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TAKEUCHI Yoshio  竹内 義雄

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Researcher Number 20111750
Other IDs
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Affiliation (based on the past Project Information) *help 2007: University of Toyama, 大学院・医学薬学研究部, 教授
2006: 富山大学, 大学院医学薬学研究部, 教授
2005: 富山大学, 薬学部, 教授
2004: 富山医科薬科大学, 薬学部, 教授
2001: 富山医薬大, 薬学部, 教授 … More
1996 – 2000: Toyama. Med. Pharm Univ. Fac. Pharm. Sci. Professor, 薬学部, 教授
1990 – 1995: 富山医科薬科大学, 薬学部, 助教授
1990: 富山医科薬科大学, 薬, 助教授
1986 – 1988: Associate Professor, 薬学部, 助教授 Less
Review Section/Research Field
Principal Investigator
Chemical pharmacy / 医薬分子機能学 / Drug development chemistry
Except Principal Investigator
Chemical pharmacy
Keywords
Principal Investigator
不斉フッ素化 / キラル誘導化試薬 / フッ化過クロリル / CFPA / DAST / 光学活性 / 多重官能性炭素化合物 / フッ素 / チロシン / トリプトファン … More / 求電子的フッ素化 / MTPA / NMR / CFTA / Isostere / イソスター / 含フッ素ペプチド / Electrophilic Fluorination / フッ素ガス / フッ素化試薬 / Molecular Design / alpha-Fluoro-alpha-amino Acid / Tertiary Alkyl Fluorides / Multifunctional Carbon Compounds / 分子設計 / α-フルオロ-α-アミノ酸 / バルビツール酸 / ジエノン / ピロロ[2,3-b]インドール / インドレニン / 安定型等価体 / 副互変異性 / サリドマイド / シュードローグ / 副互変異性体 / 光学活性体 / ^<19>F-NMR / Secondary Alkyl Fluorides / Selective Desulfonylation / Selective Denitration / Fluorinated Building Blocks / α-フルオローα-ニトロカルボン酸エステル / α-フルオロ-α-スルホニルホスホン酸エステル / α-フルオロ-α-ベンゼンスルホニルカルボン酸エステル / ビルディングブロック / 三級アルキルフルオライド / 二級アルキルフルオライド / 選択的脱エステル化 / 選択的脱ニトロ化 / 含フッ素合成素子 / chiral / fluorinating agents / asymmetric / fluorine / ケトン / 不斉・合成 / アントラサイクリン / 生物活性物質 / フッ素化剤 / 液晶 / 医薬品 / フッ素化反応剤 / フルオロケトン / 不斉 / optical resolution / multifunctional carbon / chiral fluoro compound / absolute configuration / enantiomer excess / chiral derivatizing agent / sp配座 / キラル-2級アルコール / X線結晶解析 / ab initio 計算 / ^<19>F NMR / ^1H NMR / アミノ酸 / キラル一級アミン / 絶対構造 / 光学分割 / 多重官能性炭素 / 不斉フッ素化合物 / 絶対配置 / 光学純度 / Lipase / Chiral Derivating Agent / Fluorination / Fluorine-containing Peptide / Fluoro-amino Acid / リパーゼ / フッ素化 / フルオロアミノ酸 / X-ray analysis / perchloryl fluoride / fluorine gas / N-fluorosulfonamide / alpha-phenethylamine / Benzothiazolidine / Enantioselective Fluorination / ベンズイソチアゾリジン / 2-フルオロ-2-メチル-1-テトラロン / X線解析 / N-フルオロスルホンアミド / α-フェネチルアミン / ベンズチアゾリジン / Five-membered Sultam / Fluoroindanone / Fluorotetralone / Asymmetric Fluorination / Fluorine-containing Peptides / N-Fluoroproline / TRH類縁体 / タイソスター / 2-(1-フルオロエテニル)ピロリジン / α-フルオロアミノ酸 / 6員環スルタム / 5員環スルタム / フルオロインダノン / フルオロテトラロン / α-フルオロプロリン / Fluorinating Reagent / New Medicinal / Stereoselectivity / Saccharin / alpha-Amino Acid / Asymmetric Fluorinaton / Heterocyclic Compound / 面選択性 / 不斉合成 / 新型医薬品 / 立体選択性 / サッカリン / α-アミノ酸 / 複素環 / Monofluoro compounds / Multifunctional carbon compounds / Optically active / DELTAdelta Values / _<19>F NMR / Reagents for ee determination / 立体的因子 / 化学シフト差 / 化学シフト差(△δ値) / 一フッ化物 / 化学シフト基(△δ値) / ^<19>FーNMR / 光学純度決定試薬 / NMAD Receptor / Fluorine-containing Medicinals / Fluorinated Tropanes / Monofluoro Building Blocks / 1,3双極付加 / トロパン / フルオロエテン / モノフルオロ化合物 / ブロモフルオロアルカン / バートン法 / 合成ブロック / NMAD受容体 / 含フッ素医薬品 / 含フッ素トロパン / 三級フッ化物 / モノフルオロ合成ブロック / セロトニン受容体作動薬 / Selectfluor / トリプタン系片頭痛治療薬 / 酵素阻害 / 安定型相似体 / 環状トリプトファン / セレクトフルオール / ジヒドロキシカルコン / フルオロエピネフリン / フルオロオキシインドール / 医薬品設計 / イミダゾール / ノルエピネフリン / フルオロジエノン型 / インドレニン型 / ジアステレオマ- / 不斉補助基 / カルボキシル化 / π-π相互作用 / 不斉空間 … More
Except Principal Investigator
Asymmetric Cycloaddition / Asymmetric Diels-Alder Reaction / <alpha> , <beta> -Unsaturated Sulfoxides / 高ジアステレオ選択性 / 不斉環化付加 / 不斉ディールス・アルダー反応 / α,β-不飽和スルホキシド Less
  • Research Projects

    (16 results)
  • Research Products

    (6 results)
  • Co-Researchers

    (12 People)
  •  副互変異性構造に基づく生物活性発現の機構解明と創薬化学への応用Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      2006 – 2007
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      University of Toyama
  •  副互変異性構造に起因する生物活性発現と創薬化学への新展開Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      2004 – 2005
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      University of Toyama
      Toyama Medical and Pharmaceutical University
  •  生体内における副互変異性体介在仮説の実証研究Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      2000 – 2001
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      医薬分子機能学
    • Research Institution
      Toyama Medical and Pharmaceutical University
  •  医薬品設計のための新概念と新戦略:次世紀の生命科学を指向した生体有機フッ素化学Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      1999 – 2001
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      Toyama Medical and Pharmaceutical University
  •  Efficient preparation of a highly versatile chiral derivatizing agent, CFTA, for determination of absolute configurations.Principal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1998 – 2000
    • Research Category
      Grant-in-Aid for Scientific Research (B).
    • Research Field
      Chemical pharmacy
    • Research Institution
      TOYAMA MEDICAL AND PHARMACEUTICAL UNIVERSITY
  •  Design & Synthesis of Novel Enantioselctive Fluorinationg AgentsPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1998 – 2000
    • Research Category
      Grant-in-Aid for Scientific Research (B).
    • Research Field
      Chemical pharmacy
    • Research Institution
      TOYAMA MEDICAL AND PHARMACEUTICAL UNIVERSITY
  •  Novel Fluorinated Bioorganic Molecules for the 21st CenturyPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1997 – 1998
    • Research Category
      Grant-in-Aid for international Scientific Research
    • Research Field
      医薬分子機能学
    • Research Institution
      TOYAMA MEDICAL AND PHARMACEUTICAL UNIVERSITY
  •  Synthesis and Utilization of Fluorine-containing Chiral Building Blocks for Development of the New Type of DrugsPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1995 – 1997
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      TOYAMA MEDICAL AND PHARMACEUTICAL UNIVERSITY
  •  Development of Electrophilic and Enantioselective Fluorinating Agents based on Fine Chemisty DesignPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1995 – 1996
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Grant-in-Aid for Scientific Research (C) (2)
  •  CFPA類縁体の不斉合成と絶対構造決定試薬としての応用Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      1994
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      Toyama Medical and Pharmaceutical University
  •  芳香環π-π相互作用による不斉空間の構築と光学活性CFPA合成への応用Principal Investigator

    • Principal Investigator
      竹内 義雄
    • Project Period (FY)
      1993
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      Toyama Medical and Pharmaceutical University
  •  Development of the Reagents for Electrophilic Fluorination Directing for New Type of MedicinalsPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1993 – 1994
    • Research Category
      Grant-in-Aid for General Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      TOYAMA MEDICAL AND PHARMACEUTICAL UNIVERSITY
  •  Synthesis of Monofluoro Building Blocks Designed from Fine Chemistry Viewpoint and Development of Fluorine-containing MedicinalsPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1990 – 1992
    • Research Category
      Grant-in-Aid for Developmental Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Toyama Medical & Pharmaceutical University
  •  Development of A New Reagent for Ee Determination with High Resolution Based on the Fine Chemistry DesigningPrincipal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1990 – 1991
    • Research Category
      Grant-in-Aid for General Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Toyama Medical & Pharmaceutical University
  •  Synthesis and Application of Versatile Monofluoro Building Blocks by Manipulation of the Multifunctional Carbon Compounds.Principal Investigator

    • Principal Investigator
      TAKEUCHI Yoshio
    • Project Period (FY)
      1987 – 1988
    • Research Category
      Grant-in-Aid for General Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Toyama Medical & Pharmaceutical University
  •  Studies on A Novel Asymmetric Cycloaddition Using Optically Active <alpha> , <beta> -Unsaturated Sulfoxides

    • Principal Investigator
      KOIZUMI Toru
    • Project Period (FY)
      1984 – 1986
    • Research Category
      Grant-in-Aid for General Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Toyama Medical & Pharmaceutical University

All 2007 2005

All Journal Article Presentation

  • [Journal Article] Biological Evaluation of 2-Aryl-2-Fluoropropionic Acids as Possible Platforms for New Medicinal Agents2005

    • Author(s)
      Takeuchi, Y, Fujisawa, H., Fujiwara, T., Matsuura, M., Komatsu, H., Ueno, S., Matsuzaki, T.
    • Journal Title

      Chemical & Pharmaceutical Bulletin 53・8

      Pages: 1062-1064

    • NAID

      10016656314

    • Data Source
      KAKENHI-PROJECT-16659027
  • [Journal Article] Synthesis and Optical Resolution of 2-Aryl-2-fluoropropionic Acids, Fluorinated Analogues of Non-steroidal Anti-inflammatory Drugs (NSAIDs)2005

    • Author(s)
      Fujisawa, H., Fujiwara, T., Takeuchi, Y., Omata, K.
    • Journal Title

      Chemical & Pharmaceutical Bulletin 53・5

      Pages: 524-528

    • NAID

      10016653678

    • Data Source
      KAKENHI-PROJECT-16659027
  • [Presentation] トリプトファンの安定型副互変異性等価体の合成研究2007

    • Author(s)
      尹 斌(竹内 義雄)
    • Organizer
      シンポジウム「モレキュラー・キラリティー2007」
    • Place of Presentation
      東京
    • Year and Date
      2007-05-15
    • Data Source
      KAKENHI-PROJECT-18659026
  • [Presentation] キラル含フッ素インドール誘導体の設計と合成2007

    • Author(s)
      関 孝行(竹内 義雄)
    • Organizer
      平成19年度有機合成化学北陸セミナー
    • Place of Presentation
      金沢
    • Year and Date
      2007-10-13
    • Data Source
      KAKENHI-PROJECT-18659026
  • [Presentation] Synthetic studies on fluorine-containing pseudologs corresponding to minor tautomers of tryptophan2007

    • Author(s)
      Yin, Bin (Takeuchi, Yoshio)
    • Organizer
      15th European Symposium on Fluorine Chemistry
    • Place of Presentation
      Prague,Czech Republic
    • Year and Date
      2007-07-17
    • Data Source
      KAKENHI-PROJECT-18659026
  • [Presentation] フェノール/ジエノン互変異性現象におけるジエノン対応等価体の合成研究2007

    • Author(s)
      岡田 励(竹内 義雄)
    • Organizer
      日本薬学会北陸支部第117回例会
    • Place of Presentation
      金沢
    • Year and Date
      2007-11-11
    • Data Source
      KAKENHI-PROJECT-18659026
  • 1.  TAKAHASHI Tamiko (10115181)
    # of Collaborated Projects: 8 results
    # of Collaborated Products: 0 results
  • 2.  SHIBATA Norio (40293302)
    # of Collaborated Projects: 5 results
    # of Collaborated Products: 0 results
  • 3.  SATOH Toshio (70075943)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 4.  KIRIHARA Masayuki (40262539)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 5.  ARAI Yoshitsugu (10115157)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 6.  KOIZUMI Toru (40012611)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 7.  KOMETANI Tadashi (60042842)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 8.  藤原 朋也 (70361962)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 2 results
  • 9.  HIRAI Yoshiro (70111747)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 10.  KABUTO Kuninobu (40005799)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 11.  TAKAYAMA Hiromitsu (90171561)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 12.  TACHIBANA Shinro
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results

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