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Ishida Ryosuke  石田 良典

ORCIDConnect your ORCID iD *help
Researcher Number 10937684
Other IDs
Affiliation (Current) 2025: 名古屋市立大学, 医薬学総合研究院(薬学), 助教
2025: 東京科学大学, 総合研究院, 助教
Affiliation (based on the past Project Information) *help 2022 – 2023: 東京医科歯科大学, 生体材料工学研究所, 助教
Review Section/Research Field
Principal Investigator
Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
Except Principal Investigator
Basic Section 47040:Pharmacology-related / Medium-sized Section 47:Pharmaceutical sciences and related fields
Keywords
Principal Investigator
チャネル開閉ダイナミズム / 筋疾患 / カルシウムチャネル / リアノジン受容体制御剤 / 構造活性相関 / 筋細胞異常 / リアノジン受容体
Except Principal Investigator
神経変性疾患 / ライブセルイメージング / Gタンパク質共役型受容体 … More / シグナル伝達 / シナプス / 超複合体 / 膜タンパク質 / GPCR / タンパク質ータンパク質相互作用阻害剤 / ファオルダマー / 大環状化合物 / らせん分子 / 環状構造 / らせん構造 / フォルダマー / 芳香族アミド / 創薬 / 心筋 / 機能抑制型変異 / カルシウム / 抗不整脈薬 / 不整脈 / 2型リアノジン受容体 Less
  • Research Projects

    (4 results)
  • Research Products

    (12 results)
  • Co-Researchers

    (10 People)
  •  New molecular shapes from strained aromatic foldamer macrocycles and their application to development of PPI inhibitors

    • Principal Investigator
      棚谷 綾
    • Project Period (FY)
      2023 – 2026
    • Research Category
      Fund for the Promotion of Joint International Research (International Collaborative Research)
    • Review Section
      Medium-sized Section 47:Pharmaceutical sciences and related fields
    • Research Institution
      Ochanomizu University
  •  Manipulation of membrane protein supercomplexes to elucidate their molecular dynamics and function

    • Principal Investigator
      上窪 裕二
    • Project Period (FY)
      2023 – 2025
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Review Section
      Basic Section 47040:Pharmacology-related
    • Research Institution
      Juntendo University
  •  Development of RyR2-specific inhibitors and activators and their application as antiarrhythmic agents

    • Principal Investigator
      呉林 なごみ
    • Project Period (FY)
      2022 – 2024
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Review Section
      Basic Section 47040:Pharmacology-related
    • Research Institution
      Juntendo University
  •  Development of chemical toolbox for RyR regulator and analysis of the dynamism of RyR open/close mechanismPrincipal Investigator

    • Principal Investigator
      Ishida Ryosuke
    • Project Period (FY)
      2022 – 2023
    • Research Category
      Grant-in-Aid for Early-Career Scientists
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
    • Research Institution
      Tokyo Medical and Dental University

All 2024 2023 2022

All Journal Article Presentation

  • [Journal Article] Discovery and Structure–Activity Relationship of a Ryanodine Receptor 2 Inhibitor2024

    • Author(s)
      Ryosuke Ishida, Xi Zeng, Nagomi Kurebayashi, Takashi Murayama, Shuichi Mori, Hiroyuki Kagechika
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 72 Issue: 4 Pages: 399-407

    • DOI

      10.1248/cpb.c24-00114

    • ISSN
      0009-2363, 1347-5223
    • Year and Date
      2024-04-22
    • Language
      English
    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K15244
  • [Journal Article] Screening for Novel Type 2 Ryanodine Receptor Inhibitors by Endoplasmic Reticulum Ca<sup>2+</sup>Monitoring2023

    • Author(s)
      Takenaka Mai、Kodama Masami、Murayama Takashi、Ishigami-Yuasa Mari、Mori Shuichi、Ishida Ryosuke、Suzuki Junji、Kanemaru Kazunori、Sugihara Masami、Iino Masamitsu、Miura Aya、Nishio Hajime、Morimoto Sachio、Kagechika Hiroyuki、Sakurai Takashi、Kurebayashi Nagomi
    • Journal Title

      Molecular Pharmacology

      Volume: 104 Issue: 6 Pages: 275-286

    • DOI

      10.1124/molpharm.123.000720

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K06652
  • [Journal Article] Drug development for the treatment of RyR1-related skeletal muscle diseases2023

    • Author(s)
      Takashi Murayama, Nagomi Kurebayashi, Ryosuke Ishida, Hiroyuki Kagechika
    • Journal Title

      Current Opinion in Pharmacology

      Volume: 69 Pages: 102356-102356

    • DOI

      10.1016/j.coph.2023.102356

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-22K15244, KAKENHI-PROJECT-22K06652
  • [Journal Article] A potent and selective cis-amide inhibitor of ryanodine receptor 2 as a candidate for cardiac arrhythmia treatment2023

    • Author(s)
      Ishida Ryosuke、Kurebayashi Nagomi、Iinuma Hiroto、Zeng Xi、Mori Shuichi、Kodama Masami、Murayama Takashi、Masuno Hiroyuki、Takeda Fumi、Kawahata Masatoshi、Tanatani Aya、Miura Aya、Nishio Hajime、Sakurai Takashi、Kagechika Hiroyuki
    • Journal Title

      European Journal of Medicinal Chemistry

      Volume: 262 Pages: 115910-115910

    • DOI

      10.1016/j.ejmech.2023.115910

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K06652, KAKENHI-PROJECT-22K15244
  • [Journal Article] A reconstituted depolarization-induced Ca2+ release platform for validation of skeletal muscle disease mutations and drug discovery2022

    • Author(s)
      Murayama Takashi、Kurebayashi Nagomi、Numaga-Tomita Takuro、Kobayashi Takuya、Okazaki Satoru、Yamashiro Kyosuke、Nakada Tsutomu、Mori Shuichi、Ishida Ryosuke、Kagechika Hiroyuki、Yamada Mitsuhiko、Sakurai Takashi
    • Journal Title

      Journal of General Physiology

      Volume: 154 Issue: 12

    • DOI

      10.1085/jgp.202213230

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K06652, KAKENHI-PROJECT-22K06828, KAKENHI-PROJECT-19K07105, KAKENHI-PROJECT-19H03404, KAKENHI-PROJECT-23K24067
  • [Journal Article] Mice with R2509C-RYR1 mutation exhibit dysfunctional Ca2+ dynamics in primary skeletal myocytes2022

    • Author(s)
      Tsuboi Yoshitaka、Oyama Kotaro、Kobirumaki-Shimozawa Fuyu、Murayama Takashi、Kurebayashi Nagomi、Tachibana Toshiaki、Manome Yoshinobu、Kikuchi Emi、Noguchi Satoru、Inoue Takayoshi、Inoue Yukiko U.、Nishino Ichizo、Mori Shuichi、Ishida Ryosuke、Kagechika Hiroyuki、Suzuki Madoka、Fukuda Norio、Yamazawa Toshiko
    • Journal Title

      Journal of General Physiology

      Volume: 154 Issue: 11

    • DOI

      10.1085/jgp.202213136

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-21K06789, KAKENHI-PROJECT-22K06652, KAKENHI-PROJECT-21K19929, KAKENHI-PLANNED-22H05053, KAKENHI-PLANNED-22H05054, KAKENHI-PLANNED-22H05055, KAKENHI-PROJECT-20H03421, KAKENHI-PROJECT-19K07105, KAKENHI-PROJECT-19K07306, KAKENHI-PROJECT-20K06467, KAKENHI-PROJECT-19H03404, KAKENHI-PROJECT-23K24778, KAKENHI-PROJECT-23K24067
  • [Journal Article] Development of a water-soluble ryanodine receptor 1 inhibitor2022

    • Author(s)
      Ishida Ryosuke、Mori Shuichi、Murayama Takashi、Nakamichi Ayaka、Chai Xikun、Kurebayashi Nagomi、Iinuma Hiroto、Kagechika Hiroyuki
    • Journal Title

      Bioorganic &amp; Medicinal Chemistry

      Volume: 74 Pages: 117027-117027

    • DOI

      10.1016/j.bmc.2022.117027

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K06652, KAKENHI-PROJECT-22K15244, KAKENHI-PROJECT-19K07105, KAKENHI-PROJECT-19H03404, KAKENHI-PROJECT-23K24067
  • [Presentation] A potent and selective cis-amide inhibitor of ryanodine receptor 2 as a candidate for cardiac arrhythmia treatment2024

    • Author(s)
      Xi Zeng, Ryosuke Ishida, Nagomi Kurebayashi, Hiroto Iinuma, Masami Kodama, Takashi Murayama, Hiroyuki Kagechika
    • Organizer
      24th Tetrahedron Symposium
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-22K15244
  • [Presentation] 不整脈治療への展開を指向した新規2型リアノジン受容体選択的阻害剤の開発2023

    • Author(s)
      石田良典、曾 希、森 修一、呉林なごみ、児玉 昌美、飯沼大翔、村山 尚、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第17回年会
    • Data Source
      KAKENHI-PROJECT-22K15244
  • [Presentation] 海馬スライス培養を用いたアミロイドプラーク形成と神経突起変性の経時的解析2023

    • Author(s)
      周藝瑶, 上窪裕二, 石田葉子, 日置寛之, 櫻井隆
    • Organizer
      第46回日本神経科学大会
    • Data Source
      KAKENHI-PROJECT-23K06170
  • [Presentation] 水溶性向上を意図した RyR1 阻害剤の構造展開 および結合位置特定のためのプローブ化2022

    • Author(s)
      石田良典、森 修一、飯沼大翔、柴 喜坤、村山 尚、呉林なごみ、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会 第16回年会
    • Data Source
      KAKENHI-PROJECT-22K15244
  • [Presentation] 不整脈を引き起こす変異型RyR2新規阻害剤の開発2022

    • Author(s)
      曾 希、石田良典、呉林なごみ、村山 尚、 山本優雅、森 修一、影近弘之
    • Organizer
      第66回日本薬学会関東支部大会
    • Data Source
      KAKENHI-PROJECT-22K15244
  • 1.  呉林 なごみ (50133335)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 2.  小川 治夫 (40292726)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 3.  杉原 匡美 (80648163)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 1 results
  • 4.  棚谷 綾 (40361654)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 5.  影近 弘之 (20177348)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 6.  大金 賢司 (30771092)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 7.  桑原 拓也 (60768654)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 8.  上窪 裕二 (80509670)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 1 results
  • 9.  国広 なごみ
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 4 results
  • 10.  小比類巻 生
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results

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