ENDO Yasuyuki 遠藤泰之

… Alternative Names

遠藤康之

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Researcher Number	80126002
Other IDs
External Links
Affiliation (based on the past Project Information) *help	2016 – 2019: 東北医科薬科大学, 薬学部, 教授 2014 – 2015: 東北薬科大学, 薬学部, 教授 2002 – 2012: 東北薬科大学, 薬学部, 教授 1997 – 2001: University of Tokyo, Graduate School of Pharmaceutical Sciences, Associate Professor, 大学院・薬学系研究科, 助教授 1991 – 1996: 東京大学, 薬学部, 助教授 1993: 東京大学, 薬楽部, 助教授 1986 – 1990: 東京大学, 薬学部, 講師
Review Section/Research Field	Principal Investigator Chemical pharmacy / Drug development chemistry / 医薬分子機能学 / Bioorganic chemistry Except Principal Investigator Chemical pharmacy / 医薬分子機能学 / Drug development chemistry / Biological Sciences
Keywords	Principal Investigator 発癌プロモーター / ホウ素クラスター / 疎水性相互作用 / 医薬分子設計 / 有機合成化学 / 分子設計 / テレオシジン / アンタゴニスト / アンドロゲン受容体 / エストロゲン受容体 … More / 核内受容体 / 医薬品化学 / ステロイド / hydrophobic interaction / boron cluster / receptor / 受容体 / teleocidin / フォルボールエステル / 発がんプロモーター / レチノイドX受容体 / 分子認識 / 核磁気共鳴スペクトル / 立体配座 / 立体配座解析 / 核磁気共鳴 / molecular recognition / antagonist / androgen receptor / estrogen receptor / nuclear receptor / medicinal drug design / drug design / liquid crystal / functional molecule / molecular construction / carborane / 芳香族多層構造 / 芳香族ウレア / 求核性 / 反応速度解析 / 加溶媒分解 / アセチレン / 疎水性相互 / 液晶 / 機能性分子 / 立体分子構築 / カルボラン / hydrophbic interaction / molecular Design / signal transduction / phorbol ester / benzolactam / ベンゾラクタム / 細胞内情報伝達 / バンゾラクタム / steroid / protein kinase C / chemical synthesis / molecular design / anti-HIV compound / tumor promoter / プロテインキナーゼ / 化学合成 / 抗HIV化合物 / Steroids / Molecular Design / Nuclear Magnetic Resonance / Conformational Analysis / Synthetic Chemistry / Phorbol ester / Teleocidin / Tumor promoter / 構造活性相関 / 分子動力学 / i医薬分子設計 / アゴニスト / アニオニック転位 / 反応機構 / シグマトロピック転位 / [3,3]転位 / ヒドロキシルアミン / ヒドラジン / 中員環化合物 … More Except Principal Investigator レチノイド / ビタミンA / レチノイン酸 / 分化 / 分化誘導 / 分子設計 / 核内レセプター / テレオシジン / HL60 / differentiation / retinoic acid / ビタミンA酸 / レセプター / アンタゴニスト / レチノイドレセプタ- / ベンゾラクタム / ステロイド / leukemia / vitamin A / retinoid / レチノイドアンタゴニスト / 白血病 / 反応機構 / ジカチオン / ベンゼン / アンドロゲンアンタゴニスト / シクロオキシゲナーゼ / アンドロゲン / 構造展開 / サリドマイド / 抗アンドロゲン / 生物応答調節剤 / チロキシン / 転移 / 形態形成 / 遺伝子発現 / ラジカル補足作用 / 抗腫瘍活性 / ホウ素化学 / 創薬化学 / スクリーニング / ラジカル捕捉 / ホウ素クラスター / ラジカル捕捉作用 / 抗腫瘍作用 / カルボラン / ランダムスクリーニング / 化合物ライブラリー / ホウ素化合物 / proliferation / phorbol / active vitamin D / teleocidin / retinoid, differentiation, vitamin A, retinoic acid. teleocidin retinoid / cーcmyc / ペプチド / サイトカイニン / アフィディコリン / 芳香族アミド / 血球分化 / 分化誘導物質 / 構造活性相関 / 活性ビタミンD3 / 活性ビタミンD_3 / フォルボ-ル / 増殖 / thalidomide / bioprobe / molecular design / enzyme inhibitor / antagonists / steroid hormone / structural development / nuclear receptor / 抗リウマチ活性 / 抗糖尿病活性 / 一酸化窒素 / シクロオキシゲナーゼ阻害剤 / 核内受容体 / エストロゲン / 阻害剤 / ビタミンD_3 / バチェラジン / チュブリン重合阻害剤 / 組胞分化誘導 / ビタミンDアンタゴニスト / プロテインキナーゼC / プロゲステロン / FXR / ビタミンD / PPAR / Farnesoid X Receptor (FXR) / Liver X Receptor (LXR) / 核内受容体リガンド / 蛍光プローブ / 酵素阻害剤 / ステロイドホルモン / de novo ligand design / drug design software / computer drug design / drug lead / lead generation / drug design / 受容体の立体構造 / 3次元データベース / 自動構築法 / 自動ドッキング / 3次元構造データベース / コンピュータ薬物設計 / リガンド設計 / リ-ド創製 / 医薬リ-ド / Ruthenium Porphyrin / Chiral Palladium Complex / Teleocidin Analogue / Chiral Lithium Amide / Calixarene Ester / Nuclear Magnetic Resonance / Solution Structure / Reactive Complex / 不斉Heck反応 / ルシジン / カリックスアレン / 不斉アルドール反応 / ステロイドグリコシド / キラルリチウムアミド / 膜電位変化 / 核磁気共鳴スペクトル法 / ルテニウムポルフィリン / キラルパラジウム錯体 / テレオシジン類縁体 / キラルチリウムアミド / カリックスアレーンエステル / 核磁気共鳴 / 溶液構造 / 反応活性錯体 / antagonist synergist / myeloma / tyroids / 癌 / ジベンゾジアゼピン / フオルボール / 腫瘍悪性化 / チロイドリセプター / レチノイン酸レセプター / リウマチ / チロイド / 核レセプター / Gattermann-Koch reaction / Gattermannreaction / Trifluoromethanesulfonic acid / Super acid / Carbenium ion / Iminiumbenzenium ion / Friedel-Crafts reaction / オキソニウムカチオン / エチレンジカチオン / ガッタ-マン反応 / カチオン / アセチル化 / フリ-デルクラフト反応 / 求電子試薬 / フリーデルクラフト反応 / ガッターマン・コッホ反応 / ガッターマン反応 / トリフルオルメクンスルホン酸 / 強酸 / カルベニウムイオン / イミニウムベンゼニウムイオン / フリーデル・クラフト反応 / retinoid receptor / cancer / retinoid antagonist / シリコン / 癌治療 / 核レセプタ- / レチノイドレセプター / がん / X線結晶解析 / 核中レセプター / 酸異性化 / 細胞分化 / リセプタータンパク / カルコンカルボン酸・分化 / テレフタル酸アリリド / 癌治療薬 / 分子軌道法 / ベンジルカチオン / フェノキセニウムイオン / アニレニウムイオン / 陽イオン / 芳香族化合物 / レチノイン酸結合タンパク / 白血病細胞 / DNA / ブレオマイシン / 制がん剤 / 化学療法剤 / 細胞浸潤阻害 / 耐性克服 / 前立腺がん細胞 / 一酸化窒素合成酵素 / フタルイミド / 医薬リード / フォルボール / ビタミンE / erb-A / フオルポール / 血管新生 / レチイン酸 / 分子進化 / Lーアラビノ-ス / レ-デオキシアデノシン / (dA)_6 / 三重鎖 / アンチセンスDNA / 核内レセプタ- / グルマコルケマイド / 発ガンプロモ-タ- / フオルポ-ルエステル / ビタンンA酸 / ビダミンA / 有機ゲルマニウム化合物 / 有機ケイ素化合物 / フォルボ-ルエステル / 発がんプロモ-タ- / 制がん Less

Middle up and down type medicinal chemistry based upon boron compound library
- Principal Investigator
  
  Ohta Kiminori
- Project Period (FY)
  2015 – 2019
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Drug development chemistry
- Research Institution
  Showa University
  Tohoku Medical and Pharmaceutical University
A New Development of Molecular Design Utilizing Novel Hydrophobic StructuresPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  2014 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Drug development chemistry
- Research Institution
  Tohoku Medical and Pharmaceutical University
Development of Receptor Regulators Utilizing Novel HydrophobicStructure and Its Application for Medicinal Drug DesignPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  2008 – 2012
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Tohoku Pharmaceutical University
Development and Application of Novel 3-Dimensional Hydrophobic Structures for Drug Design, Which Are Focused on Molecular Recognition between Ligand and ReceptorPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  2004 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Tohoku Pharmaceutical University
がん増悪因子を阻害する医薬リードの創製
- Principal Investigator
  
  橋本祐一
- Project Period (FY)
  2002 – 2004
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  The University of Tokyo
Design and development of biological response modifiers
- Principal Investigator
  
  HASHIMOTO Yuichi
- Project Period (FY)
  2002 – 2006
- Research Category
  
  Grant-in-Aid for Scientific Research (S)
- Research Field
  
  医薬分子機能学
- Research Institution
  The University of Tokyo
Study on Electronic and Steric Effects of Boron Cluster and Application for Construction of Functional Molecules.Principal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  2001 – 2003
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Tohoku Pharmaceutical University
  The University of Tokyo
Design and Synthesis of Cellular Signal Transduction Modulator, Benzolactam Derivatives and Related CompoundsPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  1998 – 2000
- Research Category
  
  Grant-in-Aid for Scientific Research (B).
- Research Field
  
  Chemical pharmacy
- Research Institution
  University of Tokyo
ヘテロ原子間結合の開裂による[3,3]シグマトロピック転位反応の新展開Principal Investigator
- Principal Investigator
  
  遠藤泰之
- Project Period (FY)
  1996
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  The University of Tokyo
発癌プロモーターの活性発現構造解析を目指す分子設計と合成Principal Investigator
- Principal Investigator
  
  遠藤泰之
- Project Period (FY)
  1995
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Bioorganic chemistry
- Research Institution
  The University of Tokyo
Design, Synthesis and Biological Activity of Anti-HIV Compounds Derived from TeleocidinsPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  1995 – 1997
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  医薬分子機能学
- Research Institution
  University of Tokyo
核内情報伝達系の制御分子の合成と制がん作用機構
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1994 – 1995
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
分子設計と合成による発癌プロモーターの活性発現構造の一般性の確立Principal Investigator
- Principal Investigator
  
  遠藤泰之
- Project Period (FY)
  1994
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  The University of Tokyo
Structural Studies on Reactive Complexes for Highly Selective Organic Reactions
- Principal Investigator
  
  ODASHIMA Kazunori
- Project Period (FY)
  1994 – 1995
- Research Category
  
  Grant-in-Aid for Developmental Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  University of Tokyo
Development of New Methoda for Lead Discovery Using Computer
- Principal Investigator
  
  ITAI Akiko
- Project Period (FY)
  1994 – 1995
- Research Category
  
  Grant-in-Aid for Developmental Scientific Research (B)
- Research Field
  
  医薬分子機能学
- Research Institution
  The Kitasato Institute
  The University of Tokyo
Regulatory compound of nuclear receptor functions.
- Principal Investigator
  
  SHUDO Koichi
- Project Period (FY)
  1993 – 1995
- Research Category
  
  Grant-in-Aid for Developmental Scientific Research (B)
- Research Field
  
  医薬分子機能学
- Research Institution
  University of Tokyo, Faculty of pharm.Sciences
Search for New Tumor Promoters Employing Chemical CalculationPrincipal Investigator
- Principal Investigator
  
  ENDO Yasuyuki
- Project Period (FY)
  1992 – 1993
- Research Category
  
  Grant-in-Aid for General Scientific Research (C)
- Research Field
  
  Chemical pharmacy
- Research Institution
  University of Tokyo
Participation of di- and tri-cations in Friedel-Crafts reactions.
- Principal Investigator
  
  SHUDO Koichi
- Project Period (FY)
  1991 – 1992
- Research Category
  
  Grant-in-Aid for General Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  University of Tokyo
ビタミンA酸および関連化合物による分化誘導とその機作
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1990
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
核内レセプタ-応答遺伝子の認識分子
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1990
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
臨床応用を目指すレチノイドの研究
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1990
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
Molecular design and synthesis of new retinoids
- Principal Investigator
  
  SHUDO Koichi
- Project Period (FY)
  1990 – 1992
- Research Category
  
  Grant-in-Aid for Developmental Scientific Research (B)
- Research Field
  
  Chemical pharmacy
- Research Institution
  Univ. of Tokyo
新しい作用機作をもつ抗がん剤の合成と特性
- Principal Investigator
  
  SHUDO Koichi
- Project Period (FY)
  1989
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
ビタミンA酸および関連化合物による分化誘導とその作用機作
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1989
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
新しい作用機作をもつ抗がん剤の合成と特性
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1988
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
ビタミンA酸および関連化合物による分化誘導とその作用機作
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1988
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
新しい作用機作をもつ抗がん剤の合成と特性
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1987
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Research Institution
  The University of Tokyo
Chemical studies on specific regulatory molecules of cell proliferation and differentiation.
- Principal Investigator
  
  SHUDO Koichi
- Project Period (FY)
  1987 – 1989
- Research Category
  
  Grant-in-Aid for General Scientific Research (A)
- Research Field
  
  Chemical pharmacy
- Research Institution
  The University of Tokyo
新しい作用機作をもつ新しい抗がん剤の創製
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1986
- Research Category
  
  Grant-in-Aid for Special Project Research
- Research Institution
  The University of Tokyo
ベンゼンの新反応の開発
- Principal Investigator
  
  首藤紘一
- Project Period (FY)
  1986
- Research Category
  
  Grant-in-Aid for Special Project Research
- Research Institution
  The University of Tokyo

[Journal Article] Design and Synthesis of Novel Breast Cancer Therapeutic Drug Candidates Based upon the Hydrophobic Feedback Approach of Antiestrogens2019
- Author(s)
  Ohta Kiminori、Kaise Asako、Taguchi Fumi、Aoto Sayaka、Ogawa Takumi、Endo Yasuyuki
- Journal Title
  
  Molecules
  
  Volume: 24 Issue: 21 Pages: 3966-3977
- DOI
  10.3390/molecules24213966
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-15K08029
[Journal Article] ER subtype selectivity of m-carborane-containing phenols: C-alkyl groups on the m-carborane cage enhance ERα selectivity2019
- Author(s)
  Ohta Kiminori、Ogawa Takumi、Kato Koichi、Oda Akifumi、Endo Yasuyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 29 Issue: 16 Pages: 2290-2293
- DOI
  10.1016/j.bmcl.2019.06.025
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-17K08257
[Journal Article] Anti-cancer activity of m-carborane-containing trimethoxyphenyl derivatives through tubulin polymerization inhibition2019
- Author(s)
  Kaise Asako、Endo Yasuyuki、Ohta Kiminori
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 27 Issue: 6 Pages: 1139-1144
- DOI
  10.1016/j.bmc.2019.02.018
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029
[Journal Article] Novel androgen receptor full antagonists: Design, synthesis, and a docking study of glycerol and aminoglycerol derivatives that contain p -carborane cages2018
- Author(s)
  Kaise Asako、Ohta Kiminori、Fujii Shinya、Oda Akifumi、Goto Tokuhito、Endo Yasuyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 26 Issue: 13 Pages: 3805-3811
- DOI
  10.1016/j.bmc.2018.06.007
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-17K08257, KAKENHI-PROJECT-17H03997
[Journal Article] Novel p -carborane-containing multitarget anticancer agents inspired by the metabolism of 17β-estradiol2017
- Author(s)
  Kaise Asako、Ohta Kiminori、Endo Yasuyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 25 Issue: 24 Pages: 6371-6378
- DOI
  10.1016/j.bmc.2017.10.006
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-26460151
[Journal Article] Structure-activity relations of rosmarinic acid derivatives for the amyloid beta aggregation inhibition and antioxidant properties2017
- Author(s)
  Taguchi Riho, Hatayama Koki, Takahashi Tomohito, Hayashi Takafumi, Sato Yuki, Sato Daisuke, Ohta Kiminori, Nakano Hiroto, Seki Chigusa, Endo Yasuyuki, Tokuraku Kiyotaka, Uwai Koji
- Journal Title
  
  EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
  
  Volume: 138 Pages: 1066-1075
- DOI
  10.1016/j.ejmech.2017.07.026
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16K01909, KAKENHI-PROJECT-16H03288, KAKENHI-PROJECT-26460151, KAKENHI-PROJECT-16K14704
[Journal Article] Design and synthesis of p -carborane-containing sulfamates as multitarget anti-breast cancer agents2017
- Author(s)
  Kaise Asako、Ohta Kiminori、Shirata Chinami、Endo Yasuyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 25 Issue: 24 Pages: 6417-6426
- DOI
  10.1016/j.bmc.2017.10.013
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-26460151
[Journal Article] Design and synthesis of iodocarborane-containing ligands with high affinity and selectivity toward ERβ2017
- Author(s)
  Ohta Kiminori、Ogawa Takumi、Endo Yasuyuki
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 27 Issue: 17 Pages: 4030-4033
- DOI
  10.1016/j.bmcl.2017.07.053
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-26460151
[Journal Article] BA321, a novel carborane analog that binds to androgen and estrogen receptors, acts as a new selective androgen receptor modulator of bone in male mice2016
- Author(s)
  Kenta Watanabe, Michiko Hirata Tsukasa Tominari, Chiho Matsumoto, Yasuyuki Endo, Gillian Murphy, Hideaki Nagase, Masaki Inada, Chisato Miyaura,
- Journal Title
  
  Biochem. Biophys. Res. Commun.
  
  Volume: 478 Issue: 1 Pages: 279-285
- DOI
  10.1016/j.bbrc.2016.07.027
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] BE360, a new selective estrogen receptor modulator, produces antidepressant and antidementia effects through the enhancement of hippocampal cell proliferation in olfactory bulbectomized mice.2016
- Author(s)
  Osamu Nakagawasai, Wataru Nemoto, Hiroshi Onogi, Takahiro Moriya, Jia-Rong Lin, Takayo Odaira, Fukie Yaoita, Takumi Ogawa, Kiminori Ohta, Yasuyuki Endo, Koichi Tan-No
- Journal Title
  
  Behav Brain Res
  
  Volume: 297 Pages: 315-322
- DOI
  10.1016/j.bbr.2015.10.033
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460102, KAKENHI-PROJECT-26461709, KAKENHI-PROJECT-26460151
[Journal Article] Symmetric 4,4'-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulators2016
- Author(s)
  Manabu Sato, Kiminori Ohta, Asako Kaise, Sayaka Aoto, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 24 Issue: 5 Pages: 1089-1094
- DOI
  10.1016/j.bmc.2016.01.035
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] Design, synthesis, and anti-proliferative activity of 1-(4-methoxyphenyl)-12-hydroxymethyl-p-carborane derivatives2016
- Author(s)
  Asako Kaise, Kiminori Ohta, Yasuyuki Endo
- Journal Title
  
  Eur. J. Med. Chem.
  
  Volume: 122 Pages: 257-263
- DOI
  10.1016/j.ejmech.2016.06.029
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-15K08029, KAKENHI-PROJECT-26460151
[Journal Article] Structure–activity relationship study of diphenylamine-based estrogen receptor (ER) antagonists2015
- Author(s)
  Kiminori Ohta, Yuki Chiba, Asako Kaise, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 23 Issue: 4 Pages: 861-867
- DOI
  10.1016/j.bmc.2014.12.022
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] Activation of RXR/PPAR; underlies neuroprotection by bexarotene in ischemic stroke2015
- Author(s)
  Michelangelo Certo, Yasuyuki Endo, Kiminori Ohta, Shinobu Sakurada, Giacinto Bagetta, Diana Amantea
- Journal Title
  
  Pharmacological Research
  
  Volume: 102 Pages: 298-307
- DOI
  10.1016/j.phrs.2015.10.009
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] Design and Synthesis of Carborane-containing Estrogen Receptor-beta (ERβ)-Selective Ligands2015
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Akifumi Oda, Asako Kaise, Yasuyuki Endo
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters
  
  Volume: 25 Issue: 19 Pages: 4174-4178
- DOI
  10.1016/j.bmcl.2015.08.007
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460034, KAKENHI-PROJECT-26460151, KAKENHI-PUBLICLY-15H01064
[Journal Article] Synthesis and biological evaluation of novel m-carborane-containing estrogen receptor partial agonists as SERM candidates2015
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Asako Kaise, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 25 Issue: 16 Pages: 3213-3216
- DOI
  10.1016/j.bmcl.2015.05.083
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] Estrogenic activity of bis(4-hydroxyphenyl)methanes with cyclic hydrophobic structure2015
- Author(s)
  Tomohiro Kojima, Takumi Ogawa, Souichiro Kitao, Manabu Sato, Akifumi Oda, Kiminori Ohta, Yasuyuki Endo
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 23 Issue: 21 Pages: 6900-6911
- DOI
  10.1016/j.bmc.2015.09.046
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-26460034, KAKENHI-PROJECT-26460151, KAKENHI-PUBLICLY-15H01064
[Journal Article] Novel estrogen receptor (ER) modulators containing various2014
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Asako Kaise, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 13 Pages: 3508-3514
- DOI
  10.1016/j.bmc.2014.04.022
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24790115, KAKENHI-PROJECT-26460151
[Journal Article] Aliphatic Substitution of o-Carboranyl Phenols Enhances Estrogen Receptor Beta Selectivity.2014
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Asako Kaise, Akifumi Oda, Yasuyuki Endo
- Journal Title
  
  Chem. Pharm. Bull.
  
  Volume: 62 Pages: 386-391
- NAID
  130003390780
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-26460151
[Journal Article] Estrogenic Activity of B-Fluorinated o-Carborane-1,2-bisphenol Synthesized via SNAr Reaction2012
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 22 Issue: 14 Pages: 4728-4730
- DOI
  10.1016/j.bmcl.2012.05.068
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-24790115
[Journal Article] Development of Androgen Recby Application of Ten-vertex p-Carborane as a Novel Hydrophobic Core Structure2012
- Author(s)
  Shinya Fujii, Kiminori Ohta, Tokuhito Goto, Akifumi Oda, Hiroyuki Masuno, Ysuyuki Endo, Hiroyuki Kagechika
- Journal Title
  
  Med. Chem. Commun
  
  Volume: 3 Issue: 6 Pages: 680-684
- DOI
  10.1039/c2md00294a
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128, KAKENHI-PROJECT-23790137, KAKENHI-PROJECT-24790115, KAKENHI-PLANNED-22136013
[Journal Article] Facile Synthesis and EstArylpyrrole-based Bisphenol Derivatives2012
- Author(s)
  Fumi Taguchi, Yasuyuki Endo
- Journal Title
  
  Heterocycles
  
  Volume: 86 Issue: 1 Pages: 165-170
- DOI
  10.3987/com-12-s(n)56
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-24790115
[Journal Article] RXR-gamma isDocosahexaenoic Acid Modulation of Despair Behaviors and Working Memory in Mice2011
- Author(s)
  Marta Wietrzych-Schindler, MSzyszka-Niagolov, Kiminori Ohta, Yasuyuki Endo, Efren Perez Angel R. de Lera, Pierre Chambon, Wojciech Krezel
- Journal Title
  
  Biological Psychiatry
  
  Volume: 69 Issue: 8 Pages: 788-794
- DOI
  10.1016/j.biopsych.2010.12.017
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Boron Cluster-based DevNon-Secosteroidal Vitamin D Receptor Ligands: Direct Observation of Hydrophobic Interaction between Protein Surface and Carborane2011
- Author(s)
  Shinya Fujii, Hiroyuki Masuno, Yoshiyuki Taoda, Atsushi Kano, Angsuma Wongmayura, Makoto Nakabayashi, Nobutoshi Ito, Masato Shimizu, Emiko Kawachi, Tomoya Hirano, YasuyukiEndo, Aya Tanatani, Hiroyuki Kagechika
- Journal Title
  
  J. Am. Chem. Soc
  
  Volume: 133 Issue: 51 Pages: 20933-20941
- DOI
  10.1021/ja208797n
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-22790106, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128
[Journal Article] p-Carborane Based AndrogenActive in LNCaP Cells with a Mutated Androgen Receptor2011
- Author(s)
  Shinya Fujii, Ayumi Yamada, Keiko Tomita, Mao Nagano, Tokuhito Goto, Kiminori Ohta, Takashi Harayama, Yasuyuki Endo, Hiroyuki Kagechika
- Journal Title
  
  Med. Chem. Commun
  
  Volume: 2 Issue: 9 Pages: 877-880
- DOI
  10.1039/c1md00001b
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116, KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128
[Journal Article] Crystal Structure, Docking SStructure-activity Relationship of Carborane-containing Androgen2011
- Author(s)
  Kiminori Ohta, Tokuhito Goto, Synya Fujii, Masatoshi Kawahata, Akifumi Oda, Shigeru Ohta, Kentaro Yamaguchi, Shuichi Hirono,Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 19 Issue: 11 Pages: 3540-3548
- DOI
  10.1016/j.bmc.2011.04.017
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116, KAKENHI-PROJECT-23790128
[Journal Article] Synthesis of 3-Aryl-1,2-dicarba-closo-dodecaboranes by Suzuki-Miyaura Coupling Reaction2010
- Author(s)
  Koei Aizawa, Kiminori Ohta, Yasuyuki Endo
- Journal Title
  
  Heterocycles
  
  Volume: 80 Issue: 1 Pages: 369-377
- DOI
  10.3987/com-09-s(s)32
- NAID
  40016900113
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Design and Synthesis oReceptor (AR) Antagonists Bearing a p-Carborane Cage: Promising Ligand for Antiandrogen Withdrawal Syndrome2010
- Author(s)
  Tokuhito Goto, Kiminori Ohta, Shinya Fujii, Tomoharu Suzuki, Shigeru Ohta, Yasuyuki Endo
- Journal Title
  
  J. Med. Chem
  
  Volume: 53 Issue: 13 Pages: 4917-4926
- DOI
  10.1021/jm100316f
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Design and Synthesis of Potent Androgen Receptor (AR) Antagonists Bearing a p-Carborane Cage : Promising Ligand for Antiandrogen Withdrawal Syndrome.2010
- Author(s)
  Goto, T., Ohta, K., Fujii, S., Suzuki, T., Ohta, S., Endo, Y.
- Journal Title
  
  J.Med.Chem. 53
  
  Pages: 4917-4926
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Conformational Control of Benzyl-o-carboranylbenzene Derivatives and Molecular Encapsulation of Acetone into the Dynamically-formed Space of 1,3,5-Tris(2-benzyl-o-carboran-1-yl)benzene2010
- Author(s)
  Chermkiat Songkram, Kiminori Ohta, Kentaro Yamaguchi, Fabio Pichierri, Yasuyuki Endo
- Journal Title
  
  Inorg. Chem
  
  Volume: 49 Issue: 23 Pages: 11174-11183
- DOI
  10.1021/ic101862n
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] A novel carborane acarbon-containing polyhedral boron-cluster is a new selective estrogen receptor modulator for bone2009
- Author(s)
  MichikoMorichika Takita, Takumi Ogawa, Yasuyuki Endo, Chisato Miyauraa
- Journal Title
  
  Biochem. Biophys. Res. Commun
  
  Volume: 830 Pages: 218-222
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Synthesis and biological evaluationof p-carborane bisphenols and their derivatives: Structure-activity relationship for estrogenic activity2009
- Author(s)
  Takumi Ogawa, Kiminori Ohta, Toru Iijima, Tomoharu Suzuki, Shigeru Ohta, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 17 Issue: 3 Pages: 1109-1117
- DOI
  10.1016/j.bmc.2008.12.044
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure2009
- Author(s)
  Shinya Fujii, Kiminori Ohta, TokuhitoGoto, Hiroyuki Kagechika, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 17 Issue: 1 Pages: 344-350
- DOI
  10.1016/j.bmc.2008.10.060
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Novel estrogen receptor (ECarbamate and thiocarbamate derivatives with m-carborane bisphenol structure2009
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Tomoharu Suzuki, Shigeru Ohta, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 17 Issue: 23 Pages: 7958-7963
- DOI
  10.1016/j.bmc.2009.10.018
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
[Journal Article] Novel estrogen receptor (ER) modulators : Carbamate and thiocarbamate derivatives with m-carborane bisphenol structure2009
- Author(s)
  U, Ogawa, T., Suzuki,, T., Ohta, S., Endo, Y.
- Journal Title
  
  Bioorg.Med.Chem. 17
  
  Pages: 7958-7963
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Synthesis and biological evaluation of p-carborane bisphenols and their derivatives : Structure-activity relationship for estrogenic activity2009
- Author(s)
  Ogawa, T., Ohta, K., Iijima, T., Suzuki, T., Ohta, S., Endo, Y.
- Journal Title
  
  Bioorg.Med.Chem. 17
  
  Pages: 1109-1117
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] A novel carborane analog, BE360, with a carbon-containing polyhedral boron-cluster is a new selective estrogen receptor modulator for bone.2009
- Author(s)
  Hirata, M., Inada, M., Matsumoto, C., Takita, M., Ogawa, T., Endo, Y., Miyaura, C.
- Journal Title
  
  Biochem.Biophys.Res.Commun. 930
  
  Pages: 218-222
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Identification of an intermediate in the deboronation of ortho-carborane: an adduct of ortho-carborane with two nucleophiles on one boron atom2008
- Author(s)
  Yoshiyuki Taoda, Takehiko Sawabe, Yasuyuki Endo, Kentaro Yamaguchi, Shinya Fujii, Hiroyuki Kagechika
- Journal Title
  
  Chem. Commun
  
  Issue: 17 Pages: 2049-2051
- DOI
  10.1039/b716079h
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Design and synthesis of carborane-containing androgen receptor (AR) antagonist bearing a ryridine ring2008
- Author(s)
  Ohta, K., Goto, T., Fijii, S., Suzuki, T., Ohta, S., Endo, Y.
- Journal Title
  
  Bioorg.Med.Chem. 16
  
  Pages: 8022-8028
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Design and synthesis of carborane-containing androgen receptor (AR) antagonist bearing a ryridine ring2008
- Author(s)
  Kiminori Ohta, Tokuhito Goto, Sinya Fijii, Tomoharu Suzuki, Shigeru Ohta, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem
  
  Volume: 16 Issue: 17 Pages: 8022-8028
- DOI
  10.1016/j.bmc.2008.07.055
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Identification of an Intermediate in the Deboronation of ortho-Carborane : an Adduct of ortho-Carborane with Two Mucleophiles on One Boron Atom2008
- Author(s)
  Taoda, Y., Sawabe, T., Endo, Y.*, Yamaguchi, K., Fujii, S., Kagechika, H.*
- Journal Title
  
  Chem. Commun
  
  Pages: 2049-2051
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Promising core structure for nuclear receptor ligands: Design and synthesis of novel estrogen receptor ligands based on diphenylamine skeleton2008
- Author(s)
  Kiminori Ohta , Yuki Chiba, Takumi Ogawa, Yasuyuki Endo
- Journal Title
  
  Bioorg. Med. Chem. Lett
  
  Volume: 18 Issue: 18 Pages: 5050-5053
- DOI
  10.1016/j.bmcl.2008.08.004
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Symmetric Bent-core Mesogens with m-Carborane and Adamantane As the Central Units2008
- Author(s)
  Pociecha, D., Ohta, K., Januszko, A., Kaszynski, P.*, Endo, Y
- Journal Title
  
  J. Mater. Chem (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Complexation of b-cyclodextrin with carborane derivatives in aqueous solution2008
- Author(s)
  Kiminori Ohta, Shunsuke Konno, Yasuyuki Endo
- Journal Title
  
  TetrahedronLett
  
  Volume: 49 Issue: 46 Pages: 6525-6528
- DOI
  10.1016/j.tetlet.2008.08.107
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20390035
[Journal Article] Facile and Efficient Synthesis of C-Hydroxycarboranes and C, C'-Dihydroxycarboranes2007
- Author(s)
  Ohta, K., Goto, T., Yamazaki, H., Pichierri, F. : Endo, Y.*
- Journal Title
  
  Inorg. Chem 46
  
  Pages: 3966-3970
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] ホウ素クラスター:カルボランの有機化学-合成、構造、立体分子構築への応用2007
- Author(s)
  遠藤泰之
- Journal Title
  
  有機合成化学協会誌 65
  
  Pages: 320-333
- NAID
  10018898672
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Solid-state Supramolecular Array through Cooperative tt-it Interactions of -(2-Methoxyphenyl)-o-carborane2007
- Author(s)
  Ohta, K., Yamazaki, H., Pichierri, F., Kawahata, M., Yamaguchi, K., Endo, Y.*
- Journal Title
  
  Tetrahedron 63
  
  Pages: 12160-12165
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Proton-Driven Conformational Change in a 2-Aryl-p-carborane Constrained by an Intramolecular C-H-O Hydrogen Bond2007
- Author(s)
  K. Ohta, K., Yamazaki, H., Kawahata, M., Yamaguchi, K., Pichierri, F., Endo. Y.*
- Journal Title
  
  Tetrahedron. Lett 48
  
  Pages: 5231-5234
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Genetic and Pharmacological Evidence that a Retinoic Acid Cannot be the RXR-activating Ligand in Mouse Epidermis Keratinocytes2006
- Author(s)
  Calleja, C., Messaddeq, N., Chapellier, B., Yang, H., Krezel, W., Li, M., Metzger, D., Marcrez, B., Ohta, K., kagechika H, Endo, Y., Mark, M., Ghyselinck, N. B., Chambon, P.*
- Journal Title
  
  Genes Dev 20
  
  Pages: 1525-1538
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] 創薬化学における新規3次元的疎水性構造単位の開発と応用2006
- Author(s)
  遠藤泰之
- Journal Title
  
  ファルマシア 42
  
  Pages: 421-425
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] m-Carborane Bisphenol Structure as a Pharmacophore for Selective Estrogen Receptor Modulators2006
- Author(s)
  Ogawa, T., Ohta K, Yoshimi, T., Yamazaki, H., Suzuki, T., Ohta, S., Endo, Y.*
- Journal Title
  
  Bioorg. Med. Chem. Lett 16
  
  Pages: 3943-3946
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A Distorted Benzene Bearing Two Bulky Substituents on Adjacent Positions : Structure of 1, 2-Bis(I, 2-Dicarba-closo-dodecaboran-1-yl)benzene2005
- Author(s)
  Endo, Y.*, Songkram, C., Ohta, K., Kaszynski, P., Yamaguchi, K
- Journal Title
  
  Tetrahedron Lett 46
  
  Pages: 699-702
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Potent Estrogen Receptor Ligands Based on Bisphenols with Globular Hydrophobic Cores2005
- Author(s)
  Endo, Y*., Yoshimi, T., Ohta, K., Suzuki, T., Ohta, S
- Journal Title
  
  J. Med. Chem 48
  
  Pages: 3941-3944
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] 1, 2-Dicarba-closo-dodecaboran-1-yl Naphthalene Derivatives2005
- Author(s)
  Ohta, K., Goto, T., Endo, Y.*
- Journal Title
  
  Inorg. Chem 44
  
  Pages: 8569-8573
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Synthesis of Distorted Molecules Based on Spatial Control with Icosahedral Carboranes2005
- Author(s)
  Endo, Y.*, Songkram, C., Ohta, K., Yamaguchi, K
- Journal Title
  
  J. Organomet. Chem 690
  
  Pages: 2750-2756
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Potent Estrogen Receptor Ligands Based on Bisphenols with Globular Hydrophobic Cores2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  J.Med.Chem 48
  
  Pages: 3941-3944
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A new class androgen receptor antagonists bearing carborane in place of a steroidal skeleton.2005
- Author(s)
  S.Fujii, Y.Hashimoto, T.Suzuki, Ohta, Y.Endo
- Journal Title
  
  Bioorganic & Medicinal Chemistry Letters 15・1
  
  Pages: 227-230
- Data Source
  KAKENHI-PROJECT-14103018
[Journal Article] A Distorted Benzene Bearing Two Bulky Substituents on Adjacent Positions: Structure of 1,2-Bis(1,2-Dicarba-closo-dodecaboran-l-yl)benzene2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  Tetrahedron Lett 46
  
  Pages: 699-702
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A Distorted Benzene Bearing Two Bulky Substituents on Adjacent Positions : Structure of 1,2-Bis(1,2-Dicarba-closo-dodecaboran-1-vl)benzene2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  Tetrahedron Lett. 46
  
  Pages: 699-702
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Regioselective Synthesis of Triiodo-o-carboranes and Tetraiodo-o-carborane2005
- Author(s)
  Yamazaki, H., Ohta, K., Endo, Y.*
- Journal Title
  
  Tetrahedron Lett 46
  
  Pages: 3119-3122
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A comparison of Mesogenic Properties of p-Carborane-1, 12-dicarbaldehyde Schiff Bases with Their Terephthaldehyde Analogues2005
- Author(s)
  Nagamine, T., Januszko, A., Ohta, K., Kaszynski, P., Endo, Y
- Journal Title
  
  Liq. Cryst 32
  
  Pages: 985-995
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Synthesis of Distorted Molecules Based on Spatial Control with Icosahedral Carboranes2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  J.Organomet.Chem. 690
  
  Pages: 2750-2756
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] New Synthetic Method of 1, 2-Diaryl-1, 2-dicarba-closo-dodecaboranes Employing Aromatic Nucleophilic Substitution(SNAr) Reaction2005
- Author(s)
  Ohta, K., Goto, T., Endo, Y.*
- Journal Title
  
  Tetrahedron Lett 46
  
  Pages: 483-485
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Potent Androgen Antagonists Based on Carborane As a Hydrophobic Core Structure.2005
- Author(s)
  Fujii, S., Goto, T., Ohta, K., Hashimoto, Y., Suzuki, T., Ohta, S., Endo, Y.*
- Journal Title
  
  J. Med. Chem 48
  
  Pages: 4654-4662
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Synthesis of Distorted Molecules Based on Spatial Control with Icosahedral Carboranes2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  J.Organomet.Chem 690
  
  Pages: 2750-2756
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] NMR Study of 1, 2-Dicarba-closo-dodecaboranes : Intramolecular C-H-O Hydrogen Bonding in Solution2005
- Author(s)
  Ohta, K., Yamazaki, H., Endo, Y.*
- Journal Title
  
  Tetrahedron. Lett 47
  
  Pages: 1937-1940
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Potent Estrogen receptor Ligands Based on Bisphenols with Globular Hydrophobic Cores.2005
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  J.Med.Chem. 48
  
  Pages: 3941-3944
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Design and Synthesis of Novel Androgen Receptor(AR) Antagonists with Sterically Bulky Icosahedral Carboranes2005
- Author(s)
  Goto, T., Ohta, K., Suzuki, T., Ohta, S., Endo, Y.*
- Journal Title
  
  Bioorg. Med. Chem 13
  
  Pages: 6414-6424
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Novel Retinoid X Receptor(RXR) Antagonists Having a Dicarba-closo-dodecaborane as a Hydrophobic Moiety2004
- Author(s)
  Ohta, K., Iijima, T., Kawachi, E., Kagechika, H., Endo, Y*
- Journal Title
  
  BioMed. Chem. Lett 14
  
  Pages: 5913-5918
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A New Application of Inorganic Cluster,Carboranes for Medicinal Drug Design and Molecular Construction2004
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  Phosphorous, Sulfur, and Silicon 179
  
  Pages: 799-802
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A New Application of Inorganic Cluster, Carboranes for Medicinal Drug Design and Molecular Construction2004
- Author(s)
  Yasuyuki Endo
- Journal Title
  
  Phosphorous, Sulfur, and Sillicon 179
  
  Pages: 799-802
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A New Application of Inorganic Cluster, Carboranes for Medicinal Drug Design and Molecular Construction2004
- Author(s)
  Endo, Y.*, Ohta, K., Yoshimi, T., Yamaguchi, K
- Journal Title
  
  Phosphorous, Sulfur, and Silicon 179
  
  Pages: 799-802
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] A new Class of Androgen Receptor Antagonists Bearing Carborane in Place of a Steroidal Skeleton2004
- Author(s)
  Fujii, S., Hashimoto, Y., Suzuki, T., Ohta, S., Endo, Y*
- Journal Title
  
  BioMed. Chem. Lett 15
  
  Pages: 227-230
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Journal Article] Structural Effects in Three-Ring Mesogenic Derivatives of p-Carborane and Their Hydrocarbon Analogs2004
- Author(s)
  Ohta, K., Januszko, A., Kaszynski, P., Nagamine, T., Sasnouski, G., Endo, Y
- Journal Title
  
  Liq. Cryst 31
  
  Pages: 1-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 抗腫瘍活性を示すm-カルボラン含有トリメトキシフェニル誘導体2020
- Author(s)
  皆瀬麻子、太田公規、遠藤泰之
- Organizer
  日本薬学会第１４０年会
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] 球状ホウ素クラスターを基盤とする新規エストロゲン受容体リガンドの設計と合成2019
- Author(s)
  皆瀬麻子、大山美優、吉見友弘、太田公規、遠藤泰之
- Organizer
  第３７回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] ホウ素クラスター誘導体の抗腫瘍活性とそのメカニズムについて2018
- Author(s)
  皆瀬麻子，白田智七美, 太田公規，遠藤泰之
- Organizer
  日本薬学会第138年会、金沢
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] マルチターゲット型抗腫瘍活性を示す新規カルボラン誘導体の創製2018
- Author(s)
  皆瀬麻子、太田公規、白田智七美、遠藤泰之
- Organizer
  第36回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] ホウ素クラスター誘導体の抗腫瘍活性とそのメカニズムについて2018
- Author(s)
  皆瀨麻子、白田智七美、太田公規、遠藤泰之
- Organizer
  日本薬学会　第138年会
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] 卵巣摘出マウスのうつ様行動に対する新規選択的エストロゲン受容体モジュレーターBE360の効果2017
- Author(s)
  佐久間若菜，中川西　修，根本　亙，小平貴代，小川卓巳，太田公規，遠藤泰之，只野武，丹野孝一
- Organizer
  第21回活性アミンに関するワークショップ，京都
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] Structural differences of the ligand binding pockets between estrogen receptor alpha and beta2017
- Author(s)
  Koichi Kato, Kenichiro Fujii, Tomoki Nakayoshi, Yurie Watanabe, Shuichi Fukuyoshi, Kiminori Ohta, Yasuyuki Endo, Noriyuki Yamaotsu, Shuichi Hirono, Eiji Kurimoto, Akifumi Oda
- Organizer
  XXIX IUPAP conference on computational physics
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] カルボラン含有新規選択的エストロゲン受容体抑制薬（SERD）化合物の探索2017
- Author(s)
  皆瀨麻子、吉見友弘、太田公規、遠藤泰之
- Organizer
  平成29年度東北医科薬科大学　創薬研究センターシンポジウム
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] トロポロン骨格を有する新規キサンチンオキシダーゼ阻害剤の探索とそのメカニズム解析2017
- Author(s)
  佐藤大輔, 氣仙拓也, 太田公規, 遠藤泰之
- Organizer
  平成29年度東北医科薬科大学創薬研究センターシンポジウム, 仙台
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] フェニルアゾトロポロン誘導体のキサンチンオキシダーゼ阻害活性とそのメカニズム解析2017
- Author(s)
  佐藤大輔、氣仙拓也、太田公規、遠藤泰之
- Organizer
  日本薬学会第137年会
- Place of Presentation
  仙台国際センター（仙台）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 更年期うつ病モデルマウスにおける新規選択的エストロゲン受容体モジュレーターBE360の抗うつ効果2017
- Author(s)
  佐久間若菜，中川西　修，根本　亙，小平貴代，八百板富紀枝，小川卓巳，太田公規，遠藤泰之，丹野孝一
- Organizer
  平成29年度東北医科薬科大学創薬研究センターシンポジウム, 仙台
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 新規SERD 化合物の探索：カルボラン含有ER リガンドによるER ダウンレギュレーション2017
- Author(s)
  皆瀨麻子、吉見友弘、太田公規、遠藤泰之
- Organizer
  日本薬学会第137年会
- Place of Presentation
  仙台国際センター（仙台）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 新規SERD化合物の探索：カルボラン含有ERリガンドによるERダウンレギュレーション2017
- Author(s)
  皆瀨麻子、吉見友弘、太田公規、遠藤泰之
- Organizer
  日本薬学会第137年会
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2017-03-24
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] Hydrophobicity and electronic effects of carborane for application in medicinal drug design2017
- Author(s)
  Yasuyuki Endo, Keisuke Yamamoto, Kiminori Ohta, Hiroto Yamazaki, Asako Kaise
- Organizer
  16th International Meeting on Boron Chemistry (IMEBORON XVI) , Hong Kong
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] Structural differences of the ligand　binding pockets between estrogen receptor-alpha and beta2017
- Author(s)
  Koichi Kato, Kenichiro Fujii, Tomoki Nakayoshi, Yurie Watanabe, Shuichi Fukuyoshi, Kiminori Ohta, Yasuyuki Endo, Noriyuki Yamaotsu, Shuichi Hirono, Eiji Kurimoto, Akifumi Oda
- Organizer
  XXIX IUPAP Conference on Computational Physics, CCP20, Ｐａｒｉｓ17
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラン含有非ステロイド型2-methoxyestradiol誘導体の抗腫瘍活性2017
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  ケミカルバイオロジー学会　第12回年会
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] キサンチンオキシダーゼ阻害活性を示すフェニルアゾトロポロン誘導体の探索2016
- Author(s)
  佐藤大輔、氣仙拓也、太田公規、遠藤泰之
- Organizer
  第55回日本薬学会東北支部大会
- Place of Presentation
  奥羽大学（郡山）
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] ホウ素クラスターを中心骨格とする新規選択的エストロゲン受容体抑制薬（SERD）の開発2016
- Author(s)
  皆瀨麻子、吉見友弘、太田公規、遠藤泰之
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Place of Presentation
  つくば国際会議場（つくば）
- Year and Date
  2016-11-30
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] フェニルアゾトロポロン誘導体のキサンチンオキシダーゼ阻害活性2016
- Author(s)
  佐藤大輔，氣仙拓也，太田公規，遠藤泰之
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Place of Presentation
  つくば国際会議場（つくば）
- Year and Date
  2016-11-30
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラン含有グリセロール誘導体の抗アンドロゲン活性2016
- Author(s)
  皆瀨麻子、太田公規、小田彰史、遠藤泰之
- Organizer
  日本薬学会第１３６年会
- Place of Presentation
  みなとみらい（神奈川県横浜市）
- Year and Date
  2016-03-27
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] 新規XO 阻害剤の定量的構造活性相関と結合様式の解析2016
- Author(s)
  太田公規, 佐藤匠, 石井康博, 遠藤泰之
- Organizer
  日本薬学会第136年会
- Place of Presentation
  パシフィコ横浜（横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラン含有グリセロール誘導体の抗アンドロゲン活性2016
- Author(s)
  皆瀨麻子, 太田公規, 小田彰史, 遠藤泰之
- Organizer
  日本薬学会第136年会
- Place of Presentation
  パシフィコ横浜（横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 更年期障害モデルマウスのうつ状態に対する新規選択的エストロゲン受容体モジュレターBE360の効果2016
- Author(s)
  佐久間若菜，中川西修，根本亙，八百板富紀枝，小川卓巳，太田公規，遠藤泰之，丹野孝一
- Organizer
  生体機能と創薬シンポジウム2016
- Place of Presentation
  東北大学川内北キャンパス(仙台）
- Year and Date
  2016-08-25
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] ランダムスクリーニングから見出されたトロポロン誘導体の多様な生物活性2016
- Author(s)
  太田公規、佐藤友紀、皆瀨麻子、遠藤泰之
- Organizer
  第55回日本薬学会東北支部大会
- Place of Presentation
  奥羽大学（郡山）
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 変異ARに対するカルボラン含有グリセロール誘導体の活性評価2016
- Author(s)
  皆瀨麻子、阿部孝俊、太田公規、小田彰史、遠藤泰之
- Organizer
  平成28年度創薬研究センターシンポジウム
- Place of Presentation
  東北医科薬科大学（宮城県仙台市）
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] ホウ素クラスターを中心骨格とする新規選択的エストロゲン受容体制御薬（SERD）の開発2016
- Author(s)
  皆瀨麻子、吉見友弘、太田公規、遠藤泰之
- Organizer
  第３４回メディシナルケミストリーシンポジウム
- Place of Presentation
  つくば国際会議場（茨城県つくば市）
- Year and Date
  2016-11-30
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] 新規カルボラン含有医薬化合物創製への挑戦2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第54回日本薬学会東北支部大会
- Place of Presentation
  岩手医科大学（岩手県紫波郡矢巾町）
- Year and Date
  2015-09-26
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 新規チオフェン含有エストロゲン受容体制御化合物の開発2015
- Author(s)
  青砥沙也加、田口史、皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラン含有2-methoxyestradiol誘導体の細胞増殖抑制作用とメカニズム解析2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第３３回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県千葉市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] トリアジン構造を有する新規キサンチンオキシダーゼ阻害剤の創製2015
- Author(s)
  太田公規，佐藤匠，石井康博，遠藤泰之
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 新規カルボラン含有医薬化合物創製への挑戦2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第５４回日本薬学会東北支部大会
- Place of Presentation
  岩手医科大学（岩手県紫波郡矢巾町））
- Year and Date
  2015-09-26
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] エストロゲン代謝物を基にデザインした球状ホウ素クラスター含有新規抗腫瘍性化合物の開発とメカニズム解析2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  日本ケミカルバイオロジー学会第10回年会
- Place of Presentation
  東北大学（仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラン含有2-methoxyestradiol誘導体の細胞増殖抑制作用とメカニズム解析2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] バナナ型構造を持つエストロゲン受容体リガンドにおけるアゴニスト－アンタゴニストバランスの制御2015
- Author(s)
  皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第１０回日本ケミカルバイオロジー学会
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2015-06-11
- Data Source
  KAKENHI-PROJECT-15K08029
[Presentation] バナナ型構造を持つエストロゲン受容体リガンドにおけるアゴニスト－アンタゴニストバランスの制御2015
- Author(s)
  太田公規、皆瀨麻子、遠藤泰之
- Organizer
  日本ケミカルバイオロジー学会第10回年会
- Place of Presentation
  東北大学（仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 嗅球摘出マウスの短期記憶障害と海馬神経新生抑制に対する新規選択的エストロゲン受容体モジュレーターBE360の改善効果2014
- Author(s)
  川西修、佐々木俊裕、斎藤智恵、深澤鈴、星杏奈、根本亙、八百板富紀枝、小川卓巳、太田公規、遠藤泰之、丹野孝一
- Organizer
  平成26年度東北薬科大学創薬研究センターシンポジウム
- Place of Presentation
  仙台
- Year and Date
  2014-06-14
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 2-メトキシエストラジオールをリード化合物とした新規疎水性骨格を有するチューブリン重合阻害剤の開発2013
- Author(s)
  皆瀬麻子、太田公規、遠藤泰之
- Organizer
  日本薬学会第133年会
- Place of Presentation
  横浜
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] エストロゲン代謝物を基にデザインした新規カルボラン含有チューブリン重合阻害剤2012
- Author(s)
  皆瀬麻子、太田公規、遠藤泰之
- Organizer
  第30回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 新規キサンチンオキシダーゼ(XO)阻害剤の探索2012
- Author(s)
  太田公規、小川真澄、伊藤将、遠藤泰之
- Organizer
  第30回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] カルボラン化合物BA321の新規選択的アンドロゲン受容体モジュレーターとしての作用2012
- Author(s)
  上部良輔,松本千穂,富成司,稲田全規, 遠藤泰之,宮浦千里
- Organizer
  第85回日本生化学会大会
- Place of Presentation
  福岡
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] エストロゲン活性を有するジフェニルメタン誘導体の疎水性構造活性相関2012
- Author(s)
  佐藤学、北尾聡一朗、太田公規、遠藤泰之
- Organizer
  日本薬学会第132年会
- Place of Presentation
  札幌
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of Diphenylamine-based Novel Anion Receptors Bearing o-Carborane Cages2012
- Author(s)
  Shuhei Takahashi, Hiroto Yamazaki, Kiminori Ohta, Yasuyuki Endo
- Organizer
  IME Boron XIV
- Place of Presentation
  Niagara falls, Canada
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 変異アンドロゲン受容体(AR)にも有効な新規カルボラン含有ARアンタゴニストの創製2012
- Author(s)
  皆瀬麻子、後藤徳仁、藤井晋也、太田公規、遠藤泰之
- Organizer
  日本薬学会第132年会
- Place of Presentation
  札幌
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of Novel AR Antagonists having a glycerol moiety2011
- Author(s)
  Asako Kaise, Tokuhito Goto, Shinya Fujii , Kiminori Ohta, Yasuyuki Endo
- Organizer
  IME Boron XIV
- Place of Presentation
  Niagara falls, Canada
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] ジフェニルメタン骨格への新規疎水性部位導入によるERリガンドの創製2011
- Author(s)
  佐藤学、北尾聡一朗、太田公規、遠藤泰之
- Organizer
  第50回日本薬学会東北支部大会
- Place of Presentation
  仙台
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of Estrogen ReceptorModulators: Controlling of the Agonist/Antagonist Balance in m-Carborane Bisphenol Derivatives2011
- Author(s)
  Kiminori Ohta, Takumi Ogawa, Shigeru Ohta, Yasuyuki Endo
- Organizer
  AIMECS11
- Place of Presentation
  Tokyo, Japan
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] ベンジル-o-カルボラニルベンゼンのコンフォメーション制御とアセトン分子の包接2011
- Author(s)
  太田公規、Songkram Chalermkiat、Fabio Pichierri、山口健太郎、遠藤泰之
- Organizer
  第7回ホスト・ゲスト化学シンポジウム
- Place of Presentation
  広島
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of Novel Carboranecontaining AR Antagonists Having a Glycerol Moiety Based on the Co-crystal Structure of Bicalutamide with hAR LBD2011
- Author(s)
  Asako Kaise, Tokuhito Goto, Shinya Fujii , Kiminori Ohta, Yasuyuki Endo
- Organizer
  AIMECS11
- Place of Presentation
  Tokyo, Japan
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Application of Carboranes for MedicinalDrug Design Utilizing Their Globular Geometry and Hydrophobicity.2010
- Author(s)
  Yasuyuki Endo
- Organizer
  JSPS Japan-Spain Joint Research Project, Institutde Ciencia de Materials de Barcelona (C.S.I.C.) Campus U.A.B
- Place of Presentation
  Barceloan, Spain
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 新規立体的疎水性構造の活用による受容体機能制御とその創薬への応用(招待講演)2010
- Author(s)
  遠藤泰之
- Organizer
  創薬懇話会
- Place of Presentation
  2010 in 蔵王
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Conformational Controls of Benzyl-o-carboranylbenzene Derivatives and Molecular Encapsulation of Acetone2010
- Author(s)
  Kiminori Ohta, Chalermkiat ng So kram, Masatoshi Kawahata, Kentaro Yamaguchi, Pichierri Fabio, Yasuyuki Endo
- Organizer
  5th International Symposium on Macrocyclic & Supramolecular Chemistry
- Place of Presentation
  Nara, Japan
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 新規立体的疎水性構造の活用による受容体機能制御とその創薬への応用2010
- Author(s)
  遠藤泰之
- Organizer
  創薬懇話会2010in蔵王
- Place of Presentation
  蔵王ロイヤルホテル(招待講演)
- Year and Date
  2010-11-12
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 変異受容体にも有効な新規アンドロゲンアンタゴニストの創製2010
- Author(s)
  山田歩、冨田景子、長野也麻央、藤井晋、原山尚、太田公規、遠藤泰之、影近弘之
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Application of Carboranes for Medicinal Drug Design Utilizing Their Globular Geometry and Hydrophobicity2010
- Author(s)
  Yasuyuki Endo
- Organizer
  JSPS Japan-Spain Joint Research Project, Institut de Ciencia de Materials de Barcelona (C.S.I.C.) Campus U.A.B
- Place of Presentation
  Barceloan, Spain(Invited Lecture)
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] ジフェニルメタン骨格を利用したエストロゲン受容体制御化合物の探索2010
- Author(s)
  北尾聡一朗、小川卓巳、太田公規、猪股浩平、遠藤泰之
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Application of Carboranes for Medicinal Drug Design Utilizing Their Globular Geometry and Hydrophobicity.2010
- Author(s)
  Endo, Y.
- Organizer
  JSPS Japan-Spain Joint Research Project
- Place of Presentation
  Institut de Ciencia de Materials de Barcelona (C.S.I.C.) Campus U.A.B., Barcelona, Spain,
- Year and Date
  2010-09-25
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 新規立体的疎水性構造の活用による受容体機能制御とその創薬への応用2010
- Author(s)
  遠藤泰之
- Organizer
  創薬懇話会2010 in蔵王
- Place of Presentation
  蔵王(招待講演)
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] エストロゲン受容体リガンドの創製:m-カルボランビスフェノール誘導体におけるアゴニスト-アンタゴニストバランスの制御2010
- Author(s)
  太田公規、小川卓巳、太田茂、遠藤泰之
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] ジフェニルメタン骨格を有するエストロゲン受容体リガンドの創製2009
- Author(s)
  北尾聡一朗、小川卓巳、太田公規、猪股浩平、遠藤泰之
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 10-vertex カルボランを用いたアンドロゲン受容体リガンドの創製2009
- Author(s)
  藤井晋也、太田公規、遠藤泰之、影近弘之
- Organizer
  日本薬学会第129年会
- Place of Presentation
  京都
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 性ホルモンのアゴニスト/アンタゴニストの合成と活性2008
- Author(s)
  遠藤泰之
- Organizer
  東京農工大学工学部
- Place of Presentation
  小金井
- Year and Date
  2008-03-28
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 核内受容体リガンドに対する新規Privileged structure の探索: ジフェニルアミン骨格を用いたER リガンドの創薬2008
- Author(s)
  千葉由紀、小川卓巳、太田公規、遠藤泰之
- Organizer
  第27回メディシナルケミストリーシンポジウム
- Place of Presentation
  大阪
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of halogenated carboranylphenols as estrogen receptor b selective ligands2008
- Author(s)
  Takumi Ogawa, Kiminori Ohta, Motoshi Miyazawa, Yasuyuki Endo
- Organizer
  13th International Conference on Boron Chemistry
- Place of Presentation
  Platja d'Aro, Spain
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Utility of boron cluster for drug design : Design of androgen receptor/ estrogen receptor dual ligands bearing carborane for anti-prostate cancer drug2008
- Author(s)
  Yasuyuki Endo
- Organizer
  13th International Conference on Boron Chemistry (Keynote Lecture)
- Place of Presentation
  Platja d'Aro, Spain
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Diarylcarborane 構造を利用したエストロゲン活性および抗アンドロゲン活性を併せ持つ化合物の創製2008
- Author(s)
  太田公規,後藤徳仁,小川卓巳,藤井晋也,鈴木智晴,太田茂,遠藤泰之
- Organizer
  第19回日本レチノイド研究会学術集会
- Place of Presentation
  東京
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] ジフェニルアミン骨格を有するエストロゲン受容体(ER)制御化合物の構造活性相関2008
- Author(s)
  千葉由紀、小川卓巳、太田公規、遠藤泰之
- Organizer
  第128回日本薬学会年会
- Place of Presentation
  横浜
- Year and Date
  2008-03-29
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] カルボラン骨格を利用したアンドロゲン受容体変異に対しても有効な拮抗剤の創製2008
- Author(s)
  太田公規、後藤徳仁、藤井晋也、鈴木智晴、太田茂、遠藤泰之
- Organizer
  第27回メディシナルケミストリーシンポジウム
- Place of Presentation
  大阪
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Utility of boron cluster for drug design:Design of androgen receptor/ estrogen receptor dual ligands bearing carborane for anti-prostate cancer drug2008
- Author(s)
  Yasuyuki Endo , Tokuhito Goto, Kiminori Ohta, Shinya Fujii, Hiroyuki Kagechika
- Organizer
  13th International Conferenceon Boron Chemistry
- Place of Presentation
  Platja d'Aro, Spain
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Androgen receptor antagonists based on boron cluster as a hydrophobic core structure2008
- Author(s)
  Shinya Fujii, Kiminori Ohta, Tokuhito Goto, Tomoharu Suzuki, Shigeru Ohta, Yuichi Hashimoto, Hiroyuki Kagechika, Yasuyuki Endo
- Organizer
  13th International Conference on Boron Chemistry
- Place of Presentation
  Platja d'Aro, Spain
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] Design and Synthesis of halogenated carboranylphenols as estrogen receptor β selective ligands.2008
- Author(s)
  小川卓巳, 太田公規, Miyazawa, M., 遠藤泰之
- Organizer
  13th International Conference on Boron Chemistry
- Place of Presentation
  Platja d'Aro, Spain.
- Year and Date
  2008-09-23
- Data Source
  KAKENHI-PROJECT-20390035
[Presentation] 球状疎水性分子とシクロデキストリンにおける相互作用の解析2007
- Author(s)
  遠藤泰之
- Organizer
  日本化学会第87春季年会
- Place of Presentation
  大阪
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Application of Inorganic Boron Cluster, Carboranes for Medicinal Drug Design2006
- Author(s)
  Yasuyuki, Endo
- Organizer
  Department of Chemistry, University of Washington
- Place of Presentation
  Seattle, WA, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Potent Estrogen Receptor Modulators Based on 3-Dimensional Hydropho bic Core Structure2006
- Author(s)
  Endo, Y.
- Organizer
  The 30th National Medicinal Chemistry Symposium
- Place of Presentation
  Seattle,WA,US
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 薬物受容体の形状認識に焦点を当てた新規立体的疎水性構造単位の開発と応用2006
- Author(s)
  遠藤泰之
- Organizer
  Department of Chemistry, Washington University
- Place of Presentation
  Seattle,WA,US
- Year and Date
  2006-06-29
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Potent Estrogen Receptor Modulators Based on 3-Dimensional Hydrophobic Core Structure2006
- Author(s)
  Endo, Y., Ogawa, T., Yoshimi, T., Ohta, K., Suzuki, T., Ohta, S
- Organizer
  The 30th National Medicinal Chemistry Symposium
- Place of Presentation
  Seattle, WA, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 薬物受容体の形状認識に焦点を当てた新規立体的疎水性構造単位の開発と応用2005
- Author(s)
  遠藤泰之
- Organizer
  東レ医薬研究所
- Place of Presentation
  鎌倉
- Year and Date
  2005-12-09
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 薬物-受容体の形状認識に焦点を当てた新規立体的疎水性構造単位の開発と応用2005
- Author(s)
  遠藤泰之
- Organizer
  日本薬学会北海道支部大会特別講演会
- Place of Presentation
  札幌
- Year and Date
  2005-12-03
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Application of Inorganic Boron Cluster, Carboranes for Medicinal Drug Design2005
- Author(s)
  Yasuyuki, Endo
- Organizer
  Department of Chemistry, University of Utah
- Place of Presentation
  Salt Lake City, UT, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Structure-activity study of nuclear androgen receptor(AR) antagonistd bearing carborane as a hydrophobic pharmacophore2005
- Author(s)
  Goto, T., Ohta, K., Endo, Y., Suzuki, T., Ohta, S
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 受容体構造に基づく新規坑エストロゲン薬、坑アンドロゲン薬の創製2005
- Author(s)
  遠藤泰之
- Organizer
  東北薬科大学生涯教育セミナー
- Place of Presentation
  仙台
- Year and Date
  2005-11-19
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 1-Aryl-1, 2-dicarba-closo-dodecaboranes : Evaluation of the ability of intranolecular C-H-O hydrogen bonds in solution2005
- Author(s)
  Ohta, K., Yamazaki, H., Endo, Y
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Application of Inorganic Boron Cluster, Carboranes for Medicinal Drug Design2005
- Author(s)
  Yasuyuki, Endo
- Organizer
  Department of Chemistry, Vanderbilt University
- Place of Presentation
  Nashville, TN, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Design, Synthesis and biological evaluation of estrogen receptor modulators with m-carborane as a hydrophobic pharmacophore2005
- Author(s)
  Ogawa, T., Ohta, K., Endo, Y., Suzuki, T., Ohta, S
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] The effect of the linking group on mesogenic properties of three-ring mesegenic derivatives of p-carborane2005
- Author(s)
  Nagamine, T., Ohta, K., Endo. Y., Januszko, A., Kaszynski, P
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 薬物受容体の形状認識に焦点を当てた新規立体的疎水性構造単位の開発と応用2005
- Author(s)
  遠藤泰之
- Organizer
  東京医科歯科大学
- Place of Presentation
  東京
- Year and Date
  2005-03-11
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Application of Inorganic Boron Cluster,Carboranes for Medicinal Drug Design2005
- Author(s)
  Yasuyuki Endo
- Organizer
  Department of Chemistry, Vanderbilt University
- Place of Presentation
  Nashville,TN,US
- Year and Date
  2005-07-06
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Identification of A Possible Intermediate for the Deboronation of ortho-Carborane2005
- Author(s)
  Taoda, Y., Endo, Y., Yamaguchi, K., Kagechika, H
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Regioselective iodination of o-carborane and construction of carboracycle utilyzed acidity of o-carborane C-Ht2005
- Author(s)
  Yamazaki, H., Ohta, K., Endo, Y
- Organizer
  The 12th International Conference on Boron Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] New Estrogen Receptor Modulators Bearing Carborane As A Hydrophobic Skeletal Structure2004
- Author(s)
  Endo Y, Yoshimi, T., Ohta, K., Miyaura, C
- Organizer
  The 7th French-Japanese Symposium on Medicinal and Fine Chemistry
- Place of Presentation
  Sendai, Japan
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] 球状疎水性構造を基本骨格とした選択的エストロゲン受容体リガンドの設計、合成と活性評価2004
- Author(s)
  遠藤泰之
- Organizer
  第23回メディシナルケミストリーシンポジウム/第12回日本薬学会医薬化学部会年会
- Place of Presentation
  つくば
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Construction of Three-dimensional Structures Based on Globular Icosahedral Carboranes and Planar Aromatic Species2004
- Author(s)
  Endo, Y
- Organizer
  70th Birthday Symposium for Leo Paquette
- Place of Presentation
  Columbus, OH, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Distorted Molecules Based on Spatial Definition of Carboranes2004
- Author(s)
  Endo, Y.
- Organizer
  The 3rd European Meeting on Boron Chemistry
- Place of Presentation
  Prague,Czech Republic
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Construction of Three-dimensional Structures Based on Globular Icosahedral Carboranes and Planar Aromatic Species2004
- Author(s)
  Endo, Y.
- Organizer
  70th Birthday Symposium for Leo Paquette
- Place of Presentation
  Columbus,OH US
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Utility of Boron Clusters for Drug Design. QSAR between Estrogen Receptor Binding Affinity and Hydrophobicity of Carboranylphenols2004
- Author(s)
  Ohta, K., Yamamoto, K., Endo, Y
- Organizer
  29th National Medicinal Chemistry Symposium
- Place of Presentation
  Madison, WI, US
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] New Estrogen Receptor Modulators Bearing Carborane As A Hydrophobic Skeletal Structure2004
- Author(s)
  Endo, Y.
- Organizer
  The 7th French-Japanese Symposium on Medicinal and Fine Chemistry
- Place of Presentation
  Sendai
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] Distorted Molecules Based on Spatial Definition of Carboranes2004
- Author(s)
  Endo, Y., Songkram, C., Ohta, K., Yamaguchi, K
- Organizer
  The 3rd European Meeting on Boron Chemistry
- Place of Presentation
  Prague, Czech Republic
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-16390032
[Presentation] トロポロン誘導体の抗腫瘍活性における構造活性相関
- Author(s)
  太田公規、皆瀬麻子、遠藤泰之
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] m-カルボランを中心骨格とする新規抗腫瘍性化合物の開発
- Author(s)
  皆瀨麻子, 遠藤泰之
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 硫黄含有複素環を用いた新規エストロゲン受容体リガンドの探索
- Author(s)
  青砥沙也加、田口史, 皆瀨麻子, 太田公規, 遠藤泰之
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] カルボラニルフェノールグリセロール誘導体の抗アンドロゲン活性とその構造活性相関
- Author(s)
  皆瀬麻子、阿部孝俊、太田公規、小田彰史、遠藤泰之
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 新規アゾトロポロン誘導体の細胞増殖抑制活性
- Author(s)
  太田公規, 皆瀨麻子, 遠藤泰之
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] 含硫黄複素環を有する新規エストロゲン受容体リガンドの合成と活性評価
- Author(s)
  青砥沙也加、田口史、皆瀨麻子、太田公規、遠藤泰之
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-26460151
[Presentation] サブタイプ選択性を有したSERM を目指したジフェニルメタン誘導体の疎水性構造変換
- Author(s)
  小島友寛、佐藤学、小川卓巳、太田公規、遠藤泰之
- Organizer
  日本薬学会第135年会
- Place of Presentation
  神戸
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-26460151

1. SHUDO Koichi (50012612)

# of Collaborated Projects: 16 results

# of Collaborated Products: 0 results
2. KAGECHIKA Hiroyuki (20177348)

# of Collaborated Projects: 15 results

# of Collaborated Products: 9 results
3. OHWADA Tomohiko (20177025)

# of Collaborated Projects: 9 results

# of Collaborated Products: 0 results
4. HASHIMOTO Yuichi (90164798)

# of Collaborated Projects: 9 results

# of Collaborated Products: 1 results
5. OHTA Kiminori (90347906)

# of Collaborated Projects: 5 results

# of Collaborated Products: 128 results
6. INOMATA Kohei (60221785)

# of Collaborated Projects: 4 results

# of Collaborated Products: 2 results
7. NAGASAWA Kazuo (10247223)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
8. SODEOKA Mikiko (60192142)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
9. FUJII Shinya (60389179)

# of Collaborated Projects: 1 results

# of Collaborated Products: 17 results
10. FABIO Pichierri (40374920)

# of Collaborated Projects: 1 results

# of Collaborated Products: 3 results
11. TAN-NO Koichi (20207260)

# of Collaborated Projects: 1 results

# of Collaborated Products: 5 results
12. NAKAGAWASAI Osamu (50296018)

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
13. ODASHIMA Kazunori (30152507)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
14. HIGUCHI Tsunehiko (50173159)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
15. NOGUCHI Hiroshi (60126141)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
16. ITAI Akiko (60012647)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
17. TOMIOKA Nobuo (20202202)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
18. IWAI Yuzuru (70099977)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
19. MIYACHI Hiroyuki (20376643)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
20. TANATANI Aya (40361654)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
21. OHNO Masaji (00111550)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
22. IITAKA Yoichi (90012591)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
23. KOGA Kenji (10012600)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
24. SANKAWA Ushio (60012613)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
25. 小林久芳 (80225531)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
26. 小磯邦子 (50092200)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
27. 斉藤昭一 (80231330)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
28. 浦野泰照 (20292956)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
29. 皆瀬麻子 (30710397)

# of Collaborated Projects: 1 results

# of Collaborated Products: 8 results
30. IMANARI Mamoru

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
31. 張ヶ谷泰二

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
32. ODA Akifumi

# of Collaborated Projects: 0 results

# of Collaborated Products: 2 results
33. TOKURAKU Kiyotaka

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
34. HAYASHI Takafumi

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
35. 上井幸司

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
36. 根本亙

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
37. 小野木弘志

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

ENDO Yasuyuki 遠藤 泰之

遠藤 康之

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A New Development of Molecular Design Utilizing Novel Hydrophobic StructuresPrincipal Investigator

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Development of Receptor Regulators Utilizing Novel HydrophobicStructure and Its Application for Medicinal Drug DesignPrincipal Investigator

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Development and Application of Novel 3-Dimensional Hydrophobic Structures for Drug Design, Which Are Focused on Molecular Recognition between Ligand and ReceptorPrincipal Investigator

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Study on Electronic and Steric Effects of Boron Cluster and Application for Construction of Functional Molecules.Principal Investigator

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Design and Synthesis of Cellular Signal Transduction Modulator, Benzolactam Derivatives and Related CompoundsPrincipal Investigator

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ヘテロ原子間結合の開裂による[3,3]シグマトロピック転位反応の新展開Principal Investigator

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発癌プロモーターの活性発現構造解析を目指す分子設計と合成Principal Investigator

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Design, Synthesis and Biological Activity of Anti-HIV Compounds Derived from TeleocidinsPrincipal Investigator

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分子設計と合成による発癌プロモーターの活性発現構造の一般性の確立Principal Investigator

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ENDO Yasuyuki 遠藤泰之

遠藤康之