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Fukuda Hayato  福田 隼

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… Alternative Names

FUKUDA Hayato  福田 隼

福田 隼  フクダ ハヤト

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Researcher Number 30434450
Other IDs
Affiliation (Current) 2022: 長崎大学, 医歯薬学総合研究科(薬学系), 准教授
Affiliation (based on the past Project Information) *help 2017 – 2020: 長崎大学, 医歯薬学総合研究科(薬学系), 准教授
2016: 北海道大学, 薬学研究院, 助教
2015: 北海道大学, 大学院薬学研究院, 助教
2013 – 2015: 北海道大学, 薬学研究科(研究院), 助教
2012: 北海道大学, 大学院・薬学研究院, 助教
2009: 東北大学, 大学院・薬学研究科, 助手
Review Section/Research Field
Principal Investigator
Drug development chemistry / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
Except Principal Investigator
Drug development chemistry / Chemical pharmacy
Keywords
Principal Investigator
レゾルビン / 安定等価体 / 不飽和脂肪酸 / シクロプロパン / 構造活性相関 / 全合成 / レゾルビンE2 / 標的タンパク質 / 炎症収束 / 抗炎症活性 … More / 標的タンパク / 炎症 / 創薬 / 天然物合成 / 脂質メディエーター / エイコサペンタエン酸 / デオキシレゾルビン / レゾルビン類 / 分子プローブ / レゾルビンE3 / レゾルビンT4 / 構造決定 / 細菌感染症 / レゾルビンT … More
Except Principal Investigator
ニトロキシルラジカル / アザアダマンタン / シクロプロパン / 酸化ストレス / ラジカル消去 / アダマンタン / レドックス / オキソアンモニウム / 脳保護薬 / 有機触媒 / 酸化反応 / オキソアンモニウム塩 / ニトロキシド / 不斉反応 / 不斉酸化 / アルコール酸化 / 不斉触媒 / 分子認識 / 配座制御 / 三次元的多様性 / 分子設計 / BGT-1 阻害剤 / プロテアソーム阻害剤 / BASE阻害剤 / ホスファチジルセリン / ファゴサイトーシス / 二量等価体 / クアトロフェニル / 三次元多様性 / レゾルビン / ヌクレオシド / ペプチドミメティクス / ライブラリー / ペプチドミイメティクス / レジデンスタイム / リン脂質 / トルテロジン / ムスカリン受容体 Less
  • Research Projects

    (10 results)
  • Research Products

    (93 results)
  • Co-Researchers

    (36 People)
  •  新規脂肪酸代謝物レゾルビンTシリーズの構造決定と安定等価体の創製Principal Investigator

    • Principal Investigator
      福田 隼
    • Project Period (FY)
      2020 – 2022
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
    • Research Institution
      Nagasaki University
  •  Development of a tool for analyzing the mechanism of action of resolvins based on the molecular structure of unsaturated fatty acidsPrincipal Investigator

    • Principal Investigator
      FUKUDA Hayato
    • Project Period (FY)
      2017 – 2019
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Drug development chemistry
    • Research Institution
      Nagasaki University
  •  A Versatile Strategy for Developing Long-Acting Ligands by Ligand-Phospholipid Conjugation

    • Principal Investigator
      SHUTO Satoshi
    • Project Period (FY)
      2016 – 2017
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Search for target proteins utilizing the stable equivalents of resorvins, pro-resolving lipid mediatorsPrincipal Investigator

    • Principal Investigator
      FUKUDA Hayato
    • Project Period (FY)
      2015 – 2016
    • Research Category
      Grant-in-Aid for Young Scientists (B)
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Medicinal chemistry studies based on the three-dimensional structural diversity-oriented molecular design of pharmacologically active compounds

    • Principal Investigator
      Shuto Satoshi
    • Project Period (FY)
      2015 – 2019
    • Research Category
      Grant-in-Aid for Scientific Research (A)
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Design and synthesis of phosphatidylserine dimers with antitumor effect via the phagocytosis-inducing property

    • Principal Investigator
      SHUTO satoshi
    • Project Period (FY)
      2013 – 2014
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Discovery of a stable equivalent of resolvins with potent anti-inflammatory actionPrincipal Investigator

    • Principal Investigator
      FUKUDA HAYATO
    • Project Period (FY)
      2013 – 2014
    • Research Category
      Grant-in-Aid for Young Scientists (B)
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Medicinal chemical study by the three-dimensional structural diversity-oriented strategy based on the characteristic steric and stereoelectronic features of cyclopropane

    • Principal Investigator
      SHUTO Satoshi
    • Project Period (FY)
      2012 – 2014
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Drug development chemistry
    • Research Institution
      Hokkaido University
  •  Development of oxoammonium-salt-type catalysts for highly enantioselective oxidation of alcohols

    • Principal Investigator
      IWABUCHI Yoshiharu
    • Project Period (FY)
      2009 – 2011
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Tohoku University
  •  有機ニトロキシルラジカルをモチーフとする酸化ストレス防御活性薬剤の創製

    • Principal Investigator
      IWABUCHI Yoshiharu
    • Project Period (FY)
      2008 – 2009
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Tohoku University

All 2021 2020 2019 2018 2017 2016 2015 2014 2013 Other

All Journal Article Presentation

  • [Journal Article] Synthesis of Resolvin E1 and Its Conformationally Restricted Cyclopropane Congeners with Potent Anti-Inflammatory Effect2021

    • Author(s)
      Ishimura Kohei、Fukuda Hayato、Fujiwara Koichi、Muromoto Ryuta、Hirashima Koki、Murakami Yuto、Watanabe Mizuki、Ishihara Jun、Matsuda Tadashi、Shuto Satoshi
    • Journal Title

      ACS Medicinal Chemistry Letters

      Volume: 12 Pages: 256-261

    • DOI

      10.1021/acsmedchemlett.0c00639

    • NAID

      120007186305

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06965, KAKENHI-PROJECT-20K06941
  • [Journal Article] Formal Synthesis of (?)-Haliclonin A: Stereoselective Construction of an Azabicyclo[3.3.1]nonane Ring System by a Tandem Radical Reaction2020

    • Author(s)
      Komine Keita、Urayama Yasuhiro、Hosaka Taku、Yamashita Yuki、Fukuda Hayato、Hatakeyama Susumi、Ishihara Jun
    • Journal Title

      Organic Letters

      Volume: 22 Pages: 5046-5050

    • DOI

      10.1021/acs.orglett.0c01627

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20K06941, KAKENHI-PROJECT-18K05126, KAKENHI-PROJECT-19K15568
  • [Journal Article] Concise Synthesis of TPCA-1 and Related Thiophene-carboxamides by Cross Coupling2020

    • Author(s)
      Ishihara Jun、Kawasaki Norihiko、Fukuda Hayato
    • Journal Title

      HETEROCYCLES

      Volume: 101 Pages: 707-707

    • DOI

      10.3987/com-19-s(f)43

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-18K05126
  • [Journal Article] Design and Synthesis of Benzene Congeners of Resolvin E2, a Proresolving Lipid Mediator, as Its Stable Equivalents2020

    • Author(s)
      Y. Murakami, H. Fukuda, R. Muromoto, K. Hirashima, K. Ishimura, K. Fujiwara, J. Ishihara, T. Matsuda, M. Watanabe, S. Shuto,
    • Journal Title

      ACS Medicinal Chemistry Letters

      Volume: 11 Pages: 479-484

    • DOI

      10.1021/acsmedchemlett.9b00596

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19H01014, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-19K06965, KAKENHI-PROJECT-20K06941
  • [Journal Article] Catalytic Asymmetric Total Synthesis of Exiguolide2020

    • Author(s)
      Oka Kengo、Fuchi Shunsuke、Komine Keita、Fukuda Hayato、Hatakeyama Susumi、Ishihara Jun
    • Journal Title

      Chemistry- A European Journal

      Volume: 26 Pages: 12862-12867

    • DOI

      10.1002/chem.202001773

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20K06941, KAKENHI-PROJECT-18K05126, KAKENHI-PROJECT-19K15568
  • [Journal Article] Synthesis of Resolvin E3, a Proresolving Lipid Mediator, and Its Deoxy Derivatives: Identification of 18-Deoxy-resolvin E3 as a Potent Anti-Inflammatory Agent2020

    • Author(s)
      Fukuda Hayato、Ikeda Hiroyuki、Muromoto Ryuta、Hirashima Koki、Ishimura Kohei、Fujiwara Koichi、Aoki-Saito Haruka、Hisada Takeshi、Watanabe Mizuki、Ishihara Jun、Matsuda Tadashi、Shuto Satoshi
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 85 Pages: 14190-14200

    • DOI

      10.1021/acs.joc.0c01701

    • NAID

      120007168587

    • Peer Reviewed / Open Access / Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-18K08382, KAKENHI-PROJECT-18K08404, KAKENHI-PROJECT-19K06965, KAKENHI-PROJECT-20K06941, KAKENHI-PROJECT-19H03364
  • [Journal Article] Synthetic Studies on Marineosins Based on a Direct Coupling Reaction of Pyrrole and δ-Lactone2020

    • Author(s)
      Ishihara Jun、Hatakeyama Susumi、Yamamoto Kohei、Morii Yuki、Suga Akihisa、Komine Keita、Fukuda Hayato
    • Journal Title

      HETEROCYCLES

      Volume: 100 Pages: 46-46

    • DOI

      10.3987/com-19-14123

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K15568, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-18K05126
  • [Journal Article] New entry to the enantioselective formation of substituted cyclohexenes bearing an all‐carbon quaternary stereogenic center2020

    • Author(s)
      Komine Keita、Urayama Yasuhiro、Hosaka Taku、Fukuda Hayato、Hatakeyama Susumi、Ishihara Jun
    • Journal Title

      Chirality

      Volume: 32 Pages: 273-281

    • DOI

      10.1002/chir.23173

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K15568, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-18K05126
  • [Journal Article] Synthesis of Oxytocin Derivatives Lipidated via a Carbonate or Carbamate Linkage as a Long-Acting Therapeutic Agent for Social Impairment-Like Behaviors2019

    • Author(s)
      Cherepanov Stanislav M.、Miura Risako、Shabalova Anna A.、Ichinose Wataru、Yokoyama Shigeru、Fukuda Hayato、Watanabe Mizuki、Higashida Haruhiro、Shuto Satoshi
    • Journal Title

      Bioorg. Med. Chem

      Volume: 27 Pages: 3358-3363

    • DOI

      10.1016/j.bmc.2019.06.018

    • NAID

      120007126060

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06965, KAKENHI-PROJECT-19H01014, KAKENHI-PROJECT-17K08360
  • [Journal Article] Resolvin E3 attenuates allergic airway inflammation via the interleukin‐23‐interleukin‐17A pathway2019

    • Author(s)
      Sato M, Aoki-Saito H, Fukuda H, Ikeda H, Koga Y, Yatomi M, Tsurumaki H, Maeno T, Saito T, Nakakura T, Mori T, Yanagawa M, Abe M, Sako Y, Dobashi K, Ishizuka T, Yamada M, Shuto S, Hisada T.
    • Journal Title

      FASEB J

      Volume: Nov;33(11) Pages: 12750-12759

    • DOI

      10.1096/fj.201900283r

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-18K06677, KAKENHI-PROJECT-18K08382, KAKENHI-PROJECT-18K08404, KAKENHI-PROJECT-19K07257, KAKENHI-PROJECT-19H01014, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-16K18982, KAKENHI-PROJECT-19H05647
  • [Journal Article] Synthesis of 1,1,2-trisubstituted cyclopropane nucleosides in enantiomerically pure forms2019

    • Author(s)
      D. Fushihara, H. Fukuda, H. Abe, S. Shuto
    • Journal Title

      Nucleosides, Nucleotides & Nucleic Acids

      Volume: 38 Pages: 921-941

    • DOI

      10.1080/15257770.2019.1625380

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19H01014, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-16H05106
  • [Journal Article] Synthesis of Enantiomerically Pure 1,2,3-Trisubstituted Cyclopropane Nucleosides Using Pd-Catalyzed Substitution via Directing Group-Mediated C(sp3)- H Activation as a Key Step2019

    • Author(s)
      Minami Takaaki、Fukuda Kohtaro、Hoshiya Naoyuki、Fukuda Hayato、Watanabe Mizuki、Shuto Satoshi
    • Journal Title

      Org. Lett.

      Volume: 21 Pages: 656-659

    • DOI

      10.1021/acs.orglett.8b03785

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-17K15476, KAKENHI-PROJECT-19H01014, KAKENHI-PROJECT-16H05106
  • [Journal Article] Synthesis of chiral cis-cyclopropane bearing indole and chromone as potential TNF-α inhibitors2018

    • Author(s)
      Kanada Ryutaro、Tanabe Makoto、Muromoto Ryuta、Sato Yukina、Kuwahara Tomoki、Fukuda Hayato、Arisawa Mitsuhiro、Matsuda Tadashi、Watanabe Mizuki、Shuto Satoshi
    • Journal Title

      J. Org. Chem.

      Volume: 83 Pages: 7672-7682

    • DOI

      10.1021/acs.joc.8b00466

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-17K15476, KAKENHI-PROJECT-16H05106, KAKENHI-PROJECT-15KT0063, KAKENHI-PUBLICLY-18H04260, KAKENHI-PROJECT-26288051
  • [Journal Article] Resolvin E3 attenuates lipopolysaccharide-induced depression-like behavior in mice2018

    • Author(s)
      Deyama Satoshi、Shimoda Kento、Ikeda Hiroyuki、Fukuda Hayato、Shuto Satoshi、Minami Masabumi
    • Journal Title

      J. Pharmacol. Sci.

      Volume: 138 Pages: 86-88

    • DOI

      10.1016/j.jphs.2018.09.006

    • NAID

      120006540074

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-15H02495
  • [Journal Article] Design and synthesis of cyclopropane-based conformationally restricted GABA analogues as selective inhibitors for betaine/GABA transporter 12018

    • Author(s)
      Suemasa Akihiro、Watanabe Mizuki、Kobayashi Takaaki、Suzuki Hiroe、Fukuda Hayato、Minami Masabumi、Shuto Satoshi
    • Journal Title

      Bioorg. Med. Chem. Lett

      Volume: 28 Pages: 3395-3399

    • DOI

      10.1016/j.bmcl.2018.08.031

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-17K15476
  • [Journal Article] Resolvin E1, but not resolvins E2 and E3, promotes fMLF-induced ROS generation in human neutrophils2018

    • Author(s)
      Unno Yuka、Sato Yoshinori、Fukuda Hayato、Ishimura Kohei、Ikeda Hiroyuki、Watanabe Mizuki、Tansho-Nagakawa Shigeru、Ubagai Tsuneyuki、Shuto Satoshi、Ono Yasuo
    • Journal Title

      FEBS Lett

      Volume: 592 Pages: 2706-2715

    • DOI

      10.1002/1873-3468.13215

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K00883, KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-17K15476
  • [Journal Article] Design and Synthesis of Histamine H3/H4 Receptor Ligands with a Cyclopropane Scaffold. Bioorg2018

    • Author(s)
      Watanabe, T. Kobayashi, Y. Ito, H. Fukuda, S. Yamada, M. Arisawa, S. Shuto,
    • Journal Title

      Bioorg. Med. Chem. Lett

      Volume: 28 Pages: 3630-3633

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Journal Article] Resolvin E1/E2 ameliorate lipopolysaccharide-induced depression-like behaviors via ChemR23.2018

    • Author(s)
      K. Deyama, Y. Shimoda, K. Ishikawa, H. Ishimura, H. Fukuda, S. Ide, M. Satoh, S. Shuto
    • Journal Title

      Psychopharmacology (Berl)

      Volume: 235 Pages: 329-336

    • DOI

      10.1007/s00213-017-4774-7

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-15K06765, KAKENHI-PROJECT-15K08670
  • [Journal Article] Design and synthesis of histamine H3/H4 receptor ligands with a cyclopropane scaffold2018

    • Author(s)
      Watanabe Mizuki、Kobayashi Takaaki、Ito Yoshihiko、Fukuda Hayato、Yamada Shizuo、Arisawa Mitsuhiro、Shuto Satoshi
    • Journal Title

      Bioorganic & Medicinal Chemistry Letters

      Volume: 28 Pages: 3630-3633

    • DOI

      10.1016/j.bmcl.2018.10.041

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08360, KAKENHI-PROJECT-17K15476, KAKENHI-PROJECT-15KT0063, KAKENHI-PUBLICLY-18H04260, KAKENHI-PROJECT-26288051
  • [Journal Article] An Entry to Chiral 1,1,2,3-Tetrasubstituted Arylcyclopropanes by Pd(II)-Catalyzed Arylation via Directing Group-Mediated C(sp3)-H Activation2017

    • Author(s)
      Hoshiya Naoyuki、Kondo Moemi、Fukuda Hayato、Arisawa Mitsuhiro、Uenishi Jun’ichi、Shuto Satoshi
    • Journal Title

      J. Org. Chem

      Volume: 82 Pages: 2535-2544

    • DOI

      10.1021/acs.joc.6b02935

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PUBLICLY-16H01026, KAKENHI-PROJECT-15H02495
  • [Journal Article] Identification of a Potent and Selective GPR4 Antagonist as a Drug Lead for the Treatment of Myocardial Infarction2016

    • Author(s)
      Hayato Fukuda, Saki Ito, Kenji Watari, Chihiro Mogi, Mitsuhiro Arisawa, Fumikazu Okajima, Hitoshi Kurose, Satoshi Shuto
    • Journal Title

      ACS Medicinal Chemistry Letters

      Volume: 7 Pages: 493-497

    • DOI

      10.1021/acsmedchemlett.6b00014

    • Peer Reviewed / Acknowledgement Compliant / Open Access
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-13J03105, KAKENHI-PROJECT-26288051, KAKENHI-PUBLICLY-16H01026, KAKENHI-PROJECT-25253011, KAKENHI-PROJECT-15H04641, KAKENHI-PROJECT-16K15136
  • [Journal Article] Design, Synthesis, and Identification of 4”α-Azidoethyl-Cyclic ADP-Carbocyclic-Ribose as a Highly Potent Analogue of Cyclic ADP-Ribose, a Ca2+-mobilizing Second Messenger.2016

    • Author(s)
      Sato, T.; Watanabe, M.; Tsuzuki, T.; Takano, S.; Murayama, T.; Sakurai, T.; Kameda, T.; Arisawa, M.; Fukuda, H.; Shuto, S.
    • Journal Title

      J. Med. Chem.

      Volume: 59 Pages: 7282-7286

    • DOI

      10.1021/acs.jmedchem.6b00437

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PUBLICLY-16H01026, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-26288051, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-16K15136
  • [Journal Article] Design and synthesis of cyclopropane congeners of resolvin E2, an endogenous proresolving lipid mediator, as its stable equivalents.2016

    • Author(s)
      Fukuda, H; Muromoto, R.; Takakura, Y.; Ishimura, K.; Kanada, R.; Fushihara, D.; Tanabe, M.; Matsubara, K.; Hirao, T.; Hirashima, K.; Abe, Arisawa, M.; Matsuda, T.; Shuto, S.
    • Journal Title

      Organic Letters

      Volume: 18 Pages: 6224-6227

    • DOI

      10.1021/acs.orglett.6b02612

    • Peer Reviewed / Acknowledgement Compliant / Int'l Joint Research
    • Data Source
      KAKENHI-PUBLICLY-16H01026, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-26288051, KAKENHI-PROJECT-15K12751, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15K18898, KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-16K15136
  • [Journal Article] Safe Removal of the Allyl Protecting Groups of Allyl Esters using a Recyclable, Low-leaching and Ligand-free Palladium Nanoparticle Catalyst2015

    • Author(s)
      Koji Takagi, Hayato Fukuda, Satoshi Shuto, Akira Otaka, Mitsuhiro Arisawa
    • Journal Title

      Adv. Synth. Catal

      Volume: 357 Pages: 2119-2124

    • DOI

      10.1002/adsc.201500055

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-26288051
  • [Journal Article] Synthesis of 7-Deaza-cyclic Adenosine-5′-diphosphate-carbocyclic-ribose and Its 7-Bromo Derivative as Intracellular Ca2+-Mobilizing Agents2015

    • Author(s)
      Satoshi Takano, Takayoshi Tsuzuki, Takashi Murayama, Takashi Sakurai, Hayato Fukuda, Mitsuhiro Arisawa, Satoshi Shuto
    • Journal Title

      J. Org. Chem

      Volume: 80 Pages: 6619-6627

    • DOI

      10.1021/acs.joc.5b00723

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-26288051
  • [Journal Article] Construction of a chiral quaternary carbon center by a radical cyclization/ring-enlargement reaction: synthesis of 4α-azidoethyl carbocyclic ribose, a key unit for the synthesis of cyclic ADP- ribose derivatives of biological importance2015

    • Author(s)
      Takatoshi Sato, Takayoshi Tsuzuki, Satoshi Takano, Kohtaro Kato, Hayato Fukuda, Mitsuhiro Arisawa, Satoshi Shuto
    • Journal Title

      Tetrahedron

      Volume: 71 Pages: 5403-5413

    • DOI

      10.1016/j.tet.2015.05.084

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-26288051
  • [Journal Article] Characterization of imidazopyridine compounds as negative allosteric modulators of proton-sensing GPR4 in extracellular acidification-induced responses.2015

    • Author(s)
      Ayaka Tobo, Masayuki Tobo, Takashi Nakakura, Masashi Ebara, Hideaki Tomura, Chihiro Mogi, Dong-Soon Im, Naoya Murata, Atsushi Kuwabara, Saki Ito, Hayato Fukuda, Mitsuhiro Arisawa, Satoshi Shuto, Michio Nakaya, Hitoshi Kurose, Koichi Sato, Fumikazu Okajima
    • Journal Title

      PLoS ONE

      Volume: 10

    • DOI

      10.1371/journal.pone.0129334

    • Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-15KT0063, KAKENHI-PROJECT-15K06767, KAKENHI-PROJECT-15K07772, KAKENHI-PROJECT-15K14976, KAKENHI-PROJECT-15H02495, KAKENHI-PROJECT-25253011, KAKENHI-PROJECT-15H04641, KAKENHI-PROJECT-24500435, KAKENHI-PROJECT-24591349, KAKENHI-PROJECT-26640087, KAKENHI-PROJECT-26288051, KAKENHI-PROJECT-25713007
  • [Journal Article] Nickel-Catalyzed Suzuki–Miyaura Coupling of a Tertiary Iodocyclopropane with Wide Boronic Acid Substrate Scope: Coupling Reaction Outcome Depends on Radical Species Stability.2015

    • Author(s)
      Keisuke Yotsuji, Naoyuki Hoshiya, Takaaki Kobayashi, Hayato Fukuda, Hiroshi Abe, Mitsuhiro Arisawa and Satoshi Shuto
    • Journal Title

      Advanced Synthesis & Catalysis

      Volume: 357 Pages: 1022-1028

    • DOI

      10.1002/adsc.201401000

    • Peer Reviewed / Acknowledgement Compliant / Open Access
    • Data Source
      KAKENHI-PROJECT-23246013, KAKENHI-PROJECT-24390023, KAKENHI-PUBLICLY-25105702, KAKENHI-PROJECT-25282240, KAKENHI-PROJECT-25670049, KAKENHI-PROJECT-26288051, KAKENHI-PROJECT-26860003, KAKENHI-PROJECT-15H02495
  • [Journal Article] Determination of ω-6 and ω-3 PUFA metabolites in human urine samples using UPLC/MS/MS.2015

    • Author(s)
      A. Sasaki, H. Fukuda, N. Shiida, N. Tanaka, A. Furugen, J. Ogura, S. Shuto, N. Mano, H. Yamaguchi
    • Journal Title

      Analytical and Bioanalytical Chemistry

      Volume: 407 Pages: 1625-1639

    • DOI

      10.1007/s00216-014-8412-5

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-24390023, KAKENHI-PROJECT-25460184, KAKENHI-PROJECT-15H02495
  • [Journal Article] Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor.2014

    • Author(s)
      Takaaki Kobayashi, Akihiro Suemasa, Arisa Igawa, Soichiro Ide, Hayato Fukuda, Hiroshi Abe, Mitsuhiro Arisawa, Masabumi Minami, Satoshi Shuto
    • Journal Title

      ACS Med. Chem. Lett

      Volume: 5 Pages: 889-893

    • DOI

      10.1021/ml500134k

    • Peer Reviewed / Acknowledgement Compliant / Open Access
    • Data Source
      KAKENHI-PROJECT-23246013, KAKENHI-PROJECT-24390023, KAKENHI-PUBLICLY-25105702, KAKENHI-PROJECT-25670049, KAKENHI-PROJECT-26288051
  • [Journal Article] Preparation of chiral bromomethylenecyclopropane and its use in Suzuki-Miyaura coupling; synthesis of the arylmethyl-Z-cyclopropane structure core2013

    • Author(s)
      Makoto TANABE
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 78 Pages: 11714-11720

    • DOI

      10.1021/jo401675z

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23246013, KAKENHI-PROJECT-24390023, KAKENHI-PROJECT-24710260, KAKENHI-PUBLICLY-25105702
  • [Presentation] 海産天然物ビスケルソラノリドの合成研究2021

    • Author(s)
      川﨑 則彦、小嶺 敬太、福田 隼、石原 淳
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] アンサマイシン系天然物サイトトリエニン Aの合成研究2021

    • Author(s)
      坂田 淳、佐藤 晋平、小嶺 敬太、福田 隼、渡邉 瑞貴、周東 智、石原 淳
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] 海産天然物ギムノジミンの合成研究2021

    • Author(s)
      久保田 健斗、山中 未歩、小嶺 敬太、福田 隼、石原 淳
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] ツガシン cmc-Aの合成研究2021

    • Author(s)
      堤 智寛、松本 萌、岩崎 瞳、富澤 慧、Eustache Jacques、小嶺 敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] (-)-Haliclonin Aの形式合成2020

    • Author(s)
      小嶺 敬太, 浦山 泰洋, 保坂 拓, 山下 裕貴, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      第49回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] ビスケルソラノリドの合成研究2020

    • Author(s)
      川﨑 則彦、小嶺 敬太、福田 隼、石原 淳
    • Organizer
      第117回有機合成シンポジウム
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] ツガシンcmc-Aの合成研究2020

    • Author(s)
      堤 智寛、松本 萌、岩崎 瞳、富澤 慧、Eustache Jacques、小嶺 敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] ビスゲルソラノリドの合成研究2020

    • Author(s)
      川﨑 則彦、小嶺 敬太、福田 隼、石原 淳
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性天然物(+)-イグジグオリドの全合成2020

    • Author(s)
      岡 賢吾, 淵 駿介, 小嶺敬太, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      第62回天然有機化合物討論会
    • Data Source
      KAKENHI-PROJECT-20K06941
  • [Presentation] Formal Synthesis of Haliclonin A Using Tandem Radical Reaction2019

    • Author(s)
      Keita Komine, Yasuhiro Urayama, Taku Hosaka, Yuki Yamashita, Hayato Fukuda, Susumi Hatakeyama, Jun Ishihara
    • Organizer
      27th International Society of Heterocyclic Chemistry Congress
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] ビスゲルソラノリドの全合成研究2019

    • Author(s)
      川﨑則彦、小嶺敬太、福田 隼、石原 淳
    • Organizer
      第36回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] サイトトリエニンAの全合成研究2019

    • Author(s)
      佐藤 晋平、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物(+)-イグジグオリドの合成研究2019

    • Author(s)
      岡 賢吾, 淵 駿介, 小嶺敬太, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] ジテルペン天然物クルチオリドの合成研究2019

    • Author(s)
      福島大貴、坂井良輔、水流裕明、小嶺敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      第36回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] ジテルペン天然物クルチオリドの合成研究2019

    • Author(s)
      福島大貴, 坂井良輔, 水流裕明, 小嶺敬太, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物イグジグオリドの全合成2019

    • Author(s)
      岡 賢吾、淵 駿介、大園 侑花、小嶺 敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      第36回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物(+)-イグジグオリドの合成研究2019

    • Author(s)
      岡 賢吾、淵 駿介、小嶺 敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] ジテルペン天然物クルチオリドの合成研究2019

    • Author(s)
      福島 大貴、坂井 良輔、水流 裕明、小嶺 敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物イグジグオリドの合成研究2019

    • Author(s)
      岡 賢吾, 淵 駿介, 大園侑花,小嶺敬太, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      第29回万有福岡シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 炎症収束脂質レゾルビンE2のスキップジエン構造をベンゼン環で置換した安定等価体創製研究2019

    • Author(s)
      村上 侑斗、福田 隼、石村 航平、平島 洸基、室本 竜太、渡邉 瑞貴、松田 正、 周東 智
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] Progress toward the Total Synthesis of Exiguolide, an Antitumor Macrolide2019

    • Author(s)
      Jun Ishihara, Kengo Oka, Shunsuke Fuchi, Yuka Ohzono, Keita Komine, Hayato Fukuda, Susumi Hatakeyama
    • Organizer
      the 27th French-Japanese Society of Medicinal and Fine Chemistry
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] コーディアクロム類天然物グラジオビアノールの合成研究2019

    • Author(s)
      山本 純、小嶺敬太、福田 隼、石原 淳
    • Organizer
      第36回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物イグジグオリドの合成研究2019

    • Author(s)
      岡 賢吾, 淵 駿介, 大園侑花,小嶺敬太, 福田 隼, 畑山 範, 石原 淳
    • Organizer
      第45回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 海産天然物ポルチミンの合成研究2019

    • Author(s)
      大森一樹、下岡巧弥、小嶺敬太、福田 隼、畑山 範、石原 淳
    • Organizer
      第36回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] タンデムラジカル反応を基軸とするハリクロニンAの形式合成2018

    • Author(s)
      浦山 泰洋、小嶺 敬太、保坂 拓、山下 裕貴、福田 隼、石原 淳、畑山 範
    • Organizer
      第60回天然有機化合物討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] セコラブダン型ジテルペン天然物クルチオリドの合成研究2018

    • Author(s)
      福島 大貴、坂井 良輔、水流 裕明、宮原 哲哉、福田 隼、畑山 範、石原 淳
    • Organizer
      第62回香料・テルペン及び精油化学に関する討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] trans-1, 2-シクロプロパンジアミンおよびジカルボン酸からなるオリゴアミドの合成研究2018

    • Author(s)
      山田 圭恭, 一ノ瀬 亘, 福田 隼, 渡邉 瑞貴, 周東智
    • Organizer
      日本薬学会 第138年会
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] シクロプロパンの構造特性に基づく膜透過性環状ペプチドの設計と合成2018

    • Author(s)
      植村 真衣, 加藤 七海,松井 耕平, 桑原 智希, 渡邉 瑞貴, 福田 隼, 竹内 恒, 広川 貴次, 武隈 洋, 菅原 満, 周東 智
    • Organizer
      日本薬学会第138年会
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] コーディアクロム類天然物グラジオビアノールの合成研究2018

    • Author(s)
      山本 純、福田 隼、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] サイトトリエニンAの合成研究2018

    • Author(s)
      佐藤 晋平、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      第44回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 抗腫瘍活性マクロリド天然物イグジグオリドの合成研究2018

    • Author(s)
      岡 賢吾、淵 駿介、福田 隼、畑山 範、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 多環状マクロ環アルカロイドポルチミンの合成研究2018

    • Author(s)
      大森 一樹、下岡 巧弥、福田 隼、畑山 範、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] スピロリドBの環状イミン部位の合成研究2018

    • Author(s)
      碓井 風馬、黒瀬 朋浩、川口 康徳、福田 隼、畑山 範、石原 淳
    • Organizer
      第35回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] GABAトランスポーターサブタイプ選択的阻害剤の創出を目的とするGABA配座制限誘導体の設計と合成2018

    • Author(s)
      末政亮大、中田和彰、小林嵩明、福田隼、渡邉瑞貴、井手聡一郎、人羅菜津子、南雅文、周東智
    • Organizer
      日本薬学会第138年会
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] スピロ環状イミン天然物ギムノジミンの合成研究2018

    • Author(s)
      山中 未歩、仲達 偲乃、渡邊 由貴、福田 隼、畑山 範、石原 淳
    • Organizer
      第35回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] スピロ環状イミン天然物ギムノジミンの合成研究2018

    • Author(s)
      山中 未歩、仲達 偲乃、渡邊 由貴、福田 隼、畑山 範、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] サイトトリエニンA の合成研究2018

    • Author(s)
      佐藤 晋平、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      第30回万有札幌シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] Improvement of Membrane Permeability of Cyclic Peptides by Conformational Restriction Using Cyclopropane2018

    • Author(s)
      Mizuki Watanabe, Yukina Sato, Mai Uemura, Nanami Kato, Kouhei Matsui, Hayato Fukuda, Yoh Takekuma, Mitsuru Sugawara, Satoshi Shuto
    • Organizer
      10th International Peptide Symposium
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] グラジオビアノールの合成研究2018

    • Author(s)
      山本 純、福田 隼、石原 淳
    • Organizer
      創薬懇話会2018 in 志賀島
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] セコラブダン型ジテルペンクルチオリドの合成研究2018

    • Author(s)
      福島 大貴、坂井 良輔、水流 裕明、福田 隼、畑山 範、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] IKK-2 inhibitor VI 類縁体の短段階合成2018

    • Author(s)
      川﨑 則彦、福田 隼、石原 淳
    • Organizer
      創薬懇話会2018 in 志賀島
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 大環状スピロイミナールアルカロイドマリネオシンA及びBの合成研究2018

    • Author(s)
      森井 優樹、菅 晃久、山元 広平、福田 隼、畑山 範、石原 淳
    • Organizer
      第35回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] タンデムラシジカル反応を基軸とする(-)-ハリクロニン A の形式合成2018

    • Author(s)
      浦山 泰洋、小嶺 敬太、保坂 拓、山下 裕貴、福田 隼、石原 淳,畑山 範
    • Organizer
      第35回日本薬学会九州支部大会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 大環状スピロイミナールアルカロイドマリネオシン類の合成研究2018

    • Author(s)
      森井 優樹、菅 晃久、山元 広平、福田 隼、畑山 範、石原 淳
    • Organizer
      第44回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 大環状スピロイミナール天然物マリネオシン類の合成研究2018

    • Author(s)
      森井 優樹、菅 晃久、山元 広平、福田 隼、畑山 範、石原 淳
    • Organizer
      第28回万有福岡シンポジウム
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] Synthesis and Biological Evaluation of Cyclopropane Analogues of Resolvin E2 and Deoxy-Resolvin E22018

    • Author(s)
      Hayato Fukuda, Ryuta Muromoto, Toru Hirao, Koki Hirashima, Mizuki Watanabe, Hiroshi Abe, Mitsuhiro Arisawa, Jun Ishihara, Tadashi Matsuda, Satoshi Shuto
    • Organizer
      14th International Kyoto Conference on New Aspects of Organic Chemistry
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] 多置換チオフェンを有するIKK-2 inhibitor VI 類縁体の合成2018

    • Author(s)
      川﨑 則彦、福田 隼、石原 淳
    • Organizer
      第48回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-17K08360
  • [Presentation] シクロプロパン構造特性に基づくレゾルビンE2の安定等価体の創製研究2017

    • Author(s)
      松原 光太郎、池田 紘之、石村 航平、平島 洸基、室本 竜太、松田 正、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      日本薬学会第137年会
    • Place of Presentation
      東北大学川内地区(宮城県仙台市)
    • Year and Date
      2017-03-24
    • Data Source
      KAKENHI-PROJECT-15K18898
  • [Presentation] 炎症収束性脂質レゾルビンE1配座制限誘導体の設計と合成2017

    • Author(s)
      石村 航平,福田 隼,渡邉 瑞貴,周東 智
    • Organizer
      第15回次世代を担う有機化学シンポジウム
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] 光学活性1,2,3-三置換シクロプロパンヌクレオシドの合成2017

    • Author(s)
      南貴覚、福多洸太朗、星谷尚亨、福田隼、渡邉瑞貴、周東智
    • Organizer
      第29回万有札幌シンポジウム
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] Spiro-cyclopropane type α-helix/β-strand mimimetics targeting protein-protein interactions2017

    • Author(s)
      Tomoki Kuwahara, Akira Mizuno, Hayato Fukuda, Mizuki Watanabe, Satoshi Shuto
    • Organizer
      254th ACS National Meeting & Exposition
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] シクロプロパンの立体及び立体電子特性に基づくペプチドミメティクス2017

    • Author(s)
      桑原智希,植村真衣,水野彰,一ノ瀬亘,松井耕平,福田隼,渡邉瑞貴,周東智
    • Organizer
      第43回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-15H02495
  • [Presentation] シクロプロパン構造特性に基づくレゾルビンE2の安定等価体の創製研究2016

    • Author(s)
      松原 光太郎、池田 紘之、石村 航平、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      日本薬学会北海道支部 第143回例会
    • Place of Presentation
      札幌コンベンションセンター(北海道札幌市)
    • Data Source
      KAKENHI-PROJECT-15K18898
  • [Presentation] EFFICIENT SYNTHESIS OF ANTI-INFLAMMATORY LIPID MEDIATOR RESOLVIN E1 AND ITS ANALOGUES2016

    • Author(s)
      石村 航平、福田 隼、渡邉 瑞貴、周東 智
    • Organizer
      The XXIV EFMC International Symposium on Medicinal Chemistry
    • Place of Presentation
      マンチェスター(イギリス)
    • Year and Date
      2016-08-28
    • Data Source
      KAKENHI-PROJECT-15K18898
  • [Presentation] 内因性炎症収束脂質レゾルビン類の創薬化学研究2016

    • Author(s)
      池田 紘之、福田 隼、高倉 夕季、石村 航平、平島 洸基、平尾 徹、室本 竜太、渡邉 瑞貴、松田 正、周東 智
    • Organizer
      第34回メディシナルケミストリーシンポジウム
    • Place of Presentation
      つくば国際会議場(茨城県つくば市)
    • Year and Date
      2016-11-30
    • Data Source
      KAKENHI-PROJECT-15K18898
  • [Presentation] 内因性炎症収束脂質レゾルビンE2安定等価体の創製2015

    • Author(s)
      福田隼,髙倉夕季,石村航平,金田龍太郎,平尾徹, 平島洸基,室本竜太,松田正,阿部洋,有澤光弘,周東智
    • Organizer
      第41回反応と合成の進歩シンポジウム
    • Place of Presentation
      近畿大学11月ホール(大阪府東大阪市)
    • Year and Date
      2015-10-26
    • Data Source
      KAKENHI-PROJECT-15K18898
  • [Presentation] Synthesis and SAR study of resolvin E22014

    • Author(s)
      福田 隼
    • Organizer
      247th American Chemical Society National Meeting & Exposition
    • Place of Presentation
      Dallas Convention Center, Dallas, USA
    • Data Source
      KAKENHI-PROJECT-25860087
  • [Presentation] ddntification of the first highly selective BGT-I inhibitor based on conformational restriction of GABA.

    • Author(s)
      末政亮大、中田和彰、小林嵩明、井川ありさ、福田隼、阿部洋、有澤光弘、井手聡一郎、南雅文、周東智
    • Organizer
      The 12th International Symposium for Future Drug Discovery and Medical Care
    • Place of Presentation
      札幌
    • Year and Date
      2014-09-04 – 2014-09-05
    • Data Source
      KAKENHI-PROJECT-24390023
  • [Presentation] Synthesis and SAR study of resolvin E2

    • Author(s)
      Hayato Fukuda
    • Organizer
      DPhG Annual Meeting 2014
    • Place of Presentation
      Frankfurt
    • Year and Date
      2014-09-24 – 2014-09-26
    • Invited
    • Data Source
      KAKENHI-PROJECT-25860087
  • [Presentation] ファゴサイトーシス誘導性ホスファチジルセリン二量体類縁化合物の創製研究

    • Author(s)
      佐藤耀、川村周平、平尾徹、室元竜太、福田隼、阿部洋、松田正、周東智
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-25 – 2015-03-28
    • Data Source
      KAKENHI-PROJECT-25670048
  • [Presentation] PdおよびNi触媒によるシクロプロパン第三級炭素上への芳香環導入反応―効率的化学空間探索型創薬ライブラリーの構築を目指して―

    • Author(s)
      星谷尚亨、四辻慶佑、小林嵩明、福田 隼、阿部 洋、有澤光弘、周東 智
    • Organizer
      第40回反応と合成の進歩シンポジウム
    • Place of Presentation
      仙台
    • Year and Date
      2014-11-10 – 2014-11-11
    • Data Source
      KAKENHI-PROJECT-24390023
  • [Presentation] GABA配座制限に基づく初のGABAトランスポーターBGT-1サブタイプ高選択的阻害剤の創製

    • Author(s)
      末政亮大、小林嵩明、井川ありさ、福田隼、阿部洋、井手聡一郎、南雅文、周東智
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PROJECT-24390023
  • 1.  SHUTO Satoshi (70241346)
    # of Collaborated Projects: 4 results
    # of Collaborated Products: 34 results
  • 2.  IWABUCHI Yoshiharu (20211766)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 3.  SHIBUYA Masatoshi (40359534)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 4.  有澤 光弘 (40312962)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 16 results
  • 5.  MINAMI Masabumi (20243040)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 3 results
  • 6.  HIGASHIDA Haruhiro (30093066)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 7.  HIROKAWA Takatugu (20357867)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 8.  ASAI Akira (60381737)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 9.  MATSUDA Tadashi (20212219)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 2 results
  • 10.  小松 康雄 (30271670)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 11.  山口 浩明 (80400373)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 1 results
  • 12.  一ノ瀬 亘 (00636409)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 2 results
  • 13.  MOGI Chihiro
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 3 results
  • 14.  ABE Mitsuhiro
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 15.  HISADA Takeshi
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 2 results
  • 16.  NAKAYA Michio
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 17.  IDE Soichiro
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 18.  MUROMOTO Ryuta
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 19.  渡邉 瑞貴
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 10 results
  • 20.  石原 淳
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 5 results
  • 21.  小嶺 敬太
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 4 results
  • 22.  黒瀬 等
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 2 results
  • 23.  岡島 史和
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 2 results
  • 24.  青木 悠
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 2 results
  • 25.  中倉 敬
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 26.  佐甲 靖志
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 27.  阿部 洋
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 2 results
  • 28.  海野 雄加
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 29.  藤原 広一
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 30.  佐藤 幸市
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 31.  戸村 秀明
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 32.  村田 直哉
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 33.  金田 勝幸
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 34.  佐藤 公道
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 35.  人羅 菜津子
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results
  • 36.  星谷 尚亨
    # of Collaborated Projects: 0 results
    # of Collaborated Products: 1 results

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