cyclisation and Oxidation2009
- Author(s)
  Ohta, Y., Ohno, H., et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 6299-6302
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-Catalyzed Direct Synthesis of Carbazoles via One-Pot N-Arylation and Oxidative Biaryl Coupling : Synthesis and Mechanistic Study2009
- Author(s)
  Watanabe T. and Ohno H., et.al.
- Journal Title
  
  J. Org. Chem. 74
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcoholassisted nucleophilic trifluoromethylation and organozinc-ccopper-mediated SN2' alkylation2009
- Author(s)
  Kobayashi K, Oishi S, Ohno H, Fujii N, et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 4626-4629
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Facile Synthesis of 1,2,3,4-Tetrahydro-β-carbolines by One-Pot Domino Three-Component Indole Formation and Nucleophilic Cyclization.2009
- Author(s)
  Y.Ohta, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett. 11(9)
  
  Pages: 1979-1982
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-Catalyzed Direct Synthesis of Carbazoles via One-Pot N-Arylation and Oxidative Biaryl Coupling: Synthesis and Mechanistic Study.2009
- Author(s)
  T.Watanabe, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  J.Org.Chem. 74(13)
  
  Pages: 4720-4726
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes2009
- Author(s)
  Inuki, S., Ohno, H., et al.
- Journal Title
  
  Org.Lett.
  
  Volume: 11 Pages: 4478-4481
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Facile Synthesis of 1,2,3,4-Tetrahydro-β-carbolines by One-Pot Domino -Three-Component Indole Formation and Nucleophilic Cyclization2009
- Author(s)
  Ohta Y. and Ohno H., et al.
- Journal Title
  
  Org. Lett. 11
  
  Pages: 1979-1982
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-catalyzed sp^3 C-H activation of simple alkyl groups : direct preparation of indoline derivatives from N-alkyl-2-bromoanilines2008
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 1759-1762
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Facile Synthesis of 3-(Aminomethyl)isoquinoline by Copper-Catalysed Domino Four-Component Coupling and Cyclisation.2008
- Author(s)
  Y.Ohta, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Chem.Commun 7
  
  Pages: 835-837
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides.2008
- Author(s)
  Ohno H., et. al.
- Journal Title
  
  Ore. Lett. (In press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid-derived allylic carbonates2008
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  J. Org. Chem. (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group.2008
- Author(s)
  S.Inuki, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett 10(22)
  
  Pages: 5239-5242
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic2008
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Tetrahedron 64
  
  Pages: 4332-4346
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Concise Synthesis of Indole-Fused 1,4-Diazepines through Copper(I)-Catalyzed Domino Three-Component Coupling-Cyclization-N-Arylation under Microwave Irradiation.2008
- Author(s)
  Y.Ohta, H.Chiba, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett. 10(16)
  
  Pages: 3535-3538
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity2008
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  J. Med. Chem. 51
  
  Pages: 388-391
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides2008
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 1171-1174
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-Catalyzed sp^3 C-H Activation of Simple Alkyl Groups: Direct Preparation of Indoline Derivatives from N-Alkyl-2-bromoanilines.2008
- Author(s)
  T.Watanabe, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett 10(9)
  
  Pages: 1759-1762
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Total Synthesis of(±)-Lysergic Acid, Lysergol, and Isolysergol Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group2008
- Author(s)
  Inuki S. and Ohno H., et.al.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 5239-5242
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-catalyzed sp3 C-H activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines2008
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  Org. Lett. (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation2008
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Chem. Commun. 7
  
  Pages: 835-837
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Samarium(II)-Mediated Spirocyclization by Intramolecular Aryl Radical Addition onto an Aromatic Ring2008
- Author(s)
  Inuki S. and Ohno H,., et.al.
- Journal Title
  
  J.Org.Chem. 10
  
  Pages: 7145-7152
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] N.Fujii.Palladium-Catalysed Biscyclisation of Allenic Bromoalkenes through Zipper-Mode Cascade.2008
- Author(s)
  A.Okano, T.Mizutani, S.Oishi, T.Tanaka, H.Ohno
- Journal Title
  
  Chem.Commun 30
  
  Pages: 3534-3536
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Facile synthesis of 3-(aminomethyl) isoquinolines by copper-catalysed domino four-component coupling and cyclisation2008
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  Chem. Commun. 7
  
  Pages: 835-837
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides2008
- Author(s)
  Fujii N., Ohno H., et. al.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 1171-1174
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic2008
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  Tetrahedron (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Direct Construction of Bicyclic Heterocycles by Palladium-Catalyzed Tandem Cyclization of Propargyl Bromides.2008
- Author(s)
  H.Ohno, A.Okano, S.Kosaka, K.Tsukamoto, M.Ohata, K.Ishihara, H.Maeda, T.Tanaka, N.Fujii.
- Journal Title
  
  Org.Lett 10(6)
  
  Pages: 1171-1174
- NAID
  130006995906
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Concise Synthesis of Indole-Fused 1,4-Diazepines through Copper(I)-Catalyzed Domino Three-Component Coupling-Cyclization-N-Arylation2008
- Author(s)
  Ohta Y. and Ohno H., et.al.
- Journal Title
  
  Org. Lett 10
  
  Pages: 3535-3538
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-Catalyzed sp3 C-H Activation of Simple Alkyl Groups : Direct Preparation of Indoline Derivatives from N-Alkyl-2-bromoanilines2008
- Author(s)
  Watanabe T. and Ohno H., et.al.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 1759-1762
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Structure-Activity Relationship of Pyrazine-Based CK2 Inhibitors : Synthesis and Evaluation of 2,6-Disubstituted Pyrazines and 4,6-Disubstituted Pyrimidines2008
- Author(s)
  Suzuki Y. and Ohno H., et.al.
- Journal Title
  
  Arch. Pharm. 349
  
  Pages: 554-561
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid-derived allylic carbonates2008
- Author(s)
  Ohno H., et al.
- Journal Title
  
  J. Org. Chem. 73
  
  Pages: 3942-3945
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Palladium-Catalysed Biscyclisation of Allenic Bromoalkenes through Zipper-Mode Cascade2008
- Author(s)
  Okano A. and Ohno H., et.al.
- Journal Title
  
  Chem. Commun.
  
  Pages: 3534-3536
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Zipper-Mode Double C-H Activation: Palladium-Catalyzed Direct Construction of Highly-Fused Heterocyclic Systems.2007
- Author(s)
  H.Ohno, M.Iuchi, N.Fujii, T.Tanaka.
- Journal Title
  
  Org.Lett 9(23)
  
  Pages: 4813-4815
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Fmoc-based Solid-phase Synthesis of GPR54-agonistic Pentapeptide Derivatives Containing Alkene- and Fluoroalkene-dipeptide Isosteres2007
- Author(s)
  K.Tomita, H.Ohno, N.Fujii, et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 947-950
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Zipper-mode double C-H activation : palladium-catalyzed direct construction of highly-fused heterocyclic systems2007
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 4813-4815
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling2007
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  Chem. Commun. 43
  
  Pages: 4516-4518
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] A Highly Regio- and Stereoselective Formation of Bicyclo[4.2.0]oct-5-ene Derivatives through Thermal Intramolecular [2+2] Cycloaddition2007
- Author(s)
  Ohno, H., Fujii, N., Tanaka, T.
- Journal Title
  
  J.Ore.Chem. (in press)
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions.2007
- Author(s)
  Ohno, H., Fujii, N.et al.
- Journal Title
  
  Angew.Chem.Int.Ed.Engl. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems.2007
- Author(s)
  Ohno H., et. al.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 4813-4815
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] One-Pot Synthesis of Carbazoles by Palladium-Catalyzed N-Arylation and Oxidative Coupling.2007
- Author(s)
  T.Watanabe, S.Ueda, S.Inuki, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Chem.Commun. 43
  
  Pages: 4516-4518
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Structure-activity relationships of cyclic Peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone functionalities.2007
- Author(s)
  Ueda, S., Ohno, H., Fujii, N.et al.
- Journal Title
  
  J.Med.Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] A Highly Regio- and Stereoselective Formation of Bicyclo[4.2.0]oct-5-ene Derivatives through Thermal Intramolecular [2+2] Cycloaddition of2007
- Author(s)
  H.Ohno, N.Fujii, T.Tanaka, et al.
- Journal Title
  
  J.Org.Chem. (印刷中)
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides2007
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 3465-3468
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions.2007
- Author(s)
  Ohno, H., Fujii, N.et al.
- Journal Title
  
  Angew.Chem.Int.Ed.Engl. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] A Novel Oxazolidine Linker for the Synthesis of Peptide Aldehydes2007
- Author(s)
  M.Tanaka, H.Ohno, N.Fujii, et al.
- Journal Title
  
  Int. J. Pep. Res. Ther. (印刷中)
- NAID
  10020528946
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Bromoallenes as allyl dication equivalents in the presence or absence of palladlum(O) : direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes2007
- Author(s)
  Hamaguchu, H., Ohno, H., Fujii, N., Tanaka, T.et al.
- Journal Title
  
  Chem.Eur.J. 13・6
  
  Pages: 1692-1708
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Structure-activity relationships of cyclic Peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone functionalities.2007
- Author(s)
  Ueda, S., Ohno, H., Fujii, N.et al.
- Journal Title
  
  J.Med.Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone2007
- Author(s)
  S.Ueda, H.Ohno, N.Fujii, et al.
- Journal Title
  
  J. Med. Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR542007
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  J. Med. Chem. 50
  
  Pages: 3222-3228
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Gold-Catalyzed Hydroarylation of Allenes: A Highly Regioselective Carbon-Carbon Bond Formation Producing Six-Membered Rings.2007
- Author(s)
  T.Watanabe, S.Oishi, N.Fujii, H.Ohno.
- Journal Title
  
  Org.Lett 9(23)
  
  Pages: 4821-4824
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Heck-type cyclization of oxime ethers: stereoselective carbon-carbonbond formation with aryl halides to produce heterocyclic oximes.2007
- Author(s)
  Ohno H., et. al.
- Journal Title
  
  Angew. Chem. Int. Ed. 46
  
  Pages: 6325-6328
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] A highly regio- and stereoselective formation of bicyclo [4.2.0] oct-5-ene derivatives through thermal intramolecular [2+2] cycloaddition of allenes.2007
- Author(s)
  Ohno H., et. al.
- Journal Title
  
  J. Org. Chem. 72
  
  Pages: 4378-4389
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions2007
- Author(s)
  H.Ohno, N.Fujii, et al.
- Journal Title
  
  Angew. Chem. Int. Ed. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] A Highly Regio- and Stereoselective Formation of Bicyclo[4.2.0]oct-5-ene Derivatives through Thermal Intramolecular [2 + 2] Cycloaddition2007
- Author(s)
  Ohno, H., Fujii, N., Tanaka, T.
- Journal Title
  
  J.Org.Chem. (in press)
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Heck-type cyclization of oxime ethers : stereoselective carbon-carbon bond formation with aryl halides to produce heterocvclic oximes2007
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Angew. Chem. Int. Ed. 46
  
  Pages: 6325-6328
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita, K., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 272-278
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Heck-Type Cyclization of Oxime Ethers: Stereoselective Carbon-Carbon Bond Formation with Aryl Halides to Produce Heterocyclic Oximes2007
- Author(s)
  H.Ohno, A.Aso, Y.Kadoh, N.Fujii, T.Tanaka
- Journal Title
  
  Angew.Chem.Int.Ed. 46(33)
  
  Pages: 6325-6328
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems2007
- Author(s)
  Fujii N., Ohno H., et. al.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 4813-4815
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita, K., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 272-278
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Bromoallenes as allyl dication equivalents in the presence or absence of palladium(O) : direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes.2007
- Author(s)
  Hamaguchu, H., Ohno, H., Fujii, N., Tanaka, T.et al.
- Journal Title
  
  Chem.Eur.J. 13・6
  
  Pages: 1692-1708
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling2007
- Author(s)
  Ohno H., et al.
- Journal Title
  
  Chem. Commun. 43
  
  Pages: 4516-4518
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Journal Article] Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides2007
- Author(s)
  Fujii N., Ohno H., Oishi, S., et. al.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 3465-3468
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Heck-type cyclization of oxime ethers: stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes2007
- Author(s)
  Fujii N., Ohno H., et. al.
- Journal Title
  
  Angew. Chem. Int. Ed. 46
  
  Pages: 6325-6328
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Bromoallenes as Allyl Dication Equivalents in the Presence or Absence of Palladium(O):Direct Construction of Bicyclic Sulfamides Containing Five- to Eight-membered Ring by Tandem Cyclization of Bromoallenes2007
- Author(s)
  H.Ohno, N.Fujii, T.Tanaka, et al.
- Journal Title
  
  Chem.Eur.J. 13・6
  
  Pages: 1692-1708
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita, K., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Bioorg.Med.Chem. 45・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres2006
- Author(s)
  Narumi, T., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Chem.Commun. 45
  
  Pages: 4720-2722
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Potassium Carbonate-Promoted Stereospecific 5-Endo-Trig Cyclization of Unactivated Allenes in the Absence of Any Transition Metals2006
- Author(s)
  H.Ohno, N.Fujii, T.Tanaka, et al.
- Journal Title
  
  Org.Lett. 8・5
  
  Pages: 947-950
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita, K., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Bioorg.Med.Chem. 45・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Synthesis of (Z)-alkene and (E)- fluoroalkene-containing diketopiperazine mimetics utili-zing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations2006
- Author(s)
  Niida, A., Ohno, H., Fujii, N.et al.
- Journal Title
  
  J.Org.Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-18015027
[Journal Article] Syntnesis of (Z)-alkene and (E)-fluoroalkene-containing diketoplperazine mimetics utin-zing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations2006
- Author(s)
  Niida, A., Ohno, H., Fujii, N.et al.
- Journal Title
  
  J.Org.Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/.D-ring system2006
- Author(s)
  Tanaka, T., Ohno, H.
- Journal Title
  
  Chem.Phram.Bull 54・8
  
  Pages: 1138-1143
- NAID
  110004847232
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Synthesis of (Z)-Alkene and (E)-Fluoroalkene-Containing Diketopiperazine Mimetics Utilizing Organocopper-Mediated Reduction-Alkylation and Diastereoselectivity Examination Using DFT Calculations.2006
- Author(s)
  A.Niida, H.Ohno, N.Fujii, et al.
- Journal Title
  
  J.Org.Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] A-nover one-pot reaction involving orgamcopper-mediated reduction/transmealation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres2006
- Author(s)
  Narumi, T., Ohno, H., Fujii, N.et al.
- Journal Title
  
  Chem.Commun. 45
  
  Pages: 4720-2722
- Data Source
  KAKENHI-PROJECT-18659027
[Journal Article] Construction of Tricyclic Enone, a Common Precursor for Aphidicolane and Stemodane B/C/D-Ring System2006
- Author(s)
  H.Ohno, T.Tanaka, et al.
- Journal Title
  
  Chem.Pharm.Bull. 54・8
  
  Pages: 1138-1143
- NAID
  110004847232
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Structure-Activity Relationship Study on Amall Peptidic GPR54 Agonists2006
- Author(s)
  K.Tomita, H.Ohno, N.Fujii, et al.
- Journal Title
  
  Bioorg.Med.Chem. 14・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Stereoselective Synthesis of 3,6-Disubstituted-3,6-dihydropyridin-2-ones as Potential Diketopiperazine Mimetics Using Organocopper-Mediated anti -S_N2' Reactions and Their Use in the Preparation of Low-Molecule CXCR4 Antagonists2006
- Author(s)
  A.Niida, H.Ohno, N.Fujii, et al.
- Journal Title
  
  J.Org.Chem. 71・10
  
  Pages: 3942-3951
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Novel One-Pot Reaction Involving Organocopper-Mediated Reduction/transmetalation/asymmetric Alkylation, Leading to the Diastereoselective Synthesis of Functionalized (Z)-Fluoroalkene Dipeptide Isosteres2006
- Author(s)
  T.Narumi, H.Ohno, N.Fujii, et al.
- Journal Title
  
  Chem. Commun. 45
  
  Pages: 4720-4722
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Palladium-Catalyzed Tandem Cyclization of Bromoenynes through Aromatic C-H Bond Functionalization2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Angewandte Chemie, International Edition 44・32
  
  Pages: 5233-5236
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Development of Useful Reactions Involving Tandem Cyclizations Based on the Novel Reactivities of Allenic Compounds2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Chemical & Pharmaceutical Bulletin 53・10
  
  Pages: 1211-1226
- NAID
  110003666248
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Palladium(0)-Catalyzed Tandem Cyclization of Allenenes : Direct Construction of Tricyclic Heterocycles through Aromatic C-H Bond Functionalization2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Chemistry-European Journal (in press)
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Thermal Intramolecular [2 + 2] Cycloaddition of Allenenes and Allenynes : Diastereoselective Access to Bicyclic Nitrogen Heterocycles2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Angewandte Chemie, International Edition 44・32
  
  Pages: 5113-5115
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Synthesis of Bicyclic Sulfamides by Tandem Cyclization of Bromoallenes2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Angewandte Chemie, International Edition 44・10
  
  Pages: 1513-1517
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Development of Useful Reactions Based on the Novel Reactivities of Allenic Compounds and Their Application to Tandem Cyclizations2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Yakugaku Zasshi 125・12
  
  Pages: 899-925
- NAID
  110004042077
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Palladium(0)-Catalyzed Tandem Cyclization of Allenenes : Direct Construction of Tricyclic Heterocycles through Aromatic C-H Activation2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Chemistry- European Journal 11・12
  
  Pages: 3728-3741
- Data Source
  KAKENHI-PROJECT-17790013
[Journal Article] Bromoallenes as Allyl Dication Equivalents in the Absence of Palladium(0) : Synthesis of Bicyclic Sulfamides by Tandem Cyclization of Bromoallenes2005
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Angewandte Chemie, International Edition 44・10
  
  Pages: 1513-1517
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Palladium(0)-Catalyzed Synthesis of Medium-Sized Heterocycles by Using Bromoallenes as an Allyl Dication Equivalent2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  The Journal of the American Chemical Society 126・28
  
  Pages: 8744-8754
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Stereodivergent Synthesis of Chiral 2-Alkenylaziridines : Palladium(0)-Catalyzed 2,3-cis-Selective Aziridination and Base-Mediated 2,3-trans-Selective Aziridination2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Chemcal & Pharmaceutical Bulletin 52・1
  
  Pages: 111-120
- NAID
  110003615486
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Palladium(0)-Catalyzed Stereoselective Cyclization of Allenenes ; Divergent Synthesis of Pyrrolidines and 3-Azabicyclo[3,1,0]hexanes from Single Allenenes2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  The Journal of Organic Chemistry 69・13
  
  Pages: 4541-4544
- Data Source
  KAKENHI-PROJECT-15659003
[Journal Article] Palladium(0)-Catalyzed Synthesis of Medium-Sized Heterocycles by Using Bromoallenes as an Allyl Dication Equivalent2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  The Journal of the American Chemical Society 126・28
  
  Pages: 8744-8754
- Data Source
  KAKENHI-PROJECT-15659003
[Journal Article] The First Samarium(II)-Mediated Aryl Radical Cyclization onto an Aromatic Ring2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  Chemical Communication 19
  
  Pages: 2228-2229
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] Palladium(0)-Catalyzed Stereoselective Cyclization of Allenenes : Divergent Synthesis of Pyrrolidines and 3-Azabicyclo[3.1.0]hexanes from Single Allenenes2004
- Author(s)
  Hiroaki Ohno
- Journal Title
  
  The Journal of Organic Chemistry 69・13
  
  Pages: 4541-4544
- Data Source
  KAKENHI-PROJECT-15790010
[Journal Article] N.Fujii.Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Palladium-catalyzed Carbonylation of Amino Acid-derived Allylic Carbonates.
- Author(s)
  E.Inokuchi, T.Narumi, A.Niida, K.Kobayashi, K.Tomita, S.Oishi, H.Ohno
- Journal Title
  
  J.Org.Chem.
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-19689001
[Patent] ベンゾイソチアゾロピリミジン誘導体またはその塩,およびウイルス感染阻害剤ならびに医薬品2014
- Inventor(s)
  松岡雅雄、　志村和也、藤井信孝、大野浩章、大石真也、岡崎志穂　他
- Industrial Property Rights Holder
  松岡雅雄、　志村和也、藤井信孝、大野浩章、大石真也、岡崎志穂　他
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2014-206613
- Filing Date
  2014-10-07
- Data Source
  KAKENHI-PROJECT-23390025
[Patent] ＣＸＣＲ７結合剤およびＣＸＣＲ７結合剤を含有する医薬組成物2014
- Inventor(s)
  藤井信孝、大野浩章、大石真也、黒柳友子、久保達彦他
- Industrial Property Rights Holder
  京都大学
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2014-195189
- Filing Date
  2014-09-25
- Data Source
  KAKENHI-PROJECT-23390025
[Patent] Eg5阻害剤2014
- Inventor(s)
  藤井信孝、大野浩章、大石真也、竹内智起、浅井章良、澤田潤一
- Industrial Property Rights Holder
  京都大学、ファルマバレープロジェクト支援機構
- Industrial Property Rights Type
  特許
- Filing Date
  2014-02-25
- Overseas
- Data Source
  KAKENHI-PROJECT-23390025
[Patent] 新規ケモカイン受容体拮抗剤2012
- Inventor(s)
  藤井信孝、大野浩章、大石真也、他
- Industrial Property Rights Holder
  京都大学
- Industrial Property Rights Type
  特許
- Filing Date
  2012-02-29
- Overseas
- Data Source
  KAKENHI-PROJECT-23390025
[Patent] キナーゼ阻害剤2012
- Inventor(s)
  大野浩章、辻本豪三, 他
- Industrial Property Rights Holder
  京都大学, 他
- Filing Date
  2012-03-02
- Overseas
- Data Source
  KAKENHI-PUBLICLY-22106521
[Patent] キナーゼ阻害剤2012
- Inventor(s)
  大野浩章、辻本豪三, 他
- Industrial Property Rights Holder
  京都大学, 他
- Filing Date
  2012-03-02
- Overseas
- Data Source
  KAKENHI-PROJECT-22590005
[Patent] キナーゼ阻害剤2012
- Inventor(s)
  大野浩章、辻本豪三、他10名
- Industrial Property Rights Holder
  京都大学, 他
- Filing Date
  2012-03-02
- Overseas
- Data Source
  KAKENHI-PROJECT-22590005
[Patent] CK2阻害剤2011
- Inventor(s)
  大野浩章、辻本豪三、他8名
- Industrial Property Rights Holder
  京都大学, 他
- Filing Date
  2011-03-04
- Data Source
  KAKENHI-PROJECT-22590005
[Patent] CK2阻害剤2011
- Inventor(s)
  大野浩章、辻本豪三, 他
- Industrial Property Rights Holder
  京都大学・近畿大学、大阪府立大学
- Industrial Property Number
  2011-048325
- Filing Date
  2011-03-04
- Data Source
  KAKENHI-PROJECT-22590005
[Patent] CK2阻害剤2011
- Inventor(s)
  大野浩章、辻本豪三, 他
- Industrial Property Rights Holder
  京都大学, 他
- Industrial Property Number
  2011-048325
- Filing Date
  2011-03-04
- Data Source
  KAKENHI-PUBLICLY-22106521
[Patent] Eg5阻害剤2009
- Inventor(s)
  藤井信孝、大野浩章、大石真也, 他
- Industrial Property Rights Holder
  京都大学
- Filing Date
  2009-12-25
- Overseas
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] Eg5阻害剤2008
- Inventor(s)
  藤井信孝、大石真也、大野浩章、他
- Industrial Property Rights Holder
  京都大学・ファルマIP
- Industrial Property Number
  2008-331963
- Filing Date
  2008-12-26
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 金触媒を用いたアジドアルキンの連続環化反応による八員環縮環インドールの構築2024
- Author(s)
  長谷川大輝、有地法人、井貫晋輔、大野浩章
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] スルホニルアジドへの可視光誘起エネルギー移動を利用するスルフィルイミンの合成2024
- Author(s)
  呉舒涵, 天野剛, 有地法人, 井貫晋輔, 大野浩章
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 金触媒を用いたアジドアルキンの連続環化反応による八員環縮環インドールの構築2024
- Author(s)
  長谷川大輝, 有地法人, 井貫晋輔, 大野浩章
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 計算化学的アプローチによるMR1細胞表面発現に重要な因子の特定2024
- Author(s)
  藤井俊樹, 荒木望嗣, 松本篤幸, 馬彪, 大塚教雄, 大野浩章, 井貫晋輔, 奥野恭史
- Organizer
  日本薬学会第144年会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] ビススルホンアミド構造を持つミトコンドリアNADH-キノン酸化還元酵素（複合体-I）新規阻害剤の同定2023
- Author(s)
  辻諄人、桝谷貴洋、有地法人、井貫晋輔、村井正俊、三芳秀人、大野浩章
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 金触媒を用いたアジドアルキンの連続環化反応による八員環縮環インドールの構築2023
- Author(s)
  長谷川大輝、有地法人、井貫晋輔、大野浩章
- Organizer
  第73回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 細胞表面のMR1存在量に基づくリガンドスクリーニング法の開発とMAIT細胞制御分子の同定2023
- Author(s)
  松岡巧朗、服部明、大石真也、荒木望嗣、馬彪、藤井俊樹、有地法人、奥野恭史、掛谷秀昭、山崎晶、大野浩章、井貫晋輔
- Organizer
  第65回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 可視光レドックス触媒を用いたhetisine型及びvakognavine型アルカロイドの縮環ピロリジン骨格の構築2023
- Author(s)
  黒田慈瑛、有地法人、井貫晋輔、大野浩章
- Organizer
  第73回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 金触媒連続環化反応を基盤としたAspidophylline Aの全合成研究2023
- Author(s)
  笠置拓実、田口淳一、奥村怜司、大原礼子、橋本直季、大石真也、有地法人、井貫晋輔、大野浩章
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 金触媒連続環化反応を基盤としたAspidophylline Aの全合成研究2023
- Author(s)
  笠置拓実、田口淳一、奥村怜司、大原礼子、橋本直季、大石真也、有地法人、井貫晋輔、大野浩章
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] ルマジン構造を基盤とする新規MAIT細胞活性化剤の創製研究2023
- Author(s)
  高崎亮助、松岡巧朗, 有地法人, 山崎晶, 大野浩章, 井貫晋輔
- Organizer
  ケミカルバイオロジー学会第17回年会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] MR1の細胞表面量を指標とするリガンドスクリーニング法の開発とMAIT細胞モジュレーターの同定2023
- Author(s)
  松岡巧朗、服部明、大石真也、有地法人、掛谷秀昭、山崎晶、大野浩章、井貫晋輔
- Organizer
  ケミカルバイオロジー学会第17回年会
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 現代創薬を加速する創発的有機化学研究の実現に向けて2023
- Author(s)
  大野浩章
- Organizer
  第9回薬学の未来を考える京都シンポジウム
- Invited
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 可視光酸化還元触媒を用いたラジカルカスケード反応によるビシクロ[2.2.2]オクテン骨格構築反応の開発2023
- Author(s)
  井貫晋輔、吉田悠生、竹内春佳、中川航平、藤井俊樹、有地法人、大石真也、大野浩章
- Organizer
  第49回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 分子シミュレーションによるMR1細胞表面発現に重要な因子の特定2023
- Author(s)
  藤井俊樹, 荒木望嗣, 松本篤幸, 馬彪, 大野浩章, 井貫晋輔, 奥野恭史
- Organizer
  第40回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-23K27294
[Presentation] 金触媒を用いたアジドアルキンの連続環化反応による八員環縮環インドールの構築2023
- Author(s)
  長谷川大輝、有地法人、井貫晋輔、大野浩章
- Organizer
  第73回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 金触媒を用いたアレンインの連続環化反応による多環式芳香族化合物の構築2022
- Author(s)
  津野仁美、沈靖豊、小松紘樹、有地法人、井貫晋輔、大野浩章
- Organizer
  第72回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] アクアミリンアルカロイドの多様性指向型合成に向けた金触媒環化反応の開発と合成展開2022
- Author(s)
  橋本直季、有地法人、井貫晋輔、大野浩章
- Organizer
  第51回複素環化学討論会
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 金触媒を用いたアレンインの連続環化反応による多環式骨格の構築2022
- Author(s)
  津野仁美、小松紘樹、有地法人、井貫晋輔、大野浩章
- Organizer
  第48回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-22K19028
[Presentation] 生合成を模倣しない戦略によるインドールアルカロイドの全合成研究2021
- Author(s)
  大野浩章
- Organizer
  日本薬学会第141年会
- Invited
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒連続環化反応を基盤としたPicrinineの合成研究2021
- Author(s)
  橋本直季, 田口淳一, 大石真也, 井貫晋輔, 大野浩章
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いたアルキンのヒドロアリール化による縮環型インドレニン骨格の構築2021
- Author(s)
  島恭平, 大石真也, 井貫晋輔, 大野浩章
- Organizer
  日本薬学会第141年会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 可視光レドックス触媒を用いたラジカルipso環化反応を鍵とするZephycarinatine CおよびDの全合成2020
- Author(s)
  井貫晋輔, 竹内春佳, 中川航平, 川邊隆彰, 市村敦彦, 大石真也, 大野浩章
- Organizer
  反応と合成の進歩2020特別企画シンポジウム
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いたアレンインの連続環化反応による含窒素複素環骨格の構築2020
- Author(s)
  小松紘樹, 池内貴哉, 大石真也, 井貫晋輔, 大野浩章
- Organizer
  第70回日本薬学会関西支部大会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 可視光レドックス触媒によるβ開裂・C(sp3)-C(sp3)1,5-HAT連続反応を利用した(+)-polyoxamic acidの全合成2020
- Author(s)
  松岡巧朗, 井貫晋輔, 宮川貴吏, 大石真也, 大野浩章
- Organizer
  第62回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring Fused Indoles and Propellane-Type Indolines2019
- Author(s)
  Ayuta Yamaguchi, Shinsuke Inuki, Yusuke Tokimizu, Shinya Oishi, Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Total synthesis of dictyodendrins by the gold-catalyzed cascade cyclization of conjugated diynes with pyrroles2019
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 11th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed C-C bond Formation and Its Application to Alkaloid Synthesis2019
- Author(s)
  Hiroaki Ohno
- Organizer
  Technische Universitat Wien Special Lecture
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Gold-Catalyzed Cascade Cyclization for Fused Ring Construction2019
- Author(s)
  Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒を用いた分子内連続環化反応を基盤としたAspidophylline Aの全合成研究2019
- Author(s)
  田口淳一, 奥村怜司, 大原礼子, 井貫晋輔, 大石真也, 大野浩章
- Organizer
  第39回有機合成若手セミナー
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed Cascade Cyclization Reactions via C-H Bond Cleavage2019
- Author(s)
  Hiroaki Ohno
- Organizer
  The 47th Naito Conference
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Total synthesis of dictyodendrins by the gold-catalyzed cascade cyclization of conjugated diynes with pyrroles2019
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 11th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Gold-Catalyzed Cascade Cyclization of Alkynyl Tryptophol Derivatives: Synthetic Strategy for Aspidophylline A2019
- Author(s)
  Junichi Taguchi, Reiji Okumura, Ayako Ohara, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Gold-Catalyzed Cascade Cyclization of Alkynyl Tryptophol Derivatives: Synthetic Strategy for Aspidophylline A2019
- Author(s)
  Junichi Taguchi, Reiji Okumura, Ayako Ohara, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Dictyodendrin 類の多様性志向型全合成2019
- Author(s)
  松岡純平、松田優佳、川田惟樹、井貫晋輔、大石真也、大野浩章
- Organizer
  第69回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Controllable Formation of Oxocine-Fused Indoles and Propellane-Type Indolines via Gold-Catalyzed Cascade Cyclization2019
- Author(s)
  Ayuta Yamaguchi, Shinsuke Inuki, Yusuke Tokimizu, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Dictyodendrin 類の多様性志向型全合成2019
- Author(s)
  松岡純平、松田優佳、川田惟樹、井貫晋輔、大石真也、大野浩章
- Organizer
  第61回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed C-C bond Formation and Its Application to Alkaloid Synthesis2019
- Author(s)
  Hiroaki Ohno
- Organizer
  Technische Universitat Wien Special Lecture
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Synthetic Study of Aspidophylline A Based on Gold(I)-Catalyzed Cascade Cyclization2019
- Author(s)
  Junichi Taguchi, Reiji Okumura, Ayako Ohara, Shinsuke Inuki, Shinya Oishi and Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒連続環化反応を基盤としたAspidophylline Aの全合成研究2019
- Author(s)
  田口淳一、奥村怜司、大原礼子、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Synthetic Study of Aspidophylline A Based on Gold(I)-Catalyzed Cascade Cyclization2019
- Author(s)
  Junichi Taguchi, Reiji Okumura, Ayako Ohara, Shinsuke Inuki, Shinya Oishi and Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Dictyodendrin 類の多様性志向型全合成2019
- Author(s)
  松岡純平、松田優佳、川田惟樹、井貫晋輔、大石真也、大野浩章
- Organizer
  第61回天然有機化合物討論会
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles2019
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒連続環化反応を基盤としたAspidophylline Aの全合成研究2019
- Author(s)
  田口淳一, 奥村怜司, 大原礼子, 井貫晋輔, 大石真也, 大野浩章
- Organizer
  第39回有機合成若手セミナー
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Dictyodendrin 類の多様性志向型全合成2019
- Author(s)
  松岡純平、松田優佳、川田惟樹、井貫晋輔、大石真也、大野浩章
- Organizer
  第69回日本薬学会関西支部総会・大会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles2019
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒連続環化反応を基盤としたAspidophylline Aの全合成研究2019
- Author(s)
  田口淳一、奥村怜司、大原礼子、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed Cascade Cyclization for Fused Ring Construction2019
- Author(s)
  Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring Fused Indoles and Propellane-Type Indolines2019
- Author(s)
  Ayuta Yamaguchi, Shinsuke Inuki, Yusuke Tokimizu, Shinya Oishi, Hiroaki Ohno
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Gold-Catalyzed Cascade Cyclization Reactions via C-H Bond Cleavage2019
- Author(s)
  Hiroaki Ohno
- Organizer
  The 47th Naito Conference
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Controllable Formation of Oxocine-Fused Indoles and Propellane-Type Indolines via Gold-Catalyzed Cascade Cyclization2019
- Author(s)
  Ayuta Yamaguchi, Shinsuke Inuki, Yusuke Tokimizu, Shinya Oishi, Hiroaki Ohno
- Organizer
  The 8th Japanese-Sino Symposium on Organic Chemistry for Young Scientists
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] カプシドタンパク質の化学合成と粒子形成の最適化2018
- Author(s)
  佐々木順平, 石場勲之, 津田修吾, 西尾秀喜, 片岡紀代, 渡士幸一, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 金触媒を用いた複素環骨格の構築とアルカロイドの全合成2018
- Author(s)
  大野浩章
- Organizer
  第53回天然物化学談話会
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] グルタミン酸ラセマーゼMurIの化学合成法の確立2018
- Author(s)
  大原拓己, 野口太朗, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Synthetic Study of Akuammiline Alkaloids Based on Gold(I)-Catalyzed Cascade Cyclization2018
- Author(s)
  田口淳一、奥村怜司、大原礼子、井貫晋輔、大石真也、大野浩章
- Organizer
  JGP Chem & ChemEn International Workshop: Sustainability-Oriented Organic Synthesis
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] Synthesis of Fused Cyclopropanes via Gold-Catalyzed Cascade Cyclization of Allenynes2018
- Author(s)
  池内貴哉、井貫晋輔、大石真也、大野浩章
- Organizer
  JGP Chem & ChemEn International Workshop: Sustainability-Oriented Organic Synthesis
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Gold-Catalyzed C-C bond Formation and Its Application to Alkaloid Synthesis2018
- Author(s)
  Hiroaki Ohno
- Organizer
  1st NCTU Conference on Advanced Organic Synthesis
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒を用いた複素環骨格の構築とアルカロイドの全合成2018
- Author(s)
  大野浩章
- Organizer
  第53回天然物化学談話会
- Invited
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed C-C bond Formation and Its Application to Alkaloid Synthesis2018
- Author(s)
  Hiroaki Ohno
- Organizer
  1st NCTU Conference on Advanced Organic Synthesis
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Pd触媒を用いたTHF環構築によるJaspine B 位置異性体の合成研究2018
- Author(s)
  宮川貴吏、本田真歩、中村真也、仲西功、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dictyodendrin類の多様性志向型全合成2018
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  「有機合成化学を起点とするものづくり戦略」最終シンポジウム
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Dictyodendrin類の多様性志向型全合成2018
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  「有機合成化学を起点とするものづくり戦略」最終シンポジウム
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 天然物骨格一挙構築法の開発と応用2018
- Author(s)
  大野浩章
- Organizer
  京大テックフォーラム
- Invited
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Synthesis of Fused Cyclopropanes via Gold-Catalyzed Cascade Cyclization of Allenynes2018
- Author(s)
  池内貴哉、井貫晋輔、大石真也、大野浩章
- Organizer
  JGP Chem & ChemEn International Workshop: Sustainability-Oriented Organic Synthesis
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いた複素環骨格の構築とアルカロイドの全合成2018
- Author(s)
  大野浩章
- Organizer
  第53回天然物化学談話会
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Synthetic Study of Akuammiline Alkaloids Based on Gold(I)-Catalyzed Cascade Cyclization2018
- Author(s)
  田口淳一、奥村怜司、大原礼子、井貫晋輔、大石真也、大野浩章
- Organizer
  JGP Chem & ChemEn International Workshop: Sustainability-Oriented Organic Synthesis
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Gold-Catalyzed C-C bond Formation and Its Application to Alkaloid Synthesis2018
- Author(s)
  Hiroaki Ohno
- Organizer
  1st NCTU Conference on Advanced Organic Synthesis
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いたアレンインの連続環化反応による縮環シクロプロパンの合成2018
- Author(s)
  池内貴哉、井貫晋輔、大石真也、大野浩章
- Organizer
  第44回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 天然物骨格一挙構築法の開発と応用2018
- Author(s)
  大野浩章
- Organizer
  京大テックフォーラム
- Invited
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒を用いたアルカロイド型骨格の構築と応用2018
- Author(s)
  大野浩章
- Organizer
  千葉大学薬学研究科特別講演会
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Synthesis of Fused Cyclopropanes via Gold-Catalyzed Cascade Cyclization of Allenynes2018
- Author(s)
  池内貴哉、井貫晋輔、大石真也、大野浩章
- Organizer
  JGP Chem & ChemEn International Workshop: Sustainability-Oriented Organic Synthesis
- Int'l Joint Research
- Data Source
  KAKENHI-PUBLICLY-18H04408
[Presentation] 金触媒による共役ジインと置換ベンゼンの連続環化反応を利用したベンゾカルバゾール骨格の構築2017
- Author(s)
  大村駿介、川田惟樹、吉田勇介、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  仙台国際センター（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒による共役ジインとピロールを用いたPyrrolo[2,3-c]carbazole骨格の構築2017
- Author(s)
  川田惟樹、松田優佳、藤井信孝、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Dictyodendrin類の多様性志向型全合成2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  第15回次世代を担う有機化学シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いたスキップジインの連続反応の開発―シクロヘプタ［b］ピロール骨格の構築―2017
- Author(s)
  濱田直佳、吉田勇介、大石真也、大野浩章
- Organizer
  第67回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒によるアルカロイド型骨格の構築と全合成研究2017
- Author(s)
  大野浩章
- Organizer
  第37回有機合成若手セミナー
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒による共役ジインとピロールを用いたPyrrolo[2,3-c]carbazole骨格の構築2017
- Author(s)
  川田惟樹、松田優佳、藤井信孝、大野浩章、大石真也
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations2017
- Author(s)
  Hiroaki Ohno
- Organizer
  Nordic/Kyoto OMCOS 2017
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒による共役ジインと置換ベンゼンの連続環化反応を利用したベンゾカルバゾール骨格の構築2017
- Author(s)
  大村駿介、川田惟樹、吉田勇介、井貫晋輔、大石真也、大野浩章
- Organizer
  第67回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Total synthesis of dictyodendrins by the gold-catalyzed intermolecular cascade cyclization of conjugated diynes with pyrroles2017
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinya Oishi, Hiroaki Ohno
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dbzリンカーを用いた環状ペプチドの合成研究2017
- Author(s)
  大原拓己、金田雅仁、齋藤知、大野浩章、大石真也
- Organizer
  第49回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Intermolecular Cascade Cyclization of Conjugated Diynes with Pyrroles2017
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinya Oishi, Hiroaki Ohno
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いた分子内連続環化反応を基盤としたAspidophylline Aの全合成研究2017
- Author(s)
  奥村怜司、大原礼子、熊谷洋、大石真也、大野浩章
- Organizer
  第59回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2017
- Author(s)
  関口遼、黒柳友子、小林由佳、藤井信孝、大野浩章、大石真也
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dictyodendrin類の網羅的全合成と誘導体の活性評価2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた1,4-ジインの連続反応によるシクロヘプタ[b]ピロール骨格の構築2017
- Author(s)
  濱田直佳、吉田勇介、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  仙台国際センター（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒によるアルカロイド型骨格の構築と全合成研究2017
- Author(s)
  大野浩章
- Organizer
  第37回有機合成若手セミナー
- Invited
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒を用いた複素環骨格構築法の開発と応用2017
- Author(s)
  大野浩章
- Organizer
  中外製薬講演会
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒を用いた1,4-ジインの連続反応によるシクロヘプタ[b]ピロール骨格の構築2017
- Author(s)
  濱田直佳、吉田勇介、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  仙台国際センター（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] CXCR7受容体選択的リガンドの構造活性相関研究2017
- Author(s)
  関口遼、黒柳友子、小林由佳、小林数也、赤路健一、藤井信孝、大野浩章、大石真也
- Organizer
  第35回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いたアレンインの連続環化反応による縮環シクロプロパン骨格の合成2017
- Author(s)
  池内貴哉、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Pd触媒を用いたTHF環構築によるJaspine B 位置異性体の合成研究2017
- Author(s)
  宮川貴吏、本田真歩、中村真也、仲西功、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Dictyodendrin類の全合成研究2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Dictyodendrin類の全合成研究2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Dictyodendrin類の網羅的全合成と誘導体の活性評価2017
- Author(s)
  松岡純平，松田優佳，川田惟樹, 大石真也, 大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 金触媒による共役ジインと置換ベンゼンの連続環化反応を利用したベンゾカルバゾール骨格の構築2017
- Author(s)
  大村駿介、川田惟樹、吉田勇介、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Place of Presentation
  仙台国際センター（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた分子内連続環化反応を基盤としたAspidophylline Aの全合成研究2017
- Author(s)
  奥村　怜司、大原　礼子、熊谷　洋、大石　真也、大野　浩章
- Organizer
  第59回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒を用いたスキップジインの連続反応によるシクロヘプタ[b]ピロール骨格の構築2017
- Author(s)
  濱田直佳，吉田勇介，大石真也, 大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] Dictyodendrin類の多様性志向型全合成2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  第15回次世代を担う有機化学シンポジウム
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 鏡像体タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2017
- Author(s)
  周敬棠、野口太朗、本田香織、近藤恭光、長田裕之、大野浩章、藤井信孝、大石真也
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Development of peptide macrocyclization protocol utilizing o-aminoanilide linker for flow chemistry2017
- Author(s)
  Takumi Ohara, Masato Kaneda, Tomo Saito, Hiroaki Ohno, Shinya Oishi
- Organizer
  第54回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of novel NK3 receptor antagonists with reduced environmental impact2017
- Author(s)
  Koki Yamamoto, Hiroaki Ohno, Nobutaka Fujii, Shinya Oishi
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた分子内連続環化反応を基盤としたAspidophylline Aの全合成研究2017
- Author(s)
  奥村怜司、大原礼子、熊谷洋、大石真也、大野浩章
- Organizer
  第59回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-17H03971
[Presentation] 4-epi-Jaspine B位置異性体の合成と構造活性相関研究2017
- Author(s)
  宮川貴吏、本田真歩、小林由佳、中村真也、仲西功、藤井信孝、井貫晋輔、大石真也、大野浩章
- Organizer
  第34回有機合成化学セミナー
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いたアルカロイド型骨格の構築と応用2017
- Author(s)
  大野浩章
- Organizer
  岡山大学特別講演会
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Dictyodendrin類の全合成研究2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた分子内連続環化反応の開発―Aspidophylline A の合成研究―2017
- Author(s)
  奥村怜司、大原礼子、熊谷洋、井貫晋輔、大石真也、大野浩章
- Organizer
  第67回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Intermolecular Cascade Cyclization of Conjugated Diynes with Pyrroles2017
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinya Oishi, Hiroaki Ohno
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 4-epi-Jaspine B位置異性体の合成と構造活性相関研究2017
- Author(s)
  宮川貴吏、本田真歩、小林由佳、中村真也、仲西功、藤井信孝、井貫晋輔、大石真也、大野浩章
- Organizer
  第34回有機合成化学セミナー
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒を用いたスキップジインの連続反応によるシクロヘプタ[b]ピロール骨格の構築2017
- Author(s)
  濱田直佳，吉田勇介，大石真也, 大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations2017
- Author(s)
  Hiroaki Ohno
- Organizer
  Nordic/Kyoto OMCOS 2017
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Dbzリンカーを用いた環状ペプチドの合成研究2017
- Author(s)
  大原拓己、金田雅仁、齋藤知、大野浩章、大石真也
- Organizer
  第49回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dictyodendrin類の網羅的全合成と誘導体の活性評価2017
- Author(s)
  松岡純平，松田優佳，川田惟樹, 大石真也, 大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Strictamineの不斉形式全合成2016
- Author(s)
  熊谷　洋、西山大亮、大石真也、藤井信孝、大野浩章
- Organizer
  第42回反応と合成の進歩シンポジウム
- Place of Presentation
  清水文化会館（静岡県清水市）
- Year and Date
  2016-11-07
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 化学合成タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2016
- Author(s)
  周敬棠、大石真也、野口太朗、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第11回年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Facile access to the mirror-image library of chiral natural product derivatives: identification of MDM2-p53 interaction inhibitor2016
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Strictamineの不斉形式全合成2016
- Author(s)
  熊谷洋、西山大亮、大石真也、藤井信孝、大野浩章
- Organizer
  第42回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] プロパルギル基の転位を伴う2-アルキニルアニリンの連続環化反応を用いた高度縮環型複素環の合成2016
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第14回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール（東京都渋谷区）
- Year and Date
  2016-05-27
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Development of a screening system for Grb2 SH2 domain inhibitors using synthetic proteins2016
- Author(s)
  Taro Noguchi, Hiroyuki Ishiba, Kaori Honda, Yasumitsu Kondoh, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii, Shinya Oishi
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Strictamineの不斉形式全合成2016
- Author(s)
  熊谷　洋、西山大亮、大石真也、藤井信孝、大野浩章
- Organizer
  第42回反応と合成の進歩シンポジウム
- Place of Presentation
  清水文化会館（静岡県清水市）
- Year and Date
  2016-11-07
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒による共役ジインとピロールを用いたPyrrolo[2,3-c]carbazole骨格の構築2016
- Author(s)
  川田惟樹、松田優佳、藤井信孝、大石真也、大野浩章
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学（大阪府高槻市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いたアスピドスペルマ型アルカロイド骨格構築法の開発－Aspidosprmidineの合成研究－2016
- Author(s)
  熊谷　洋、大石真也、大野浩章
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学（大阪府高槻市）
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Strictamineの全合成研究2016
- Author(s)
  西山大亮、大原礼子、熊谷洋、千葉浩亮、藤井信孝、大石真也、大野浩章
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Place of Presentation
  つくば国際会議場（茨城県つくば市）
- Year and Date
  2016-11-30
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いたアスピドスペルマ型アルカロイド骨格構築法の開発--Aspidosprmidineの合成研究--2016
- Author(s)
  熊谷洋、大石真也、大野浩章
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Design of iron-chelating cyclic peptides2016
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  8th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of screening systems for c-Src SH2 domain inhibitors using synthetic proteins2016
- Author(s)
  Keitou Shu, Taro Noguchi, Nobutaka Fujii, Hiroaki Ohno, Shinya Oishi
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Design of Fe(II)-chelaing cyclic hexapeptide with bidentate pyridinyl-triazlole groups2016
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 長時間作用型PEG化NK3受容体作動薬の創製2016
- Author(s)
  桑井真司、大石真也、三須良介、大野浩章、山村崇、若林嘉浩、岡村裕昭、藤井信孝
- Organizer
  日本薬学会第136回年会
- Place of Presentation
  パシフィコ横浜（神奈川県横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた共役ジインの連続環化反応による1,7-縮環型インドールの構築2016
- Author(s)
  吉田勇介、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  日本薬学会第136回年会
- Place of Presentation
  パシフィコ横浜（神奈川県横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた共役ジインの連続環化反応による1,7-縮環型インドールの構築2016
- Author(s)
  吉田勇介、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  日本薬学会第136回年会
- Place of Presentation
  パシフィコ横浜（神奈川県横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Development of Novel CXCR7 Ligands: Selectivity Switch from CXCR4 Antagonists with Cyclic Pentapeptide Scaffold2016
- Author(s)
  Tomoko Kuroyanagi, Shinya Oishi, Tatsuhiko Kubo, Yuka Kobayashi, Haruka Sekiguchi, Ryosuke Misu, Hiroaki Ohno, Nicolas Montpas, Nikolaus Heveker, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Strictamineの全合成研究2016
- Author(s)
  西山大亮、大原礼子、熊谷洋、千葉浩亮、藤井信孝、大石真也、大野浩章
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いたアスピドスペルマ型アルカロイド骨格構築法の開発－Aspidosprmidineの合成研究－2016
- Author(s)
  熊谷　洋、大石真也、大野浩章
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学（大阪府高槻市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Gold-catalyzed construction of tetracyclic skeleton for aspidosperma alkaloid synthesis: Synthetic study on (±)-aspidospermidine2016
- Author(s)
  Hiroshi Kumagai, Shinya Oishi, Hiroaki Ohno
- Organizer
  ISONIS-10
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた反応の開発と応用2016
- Author(s)
  大野浩章
- Organizer
  塩野義製薬創薬科学セミナー
- Place of Presentation
  塩野義製薬医薬研究センター（大阪府豊中市）
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] MDM2タンパク質の化学合成と天然物の鏡像体化合物群からの医薬品探索への応用2016
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  第36回有機合成若手セミナー
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 多重結合の連続活性化を用いた骨格構築反応の開発と応用2016
- Author(s)
  大野浩章
- Organizer
  近畿大学薬学研究科講演会
- Place of Presentation
  近畿大学薬学研究科（大阪府東大阪市）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Strictamineの全合成研究2016
- Author(s)
  西山大亮、大原礼子、熊谷洋、千葉浩亮、藤井信孝、大石真也、大野浩章
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Place of Presentation
  つくば国際会議場（茨城県つくば市）
- Year and Date
  2016-11-30
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒による共役ジインとピロールを用いたPyrrolo[2,3-c]carbazole骨格の構築2016
- Author(s)
  川田惟樹、松田優佳、藤井信孝、大野浩章、大石真也
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Place of Presentation
  大阪薬科大学（大阪府高槻市）
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Efficient Construction of Heterocyclic Scaffolds and Its Application2016
- Author(s)
  Hiroaki Ohno
- Organizer
  AGORA Bayer Meeting
- Place of Presentation
  京都大学国際科学イノベーション棟（京都）
- Year and Date
  2016-04-14
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] ケモカイン受容体CXCR7 選択的リガンドの構造最適化研究2016
- Author(s)
  関口遼、大石真也、黒柳友子、小林由佳、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第11回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Facile access to the mirror-image library of chiral natural product derivatives: identification of MDM2-p53 interaction inhibitor2016
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 多重結合の連続活性化を用いた骨格構築反応の開発と応用2016
- Author(s)
  大野浩章
- Organizer
  近畿大学薬学研究科講演会
- Place of Presentation
  近畿大学薬学研究科（大阪府東大阪市）
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Total synthesis of a novel cytotoxic depsipeptide from Okinawan marine cyanobacteria2016
- Author(s)
  Masato Kaneda, Shinya Oishi, Kosuke Sueyoshi, Toshiaki Teruya, Hiroaki Ohno and Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] プロパルギル基の転位を伴う2-アルキニルアニリンの連続環化反応を用いた高度縮環型複素環の合成2016
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第14回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール（東京都渋谷区）
- Year and Date
  2016-05-27
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 化学合成タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2016
- Author(s)
  周敬棠、野口太朗、藤井信孝、大野浩章、大石真也
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 天然物とその誘導体の鏡像体化合物群の活用を目指した新規スクリーニング法の開発2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  名城大学特別講演会
- Place of Presentation
  名城大学薬学部（愛知県名古屋市）
- Invited
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of Novel CXCR7 Ligands by Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold2015
- Author(s)
  Shinya Oishi, Tomoko Kuroyanagi, Tatsuhiko Kubo, Nicolas Montpas, Yasushi Yoshikawa, Ryosuke Misu, Yuka Kobayashi, Hiroaki Ohno, Nikolaus Heveker, Toshio Furuya, and Nobutaka Fujii
- Organizer
  AIMECS2015
- Place of Presentation
  Jeju international convention center（韓国、済州島）
- Year and Date
  2015-10-18
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  名城大学特別講演会
- Place of Presentation
  名城大学薬学部（愛知県名古屋市）
- Year and Date
  2015-12-04
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] Identification of an MDM2-p53 interaction inhibitor from virtual mirror-image library of chiral natural product derivatives2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第52回ペプチド討論会
- Place of Presentation
  平塚市中央公民館（神奈川県平塚市）
- Year and Date
  2015-11-16
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Identification of a novel MDM2-p53 inhibitor using mirror-image-screening technology for chiral natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  SKO symposium
- Place of Presentation
  New Drug Development Center, Seoul University（韓国、ソウル）
- Year and Date
  2015-11-17
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2015
- Author(s)
  黒柳友子，大石真也，小林由佳，関口遼，三須良介，大野浩章，Montpas Nicolas，Heveker Nikolaus，藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles2015
- Author(s)
  Hiroaki Ohno
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（アメリカ、ホノルル）
- Year and Date
  2015-12-15
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] プロパルギル転位を伴う共役ジインの金触媒三連続環化反応を用いたカルバゾールの合成2015
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 天然物とその誘導体の鏡像体化合物群の活用を目指した新規スクリーニング法の開発2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2015
- Author(s)
  黒柳友子，大石真也，久保達彦，三須良介，小林由佳，大野浩章，Montpas Nicolas，Heveker Nikolaus，吉川寧，古谷利夫，藤井信孝
- Organizer
  第65回日本薬学会　近畿支部総会・大会
- Place of Presentation
  大阪大谷大学（大阪府羽曳野市）
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles2015
- Author(s)
  Hiroaki Ohno
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（アメリカ、ホノルル）
- Year and Date
  2015-12-15
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] アルキンの活性化を基盤とする連続反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  日本薬学会東海支部特別講演会
- Place of Presentation
  岐阜薬科大学（岐阜県岐阜市）
- Invited
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Novel screening approach for drug discovery from virtual mirror-image libaray of natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（米国、ホノルル市）
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] アポモルヒネによるMDM2-p53相互作用の阻害メカニズムの解明2015
- Author(s)
  石場勲之、大石真也、野口太朗、周敬棠、大野浩章、本田香織、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第65回日本薬学会近畿支部大会
- Place of Presentation
  大阪大谷大学（大阪府富田林市）
- Year and Date
  2015-10-17
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Identification of a novel MDM2-p53 inhibitor using mirror-image-screening technology for chiral natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  SKO symposium
- Place of Presentation
  ソウル国際大学（韓国、ソウル市）
- Year and Date
  2015-11-17
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] キラルな天然有機化合物の鏡像体群をリソースとしたMDM2-p53間相互作用阻害剤の探索2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Investigation of inhibitory mechanism of apomorphine against MDM2-p53 interaction2015
- Author(s)
  Hiroyuki Ishiba, Shinya Oishi, Taro Noguchi, Keito Shu, Hiroaki Ohno, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第52回ペプチド討論会
- Place of Presentation
  平塚市中央公民館（神奈川県平塚市）
- Year and Date
  2015-11-16
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] MDM2-p53タンパク質間相互作用に対するアポモルフィンの阻害メカニズムの解明2015
- Author(s)
  石場勲之、大石真也、野口太朗、周敬棠、大野浩章、藤井信孝
- Organizer
  創薬懇話会2015 in 徳島
- Place of Presentation
  グランドエクシブ鳴門ザ・ロッジ（徳島県鳴門市）
- Year and Date
  2015-07-01
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  京大有機金属化学若手勉強会
- Place of Presentation
  京都大学薬学研究科（京都府京都市）
- Invited
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 環境調和型NK3受容体拮抗剤の創製研究2015
- Author(s)
  山本昂輝、大石真也、大野浩章、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Novel screening approach for drug discovery from virtual mirror-image library of natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（アメリカ、ホノルル）
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた共役ジインの連続環化反応による縮環インドールの一挙合成2015
- Author(s)
  直江紗織、斉藤竜男、内山真伸、大石真也、藤井信孝、大野浩章
- Organizer
  第13回次世代を担う有機化学シンポジウム
- Place of Presentation
  立命館大学（滋賀県草津市）
- Year and Date
  2015-05-22
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  京大有機金属化学若手勉強会
- Place of Presentation
  京都大学薬学研究科（京都府京都市）
- Year and Date
  2015-10-31
- Invited
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  名城大学特別講演会
- Place of Presentation
  名城大学薬学部（愛知県名古屋市）
- Year and Date
  2015-12-04
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] プロパルギル転位を伴う共役ジインの金触媒三連続環化反応を用いたカルバゾールの合成2015
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] PEG修飾による長時間作用型NK3受容体作動薬の創製2015
- Author(s)
  桑井真司、大石真也、三須良介、岡崎志穂、山本昂輝、大野浩章、山村崇、若林嘉浩、岡村裕昭、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 共役ジインとピロールを用いた金触媒[4+2]型インドール合成と縮環骨格構築への展開2015
- Author(s)
  松田優佳、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles2015
- Author(s)
  Hiroaki Ohno
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（アメリカ、ホノルル）
- Year and Date
  2015-12-15
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  京大有機金属化学若手勉強会
- Place of Presentation
  京都大学薬学研究科（京都府京都市）
- Year and Date
  2015-10-31
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] プロパルギル転位を伴う共役ジインの金触媒三連続環化反応を用いたカルバゾールの合成2015
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] アルキンの活性化を基盤とする連続反応の開発と応用2015
- Author(s)
  大野浩章
- Organizer
  日本薬学会東海支部特別講演会
- Place of Presentation
  岐阜薬科大学（岐阜県岐阜市）
- Year and Date
  2015-05-29
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 共役ジインとピロールを用いた金触媒[4+2]型インドール合成と縮環骨格構築への展開2015
- Author(s)
  松田優佳、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15KT0061
[Presentation] 共役ジインとピロールを用いた金触媒[4+2]型インドール合成と縮環骨格構築への展開2015
- Author(s)
  松田優佳、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた共役ジインの連続環化反応による縮環インドールの一挙合成2014
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  日本薬学会第134年会
- Place of Presentation
  熊本大学（熊本県熊本市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] アレンやアルキンを合成素子とする連続反応の開発と応用2014
- Author(s)
  大野浩章
- Organizer
  金沢大学特別講演会
- Place of Presentation
  金沢大学（石川県金沢市）
- Year and Date
  2014-06-13
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた共役ジインの連続環化反応による縮環インドールの一挙合成2014
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  日本薬学会第134年会
- Place of Presentation
  熊本大学（熊本県熊本市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] パラジウム触媒による連続環化反応を用いた四環性スピロインドール類の合成2013
- Author(s)
  岩田顕、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部（福岡県福岡市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いたベンゾフランによる分子内ヒドロアリール化反応の検討2013
- Author(s)
  坂井由葵、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部（福岡県福岡市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] パラジウム触媒による連続反応を用いたスピロインドール類の合成2013
- Author(s)
  岩田顕、大野浩章、他
- Organizer
  日本薬学会第133年会
- Place of Presentation
  パシフィコ横浜（神奈川県）
- Year and Date
  2013-03-28
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Synthesis of the Fused Tetracyclic Spiroindoles via Palladium-Catalyzed Cascade Reaction2013
- Author(s)
  Iwata, A.; Ohno, H., et al.
- Organizer
  246th American Chemical Society National Meeting and Exposition
- Place of Presentation
  Indiana Convention Center（米国）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究2013
- Author(s)
  大野浩章
- Organizer
  天然物ケミカルバイオロジー：分子標的と活性制御地区シンポジウム
- Place of Presentation
  理化学研究所（埼玉県）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用2013
- Author(s)
  大野浩章
- Organizer
  創薬基盤科学若手セミナー
- Place of Presentation
  立命館大学（滋賀県草津市）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 付加反応を用いて中心骨格を構築する天然物合成2013
- Author(s)
  大野浩章
- Organizer
  第12回化学系薬学若手研究者セミナー（日本薬学会東北支部）
- Place of Presentation
  東北大学（宮城県仙台市）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 化合物アレイを用いた新規MDM2/MDMX-p53阻害剤探索法の開発2013
- Author(s)
  野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  日本薬学会第133年会
- Place of Presentation
  パシフィコ横浜（神奈川県）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Gold-Catalyzed Reactions for Construction of Heterocycles2013
- Author(s)
  Ohno, H.
- Organizer
  Special Lecture at Dortmund University
- Place of Presentation
  ドルトムント工科大学（ドイツ、ドルトムント）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用2013
- Author(s)
  大野浩章
- Organizer
  創薬基盤科学若手セミナー
- Place of Presentation
  立命館大学　（滋賀県草津市）
- Year and Date
  2013-12-09
- Invited
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた共役ジインの多連続環化反応による縮環インドールの一挙合成2013
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部（福岡県福岡市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Gold-Catalyzed Reactions for Construction of Heterocycles2013
- Author(s)
  Ohno, H.
- Organizer
  Special Lecture at Dortmund University
- Place of Presentation
  ドルトムント工科大学（ドイツ）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Synthesis of the Fused Tetracyclic Spiroindoles via Palladium-Catalyzed Cascade Reaction2013
- Author(s)
  Akira Iwata, Hiroaki Ohno, Nobutaka Fujii, et al.
- Organizer
  246th American Chemical Society National Meeting and Exposition
- Place of Presentation
  Indiana Convention Center（米国インディアナ州）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用2013
- Author(s)
  大野浩章
- Organizer
  創薬基盤科学若手セミナー
- Place of Presentation
  立命館大学（滋賀県草津市）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] パラジウム触媒を用いた中員環形成反応によるLaurencia族環状エーテルの構築：Laurendecumallene Bの合成研究2013
- Author(s)
  大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学（福岡県福岡市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] パラジウム触媒による連続環化反応を用いた4環姓スピロインドール類の合成2013
- Author(s)
  岩田　顕、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学（福岡県福岡市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いた共役ジインの多連続環化反応による縮環インドールの一挙合成2013
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学（福岡県福岡市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Gold-Catalyzed Reactions for Construction of Heterocycles2013
- Author(s)
  Ohno, H.
- Organizer
  Special Lecture at Heidelberg University
- Place of Presentation
  ハイデルベルク大学（ドイツ、ハイデルベルク）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた三成分環化反応によるジヒドロピラゾールの合成とCK2阻害剤開発への応用2013
- Author(s)
  大野浩章、他
- Organizer
  第43回複素環化学討論会
- Place of Presentation
  長良川国際会議場（岐阜県岐阜市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] パラジウム触媒を用いた中員環形成反応によるLaurencia族環状エーテルの構築：Laurendecumallene Bの合成研究2013
- Author(s)
  大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部（福岡県福岡市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] パラジウム触媒による連続反応を用いたスピロインドール類の合成2013
- Author(s)
  岩田顕、大野浩章、他
- Organizer
  日本薬学会第133年会
- Place of Presentation
  パシフィコ横浜（神奈川県横浜市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Gold-Catalyzed Reactions for Construction of Heterocycles2013
- Author(s)
  Ohno, H.
- Organizer
  Special Lecture at Heidelberg University
- Place of Presentation
  ハイデルベルク大学（ドイツ）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用2013
- Author(s)
  大野浩章
- Organizer
  第18回鴨叡会・生命分子化学科セミナー
- Place of Presentation
  京都府立大学（京都府京都市）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究2013
- Author(s)
  大野浩章
- Organizer
  天然物ケミカルバイオロジー：分子標的と活性制御地区シンポジウム
- Place of Presentation
  理化学研究所（埼玉県和光市）
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた三成分環化反応によるジヒドロピラゾールの合成とCK2阻害剤開発への応用2013
- Author(s)
  大野浩章、他
- Organizer
  第43回複素環化学討論会
- Place of Presentation
  長良川国際会議場（岐阜県岐阜市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 付加反応を用いて中心骨格を構築する天然物合成2013
- Author(s)
  大野浩章
- Organizer
  第12回化学系薬学若手研究者セミナー（日本薬学会東北支部）
- Place of Presentation
  東北大学（宮城県仙台市）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いたベンゾフランによる分子内ヒドロアリール化反応の検討2013
- Author(s)
  坂井由葵、大野浩章、他
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学（福岡県福岡市）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用2013
- Author(s)
  大野浩章
- Organizer
  第18回鴨叡会・生命分子化学科セミナー
- Place of Presentation
  京都府立大学（京都府京都市）
- Invited
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] ピリミドベンゾチアジン誘導体の新規合成法の開発と抗HIV剤を指向した構造活性相関研究2012
- Author(s)
  水原司、大石真也、大野浩章、志村和也、松岡雅雄、藤井信孝
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒による三成分環形成反応を用いた多置換ジヒドロピラゾールの効率的合成法の開発2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒を用いた位置選択的なカスケード型分子間/分子内付加反応による縮合ベンゼン環の一挙構築法の開発2012
- Author(s)
  直江紗織、大野浩章, 他
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Pd触媒を用いたプロパルギル化合物の連続環化反応を利用した(+)-ビオチンの合成研究2012
- Author(s)
  水嶋真吾、大野浩章, 他
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-29
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] パラジウム触媒によるプロパルギル化合物の中員環形成反応を利用したlaurendecumallene Bの合成研究2012
- Author(s)
  吉光佑二、大野浩章、他
- Organizer
  第38回反応と合成の進歩シンポジウム
- Place of Presentation
  タワーホール船堀（東京都江戸川区）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Synthetic Study of Quinocarcin2012
- Author(s)
  Chiba, H., Ohno, H., et al
- Organizer
  243rd American Chemical Society National Meeting & Exposition
- Place of Presentation
  San Diego (USA)
- Year and Date
  2012-03-25
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Enantioselective Total Syntheses of (+)-Lysergic Acid, (+)-Lysergol and (+)-Isolysergol2012
- Author(s)
  Iwata, A. and Ohno, H. et al.
- Organizer
  IKCOC-12
- Place of Presentation
  リーガロイヤルホテル京都（京都府）
- Year and Date
  2012-11-12
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] パラジウム触媒によるプロパルギル化合物の中員環形成反応を利用したlaurendecumallene Bの合成研究2012
- Author(s)
  吉光佑二、大野浩章、他
- Organizer
  第38回反応と合成の進歩シンポジウム
- Place of Presentation
  タワーホール船堀（東京都）
- Year and Date
  2012-11-05
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] 縮環型含窒素複素環の多様性指向型合成反応の開発とCK2阻害剤の構造活性相関研究への応用2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] ピリミドベンゾチアジン誘導体の合成法の開発と抗HIV 剤の構造活性相関研究への応用2012
- Author(s)
  水原司、大石真也、大野浩章、志村和也、松岡雅雄、藤井信孝
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Potent CXCR4 Antagonists Containing Amidine-type Peptide Bond Isosteres2012
- Author(s)
  Kubo T, Inokuchi E, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Jaspine B立体異性体の分岐的合成と構造活性相関研究2012
- Author(s)
  宮垣潤、吉光佑二、大石真也、大野浩章、藤井信孝
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた位置選択的なカスケード型分子間/分子内付加反応による縮合ベンゼン環の一挙構築法の開発2012
- Author(s)
  直江紗織、大野浩章、他5名
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Efficient synthesis of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives and its application to structure-activity relationship study of anti-HIV agents2012
- Author(s)
  Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  第6回武田科学振興財団薬科学シンポジウム
- Place of Presentation
  武田薬品工業研修所（大阪府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] (-)-Quinocarcinの全合成2012
- Author(s)
  千葉浩亮、大野浩章、他
- Organizer
  第38回反応と合成の進歩シンポジウム
- Place of Presentation
  タワーホール船堀（東京都江戸川区）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究2012
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B) and their sphingosine kinase inhibitory activities2012
- Author(s)
  吉光佑二、宮垣潤、大石真也、藤井信孝、大野浩章
- Organizer
  ISMC2012
- Place of Presentation
  ベルリン（ドイツ）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒による三成分環形成反応を用いた多置換ジヒドロピラゾールの効率的合成法の開発2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府）
- Year and Date
  2012-10-11
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] (-)-Quinocarcinの全合成2012
- Author(s)
  千葉浩亮、大野浩章、他
- Organizer
  第38回反応と合成の進歩シンポジウム
- Place of Presentation
  タワーホール船堀（東京都）
- Year and Date
  2012-11-05
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成2012
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学（北海道）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] アザインドール骨格またはフェニルアゾール骨格を有する新規プロテインキナーゼCK2阻害剤の開発研究2012
- Author(s)
  侯増燁、大野浩章、他
- Organizer
  第10回次世代シンポ
- Place of Presentation
  大阪大学（大阪府吹田市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B) and their sphingosine kinase inhibitory activities2012
- Author(s)
  吉光佑二、宮垣潤、大石真也、藤井信孝、大野浩章
- Organizer
  ISMC2012
- Place of Presentation
  ベルリン（ドイツ）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives2012
- Author(s)
  Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  IKCOC-12
- Place of Presentation
  リーがロイヤルホテル京都（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Synthesis and structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for development of anti-HIV agents2012
- Author(s)
  水原司、大石真也、大野浩章、志村和也、松岡雅雄、藤井信孝
- Organizer
  The 7th SKO Joint Symposium for Young Scientists
- Place of Presentation
  京都大学（京都府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] アザインドール骨格またはフェニルアゾール骨格を有する新規プロテインキナーゼCK2阻害剤の開発研究2012
- Author(s)
  侯増燁、大石真也、武井義則、安江美里、三須良介、鈴木大和、村田克美、北浦和夫、平澤明、辻本豪三、大野浩章、藤井信孝、仲西功、中村真也、呉竜英、木下誉富
- Organizer
  第10回次世代を担う有機化学シンポジウム
- Place of Presentation
  大阪大学銀杏会館（大阪府）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究2012
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒を用いた位置選択的なカスケード型分子間/分子内付加反応による縮合ベンゼン環の一挙構築法の開発2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第62回日本薬学会近畿支部総会・大会
- Place of Presentation
  武庫川女子大学（兵庫県西宮市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成2012
- Author(s)
  宮垣潤、大野浩章、他3名
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-29
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成2012
- Author(s)
  宮垣潤、大野浩章, 他
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-29
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Enantioselective Total Syntheses of (+)-Lysergic Acid, (+)-Lysergol and (+)-Isolysergol2012
- Author(s)
  Iwata, A. and Ohno, H. et al.
- Organizer
  IKCOC-12
- Place of Presentation
  リーガロイヤルホテル京都（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Synthetic Study of Quinocarcin2012
- Author(s)
  Chiba, H., Ohno, H., et al
- Organizer
  243rd American Chemical Society National Meeting & Exposition
- Place of Presentation
  San Diego (USA)
- Year and Date
  2012-03-25
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Efficient Synthesis of Highly Functionalized Dihydropyrazoles via Gold-Catalyzed Three-Component Annulation2012
- Author(s)
  Suzuki Y, Oishi S, Fujii N, Ohno H.
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた位置選択的なカスケード型分子間/分子内付加反応による縮合ベンゼン環の一挙構築法の開発2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第62回日本薬学会近畿支部総会・大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Jaspine B立体異性体の分岐的合成と構造活性相関研究2012
- Author(s)
  宮垣潤、大野浩章、他
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 縮環型含窒素複素環の多様性指向型合成反応の開発とCK2阻害剤の構造活性相関研究への応用2012
- Author(s)
  直江紗織、大野浩章、他
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府）
- Year and Date
  2012-06-07
- Data Source
  KAKENHI-PUBLICLY-24106720
[Presentation] Synthetic Study of Quinocarcin2012
- Author(s)
  H. Chiba, H. Ohno, 他2名
- Organizer
  243rd American Chemical Society National Meeting & Exposition
- Place of Presentation
  San Diego(USA)
- Year and Date
  2012-03-25
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Pd触媒を用いたプロパルギル化合物の連続環化反応を利用した(+)-ビオチンの合成研究2012
- Author(s)
  水嶋真吾、大野浩章、他3名
- Organizer
  日本薬学会第132年会
- Place of Presentation
  北海道大学(北海道)
- Year and Date
  2012-03-29
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B)2012
- Author(s)
  Yoshimitsu, Y. and Ohno, H. et al.
- Organizer
  ISMC2012
- Place of Presentation
  Estrel Hotel（ドイツ、ベルリン）
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Efficient Synthesis of Pyrimido[1,2-c]benzothiazin-6-imine and Related Tricyclic Heterocycles by Cu(II)-mediated C-H Functionalization and Aromatic Nucleophilic Substitution2011
- Author(s)
  Mizuhara T, Oishi S, Fujii N, Ohno H.
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 銅触媒による連続環化反応を用いた高度縮環型ペリミジンの合成2011
- Author(s)
  時水勇輔、大野浩章、他4名
- Organizer
  第61回日本薬学会近畿支部総会・大会
- Place of Presentation
  神戸薬科大学(兵庫県)
- Year and Date
  2011-10-23
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Jaspine Bおよびその誘導体の立体分岐合成と構造活性相関研究2011
- Author(s)
  宮垣潤、大野浩章, 他
- Organizer
  第28回有機合成化学セミナー
- Place of Presentation
  滝の湯(山形県)
- Year and Date
  2011-09-01
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒による三成分環形成反応を用いた多置換ジヒドロピラゾールの効率的合成法の開発2011
- Author(s)
  鈴木大和、大野浩章、他2名
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Synthesis and Biological Evaluation of Novel CXCR4 Antagonists Containing Amidine-type Peptide Bond Isosteres2011
- Author(s)
  Inokuchi E, Oishi S, Kubo T, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章、他2名
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Structure-activity Relationship Study on a CXCR4 Antagonist FC131 Using Alkene-type Dipeptide Isosteres2011
- Author(s)
  Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Naito T, Matsuoka M, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用2011
- Author(s)
  大野浩章
- Organizer
  6th Organic Syntheses Lectureship, University of Tokyo
- Place of Presentation
  東京大学(東京都)(招待講演)
- Year and Date
  2011-02-22
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Jaspine Bおよびその誘導体の立体分岐合成と構造活性相関研究2011
- Author(s)
  宮垣潤、大野浩章、他3名
- Organizer
  第28回有機合成化学セミナー
- Place of Presentation
  滝の湯(山形県)
- Year and Date
  2011-09-01
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたヒドロアリール化反応を基盤とする連続環化反応の開発2011
- Author(s)
  直江紗織、大野浩章, 他
- Organizer
  第28回有機合成化学セミナー
- Place of Presentation
  滝の湯(山形県)
- Year and Date
  2011-09-01
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Efficient Synthesis of Highly Functionalized Dihydropyrazoles via Gold-Catalyzed Three-Component Annulation2011
- Author(s)
  Y. Suzuki, H. Ohno, 他2名
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒による連続環化反応を用いた高度縮環型ペリミジンの合成2011
- Author(s)
  時水勇輔、大野浩章, 他
- Organizer
  第61回日本薬学会近畿支部総会・大会
- Place of Presentation
  神戸薬科大学(兵庫県)
- Year and Date
  2011-10-23
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  第53回天然有機化合物討論会
- Place of Presentation
  大阪国際交流センター(大阪府)
- Year and Date
  2011-09-28
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いたオルト無置換ベンズアミジンのアルキニル化-環化によるキナゾリンの直接的合成2011
- Author(s)
  時水勇輔、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] DIVERSITY-ORIENTED SYNTHESIS OF PYRIMIDO[1,2-c][1,3]BENZOTHIAZIN-6-IMINE AND THE RELATED TRICYCLIC HETEROCYCLES2011
- Author(s)
  Mizuhara T, Oishi S, Ohno H, Fujii N
- Organizer
  Nature Chemical Biology Symposium 2011: Cancer Chemical Biology
- Place of Presentation
  Boston（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章、他2名
- Organizer
  第53回天然有機化合物討論会
- Place of Presentation
  大阪国際交流センター(大阪府)
- Year and Date
  2011-09-28
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたアニリン誘導体の連続型分子内ヒドロアミノ化-ヒドロアリール化反応による高度縮環型カルバゾール誘導体の合成2011
- Author(s)
  稲葉祐介、大野浩章、他3名
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] リゼルグ酸および関連アルカロイドの不斉全合成2011
- Author(s)
  岩田顕、大野浩章, 他
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] リゼルグ酸および関連アルカロイドの不斉全合成2011
- Author(s)
  岩田顕、大野浩章、他3名
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたアルキンに対する分子間求核付加-環化反応によるナフタレン誘導体の合成2011
- Author(s)
  直江紗織、大野浩章, 他
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] INTERNALIZATION OF CXC CHEMOKINE RECEPTOR 4 (CXCR4) INDUCED BY POLYPHEMUSIN II-DERIVED ANTAGONIST PEPTIDES2011
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Nakase I, Futaki S, Fujii N.
- Organizer
  第48回ペプチド討論会
- Place of Presentation
  札幌コンベンションセンター（北海道）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Total Synthesis of (+)-Lysergic Acid by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group2011
- Author(s)
  Ohno, H., et al
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成2011
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第28回有機合成化学セミナー
- Place of Presentation
  滝の湯（山形県）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Efficient Synthesis of Highly Functionalized Dihydropyrazoles via Gold-Catalyzed Three-Component Annulation2011
- Author(s)
  Suzuki, Y., Ohno, H., et al
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Jaspine Bおよびその誘導体の立体分岐合成と構造活性相関研究2011
- Author(s)
  吉光佑二、大野浩章, 他
- Organizer
  第9回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール(東京都)
- Year and Date
  2011-05-28
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用2011
- Author(s)
  大野浩章
- Organizer
  6th Organic Syntheses Lectureship(University of Tokyo)
- Place of Presentation
  東京大学(東京)(招待講演)
- Year and Date
  2011-02-22
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] アミジン型ペプチド結合等価体の合成と応用2011
- Author(s)
  井ノ口恵利子、山田愛、大石真也、久保達彦、大野浩章、保住健太郎、野水基義、志村和也、松岡雅雄、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会第6回年会
- Place of Presentation
  東京工業大学大岡山キャンパス（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Synthetic Study of Quinocarcin2011
- Author(s)
  Chiba, H., Ohno, H., et al
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Goldcatalyzed three-component annulation : anefficient synthesis of 1, 2, 3, 5-tetrasubstituted dihydropyrazoles from alkynes, aldehydes, and hydrazines"2011
- Author(s)
  Y. Suzuki, H. Ohno, 他2名
- Organizer
  242rd American Chemical Society National Meeting & Exposition
- Place of Presentation
  Denver(USA)
- Year and Date
  2011-08-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用2011
- Author(s)
  大野浩章
- Organizer
  6th Organic Syntheses Lectureship, University of Tokyo
- Place of Presentation
  東京大学(東京都)
- Year and Date
  2011-02-22
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] アルケン型及びアミジン型ジペプチドイソスターの合成とCXCR4拮抗剤の構造活性相関研究への応用2011
- Author(s)
  小林数也、大石真也、井ノ口恵利子、林亮子、富田健嗣、久保達彦、棚原憲子、大野浩章、藤井信孝、吉川寧、古谷利夫、志村和也、松岡雅雄
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール（徳島県）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Gold-catalyzed three-component annulation: an efficient synthesis of 1,2,3,5-tetrasubstituted dihydropyrazoles from alkynes, aldehydes, and hydrazines2011
- Author(s)
  Suzuki Y, Oishi S, Fujii N, Ohno H.
- Organizer
  242nd American Chemical Society National Meeting & Exposition
- Place of Presentation
  Denver（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒によるアルキンのヒドロアリール化を用いた多連続環化反応の開発2011
- Author(s)
  大野浩章, 他
- Organizer
  第41回複素環化学討論会
- Place of Presentation
  熊本市民会館・(熊本県)
- Year and Date
  2011-10-20
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  第53回天然有機化合物討論会
- Place of Presentation
  大阪国際交流センター(大阪府)
- Year and Date
  2011-09-28
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒による三成分環形成反応を用いた多置換ジヒドロピラゾールの効率的合成法の開発2011
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 銅触媒を用いたオルト無置換ベンズアミジンのアルキニル化-環化によるキナゾリンの直接的合成2011
- Author(s)
  時水勇輔、大野浩章、他3名
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] エポキシドの位置選択的開環反応を用いたリゼルグ酸の不斉全合成2011
- Author(s)
  岩田顕、大野浩章、他3名
- Organizer
  第61回日本薬学会近畿支部総会・大会
- Place of Presentation
  神戸薬科大学(兵庫県)
- Year and Date
  2011-10-23
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたアニリン誘導体の連続型分子内ヒドロアミノ化-ヒドロアリール化反応による高度縮環型カルバゾール誘導体の合成2011
- Author(s)
  稲葉祐介、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒による三成分環形成反応を用いた多置換ジヒドロピラゾールの効率的合成法の開発2011
- Author(s)
  鈴木大和，大石真也，藤井信孝，大野浩章
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール（徳島県）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒によるアルキンのヒドロアリール化を用いた多連続環化反応の開発2011
- Author(s)
  大野浩章、他4名
- Organizer
  第41回複素環化学討論会
- Place of Presentation
  熊本市民会館(熊本県)
- Year and Date
  2011-10-20
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究2011
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 縮環インドール構造を有する新規Eg5阻害剤の開発2011
- Author(s)
  竹内智起、大石真也、渡部敏明、大野浩章、浅田直也、北浦和夫、澤田潤一、浅井章良、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会第6回年会
- Place of Presentation
  東京工業大学大岡山キャンパス（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] エポキシドの位置選択的開環反応を用いたリゼルグ酸の不斉全合成2011
- Author(s)
  岩田顕、大野浩章, 他
- Organizer
  第61回日本薬学会近畿支部総会・大会
- Place of Presentation
  神戸薬科大学(兵庫県)
- Year and Date
  2011-10-23
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Jaspine Bおよびその誘導体の立体分岐合成と構造活性相関研究2011
- Author(s)
  吉光佑二、大野浩章、他4名
- Organizer
  第9回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール(東京都)
- Year and Date
  2011-05-28
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] (+)-リゼルグ酸の不斉全合成研究2011
- Author(s)
  岩田顕、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-29
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Gold-catalyzed three-component annulation : an efficient synthesis of 1,2,3,5-tetrasubstituted dihydropyrazoles from alkynes, aldehydes, and hydrazines2011
- Author(s)
  Suzuki, Y., Ohno, H., et al
- Organizer
  242nd American Chemical Society National Meeting & Exposition
- Place of Presentation
  Denver (USA)
- Year and Date
  2011-08-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたアニリン誘導体の連続型分子内ヒドロアミノ化-ヒドロアリール化反応による高度縮環型カルバゾール誘導体の合成2011
- Author(s)
  稲葉祐介、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Total Synthesis of (+)-Lysergic Acid by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group2011
- Author(s)
  Ohno, H., et al
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Jaspine Bおよびその誘導体の立体分岐合成と構造活性相関研究2011
- Author(s)
  吉光佑二、大石真也、宮垣　潤、井貫晋輔、藤井信孝、大野浩章
- Organizer
  第7回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] DEVELOPMENT AND APPLICATION OF FLUORESCENT PROBES FOR MONITORING CXCR4 RECEPTOR INTERNALIZATION2011
- Author(s)
  Oishi S, Masuda R, Tanahara N, Ohno H, Yano Y, Matsuzaki K, Hirasawa A, Tsujimoto G, Fujii N.
- Organizer
  Nature Chemical Biology Symposium 2011: Cancer Chemical Biology
- Place of Presentation
  Boston（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いたヒドロアリール化反応を基盤とする連続環化反応の開発2011
- Author(s)
  直江紗織、大野浩章、他5名
- Organizer
  第28回有機合成化学セミナー
- Place of Presentation
  滝の湯(山形県)
- Year and Date
  2011-09-01
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] (+)-リゼルグ酸の不斉全合成研究2011
- Author(s)
  岩田顕、大野浩章、他3名
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡県)
- Year and Date
  2011-03-29
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Total Synthesis of(+)-Lysergic Acid by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group2011
- Author(s)
  H. Ohno, 他4名
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Gold-catalyzed three-component annulation : an efficient synthesis of 1,2,3,5-tetrasubstituted dihydropyrazoles from alkynes, aldehydes, and hydrazines2011
- Author(s)
  Suzuki, Y., Ohno, H., et al
- Organizer
  242nd American Chemical Society National Meeting & Exposition
- Place of Presentation
  Denver (USA)
- Year and Date
  2011-08-31
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒を用いたアルキンに対する分子間求核付加-環化反応によるナフタレン誘導体の合成2011
- Author(s)
  直江紗織、大野浩章、他5名
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール(徳島県)
- Year and Date
  2011-11-08
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Synthetic Study of Quinocarcin2011
- Author(s)
  H. Chiba, H. Ohno, 他2名
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル(東京都)
- Year and Date
  2011-11-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] (+)-リゼルグ酸の不斉全合成研究2011
- Author(s)
  岩田顕、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡)
- Year and Date
  2011-03-29
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Synthesis and Application of Fluorescent SDF-1 Derivatives2011
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Development of a Novel Class of ATP-competitive Kinesin Spindle Protein Inhibitors2011
- Author(s)
  Oishi S, Takeuchi T, Watanabe T, Ohno H, Sawada J, Matsuno M, Asai A, Asada N, Kitaura K, Fujii N.
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル（東京都）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 銅触媒を用いたオルト無置換ベンズアミジンのアルキニル化-環化によるキナゾリンの直接的合成2011
- Author(s)
  時水勇輔、大野浩章, 他
- Organizer
  日本薬学会第131年会
- Place of Presentation
  ツインメッセ静岡(静岡)
- Year and Date
  2011-03-31
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] パラジウム触媒によるブロモアレンとプロパルギル化合物の連続環化反応を利用したJaspine Bの全合成とその応用2010
- Author(s)
  井貫晋輔、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(名古屋)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 触媒的連続結合形成反応による複素環骨格構築法の開発研究2010
- Author(s)
  大野浩章
- Organizer
  京都大学グローバルCOEプログラム有機若手ワークショップ
- Place of Presentation
  京都大学,(京都府)
- Year and Date
  2010-09-15
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 遷移金属触媒を用いたSonogashiraカップリング-環化反応を鍵反応としたQuinocarcinの合成研究2010
- Author(s)
  千葉浩亮、大野浩章、他2名
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いたオルト無置換ベンズアミジンのアルキニル化-環化によるキナゾリンの直接的合成2010
- Author(s)
  時水勇輔、大野浩章, 他
- Organizer
  第27回有機合成化学セミナー
- Place of Presentation
  シーサイドホテル舞子ビラ神戸(兵庫県)
- Year and Date
  2010-09-23
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒によるジインおよびトリイン誘導体の連続環化反応を用いた縮環型インドール誘導体の合成2010
- Author(s)
  平野公夫、大野浩章、他3名
- Organizer
  第98回有機合成シンポジウム
- Place of Presentation
  早稲田大学国際会議場(東京都)
- Year and Date
  2010-11-06
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] アザインドール骨格を有する新規CK2阻害剤テンプレートの開発研究2010
- Author(s)
  侯増〓、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(名古屋)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いたオルト無置換ベンズアミジンのアルキニル化-環化によるキナゾリンの直接的合成2010
- Author(s)
  時水勇輔、大野浩章, 他
- Organizer
  第27回有機合成化学セミナー
- Place of Presentation
  シーサイドホテル舞子ビラ神戸(神戸)
- Year and Date
  2010-09-23
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒を用いたアニリン誘導体の分子内連続環化反応による芳香環縮環型カルバゾール誘導体の合成2010
- Author(s)
  稲葉祐介、大野浩章、他
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-28
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 金触媒による分子内連続環化反応を用いた高度縮環型カルバゾールの合成法の開発2010
- Author(s)
  稲葉祐介、大野浩章、他3名
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪府)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 触媒的連続結合形成反応による複素環骨格構築法の開発研究2010
- Author(s)
  大野浩章
- Organizer
  京都大学グローバルCOEプログラム有機若手ワークショップ
- Place of Presentation
  京都大学(京都府)(招待講演)
- Year and Date
  2010-09-15
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒によるジインおよびトリイン誘導体の連続環化反応を用いた縮環型インドール誘導体の合成2010
- Author(s)
  平野公夫、大野浩章, 他
- Organizer
  第98回有機合成シンポジウム
- Place of Presentation
  早稲田大学国際会議場(東京)
- Year and Date
  2010-11-06
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Jaspine Bおよびその誘導体の立体選択的合成研究2010
- Author(s)
  吉光佑二、大野浩章, 他
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-28
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 連続的多成分カップリング-環化反応によるピロロインドール及びジピロロピリジン誘導体の効率的合成法の開発2010
- Author(s)
  鈴木大和、大野浩章、他6名
- Organizer
  第29回メディシナルケミストリーシンポジウム
- Place of Presentation
  京都テルサ(京都府)
- Year and Date
  2010-11-18
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 触媒的連続結合形成反応による複素環骨格構築法の開発研究2010
- Author(s)
  大野浩章
- Organizer
  京都大学グローバルCOEプログラム有機若手ワークショップ
- Place of Presentation
  京都大学(京都)(招待講演)
- Year and Date
  2010-09-15
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] アザインドール骨格を有する新規CK2阻害剤テンプレートの開発研究2010
- Author(s)
  侯増華、大野浩章、他6名
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates2010
- Author(s)
  Inuki, S., Ohno, H., et al
- Organizer
  The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Place of Presentation
  大阪大学(大阪府)
- Year and Date
  2010-05-20
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] アザインドール骨格を有する新規CK2阻害剤テンプレートの開発研究2010
- Author(s)
  侯増〓、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] パラジウム触媒とイソシアネートを用いたエチニルアジリジンの環拡大-連続的環化反応による連結型複素環の構築2010
- Author(s)
  岡野晃典、大野浩章, 他
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-28
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 遷移金属触媒を用いたSonogashiraカップリングー環化反応を鍵反応としたQuinocarcinの合成研究2010
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(名古屋)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒による分子内連続環化反応を用いた高度縮環型カルバゾールの合成法の開発2010
- Author(s)
  稲葉祐介、大野浩章, 他
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いた四成分カップリング反応によるイソキノリン縮環型三環性複素環の一挙構築2010
- Author(s)
  久保田悠史、大野浩章、他5名
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪府)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine(Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates2010
- Author(s)
  S. Inuki, H. Ohno, 他3名
- Organizer
  The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Place of Presentation
  大阪大学(大阪府)
- Year and Date
  2010-05-20
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いた四成分カップリング反応によるイソキノリン縮環型三環性複素環の一挙構築2010
- Author(s)
  久保田悠史、大野浩章, 他
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪府)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 金触媒によるジインおよびトリイン誘導体の連続環化反応を用いた縮環型インドール誘導体の合成2010
- Author(s)
  平野公夫、大野浩章, 他
- Organizer
  第98回有機合成シンポジウム
- Place of Presentation
  早稲田大学国際会議場(東京都)
- Year and Date
  2010-11-06
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 銅触媒を用いたオルト無置換ベンズ0名アミジンのアルキニル化-環化によるキナゾリンの直接的合成2010
- Author(s)
  時水勇輔、大野浩章、他3名
- Organizer
  第27回有機合成化学セミナー
- Place of Presentation
  シーサイドホテル舞子ビラ神戸(兵庫県)
- Year and Date
  2010-09-23
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 銅触媒を用いた四成分カップリング反応によるイソキノリン縮環型三環性複素環の一挙構築2010
- Author(s)
  久保田悠史、大野浩章, 他
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 連続的多成分カップリング-環化反応によるピロロインドール及びジピロロピリジン誘導体の効率的合成法の開発2010
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  第29回メディシナルケミストリーシンポジウム
- Place of Presentation
  京都テルサ(京都府)
- Year and Date
  2010-11-18
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 連続的多成分カップリング-環化反応によるピロロインドール及びジピロロピリジン誘導体の効率的合成法の開発2010
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  第29回メディシナルケミストリーシンポジウム
- Place of Presentation
  京都テルサ(京都)
- Year and Date
  2010-11-18
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 遷移金属触媒を用いたSonogashiraカップリング-環化反応を鍵反応としたQuinocarcinの合成研究2010
- Author(s)
  千葉浩亮、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] Ring-Construction/Stereoselective Functionalization Cascade : Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates2010
- Author(s)
  Inuki, S., Ohno H., et al.
- Organizer
  The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Place of Presentation
  大阪大学(大阪)
- Year and Date
  2010-05-20
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] 金触媒による分子内連続環化反応を用いた高度縮環型カルバゾールの合成法の開発2010
- Author(s)
  稲葉祐介、大野浩章, 他
- Organizer
  第60回日本薬学会近畿支部総会
- Place of Presentation
  摂南大学(大阪府)
- Year and Date
  2010-10-30
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] パラジウム触媒によるブロモアレンとプロパルギル化合物の連続環化反応を利用したJaspine Bの全合成とその応用2010
- Author(s)
  井貫晋輔、大野浩章, 他
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PUBLICLY-22106521
[Presentation] 縮環インドール構造を有する新規Eg5阻害剤の開発2010
- Author(s)
  竹内智起、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-29
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] パラジウム触媒によるブロモアレンとプロパルギル化合物の連続環化反応を利用したJaspine Bの全合成とその応用2010
- Author(s)
  井貫晋輔、大野浩章、他3名
- Organizer
  第36回反応と合成の進歩シンポジウム
- Place of Presentation
  愛知県労働産業センター(愛知県)
- Year and Date
  2010-11-02
- Data Source
  KAKENHI-PROJECT-22590005
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  東京
- Year and Date
  2009-08-03
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Pd-Catalyzed Carbonylation of Amino Acid-Derived Allylic Carbonates2009
- Author(s)
  Inokuchi E, Oishi S, Ohno H, Fujii N, et al.
- Organizer
  8th Australian Peptide Conference
- Place of Presentation
  Queensland Australia
- Year and Date
  2009-10-12
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 固相上におけるペプチド鎖へのDTPAの新規標識法の開発2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] カルバゾール骨格を有する新規Eg5阻害剤のデザインと合成2009
- Author(s)
  渡部敏明、大野浩章, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-19
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] カルバゾール骨格を有する新規Eg5阻害剤のデザインと合成2009
- Author(s)
  渡部敏明、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-19
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Jaspine Bおよびその誘導体の立体選択的合成2009
- Author(s)
  吉光佑二、大野浩章, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した新規化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ピラジンを母核とするCK2阻害剤の構造活性相関研究2009
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2009-05-19
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 銅触媒によるテトラヒドロピリミジンを配位性置換基とした酸化的分子間オルトC-H官能基化反応2009
- Author(s)
  水原司、大野浩章, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 有機銅-亜鉛複合試薬を用いたトリフルオロメチルアルケンジペプチドイソスターの新規合成法の開発2009
- Author(s)
  小林数也、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第35回反応と合成の進歩シンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-16
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 銅触媒を用いた連続三成分結合形成反応による2-(アミノメチル)インドール骨格およびインドール縮環型多環式骨格構築法の開発2009
- Author(s)
  太田悠介、大野浩章, 他
- Organizer
  日本薬学会第129年会
- Place of Presentation
  京都
- Year and Date
  2009-03-27
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-18
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した新規化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] パラジウム触媒とイソシアネートを用いたエチニルアジリジンの環拡大-連続的環化反応による連結型複素環の構築2009
- Author(s)
  岡野晃典、大野浩章, 他
- Organizer
  第29回有機合成若手セミナー
- Place of Presentation
  神戸
- Year and Date
  2009-11-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第6回GPCR研究会
- Place of Presentation
  東京
- Year and Date
  2009-05-08
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  東京
- Year and Date
  2009-08-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 銅触媒による多成分カップリング反応を用いたワンポット含窒素多環式複素環骨格構築法の開発2009
- Author(s)
  太田悠介、大野浩章、他
- Organizer
  第35回反応と合成の進歩シンポジウム
- Place of Presentation
  金沢
- Year and Date
  2009-11-16
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第6回GPCR研究会
- Place of Presentation
  東京
- Year and Date
  2009-05-08
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 多成分カップリング・連続環化反応によるピロロインドール誘導体及びジピロロピリジン誘導体の合成研究2009
- Author(s)
  鈴木大和、大野浩章、他
- Organizer
  第7回次世代を担う有機化学シンポジウム
- Place of Presentation
  大阪
- Year and Date
  2009-07-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 銅触媒によるテトラヒドロピリミジンを配位性置換基とした酸化的分子間オルトC-H官能基化反応2009
- Author(s)
  水原司、大野浩章, 他
- Organizer
  第35回反応と合成の進歩シンポジウム
- Place of Presentation
  金沢
- Year and Date
  2009-11-17
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 銅触媒による多成分カップリング反応を用いた多環式インドールのワンポット構築法の開発2009
- Author(s)
  太田悠介、大野浩章, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたsp3 C-H活性化によるインドリンの合成2009
- Author(s)
  渡部敏明、大野浩章, 他
- Organizer
  日本薬学会第129年会
- Place of Presentation
  京都
- Year and Date
  2009-03-28
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Synthesis and Application of Novel Fluorescent-Labeled CXCR4 Antagonists2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第10回文部科学省特定領域研究「がん」5領域若手研究者ワークショップ
- Place of Presentation
  蓼科
- Year and Date
  2009-09-02
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 固相上におけるペプチド鎖へのDTPAの新規標識法の開発2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-18
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Synthesis and Application of Novel Fluorescent-Labeled CXCR4 Antagonists2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第10回文部科学省特定領域研究「がん」5領域若手研究者ワークショップ
- Place of Presentation
  蓼科
- Year and Date
  2009-09-02
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 縮環インドール構造を有する新規Eg5阻害剤の開発2009
- Author(s)
  竹内智起、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大野浩章, 他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 銅触媒-マイクロ波照射を用いた連続三成分カップリング-環化-N-アリール化反応によるインドール縮環型1,4-ジアゼピン合成法開発2008
- Author(s)
  太田悠介、大野浩章、他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-04
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたアレン連続環化反応を利用したErgot Alkaloid 骨格の一挙構築法開発と応用2008
- Author(s)
  井貫晋輔、大野浩章、他
- Organizer
  第6回次世代を担う有機化学シンポジウム
- Place of Presentation
  東京
- Year and Date
  2008-05-30
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 触媒的連続結合形成反応の開発とErgotアルカロイド全合成への応用2008
- Author(s)
  大野浩章
- Organizer
  第43回天然物化学討論会
- Place of Presentation
  大阪
- Year and Date
  2008-07-10
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Pd触媒によるアレン連続環化反応を利用したErgotAlkaloid骨格の一挙構築法開発と応用2008
- Author(s)
  井貫晋輔、大野浩章、他
- Organizer
  第6回次世代を担う有機化学シンポジウム
- Place of Presentation
  東京
- Year and Date
  2008-05-30
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたアレン連続環化反応を利用したErgot Alkaloid骨格の一挙構築法開発と応用2008
- Author(s)
  井貫晋輔、大野浩章, 他
- Organizer
  第6回次世代を担う有機化学シンポジウム
- Place of Presentation
  東京
- Year and Date
  2008-05-30
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 新規三環性ヘテロ芳香環構築反応の開発とキナーゼ阻害剤テンプレートへの応用2008
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  日本薬学会第129年会
- Place of Presentation
  京都
- Year and Date
  2008-03-27
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 連続三成分カップリングー環化-N-アリール化反応による銅触媒一マイクロ波照射を用いたインドール縮環型1, 4-ジアゼピン合成法の開発2008
- Author(s)
  太田悠介、大野浩章, 他
- Organizer
  第28回有機合成若手セミナー
- Place of Presentation
  大阪
- Year and Date
  2008-11-12
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたプロモエンアレンの連続的閉環反応による多環式複素環の一挙構築2008
- Author(s)
  岡野晃典、大野浩章, 他
- Organizer
  第28回有機合成若手セミナー
- Place of Presentation
  大阪
- Year and Date
  2008-11-12
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Pd触媒によるアレン連続環化反応を利用したErgotAlkaloid骨格の一挙構築法開発と応用2008
- Author(s)
  井貫晋輔、大野浩章、他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-24
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Pd触媒によるアレン連続環化反応を利用したErgot Alkaloid骨格の一挙構築法開発と応用2008
- Author(s)
  井貫晋輔、大野浩章, 他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-04
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] キナーゼ阻害剤テンプレートを指向した三環性芳香環構築反応の開発2008
- Author(s)
  鈴木大和、大野浩章, 他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたプロモエンアレンの連続環化反応による多環式複素環の一挙構築2008
- Author(s)
  岡野晃典、大野浩章, 他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-05
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 銅触媒-マイクロ波照射を用いた連続三成分カップリング-環化-N-アリール化反応によるインドール縮環型1.4-ジアゼピン合成法2008
- Author(s)
  太田悠介、大野浩章, 他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-14
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Construction of 2-(aminomethyl)indole motif by Cu-catalyzed multicomponent reaction2007
- Author(s)
  Yusuke Ohta, Hiroaki Ohno, et al.
- Organizer
  234th ACS meeting & exposition
- Place of Presentation
  ボストン
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 連続結合形成反応による縮環型芳香族化合物の一挙合成法の開発2007
- Author(s)
  大野浩章
- Organizer
  第33回反応と合成の進歩シンポジウム
- Place of Presentation
  長崎
- Year and Date
  2007-11-06
- Data Source
  KAKENHI-PROJECT-18015027
[Presentation] Construction of 2-(aminomethyl)indole motif by Cu-catalyzed multi-component reaction2007
- Author(s)
  Yusuke Ohta, Hiroaki Ohno, et al.
- Organizer
  14th IUPAC Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
- Place of Presentation
  奈良
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Pd触媒を用いたタンデム型N-アリール化-C-H 活性化によるカルバゾールの合成と反応機構の考察2007
- Author(s)
  渡部敏明、大野浩章、他
- Organizer
  第5回次世代を担う有機化学シンポジウム
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Synthesis and application of carbazoles by palladium-catalyzed tandem N-arylation of carbazoles by palladium-catalyzed tandem N-arylation and oxidative C-H activation2007
- Author(s)
  Toshiaki Watanabe, Hiroaki Ohno, et al.
- Organizer
  14th IUPAC Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
- Place of Presentation
  奈良
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] パラジウム触媒を用いたプロパルギルブロミドの連続的閉環反応による二環性複素環の一挙構築2007
- Author(s)
  岡野晃典、大野浩章、他
- Organizer
  第33回反応と合成の進歩シンポジウム
- Place of Presentation
  長崎
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] 連続結合形成反応による縮環型芳香族化合物の一挙合成法の開発2007
- Author(s)
  大野浩章、他
- Organizer
  第33回反応と合成の進歩シンポジウム
- Place of Presentation
  長崎
- Year and Date
  2007-11-06
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Synthesis and application of carbazoles by palladium-catalyzed tandem N-arylation and oxidative C-H activation2007
- Author(s)
  Toshiaki Watanabe, Hiroaki Ohno, et al.
- Organizer
  Eighth Tetrahedron Symposium
- Place of Presentation
  ベルリン
- Data Source
  KAKENHI-PROJECT-19689001
[Presentation] Direct Construction of Fused Indoles by Gold-Catalyzed Cascade Cyclization of Conjugated Diynes
- Author(s)
  Saori Naoe, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno
- Organizer
  第８回集積有機合成国際シンポジウム（ISIS-8）
- Place of Presentation
  東大寺総合文化センター (奈良県奈良市）
- Year and Date
  2013-09-23 – 2013-09-26
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 光アフィニティープローブを利用したキスペプチン類の受容体結合残基の同定
- Author(s)
  三須良介、大石真也、説田章平、野口太朗、金田雅仁、大野浩章、藤井信孝
- Organizer
  第8回ケミカルバイオロジー学会年会
- Place of Presentation
  東京医科歯科大学　（東京都文京区）
- Year and Date
  2013-06-19 – 2013-06-21
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] NK3受容体アゴニストの生体内安定性評価と新規誘導体の創製
- Author(s)
  三須良介、大石真也、山田愛、山本昂輝、野口太朗、大野浩章、山村崇、岡村裕昭、松田二子、大蔵聡、藤井信孝
- Organizer
  第11回GPCR研究会
- Place of Presentation
  日本科学未来館　みらいCANホール　（東京都江東区）
- Year and Date
  2014-05-09 – 2014-05-10
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 化合物アレイを用いた新規mdm2/mdmx-p53阻害剤の探索法の開発とその応用
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第31回メディシナルケミストリーシンポジウム
- Place of Presentation
  アステールプラザ（広島県広島市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒を用いた共役ジインの三連続環化反応による縮環カルバゾールの合成
- Author(s)
  田口将光、大野浩章、他
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸学院大学等（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Structure-activity Relationship Study of Tachykinin Peptides for Development of Novel Neurokinin-3 Receptor Selective Agonists
- Author(s)
  Ryosuke Misu, Shinya Oishi, Taro Noguchi, Ai Yamada, Hiroaki Ohno, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  23rd American Peptide Symposium
- Place of Presentation
  ヒルトンワイコロアホテル　（米国ハワイ州ワイコロワ）
- Year and Date
  2013-06-22 – 2013-06-27
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] キネシンモータータンパク質KSP阻害剤の創製研究-連続縮環型分子の変換による溶解性改善-
- Author(s)
  竹内智起、大石真也、金田雅仁、大野浩章、澤田潤一、浅井章良、藤井信孝
- Organizer
  第11回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール (東京都渋谷区）
- Year and Date
  2013-05-24 – 2013-05-25
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた共役ジインとピロールの分子間 [4 + 2] 型反応によるインドール骨格の構築
- Author(s)
  松田優佳、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  第40回反応と合成の進歩シンポジウム
- Place of Presentation
  東北大学川内萩ホール　（宮城県仙台市）
- Year and Date
  2014-11-10 – 2014-11-11
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒によるアジドイナミドの連続環化反応を用いたインドロキノリン骨格の一挙構築
- Author(s)
  時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第40回反応と合成の進歩シンポジウム
- Place of Presentation
  東北大学川内萩ホール　（宮城県仙台市）
- Year and Date
  2014-11-10 – 2014-11-11
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、岩田顕、大槻和裕、丸山透、大石真也、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学（大阪府豊中市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒を用いた三成分環化反応によるジヒドロピラゾールの合成とCK2阻害剤開発への応用
- Author(s)
  大野浩章、鈴木大和、侯増燁、呉竜英、仲西功、平澤明、大石真也、藤井信孝
- Organizer
  第43回複素環化学討論会
- Place of Presentation
  長良川国際会議場　（岐阜県岐阜市）
- Year and Date
  2013-10-17 – 2013-10-19
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Formal [4 + 2] Reaction between 1,3-Diynes and Pyrroles: Gold(I)-Catalyzed Indole Synthesis via Double Hydroarylation
- Author(s)
  Y. Matsuda, and H. Ohno, et al.
- Organizer
  ISIS-9
- Place of Presentation
  淡路夢舞台国際会議場（兵庫県淡路市）
- Year and Date
  2014-11-14 – 2014-11-15
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] パラジウム触媒による連続環化反応を用いた四環性スピロインドール類の合成
- Author(s)
  岩田　顕、井貫晋輔、大石真也、藤井信孝、大野浩章
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部百年講堂　（福岡県福岡市）
- Year and Date
  2013-11-05 – 2013-11-07
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Gold-Catalyzed Annulations and Their Medicinal Applications
- Author(s)
  Hiroaki Ohno
- Organizer
  DPhG Annual Meeting 2014
- Place of Presentation
  ゲーテ大学（ドイツ、フランクフルト）
- Year and Date
  2014-09-23 – 2014-09-26
- Invited
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 鉄(II)イオン配位性ペプチドの設計と機能評価
- Author(s)
  小林由佳、大石真也、大野浩章、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  デザイン・クリエイティブセンター神戸　（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 化合物アレイを用いた新規mdm2/mdmx-p53阻害剤の探索法の開発とその応用
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第63回日本薬学会近畿支部大会
- Place of Presentation
  同志社女子大学（京都府京田辺市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] パラジウム触媒を用いた中員環形成反応によるLaurencia族環状エーテルの構築：Laurendecumallene Bの合成研究
- Author(s)
  大野浩章、吉光佑二、井貫晋輔、大石真也、藤井信孝
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部百年講堂　（福岡県福岡市）
- Year and Date
  2013-11-05 – 2013-11-07
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Structure-activity Relationship Study of Tachykinin Peptides for Evaluation of Biological Stability of Neurokinin-3 Receptor Agonists for the Development of Novel Biostable Analogs
- Author(s)
  Ryosuke Misu, Shinya Oishi, Taro Noguchi, Ai Yamada, Hiroaki Ohno, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク　（大阪府吹田市）
- Year and Date
  2013-11-06 – 2013-11-08
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Identification of Novel CXCR7 Selective Ligands with Cyclic Pentapeptide Scaffold
- Author(s)
  Tomoko Kuroyanagi, Shinya Oishi, Tatsuhiko Kubo, Yuka Kobayashi, Ryosuke Misu, Hiroaki Ohno, Nicolas Montpas, Nikolaus Heveker, Yasushi Yoshikawa, Toshio Furuya, Nobutaka Fujii
- Organizer
  第51回ペプチド討論会
- Place of Presentation
  徳島大学　（徳島県徳島市）
- Year and Date
  2014-10-22 – 2014-10-24
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 環状ペンタペプチド骨格を有する新規CXCR7選択的リガンドの創製
- Author(s)
  黒柳友子、大石真也、久保達彦、小林由佳、三須良介、大野浩章、Montpas Nicolas、Heveker Nikolaus、吉川寧、古谷利夫、藤井信孝
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸国際会議場　（兵庫県神戸市）
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、大野浩章、他
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学（大阪府豊中市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 新規CXCR7選択的リガンドの創製：CXCR4拮抗剤からの受容体選択性の変換
- Author(s)
  黒柳友子、大石真也、久保達彦、小林由佳、三須良介、大野浩章、Montpas Nicolas、Heveker Nikolaus、吉川寧、古谷利夫、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  兵庫医療大学　（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] クロスメタセシス反応を利用したスフインゴシンキナーゼ阻害剤の創製研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、大槻和裕、丸山透、中村真也、仲西功、大石真也、大野浩章、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  兵庫医療大学　（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、岩田顕、大槻和裕、丸山透、中村真也、仲西功、大石真也、大野浩章、藤井信孝
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸国際会議場（兵庫県神戸市）
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒を用いた共役ジインの三連続反応による縮環カルバゾールの合成
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸学院大学　（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] OPTIMIZATION OF NEUROKININ-3 RECEPTOR (NK3R) SELECTIVE AGONISTS
- Author(s)
  Koki Yamamoto, Shinya Oishi, Ryosuke Misu, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Nobutaka Fujii
- Organizer
  第51回ペプチド討論会
- Place of Presentation
  徳島大学　（徳島県徳島市）
- Year and Date
  2014-10-22 – 2014-10-24
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 新規フェニルピラゾール誘導体の抗HIV活性に関する構造活性相関研究
- Author(s)
  岡崎志穂、水原司、加藤貴之、平井敦、栗原秀樹、嶋田泰宏、谷口雅彦、前田英樹、戸上博昭、志村和也、松岡雅雄、竹内智起、大野浩章、大石真也、藤井信孝
- Organizer
  第31回メディシナルケミストリーシンポジウム
- Place of Presentation
  アステールプラザ　（広島県広島市）
- Year and Date
  2013-11-20 – 2013-11-22
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 新規ニューロキニン-3受容体アゴニストの創製研究
- Author(s)
  山本昂輝、大石真也、三須良介、野口太朗、大野浩章、山村崇、岡村裕昭、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学　（大阪府吹田市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた共役ジインとピロールの分子間 [4 + 2] 型反応によるインドール骨格の構築
- Author(s)
  松田優佳、大野浩章、他
- Organizer
  第40回反応と合成の進歩シンポジウム
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2014-11-10 – 2014-11-11
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] クロスメタセシス反応を利用したスフィンゴシンキナーゼ阻害剤の創製研究
- Author(s)
  本田真歩、大野浩章、他
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸学院大学等（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Kinesin spindle protein (KSP) inhibitors with carbazole and diaryl amine scaffolds
- Author(s)
  Tomoki Takeuchi, Shinya Oishi, Masato Kaneda, Hiroaki Ohno, Jun-ichi Sawada, Akira Asai, Nobutaka Fujii
- Organizer
  246th American Chemical Society National Meeting and Exposition
- Place of Presentation
  Indiana convention center　（米国インディアナ州インディアナポリス）
- Year and Date
  2013-09-08 – 2013-09-12
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第62回日本薬学会近畿支部大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] ピリミドベンゾチアジン誘導体の新規合成法の開発と抗HIV剤を指向した構造活性相関研究
- Author(s)
  水原司、大石真也、大野浩章、志村和也、松岡雅雄、藤井信孝
- Organizer
  第62回日本薬学会近畿支部大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Identification of Novel MDM2/MDMX-p53 interaction inhibitors by chemical array technology
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Synthetic Study of (-)-Aspidophylline A
- Author(s)
  A. Ohara, and H. Ohno, et al.
- Organizer
  ISIS-9
- Place of Presentation
  淡路夢舞台国際会議場（兵庫県淡路市）
- Year and Date
  2014-11-14 – 2014-11-15
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、岩田顕、大槻和裕、丸山透、大石真也、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学　（大阪府吹田市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Development of Carbazole- and Diaryl Amine-type Kinesin Spindle Protein (KSP) Inhibitors
- Author(s)
  Tomoki Takeuchi, Shinya Oishi, Masato Kaneda, Hiroaki Ohno, Tatsuhide Kure, Shinya Nakamura, Isao Nakanishi, Jun-ichi Sawada, Akira Asai, Nobutaka Fujii
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館　（京都府京都市）
- Year and Date
  2013-10-07 – 2013-10-09
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Gold-Catalyzed Cascade Cyclization of (Azido)ynamides: an Efficient Strategy for the Construction of Indoloquinolines
- Author(s)
  Y. Tokimizu, and H. Ohno, et al.
- Organizer
  8th Asian-European Symposium on Metal-Mediated Efficient Organic Synthesis
- Place of Presentation
  Ilica Hotel（トルコ、チェシメ）
- Year and Date
  2014-09-07 – 2014-09-10
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Synthesis of the fused tetracyclic spiroindoles via palladium-catalyzed cascade reaction
- Author(s)
  Akira Iwata, Shinsuke Inuki Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  246th American Chemical Society National Meeting and Exposition
- Place of Presentation
  Indiana convention center　（米国インディアナ州インディアナポリス）
- Year and Date
  2013-09-08 – 2013-09-12
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、大野浩章、他
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸国際会議場
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] 金触媒によるアジドイナミドの連続環化反応を用いたインドロキノリン骨格の一挙構築
- Author(s)
  時水勇輔、大野浩章、他
- Organizer
  第12回次世代を担う有機化学シンポジウム
- Place of Presentation
  日本薬学会長井記念ホール（東京都渋谷区）
- Year and Date
  2014-05-23 – 2014-05-24
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Development of novel neurokinin-3 receptor selective agonists with resistance against proteolytic degradation
- Author(s)
  Ryosuke Misu, Shinya Oishi, Ai Yamada, Koki Yamamoto, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  第51回ペプチド討論会
- Place of Presentation
  徳島大学　（徳島県徳島市）
- Year and Date
  2014-10-22 – 2014-10-24
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 新規抗HIV剤を指向したベンゾイソチアゾロピリミジン誘導体の構造活性相関研究
- Author(s)
  岡崎志穂、水原司、志村和也、村山大人、松岡雅雄、大野浩章、大石真也、藤井信孝
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸国際会議場　（兵庫県神戸市）
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒を用いた共役ジインとピロールの分子間 [4 + 2] 型反応による4,7-二置換インドール骨格の構築
- Author(s)
  松田優佳、大野浩章、他
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸学院大学等（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] ペプチダーゼ耐性を有する新規NK3受容体アゴニストの創製研究
- Author(s)
  三須良介、大石真也、山田愛、山本昂輝、野口太朗、大野浩章、山村崇、岡村裕昭、松田二子、大蔵聡、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学　（大阪府吹田市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 金触媒によるアジドイナミドの連続環化反応を用いたインドロキノリン骨格の一挙構築
- Author(s)
  時水勇輔、大野浩章、他
- Organizer
  第40回反応と合成の進歩シンポジウム
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2014-11-10 – 2014-11-11
- Data Source
  KAKENHI-PROJECT-24689001
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第62回日本薬学会近畿支部大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 連続縮環型分子の修飾によるKSP阻害剤の溶解性改善
- Author(s)
  竹内智起、大石真也、金田雅仁、大野浩章、中村真也、仲西功、山根正敏、澤田潤一、浅井章良、藤井信孝
- Organizer
  第31回メディシナルケミストリーシンポジウム
- Place of Presentation
  アステールプラザ　（広島県広島市）
- Year and Date
  2013-11-20 – 2013-11-22
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Development of Photoaffinity Probes for Characterization of the Receptor Binding Residues in Kisspeptins
- Author(s)
  Shinya Oishi, Shohei Setsuda, Ryosuke Misua Taro Noguchi, Masato Kaneda, Hiroaki Ohno, Barry Evans, Jean-Marc Navenot, Stephen C. Peiper, Nobutaka Fujii
- Organizer
  23rd American Peptide Symposium
- Place of Presentation
  ヒルトンワイコロアホテル　（米国ハワイ州ワイコロワ）
- Year and Date
  2013-06-22 – 2013-06-27
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] 天然物の鏡像体化合物群の活用を目指した新規スクリーニング法の開発
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  デザイン・クリエイティブセンター神戸（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] クロスメタセシス反応を利用したスフインゴシンキナーゼ阻害剤の創製研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、大槻和裕、丸山透、中村真也、仲西功、大石真也、大野浩章、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  兵庫医療大学（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 金触媒を用いたベンゾフランによる分子内ヒドロアリール化反応の検討
- Author(s)
  坂井由葵、大石真也、藤井信孝、大野浩章
- Organizer
  第39回反応と合成の進歩シンポジウム
- Place of Presentation
  九州大学医学部百年講堂　（福岡県福岡市）
- Year and Date
  2013-11-05 – 2013-11-07
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Synthesis of IB-01212 by Site-Selective N-Methylation of Peptide Bonds
- Author(s)
  Ryota Nabika, Shinya Oishi, Ryosuke Misu, Hiroaki Ohno and Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク　（大阪府吹田市）
- Year and Date
  2013-11-06 – 2013-11-08
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] Synthetic Studies on Coibamide A
- Author(s)
  Ryota Nabika, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  The First Asian Conference for ''MONODUKURI'' Strategy by Synthetic Organic Chemistry
- Place of Presentation
  Southern Beach Hotel & Resort Okinawa（沖縄県糸満市）
- Year and Date
  2013-07-17 – 2013-07-19
- Data Source
  KAKENHI-PROJECT-23390025
[Presentation] C-H官能基化反応、及び芳香族求核置換反応によるピリミド［1,2-c］ベンゾチアジン-6-イミンとその誘導体の効率的合成法の開発
- Author(s)
  Mizuhara T, Oishi S, Fujii N, Ohno H.
- Organizer
  第31回有機合成若手セミナー「明日の有機合成を担う人のために」
- Place of Presentation
  京都大学（京都府）
- Data Source
  KAKENHI-PROJECT-23390025

1. FUJII Nobutaka (60109014)

# of Collaborated Projects: 9 results

# of Collaborated Products: 194 results
2. OISHI Shinya (80381739)

# of Collaborated Projects: 8 results

# of Collaborated Products: 125 results
3. TANAKA Tetsuaki (40116059)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
4. MAEZAKI Naoyoshi (00229296)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
5. 井貫晋輔 (70736272)

# of Collaborated Projects: 2 results

# of Collaborated Products: 36 results
6. KITAURA Kazuo (30132723)

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
7. NAKANISHI Isao (10362576)

# of Collaborated Projects: 1 results

# of Collaborated Products: 3 results
8. Saito Tamio (40260228)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
9. Kondo Yasumitsu (80333342)

# of Collaborated Projects: 1 results

# of Collaborated Products: 15 results
10. Kashiwada Yoshiki (30169429)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
11. 野田岳志 (00422410)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
12. 松本篤幸 (00753906)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
13. 有地法人 (60904935)

# of Collaborated Projects: 1 results

# of Collaborated Products: 10 results
14. UCHIYAMA Masanobu

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
15. 斉藤臣雄

# of Collaborated Projects: 0 results

# of Collaborated Products: 10 results
16. 王超

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
17. 宮本洋一

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
18. 和泉自泰

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
19. 山崎晶

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
20. 秋葉宏樹

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
21. 澤田潤一

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

Ohno Hiroaki 大野 浩章

OHNO Hiroaki 大野 浩章

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Natural product syntheses based on cascade cyclization and their applications to middle-molecule drug modalitiesPrincipal Investigator

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Synthesis of Novel Bowl-Shaped Highly pi-Conjugated Molecules Based on the Original Vinylcation FormationPrincipal Investigator

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Alkaloid Synthesis and Its Middle Molecular Strategy Based on Reaction IntegrationPrincipal Investigator

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Synthetic and medicinal studies on bioactive indole alkaloids based on direct construction of polycyclic ring systemsPrincipal Investigator

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Precise activation based on transition state control using neighboring effect and its medicinal applicationPrincipal Investigator

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原子移動型反応の高度集積化による多環式芳香族化合物の合成と創薬展開Principal Investigator

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Innovative Molecular Transformations Based on Consecutive pai-Activation and Their Medicinal ApplicationsPrincipal Investigator

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触媒的多成分反応・高原子効率反応の高度集積化と創薬展開Principal Investigator

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Divergent syntheses of biologically active compounds based on catalytic cascade cyclization reactionsPrincipal Investigator

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Ohno Hiroaki 大野浩章

OHNO Hiroaki 大野浩章