Oishi Shinya 大石真也

… Alternative Names

OISHI Shinya 大石真也

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Researcher Number	80381739
Other IDs	https://orcid.org/0000-0002-2833-2539
Affiliation (Current)	2024: 京都薬科大学, 薬学部, 教授
Affiliation (based on the past Project Information) *help	2019 – 2024: 京都薬科大学, 薬学部, 教授 2015 – 2018: 京都大学, 薬学研究科, 准教授 2017: 京都大学, 薬学部, 准教授 2016 – 2017: 京都大学, 大学院薬学研究科, 准教授 2015: 京都大学, 薬学研究科, 助教授 … More 2013 – 2014: 京都大学, 大学院薬学研究科, 講師 2011 – 2014: 京都大学, 薬学研究科(研究院), 講師 2013: 京都大学, 薬学研究科, 講師 2011: 京都大学, 薬学研究科, 講師 2009: Kyoto University, 薬学研究科, 講師 2007 – 2008: Kyoto University, Graduate School of Pharmaceutical Sciences, Assistant Professor 2005 – 2006: 京都大学, 薬学研究科, 助手 2005: 静岡県立大学, 薬学研究科, 講師 Less
Review Section/Research Field	Principal Investigator Drug development chemistry / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Medium-sized Section 47:Pharmaceutical sciences and related fields / Medium-sized Section 37:Biomolecular chemistry and related fields / Chemical pharmacy Except Principal Investigator Drug development chemistry / Biological Sciences / Basic Section 52040:Radiological sciences-related / Basic Section 37010:Bio-related chemistry / Medium-sized Section 47:Pharmaceutical sciences and related fields … More / Medium-sized Section 49:Pathology, infection/immunology, and related fields / Broad Section F / General surgery / Polymer/Textile materials / Pathological medical chemistry / Radiation science / General physiology / Basic veterinary science/Basic zootechnical science / Chemical biology Less
Keywords	Principal Investigator スクリーニング / 鏡像型タンパク質 / ペプチド / モダリティ / 抗体様分子 / 医薬品探索 / 天然物 / 創薬 / キラル化合物 / ケモカイン … More / HIV / 酵素 / 機能分子 / 化学合成タンパク質 / 抗菌薬 / 抗ウイルス薬 / BIRドメイン / カスパーゼ / SH2ドメイン / 薬らしさ / 全合成 / 二次代謝産物 / プローブ / 受容体 / ニューロキニン / GPR54 / キスペプチン / 性ホルモン / 構造活性相関 / CXCR4 / キナーゼ / 抗がん剤 / シグナル伝達 / HIV-1 / 化学合成ペプチド / gp41 / 抗HIV剤 / 膜融合 / 蛋白質-蛋白質相互作用 … More Except Principal Investigator CXCR4 / 癌 / ケモカイン / ペプチド / GPCR / 構造活性相関 / ファージディスプレイ / 抗体 / 創薬 / PDT / PET / T140 / スクリーニング / プローブ / activity-based probe / 脱ユビキチン化酵素 / ユビキチン / GPR54 / ACKR3 / ラジオセラノスティクスプローブ / ケモカイン受容体 / 免疫原性 / CDR / Nanobody / ヘリックス / 膜融合 / SARS-CoV-2 / 前腹側室周囲核（AVPV） / 弓状核 / 黄体形成ホルモン（LH） / 性腺刺激ホルモン放出ホルモン（GnRH） / 生殖中枢キスペプチンニューロン / 家畜の繁殖促進技術 / 卵胞発育・排卵制御 / 家畜（ウシ・ヤギ） / 遺伝子改変ラット / 視床下部 / エストロゲン / キスペプチン / KSP / 末梢神経障害 / 微小管阻害薬 / 乳癌 / kinesin spindle protein / 環状ペプチド / キナーゼ / 合理的分子設計 / 創薬テンプレート / 複素環 / 化学合成 / 合成化学 / キャプシド / 低分子化合物スクリーニング / 化合物スクリーニング / TBP-2 / イノベーション / アルファアレスチン / 癌抑制 / ケミカルバイオロジー / 低分子化合物 / インスリン抵抗性 / 糖尿病 / Txnip / animal / membrane potential / Cell line / SPEC / Oxygen effect / Tumor / 動物 / 膜電位 / 腫瘍細胞 / SPECT / 酸素効果 / ガン / G-protein coupled receptor / chemical proteomics / Seven transmembrane protein / Intein-splicing system / Bioluminescece Resonance Energy Transfer / 非ペプチド化 / GPR-54 / 光感受性保護基 / Cysteine-ligation / 7TMGPCR / ケミカルプロテオミクス / 7回膜貫通型受容体 / システインプロテアーゼ / 天然有機化合物 / 鏡像体 / 生物活性化合物 / アッセイ / 化合物ライブラリー / 天然物 / 性腺刺激ホルモン放出ホルモン / G蛋白質共役型受容体 / 性腺刺激ホルモン放出ホルモン / ラット / LH / GnRH / 神経ペプチド / activety-based probe / プロテオミクス解析 / アクティビティーベースドプローブ / プロテアーゼ / ユビキチン様ドメイン / 酸化ストレス / 活性制御 / 薬剤耐性 / kisspeptin / SDF-1 Less

Development of a low-molecular-weight antibody library and its application in mirror-image screening
- Principal Investigator
  
  野中元裕
- Project Period (FY)
  2024 – 2027
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 37010:Bio-related chemistry
- Research Institution
  Kyoto University
ケモカイン受容体を標的としたラジオセラノスティクスプローブの開発
- Principal Investigator
  
  木村寛之
- Project Period (FY)
  2024 – 2026
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 52040:Radiological sciences-related
- Research Institution
  Kanazawa University
Development of Platform Technlogy for Therapeutic Applications of Mirror-image Functional ProteinsPrincipal Investigator
- Principal Investigator
  
  大石真也
- Project Period (FY)
  2024 – 2026
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 47:Pharmaceutical sciences and related fields
- Research Institution
  Kyoto Pharmaceutical University
Development of antibody-mimetic libraries by CDR grafting
- Principal Investigator
  
  野中元裕
- Project Period (FY)
  2022 – 2023
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 47:Pharmaceutical sciences and related fields
- Research Institution
  Kyoto University
Development of mirror-image antibody-like scaffolds and their applicationsPrincipal Investigator
- Principal Investigator
  
  大石真也
- Project Period (FY)
  2022 – 2025
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Kyoto Pharmaceutical University
Exploration of estrogen feedback mechanisms regulating animal reproduction to improve the methods controlling ovulation and follicle development in domestic animals
- Principal Investigator
  
  束村博子
- Project Period (FY)
  2021 – 2025
- Research Category
  
  Grant-in-Aid for Scientific Research (S)
- Review Section
  
  Broad Section F
- Research Institution
  Nagoya University
コロナウイルス制圧のための新規膜融合阻害ペプチドの創出と合理的な設計法の確立
- Principal Investigator
  
  児玉栄一
- Project Period (FY)
  2021 – 2023
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 49:Pathology, infection/immunology, and related fields
- Research Institution
  Tohoku University
Development of Screening Platform for Mirror-image Antibody-like ScaffoldsPrincipal Investigator
- Principal Investigator
  
  Oishi Shinya
- Project Period (FY)
  2020 – 2022
- Research Category
  
  Grant-in-Aid for Challenging Research (Exploratory)
- Review Section
  
  Medium-sized Section 37:Biomolecular chemistry and related fields
- Research Institution
  Kyoto Pharmaceutical University
Development of Drug Discovery Technologies Using Mirror-image BiomoleculesPrincipal Investigator
- Principal Investigator
  
  Oishi Shinya
- Project Period (FY)
  2018 – 2021
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Review Section
  
  Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
- Research Institution
  Kyoto Pharmaceutical University
  Kyoto University
Develoment of a screening platform using mirror-image proteins and their application to drug discoveryPrincipal Investigator
- Principal Investigator
  
  Shinya Oishi
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Studies toward a synthesis of virus capsids
- Principal Investigator
  
  Chihiro Tsukano
- Project Period (FY)
  2015 – 2016
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Polymer/Textile materials
- Research Institution
  Kyoto University
Development of Novel Drug Discovery Technologies for Target Proteins with Elusive Molecular Basis
- Principal Investigator
  
  Fujii Nobutaka
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Potential new chemotherapy for breast cancer therapy with a novel KSP inhibitor
- Principal Investigator
  
  Ohta Yuki
- Project Period (FY)
  2015 – 2017
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  General surgery
- Research Institution
  St. Marianna University School of Medicine
Elucidation of the molecular mechanism of insulin resistance by investigating TBP-2/Txnip and chemical biology
- Principal Investigator
  
  MASUTANI Hiroshi
- Project Period (FY)
  2013 – 2015
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Pathological medical chemistry
- Research Institution
  Kyoto University
A new concept for drug discovery from peptide natural productsPrincipal Investigator
- Principal Investigator
  
  OISHI Shinya
- Project Period (FY)
  2012 – 2014
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Chemical pharmacy
- Research Institution
  Kyoto University
Development and application of a novel screening technolgy toward effective uses of chemical library
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2012 – 2014
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Mechanism of unanchored polyubiquitin chain production
- Principal Investigator
  
  HATTORI Akira
- Project Period (FY)
  2012 – 2013
- Research Category
  
  Grant-in-Aid for Challenging Exploratory Research
- Research Field
  
  General physiology
- Research Institution
  Kyoto University
Biochemical and physiological studies on deubiquitinating enzymes based on an analysis of the enzymatic activity dynamics
- Principal Investigator
  
  HATTORI Akira
- Project Period (FY)
  2011 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Chemical biology
- Research Institution
  Kyoto University
Expression profiles of G-protein coupled receptors in gonadotropin-releasing hormone neurons
- Principal Investigator
  
  UENOYAMA Yoshihisa
- Project Period (FY)
  2011 – 2013
- Research Category
  
  Grant-in-Aid for Scientific Research (C)
- Research Field
  
  Basic veterinary science/Basic zootechnical science
- Research Institution
  Nagoya University
Investigation on the molecular basis of neuropeptide receptors for the regulation of reproductive systemsPrincipal Investigator
- Principal Investigator
  
  OISHI Shinya
- Project Period (FY)
  2011 – 2014
- Research Category
  
  Grant-in-Aid for Young Scientists (A)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
多重標的創薬概念に基づくがん化学療法の新機軸Principal Investigator
- Principal Investigator
  
  大石真也, 藤井信孝
- Project Period (FY)
  2008 – 2009
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
GPCR周辺の細胞外環境解明のためのケミカルプローブの創出と応用Principal Investigator
- Principal Investigator
  
  大石真也, 藤井信孝
- Project Period (FY)
  2008 – 2009
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
Development of Novel Screening Systems for Receptor LigandsPrincipal Investigator
- Principal Investigator
  
  OISHI Shinya
- Project Period (FY)
  2008 – 2009
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
有機化学を基盤にしたGPCR細胞外環境のケミカルバイオロジー研究
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2006 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research on Priority Areas
- Review Section
  
  Biological Sciences
- Research Institution
  Kyoto University
蛋白質-蛋白質相互作用阻害剤の探索を指向した新規化合物評価システムの開発Principal Investigator
- Principal Investigator
  
  大石真也
- Project Period (FY)
  2005 – 2007
- Research Category
  
  Grant-in-Aid for Young Scientists (B)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Evolution of Drug Discovery Targeting for G-protein Coupled Receptors
- Principal Investigator
  
  FUJII Nobutaka
- Project Period (FY)
  2005 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research (A)
- Research Field
  
  Drug development chemistry
- Research Institution
  Kyoto University
Development of novel evaluation system and radiopharmaceutical for prediction of tumor treatment effect ; especially oxygen effect of tumor therapy
- Principal Investigator
  
  MAGATA Yasuhiro
- Project Period (FY)
  2005 – 2007
- Research Category
  
  Grant-in-Aid for Scientific Research (B)
- Research Field
  
  Radiation science
- Research Institution
  Hamamatsu University School of Medicine

[Book] インシリコ創薬科学2008
- Author(s)
  大石真也、藤井信孝、他
- Total Pages
  210
- Publisher
  京都廣川書店
- Data Source
  KAKENHI-PROJECT-20015021
[Book] インシリコ創薬科学2008
- Author(s)
  大石真也, 他
- Total Pages
  210
- Publisher
  京都廣川書店
- Data Source
  KAKENHI-PROJECT-20790098
[Book] インシリコ創薬科学2008
- Author(s)
  大石真也、藤井信孝、他
- Total Pages
  210
- Publisher
  京都廣川書店
- Data Source
  KAKENHI-PROJECT-20057011
[Book] ケミカルバイオロジーを基盤とするペプチド創薬2007
- Author(s)
  大石真也, 他
- Total Pages
  5
- Publisher
  メディカルドゥ
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Book] ペプチドをリードとした創薬蛋白質核酸酵素増刊ケミカルバイオロジー2007
- Author(s)
  大石真也, 他
- Total Pages
  6
- Publisher
  共立出版
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Book] インシリコ創薬科学(3.2節・3.3節)
- Author(s)
  掛谷秀昭、大石真也、矢倉徹、藤井信孝
- Publisher
  京都廣川書店
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Interferon lambda 3 in the early phase of coronavirus disease-19 can predict disease progression.2022
- Author(s)
  Tetsuya Suzuki. Noriko Iwamoto, Shinya Tsuzuki, Yuko Kakumoto, Michiyo Suzuki, Shinobu Ashida, et. al.
- Journal Title
  
  European Journal of Clinical Investigation
  
  Volume: 52 Issue: 9
- DOI
  10.1111/eci.13808
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-21K19366
[Journal Article] 化学合成タンパク質を利用したスクリーニング技術の開発 ―鏡の中に存在する化合物リソースの創薬研究への応用―2021
- Author(s)
  大石真也
- Journal Title
  
  京都薬科大学紀要
  
  Volume: 2 Issue: 2 Pages: 123-133
- DOI
  10.34445/00000277
- NAID
  120007183926
- ISSN
  2435-4112
- URL
  https://kyoto-phu.repo.nii.ac.jp/records/297
- Year and Date
  2021-11-30
- Language
  Japanese
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-20K21252, KAKENHI-PROJECT-18H02555
[Journal Article] Design of Coibamide A Mimetics with Improved Cellular Bioactivity2021
- Author(s)
  Kitamura Takashi、Suzuki Rikito、Inuki Shinsuke、Ohno Hiroaki、McPhail Kerry L.、Oishi Shinya
- Journal Title
  
  ACS Medicinal Chemistry Letters
  
  Volume: 13 Issue: 1 Pages: 105-110
- DOI
  10.1021/acsmedchemlett.1c00591
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Journal Article] Through the looking glass, and the drug candidates to be found there2021
- Author(s)
  大石真也
- Journal Title
  
  MEDCHEM NEWS
  
  Volume: 31 Issue: 3 Pages: 143-146
- DOI
  10.14894/medchem.31.3_143
- NAID
  130008070858
- ISSN
  2432-8618, 2432-8626
- Year and Date
  2021-08-01
- Language
  Japanese
- Data Source
  KAKENHI-PROJECT-20K21252, KAKENHI-PROJECT-18H02555
[Journal Article] Coibamide A Targets Sec61 to Prevent Biogenesis of Secretory and Membrane Proteins2020
- Author(s)
  Tranter Dale、Paatero Anja O.、Kawaguchi Shinsaku、Kazemi Soheila、Serrill Jeffrey D.、Kellosalo Juho、Vogel Walter K.、Richter Uwe、Mattos Daphne R.、Wan Xuemei、Thornburg Christopher C.、Oishi Shinya、McPhail Kerry L.、Ishmael Jane E.、Paavilainen Ville O.
- Journal Title
  
  ACS Chemical Biology
  
  Volume: 15 Issue: 8 Pages: 2125-2136
- DOI
  10.1021/acschembio.0c00325
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Journal Article] Isoform-selective regulation of mammalian cryptochromes2020
- Author(s)
  Miller Simon、Son You Lee、Aikawa Yoshiki、Makino Eri、Nagai Yoshiko、Srivastava Ashutosh、Oshima Tsuyoshi、Sugiyama Akiko、Hara Aya、Abe Kazuhiro、Hirata Kunio、Oishi Shinya、Hagihara Shinya、Sato Ayato、Tama Florence、Itami Kenichiro、Kay Steve A.、Hatori Megumi、Hirota Tsuyoshi
- Journal Title
  
  Nature Chemical Biology
  
  Volume: - Issue: 6 Pages: 676-685
- DOI
  10.1038/s41589-020-0505-1
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18K19171, KAKENHI-PROJECT-18H02555, KAKENHI-PROJECT-19H05463, KAKENHI-PROJECT-17H03653, KAKENHI-PROJECT-18H02402, KAKENHI-PROJECT-18K06316, KAKENHI-PROJECT-19K22693, KAKENHI-PROJECT-19H03266
[Journal Article] Development of Mirror-Image Screening Systems for XIAP BIR3 Domain Inhibitors2019
- Author(s)
  Shu Keitou、Iwamoto Naoya、Honda Kaori、Kondoh Yasumitsu、Hirano Hiroyuki、Osada Hiroyuki、Ohno Hiroaki、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  Bioconjugate Chemistry
  
  Volume: 30 Issue: 5 Pages: 1395-1404
- DOI
  10.1021/acs.bioconjchem.9b00154
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18K05366, KAKENHI-PLANNED-18H05503, KAKENHI-PROJECT-18H02555
[Journal Article] Scaffold hopping of fused piperidine-type NK3 receptor antagonists to reduce environmental impact2019
- Author(s)
  Yamamoto Koki、Inuki Shinsuke、Ohno Hiroaki、Oishi Shinya
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 印刷中 Issue: 10 Pages: 2019-2026
- DOI
  10.1016/j.bmc.2019.03.059
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17J10582, KAKENHI-PROJECT-18H02555
[Journal Article] Synthesis of Triazolo- and Oxadiazolopiperazines by Gold(I)-Catalyzed Domino Cyclization: Application to the Design of a Mitogen Activated Protein (MAP) Kinase Inhibitor2018
- Author(s)
  Yamamoto Koki、Yoshikawa Yasushi、Ohue Masahito、Inuki Shinsuke、Ohno Hiroaki、Oishi Shinya
- Journal Title
  
  Organic Letters
  
  Volume: 21 Issue: 2 Pages: 373-377
- DOI
  10.1021/acs.orglett.8b03500
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17J10582, KAKENHI-PROJECT-18H02555
[Journal Article] Easy-to-Attach/Detach Solubilizing-Tag-Aided Chemical Synthesis of an Aggregative Capsid Protein2018
- Author(s)
  Tsuda Shugo、Mochizuki Masayoshi、Ishiba Hiroyuki、Yoshizawa-Kumagaye Kumiko、Nishio Hideki、Oishi Shinya、Yoshiya Taku
- Journal Title
  
  Angewandte Chemie International Edition
  
  Volume: 57 Issue: 8 Pages: 2105-2109
- DOI
  10.1002/anie.201711546
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15H04653
[Journal Article] Head-to-Tail Macrocyclization of Cysteine-Free Peptides Using an o-Aminoanilide Linker2018
- Author(s)
  T. Ohara, M. Kaneda, T. Saito, N. Fujii, H. Ohno, S. Oishi
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 28 Issue: 8 Pages: 1283-1286
- DOI
  10.1016/j.bmcl.2018.03.027
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-15J05499
[Journal Article] Synthesis of Jaspine B Regioisomers through Palladium-Catalyzed Stereoselective Tetrahydrofuran Formation: Insight into the Ligand Recognition of Sphingosine Kinases2018
- Author(s)
  Miyagawa, S. Inuki, M. Honda, S. Nakamura, I. Nakanishi, N. Fujii, S. Oishi, H. Ohno
- Journal Title
  
  Tetrahdron
  
  Volume: 74 Issue: 15 Pages: 1802-1809
- DOI
  10.1016/j.tet.2018.02.042
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PUBLICLY-18H04408, KAKENHI-PROJECT-17H03971
[Journal Article] Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3)2018
- Author(s)
  Sekiguchi Haruka、Kuroyanagi Tomoko、Rhainds David、Kobayashi Kazuya、Kobayashi Yuka、Ohno Hiroaki、Heveker Nikolaus、Akaji Kenichi、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: 61 Issue: 8 Pages: 3745-3751
- DOI
  10.1021/acs.jmedchem.8b00336
- Peer Reviewed / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-16H05104
[Journal Article] Identification of Selective Inhibitors of Sphingosine Kinases 1 and 2 through a Structure-Activity Relationship Study of 4-epi-Jaspine B2017
- Author(s)
  H. Ohno, M. Honda, N. Hamada, J. Miyagaki, A. Iwata, K. Otsuki, T. Maruyama, S. Nakamura, I. Nakanishi, S. Inuki, N. Fujii, S. Oishi
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 25 Issue: 12 Pages: 3046-3052
- DOI
  10.1016/j.bmc.2017.03.059
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-17H03971
[Journal Article] Synthesis of Grb2 SH2 domain proteins for mirror-image screening systems.2017
- Author(s)
  Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S.
- Journal Title
  
  Bioconjugate Chemistry
  
  Volume: 28 Issue: 2 Pages: 609-619
- DOI
  10.1021/acs.bioconjchem.6b00692
- Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-26350976, KAKENHI-PROJECT-15H04653
[Journal Article] Synthesis of the Src SH2 domain and its application in bioassays for mirror-image screening2017
- Author(s)
  Shu Keitou、Noguchi Taro、Honda Kaori、Kondoh Yasumitsu、Osada Hiroyuki、Ohno Hiroaki、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  RSC Advances
  
  Volume: 7 Issue: 61 Pages: 38725-38732
- DOI
  10.1039/c7ra07445j
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-15H04653
[Journal Article] Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction.2017
- Author(s)
  Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S
- Journal Title
  
  Bioorg Med Chem Lett
  
  Volume: 印刷中 Issue: 11 Pages: 2571-2574
- DOI
  10.1016/j.bmcl.2017.03.082
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-26350976, KAKENHI-PROJECT-15H04653
[Journal Article] Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles2017
- Author(s)
  J. Matsuoka, Y. Matsuda, Y. Kawada, S. Oishi, H. Ohno
- Journal Title
  
  Angew. Chem. Int. Ed.
  
  Volume: 56 Issue: 26 Pages: 7444-7448
- DOI
  10.1002/anie.201703279
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-17H03971
[Journal Article] A Novel KSP Inhibitor, KPYB10602, Induces Mitotic Arrest and Cell Death in Breast Cancer Cells2016
- Author(s)
  Kojima-Tsuchiya Seiko, Ohta Yuki, Takenaga Mitsuko, Niimi Jun, Watanabe Daiki, Tsunoda Satoshi, Ootaki Masanori, Oishi Shinya, Fujii Nobutaka, Matsumoto Naoki, Tsugawa Koichiro
- Journal Title
  
  Journal of St.Marianna University
  
  Volume: 7 Pages: 105-116
- NAID
  130005251535
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-15K10074
[Journal Article] Development of novel NK3 receptor antagonists with reduced environmental impact2016
- Author(s)
  Yamamoto Koki、Okazaki Shiho、Ohno Hiroaki、Matsuda Fuko、Ohkura Satoshi、Maeda Kei-ichiro、Fujii Nobutaka、Oishi Shinya
- Journal Title
  
  Bioorganic & Medicinal Chemistry
  
  Volume: 24 Issue: 16 Pages: 3494-3500
- DOI
  10.1016/j.bmc.2016.05.054
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15H04654
[Journal Article] Screening of a virtual mirror-image library of natural products2016
- Author(s)
  T. Noguchi, S. Oishi, K. Honda, Y. Kondoh, T. Saito, H. Ohno, H. Osada, N. Fujii
- Journal Title
  
  Chem. Comm.
  
  Volume: 52 Issue: 49 Pages: 7653-7656
- DOI
  10.1039/c6cc03114e
- Peer Reviewed / Acknowledgement Compliant / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-26350976
[Journal Article] Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne2016
- Author(s)
  S. Naoe, Y. Yoshida, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  J. Org. Chem.
  
  Volume: 81 Issue: 13 Pages: 5690-5698
- DOI
  10.1021/acs.joc.6b00720
- NAID
  120006634624
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654
[Journal Article] Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization2016
- Author(s)
  D. Nishiyama, A. Ohara, H. Chiba, H. Kumagai, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 18 Issue: 7 Pages: 1670-1673
- DOI
  10.1021/acs.orglett.6b00536
- NAID
  120006634625
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Structure-Activity Relationship Study of 4-(Thiazol-5-yl)benzoic Acid Derivatives as Potent Protein Kinase CK2 Inhibitors2016
- Author(s)
  H. Ohno, D. Minamiguchi, S. Nakamura, K. Shu, S. Okazaki, M. Honda, R. Misu, H. Moriwaki, S. Nakanishi, S. Oishi, T. Kinoshita, I. Nakanishi, N. Fujii
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 24 Issue: 5 Pages: 1136-1141
- DOI
  10.1016/j.bmc.2016.01.043
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Enhanced antibody-mediated neutralization of HIV-1 variants that are resistant to fusion inhibitors2016
- Author(s)
  Alam, M., Kuwata, T., Shimura, K., Yokoyama, M., Ramirez Valdez, K. P., Tanaka, K., Maruta, Y., Oishi, S., Fujii, N., Sato, H., Matsuoka M. and Matsushita S.
- Journal Title
  
  Retrovirology
  
  Volume: 13 Issue: 1 Pages: 70-70
- DOI
  10.1186/s12977-016-0304-7
- NAID
  120005973385
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-26430091, KAKENHI-PROJECT-16K08824, KAKENHI-PROJECT-15H04654, KAKENHI-PROJECT-15H04870
[Journal Article] CXCL12/CXCR4 pathway is activated by oncogenic JAK2 in a PI3K-dependent manner2016
- Author(s)
  Abdelouahab Hadjer、Zhang Yanyan、Wittner Monika、Oishi Shinya、Fujii Nobutaka、Besancenot Rodolphe、Plo Isabelle、Ribrag Vincent、Solary Eric、Vainchenker William、Barosi Giovanni、Louache Fawzia
- Journal Title
  
  Oncotarget
  
  Volume: 8 Issue: 33 Pages: 54082-54095
- DOI
  10.18632/oncotarget.10789
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Journal Article] A Novel Peptide Derived from the Fusion Protein Heptad Repeat Inhibits Replication of Subacute Sclerosing Panencephalitis Virus In Vitro and In Vivo.2016
- Author(s)
  Watanabe M, Hashimoto K, Abe Y, Kodama EN, Nabika R, Oishi S, Ohara S, Sato M,Kawasaki Y, Fujii N, Hosoya M.
- Journal Title
  
  PLoS One.
  
  Volume: 11 Issue: 9 Pages: e0162823-e0162823
- DOI
  10.1371/journal.pone.0162823
- Peer Reviewed / Open Access / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-16H05346, KAKENHI-PROJECT-15H04654
[Journal Article] Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor2016
- Author(s)
  D. Nishiyama, Y. Sakai, H. Sekiguchi, H. Chiba, R. Misu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Chemical and Pharmaceutical Bulletin
  
  Volume: 64 Issue: 7 Pages: 996-1003
- DOI
  10.1248/cpb.c16-00302
- NAID
  130005160050
- ISSN
  0009-2363, 1347-5223
- Language
  English
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-15H04654
[Journal Article] Optimization of neurokinin-3 receptor (NK3R)-selective agonists2015
- Author(s)
  Yamamoto K, Oishi S, Misu R, Noguchi T, Ohno H, Yamamura T, Okamura H, Fujii N.
- Journal Title
  
  Peptide Science
  
  Volume: 2014 Pages: 241-242
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23689007
[Journal Article] Structure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists.2015
- Author(s)
  Misu R, Yamamoto K, Yamada A, Noguchi T, Ohno H, Yamamura T, Okamura H, Matsuda F, Ohkura S, Oishi S, Fujii N.
- Journal Title
  
  MedChemCommun
  
  Volume: 6 Issue: 3 Pages: 469-476
- DOI
  10.1039/c4md00514g
- Peer Reviewed / Open Access
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-24380154
[Journal Article] Development of a novel neurokinin-3 receptor selective agonist with highly biological stability2015
- Author(s)
  Misu R, Oishi S, Yamada A, Yamamoto K, Noguchi T, Ohno H, Yamamura T, Okamura H, Matsuda F, Ohkura S, Fujii N.
- Journal Title
  
  Peptide Science
  
  Volume: 2014 Pages: 23-24
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23689007
[Journal Article] Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group2015
- Author(s)
  M. Taguchi, Y. Tokimizu, S. Oishi, N. Fujii, H. Ohno
- Journal Title
  
  Org. Lett.
  
  Volume: 17 Issue: 24 Pages: 6250-6253
- DOI
  10.1021/acs.orglett.5b03254
- NAID
  120006634626
- Peer Reviewed / Acknowledgement Compliant / Open Access
- Data Source
  KAKENHI-PROJECT-15KT0061, KAKENHI-PROJECT-24689001, KAKENHI-PROJECT-15H04654
[Journal Article] Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation.2014
- Author(s)
  Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N.
- Journal Title
  
  J. Med. Chem.
  
  Volume: 57 Issue: 20 Pages: 8646-8651
- DOI
  10.1021/jm500771w
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07738, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-24380154
[Journal Article] A radiogallium-DOTA-based bivalent peptidic ligand targeting a chemokine receptor, CXCR4, for tumor imaging2014
- Author(s)
  Sano K, Masuda R, Hisada H, Oishi S, Shimokawa K, Ono M, Fujii N, Saji H, Mukai T.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 24 Issue: 5 Pages: 1386-1388
- DOI
  10.1016/j.bmcl.2014.01.031
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007
[Journal Article] Synthesis of IB-01212 by multiple N-methylations of peptide bonds.2014
- Author(s)
  Nabika R, Oishi S, Misu R, Ohno H, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 21 Pages: 6156-6162
- DOI
  10.1016/j.bmc.2014.08.036
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07872, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659004
[Journal Article] Design and synthesis of fluorescent probes for GPR54.2014
- Author(s)
  Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 22 Issue: 13 Pages: 3325-3330
- DOI
  10.1016/j.bmc.2014.04.052
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-26252046
[Journal Article] Synthesis and biological evaluation of the [D-MeAlall]-epimer of coibamide A.2014
- Author(s)
  Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 25 Issue: 2 Pages: 302-306
- DOI
  10.1016/j.bmcl.2014.11.044
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-14J07872, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659004
[Journal Article] Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes2013
- Author(s)
  Misu R, Oishi S, Setsuda S, Noguchi T, Kaneda M, Ohno H, Evans B, Navenot JM, Peiper SC, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett.
  
  Volume: 23 Issue: 9 Pages: 2628-2631
- DOI
  10.1016/j.bmcl.2013.02.098
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007
[Journal Article] Chronic Peripheral Administration of Kappa-Opioid Receptor Antagonist Advances Puberty Onset Associated with Acceleration of Pulsatile Luteinizing Hormone Secretion in Female Rats2013
- Author(s)
  中原辰夫
- Journal Title
  
  J. Reprod. Dev.
  
  Volume: 59 Issue: 5 Pages: 479-484
- DOI
  10.1262/jrd.2013-046
- NAID
  130003361050
- ISSN
  0916-8818, 1348-4400
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J05310, KAKENHI-PROJECT-23689007, KAKENHI-PLANNED-24108008
[Journal Article] Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists.2013
- Author(s)
  Misu R, Noguchi T, Ohno H, Oishi S, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 21 Issue: 8 Pages: 2413-2417
- DOI
  10.1016/j.bmc.2013.01.036
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J06309, KAKENHI-PROJECT-23689007
[Journal Article] Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors.2013
- Author(s)
  Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Kubo T, Kaneda M, Ohno H, Osada H, Fujii N
- Journal Title
  
  Bioorg Med Chem Lett
  
  Volume: 23 Issue: 13 Pages: 3802-3805
- DOI
  10.1016/j.bmcl.2013.04.094
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23510287, KAKENHI-PROJECT-24659046
[Journal Article] Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis2013
- Author(s)
  Yoshimitsu Y, Miyagaki J, Oishi S, Fujii N, Ohno H.
- Journal Title
  
  Tetrahedron
  
  Volume: 69 Issue: 21 Pages: 4211-4220
- DOI
  10.1016/j.tet.2013.03.091
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-24659046, KAKENHI-PROJECT-24689001, KAKENHI-PUBLICLY-24106720
[Journal Article] An optimized method of G-protein coupled receptor homology modeling: its application to the discovery of novel CXCR7 ligands2013
- Author(s)
  Yoshikawa Y, Oishi S, Kubo T, Tanahara N, Fujii N, Furuya T.
- Journal Title
  
  J. Med. Chem.
  
  Volume: 56 Issue: 11 Pages: 4236-4251
- DOI
  10.1021/jm400307y
- Peer Reviewed / Acknowledgement Compliant
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23689007
[Journal Article] Chronic peripheral administration of kappa-opioid receptor antagonist advances puberty onset associated with acceleration of pulsatile luteinizing hormone secretion in female rats2013
- Author(s)
  Nakahara T, Uenoyama Y, Iwase A, Oishi S, Nakamura S, Minabe S, Watanabe Y, Deura C, Noguchi T, Fujii N, Kikkawa F, Maeda K-I, Tsukamura H.
- Journal Title
  
  J Reprod Dev
  
  Volume: 59 Pages: 479-484
- NAID
  130003361050
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23580402
[Journal Article] Synthesis and functional analysis of deferriferrichrysin derivatives: application to colorimetric pH indicators2013
- Author(s)
  Kobayashi Y, Oishi S, Kobayashi K, Ohno H, Tsutsumi H, Hata Y, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 21 Issue: 14 Pages: 4296-4300
- DOI
  10.1016/j.bmc.2013.04.078
- NAID
  120005302101
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24659004
[Journal Article] Effects of Full-Length Kisspeptin Administration on Follicular Development in Japanese Black Beef Cows2013
- Author(s)
  Naniwa, Y., Nakatsukasa, K., Setsuda, S., Oishi, S., Fujii, N., Matsuda, F., Uenoyama, Y., Tsukamura, H., Maeda, K. -I. and Ohkura, S.
- Journal Title
  
  J. Reprod. Dev.
  
  Volume: 59 Issue: 6 Pages: 588-594
- DOI
  10.1262/jrd.2013-064
- NAID
  130003381852
- ISSN
  0916-8818, 1348-4400
- Language
  English
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-12J10489, KAKENHI-PROJECT-23658223, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-24380154
[Journal Article] Structure-Activity Relationship Study of a CXC Chemokine Receptor Type 4 Antagonist, FC131, Using a Series of Alkene Dipeptide Isosteres2012
- Author(s)
  Kobayashi K., et al
- Journal Title
  
  Journal of Medicinal Chemistry
  
  Volume: (in press) Issue: 6 Pages: 2746-2757
- DOI
  10.1021/jm2016914
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-10J02083, KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23570192, KAKENHI-PROJECT-23689007
[Journal Article] Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists.2012
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot J, Peiper S, Fujii N.
- Journal Title
  
  Bioconjug. Chem.
  
  Volume: 23 Issue: 6 Pages: 1259-1265
- DOI
  10.1021/bc300084h
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23659038, KAKENHI-PROJECT-23689007
[Journal Article] The metastasis suppressor KISS1 lacks antimetastatic activity in the C8161.9 xenograft model of melanoma2012
- Author(s)
  Navenot JM, Evans B, Oishi S, Setsuda S, Fujii N, Peiper SC.
- Journal Title
  
  Melanoma Res.
  
  Volume: 22 Issue: 2 Pages: 140-150
- DOI
  10.1097/cmr.0b013e328350fa07
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23689007
[Journal Article] Development and application of fluorescent SDF-1 derivatives2012
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N.
- Journal Title
  
  Future Med. Chem.
  
  Volume: 4 Issue: 7 Pages: 837-844
- DOI
  10.4155/fmc.12.31
- NAID
  120005285488
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23390025, KAKENHI-PROJECT-23590636, KAKENHI-PROJECT-23659038, KAKENHI-PROJECT-23689007
[Journal Article] Synthesis and Investigation of Novel Metal Complexes of Deferriferrichrysin2012
- Author(s)
  Kobayashi Y, Oishi S, Kobayashi K, Ohno H, Tsutsumi H, Hata Y, Fujii N.
- Journal Title
  
  Peptide Science
  
  Volume: 2012 Pages: 181-182
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-24659004
[Journal Article] CXCR4 stimulates macropinocytosis: implications for cellular uptake of arginine-rich cell-penetrating peptides and HIV2012
- Author(s)
  Gen Tanaka, Ikuhiko Nakase, et al.
- Journal Title
  
  Chemistry & Biology
  
  Volume: 19 Issue: 11 Pages: 1437-1446
- DOI
  10.1016/j.chembiol.2012.09.011
- Peer Reviewed
- Data Source
  KAKENHI-PUBLICLY-22121511, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-23790129, KAKENHI-PROJECT-24790099, KAKENHI-PROJECT-24791021
[Journal Article] Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR42011
- Author(s)
  Masuda R, Oishi S, Ohno H, Kimura H, Saji H, Fujii N.
- Journal Title
  
  Bioorg. Med. Chem.
  
  Volume: 19 Issue: 10 Pages: 3216-3220
- DOI
  10.1016/j.bmc.2011.03.059
- NAID
  120004770226
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23689007
[Journal Article] Kisspeptin neurons mediate reflex ovulation in the musk shrew (Suncus murinus)2011
- Author(s)
  Inoue N, Sasagawa K, Ikai K, Sasaki Y, Tomikawa J, Oishi S, Fujii N, Uenoyama Y, Ohmori Y, Yamamoto N, Hondo E, Maeda K, Tsukamura H.
- Journal Title
  
  Proc Natl Acad Sci U S A
  
  Volume: 108 Pages: 17527-17532
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23580402
[Journal Article] Kisspeptin neurons mediate reflex ovulation in the musk shrew (Suncus murinus).2011
- Author(s)
  Inoue, N. Sasagawa, K. Ikai, K. Sasaki, Y. Tomikawa, J. Oishi, S. Fujii, N. Uenoyama, Y. Ohmori, Y. Yamamoto, N. Hondo, E. Maeda, K. Tsukamura, H.
- Journal Title
  
  Proc Natl Acad Sci U S A.
  
  Volume: 108 Issue: 42 Pages: 17527-17532
- DOI
  10.1073/pnas.1113035108
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-23650233, KAKENHI-PROJECT-23689007, KAKENHI-PROJECT-23780292
[Journal Article] Fluorescent imaging of high grade bladder cancer using a specific antagonist for chemokine receptor CXCR42010
- Author(s)
  Nishizawa K, Oishi S, Fujii N, et al.
- Journal Title
  
  Int.J.Cancer
  
  Volume: 127 Pages: 1180-1187
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Fluorescent imaging of high grade bladder cancer using a specific antagonist for chemokine receptor CXCR42010
- Author(s)
  Nishizawa K, Oishi S, Fujii N, et al.
- Journal Title
  
  Int.J.Cancer
  
  Volume: 127 Pages: 1180-1187
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres2010
- Author(s)
  Narumi T, Ohno H, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 8 Pages: 616-621
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres.2010
- Author(s)
  Narumi T., Hayashi R., Tomita K., Kobayashi K., Tanahara N., Ohno H., Naito T., Kodama E., Matsuoka M., Oishi S., Fujii N.
- Journal Title
  
  Org.Biomol.Chem. 8(3)
  
  Pages: 616-621
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres2010
- Author(s)
  Narumi T, Ohno H, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 8 Pages: 616-621
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres2010
- Author(s)
  Narumi T, Ohno H, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 8 Pages: 616-621
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Chemokine receptor CXCR4 as a therapeutic target for neuroectodermal tumors2009
- Author(s)
  Hyunsuk S., Oishi S., Fujii N., et.al.
- Journal Title
  
  Semin. Cancer Biol 19
  
  Pages: 123-134
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] SDF-1/CXCR4 signaling is critical for the recruitment of mesenchymal stem cells to the fracture site during skeletal repair2009
- Author(s)
  Kitaori T., Oishi S., Fujii N., et.al.
- Journal Title
  
  Arthritis Rheum 60
  
  Pages: 813-823
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-ccopper-mediated SN2' alkylation2009
- Author(s)
  Kobayashi K, Oishi S, Ohno H, Fujii N, et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 4626-4629
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Chemokine receptor CXCR4 as a therapeutic target for neuroectodermal tumors.2009
- Author(s)
  Hyunsuk S., Oishi S., Fujii N.
- Journal Title
  
  Semin.Cancer Biol. 19(2)
  
  Pages: 123-134
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Prognostic value of metastin expression in human pancreatic cancer2009
- Author(s)
  Nagai K, Oishi S, Fujii N, et al.
- Journal Title
  
  J.Exp.Clin.Cancer Res.
  
  Volume: 28 Pages: 9-9
- NAID
  120004770245
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclicpentapeptide scaffold : the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids2009
- Author(s)
  Tanaka T, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem
  
  Volume: 7 Pages: 3805-3809
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution2009
- Author(s)
  Watabe T, Oishi S, et al.
- Journal Title
  
  J.Mol.Biol.
  
  Volume: 392 Pages: 657-665
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-ccopper-mediated SN2' alkylation2009
- Author(s)
  Kobayashi K, Oishi S, et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 4626-4629
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus.2009
- Author(s)
  Oishi S., Kodera Y., Nishikawa H., Kamitani H., Watabe T., Ohno H., Tochikura T., Shimane K., Kodama E., Matsuoka M., Mizukoshi F., Tsujimoto H., Fujii N.
- Journal Title
  
  Bioorg.Med.Chem. 17(14)
  
  Pages: 4916-4920
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group from recombinant protein.2009
- Author(s)
  Kajiwara K., Watanabe K., Tokiwa R., Kurose T., Ohno H., Tsutsumi H., Hata Y., Izumi K., Kodama E., Matsuoka M., Oishi S., Fujii N.
- Journal Title
  
  Bioorg.Med.Chem. 17(23)
  
  Pages: 7964-7970
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Prognostic value of metastin expression in human pancreatic cancer2009
- Author(s)
  Nagai K, Oishi S, Fujii N, et al.
- Journal Title
  
  J.Exp.Clin.Cancer Res.
  
  Volume: 28 Pages: 9-9
- NAID
  120004770245
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres : synthesis and bioevaluation of a-helical anti-HIV peptide analogues2009
- Author(s)
  Oishi S, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 7 Pages: 2872-2877
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcoholassisted nucleophilic trifluoromethylation and organozinc-ccopper-mediated SN2' alkylation2009
- Author(s)
  Kobayashi K, Oishi S, Ohno H, Fujii N, et al.
- Journal Title
  
  J.Org.Chem.
  
  Volume: 74 Pages: 4626-4629
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] SDF-1/CXCR4 signaling is critical for the recruitment of mesenchvmal stem cells to the fracture site during skeletal repair2009
- Author(s)
  Kitaori T., Oishi S., Fujii N., et.al.
- Journal Title
  
  Arthritis Rheum 60
  
  Pages: 813-823
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Expression of CXCR4, a G-protein-coupled receptor for CXCL12 in yeast identification of new-generation inverse agonists2009
- Author(s)
  Evans BJ, Oishi S, Fujii N, et al
- Journal Title
  
  Methods Enzymol.
  
  Volume: 460 Pages: 399-412
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus2009
- Author(s)
  Oishi S, et al.
- Journal Title
  
  Bioorg.Med.Chem.
  
  Volume: 17 Pages: 4916-4920
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres : synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues.2009
- Author(s)
  Oishi S., Kamitani H., Kodera Y., Watanabe K., Kobayashi K., Narumi T., Tomita K., Ohno H., Naito T., Kodama E., Matsuoka M., Fujii N.
- Journal Title
  
  Org.Biomol.Chem. 7(14)
  
  Pages: 2872-2877
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Structure-activity relationship study on polyglutamine binding peptide QBP12009
- Author(s)
  Tomita K, Oishi S, et al.
- Journal Title
  
  Bioorg.Med.Chem.
  
  Volume: 17 Pages: 1259-1263
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Expression of CXCR4, a G-protein-coupled receptor for CXCL12 in yeast identification of new-generation inverse agonists.2009
- Author(s)
  Evans B.J., Wang Z., Broach J.R., Oishi S., Fujii N., Peiper S.C.
- Journal Title
  
  Methods Enzymol. 460
  
  Pages: 399-412
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins2009
- Author(s)
  Tanaka M, Oishi S, et al.
- Journal Title
  
  Bioorg.Med.Chem.
  
  Volume: 17 Pages: 7487-7492
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold : the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids2009
- Author(s)
  Tanaka T, Oishi S, Fujii N, et al.
- Journal Title
  
  Org.Biomol.Chem.
  
  Volume: 7 Pages: 3805-3809
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyano-cysteine-mediated cleavages of recombinant proteins.2009
- Author(s)
  Tanaka M., Kajiwara K., Tokiwa R., Watanabe K., Ohno H., Tsutsumi H., Hata Y., Izumi K., Kodama E., Matsuoka M., Oishi S., Fujii N.
- Journal Title
  
  Bioorg.Med.Chem. 17(21)
  
  Pages: 7487-7492
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Expression of CXCR4, a G-protein-coupled receptor for CXCL12 in yeast identification of new-generation inverse agonists2009
- Author(s)
  Evans BJ, Oishi S, Fujii N, et al.
- Journal Title
  
  Methods Enzymol.
  
  Volume: 460 Pages: 399-412
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group2009
- Author(s)
  Kajiwara K, Oishi S, et al.
- Journal Title
  
  Bioorg.Med.Chem.
  
  Volume: 17 Pages: 7964-7970
- NAID
  120002098852
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Expression of CXCR4, a G-protein-coupled receptor for CXCL12 in yeast identification of new-generation inverse agonists2009
- Author(s)
  Evans BJ, Oishi S, Fujii N, et al.
- Journal Title
  
  Methods Enzymol.
  
  Volume: 460 Pages: 399-412
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Chemokine receptor CXCR4 as a therapeutic target for neuroectodermal tumors2009
- Author(s)
  Hyunsuk S., Oishi S., Fujii N., et.al.
- Journal Title
  
  Semin. Cancer Biol 19
  
  Pages: 123-134
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Clinical significance of plasma metastin level in pancreatic cancer patients2009
- Author(s)
  Katagiri F, Oishi S, Fujii N, et al.
- Journal Title
  
  Oncol.Rep.
  
  Volume: 21 Pages: 815-819
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Clinical significance of plasma metastin level in pancreatic cancer patients2009
- Author(s)
  Katagiri F, Oishi S, Fujii N, et al.
- Journal Title
  
  Oncol.Rep.
  
  Volume: 21 Pages: 815-819
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Novel screening systems for HIV-1 fusion mediated by two extra-virion hentad repeats of gp412008
- Author(s)
  Nishikawa H., Oishi S., et.al.
- Journal Title
  
  Antivir. Res. 80
  
  Pages: 71-76
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity.2008
- Author(s)
  Oishi S., et. al.
- Journal Title
  
  J. Med. Chem. 51
  
  Pages: 388-391
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Chemokine receptor CXCR4 as a therapeutic target for neuroectodermal tumors2008
- Author(s)
  Hyunsuk S., Oishi S., et.al.
- Journal Title
  
  Semin. Cancer Biol 19
  
  Pages: 123-134
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic2008
- Author(s)
  Narumi T., Oishi S., et.al.
- Journal Title
  
  Tetrahedron 64
  
  Pages: 4332-4346
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides2008
- Author(s)
  Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Synth. Org. Chem. Jpn 66
  
  Pages: 846-857
- NAID
  10024278609
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides2008
- Author(s)
  Oishi S., et.al.
- Journal Title
  
  J. Synth. Org. Chem. Jpn. 66
  
  Pages: 846-857
- NAID
  10024278609
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid-derived allylic carbonates.2008
- Author(s)
  Inokuchi E., Narumi T., Niida A., Kobayashi K., Tomita K., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  J. Org. Chem. 73
  
  Pages: 3942-3945
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Diastereoselective synthesis of highlyfunctionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic.2008
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Tetrahedron 64(19)
  
  Pages: 4332-4346
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis and application of fluorescein-and biotin-labeled molecular probes for chemokine receptor CXCR4.2008
- Author(s)
  Oishi S., et. al.
- Journal Title
  
  ChemBioChem. (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Synthesis and application of fluorescein- and botin-labeled molecular probes for chemokine receptor CXCR4.2008
- Author(s)
  Oishi S., et al.
- Journal Title
  
  ChemBioChem 9
  
  Pages: 1154-1158
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation.2008
- Author(s)
  Ohta Y., Oishi S., Fujii N., Ohno H.
- Journal Title
  
  Chem. Commun. 7
  
  Pages: 835-837
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Identification of novel nonpeptide CXCR4 antagonists by ligand-based design approach2008
- Author(s)
  Ueda S., Oishi S., et.al.
- Journal Title
  
  Bioorg. Med. Chem. Lett. 18
  
  Pages: 4124-4129
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic.2008
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Tetrahedron 64
  
  Pages: 4332-4346
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] dentification of novel nonpeptide CXCR4 antagonists by ligand-based design approach.2008
- Author(s)
  Ueda S., Kato M., Inuki S., Ohno H., Evans B., Wang Z., Peiper S.C., Izumi K., Kodama E., Matsuoka M., Nagasawa H., Oishi S., Fujii N.
- Journal Title
  
  Bioorg.Med.Chem.Lett. 18(14)
  
  Pages: 4124-4129
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis of highly functionalized alkene dipeptide isosteres and its application to thestructure-activity relationship study on bioactive peptides2008
- Author(s)
  Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Synth. Org. Chem. Jpn 66
  
  Pages: 846-857
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic2008
- Author(s)
  Narumi T., Oishi S., Fujii N., et.al.
- Journal Title
  
  Tetrahedron 64
  
  Pages: 4332-4346
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Identification of novel nonpeptide CXCR4 antagonists by ligand-baseddesian aporoach2008
- Author(s)
  Ueda S., Oishi S., Fujii N., et.al.
- Journal Title
  
  Bioorg. Med. Chem. Lett 18
  
  Pages: 4124-4129
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Design of a novel HIV-1fusion inhibitor that displays a minimal interface for binding affinity.2008
- Author(s)
  Oishi S., Ito S., Nishikawa H., Watanabe K., Tanaka M., Ohno H., Izumi K., Sakagami Y., Kodama E., Matsuoka M., Fujii N.
- Journal Title
  
  J. Med. Chem. 51
  
  Pages: 388-391
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis and application of fluorescein-and botin-labeled molecular probes for chemokine receptor CXCR4.2008
- Author(s)
  Oishi S., et. al.
- Journal Title
  
  ChemBioChem. (In press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres bypalladium-catalyzed carbonylation of amino acid-derived Arlie carbonates2008
- Author(s)
  Inokuchi E., Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Org. Chem 73
  
  Pages: 3942-3945
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Development of novel GPR54 agonists with resistance to degradation by matrix metalloproteinase2008
- Author(s)
  Tomita K., Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Med. Chem 51
  
  Pages: 7645-7649
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Identification of novel nonpeptide CXCR4 antagonists by ligand-based design approach2008
- Author(s)
  Ueda S., Oishi S., Fujii N., et.al.
- Journal Title
  
  Bioorg. Med. Chem. Lett 18
  
  Pages: 4124-4129
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid-derived allylic carbonates2008
- Author(s)
  Inokuchi E., Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Org. Chem 73
  
  Pages: 3942-3945
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20015021
[Journal Article] Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and itsapplication to Fmoc-based solid phase synthesis of a cyclic pentapeptide mimetic2008
- Author(s)
  Narumi T., Oishi S., Fujii N., et.al.
- Journal Title
  
  Tetrahedron 64
  
  Pages: 4332-4346
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity.2008
- Author(s)
  Oishi S., et al.
- Journal Title
  
  J. Med. Chem. 51
  
  Pages: 388-391
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Palladium-catalyzed sp3 C-H activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines.2008
- Author(s)
  Watanabe T., Oishi S., Fujii N., Ohno H.
- Journal Title
  
  Org. Lett. 10
  
  Pages: 1759-1762
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides.2008
- Author(s)
  Oishi S., Narumi T., Ohno H., Otaka A., Fujii N.
- Journal Title
  
  J.Synth.Org.Chem.Jpn. 66(9)
  
  Pages: 846-857
- NAID
  10024278609
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity2008
- Author(s)
  Oishi S., et al.
- Journal Title
  
  J. Med. Chem. 51
  
  Pages: 388-391
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis and application of fluorescein- and botin-labeled molecular probes for chemokine receptor CXCR4.2008
- Author(s)
  Oishi S., Masuda R., Evans B., Ueda S., Goto Y., Ohno H., Hirasawa A., Tsujimoto G., Wang Z., Peiper S. C., Naito T., Kodama E., Matsuoka M., Fujii N.
- Journal Title
  
  Chem BioChem 9
  
  Pages: 1154-1158
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Novel screening systems for HIV-1 fusion mediated by two extra-virion heptad repeats of gp41.2008
- Author(s)
  Nishikawa H., Kodama E., Sakakibara A., Fukudome A., Izumi K., Oishi S., Fujii N., Matsuoka M.
- Journal Title
  
  Antivir.Res. 80(1)
  
  Pages: 71-76
- NAID
  120002790066
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Synthesis and application of fluorescein- and biotin-labeled molecular probes for chemokine receptor CXCR42008
- Author(s)
  Oishi S., et al.
- Journal Title
  
  ChemBioChem. (in press)
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Development of novel GPR54 agonists with resistance to degradation by matrixmetalloproteinase2008
- Author(s)
  Tomita K., Oishi S., Fujii N., et.al.
- Journal Title
  
  J. Med. Chem 51
  
  Pages: 7645-7649
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20057011
[Journal Article] Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid-derived allylic carbonates2008
- Author(s)
  Inokuchi E., Oishi S., et.al.
- Journal Title
  
  J. Org. Chem. 73
  
  Pages: 3942-3945
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-20790098
[Journal Article] Cyclic peptide analysis of the biologically active loop region in the laminin R3 chain LG4 module demonstrates the importance of peptide conformation on biological activity.2007
- Author(s)
  Kato Takagaki, K., Oishi, S., Nomizu, M.et al.
- Journal Title
  
  Biochemistry 46・7
  
  Pages: 1952-1960
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Establishment and clinical application of enzyme immunoassays for determination of luteinizing hormone releasing hormone and metastin.2007
- Author(s)
  Katagiri F., Tomita K., Oishi S., Takeyama M., Fujii N.
- Journal Title
  
  J. Pept. Sci. 13
  
  Pages: 422-429
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions.2007
- Author(s)
  Ohno H., Ohta Y., Oishi S., Fujii N.
- Journal Title
  
  Angew. Chem. Int. Ed. 46
  
  Pages: 2295-2298
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions.2007
- Author(s)
  Ohno, H., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Angew. Chem. Int. Ed. Engl. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] The therapeutic potential of the chemokine receptor CXCR4 antagonists as multi-functional agents.2007
- Author(s)
  Tsutsumi H., Tanaka T., Ohashi N., Masuno H., Tamamura H., Hiramatsu K., Araki T., Ueda S., Oishi S., Fujii N.
- Journal Title
  
  Biopolymers 88
  
  Pages: 279-289
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] ペプチドをリードとした創薬2007
- Author(s)
  大石真也, et. al.
- Journal Title
  
  蛋白質核酸酵素増刊ケミカルバイオロジー長野哲雄・長田裕之・菊地和也・上杉志成編集 52
  
  Pages: 1696-1701
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Structure-activity relationships of cyclic Peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone functionalities.2007
- Author(s)
  Ueda, S., Oishi, H., Fujii, N.et al.
- Journal Title
  
  J.Med.Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Structureactivity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and hackbone2007
- Author(s)
  Ueda S., Oishi S., Wang Z. X., Araki T., Tamamura H., Cluzeau J., Ohno H. Kusano S., Nakashima H., Trent J. O., Peiper S. C., Fujii N.
- Journal Title
  
  J. Med. Chem. 50
  
  Pages: 192-198
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] A novel oxazolidine linker for the synthesis of peptide aldehydes2007
- Author(s)
  Tanaka, M., Oishi, H., Fujii, N.et al.
- Journal Title
  
  Int.J.Pep.Res.Ther. (in press)
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] ケミカルバイオロジーを基盤とするペプチド創薬2007
- Author(s)
  大石真也, et. al.
- Journal Title
  
  遺伝子医学MOOK8ペプチドと創薬寒川賢治・南野直人編集
  
  Pages: 87-91
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists.2007
- Author(s)
  Cluzeau J., Oishi S., Ohno H., Wang Z., Evans B., Peiper S. C., Fujii N.
- Journal Title
  
  Org. Biomol. Chem. 5
  
  Pages: 1915-1923
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Versatile use of acid-catalyzed ring-opening of □-aziridinyl-□, □ enoates to stereoselective synthesis of peptidomimetics.2007
- Author(s)
  Tamamura H., Tanaka T., Tsutsumi H., Nemoto K., Mizokami S., Ohashi N., Oishi S., Fujii N.
- Journal Title
  
  Tetrahedron 63
  
  Pages: 9243-9254
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] ペプチドをリードとした創薬2007
- Author(s)
  大石真也, et. al.
- Journal Title
  
  蛋白質核酸酵素増刊ケミカルバイオロジー長野哲雄・長田裕之・菊地和也・上杉志成編集 52
  
  Pages: 1696-1701
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 272-278
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions.2007
- Author(s)
  Ohno, H., Oishi, S., Fujii, N., et al.
- Journal Title
  
  Angew.Chem.Int.Ed.Engl. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita K., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Biopolymers 88
  
  Pages: 272-278
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the pTyr+1 position of Grb2 SH2 domain-binding tripeptides.2007
- Author(s)
  Kang, S.-U., Oishi, S., Burke, T.R., Jr.et al.
- Journal Title
  
  J.Med.Chem. 50・8
  
  Pages: 1978-1982
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] ケミカルバイオロジーを基盤とするペプチド創薬2007
- Author(s)
  大石真也, et al.
- Journal Title
  
  遺伝子医学MOOK8ペプチドと創薬寒川賢治・南野直人編集
  
  Pages: 87-91
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54.2007
- Author(s)
  Tomita K., Oishi S., Cluzeau J., Ohno H., Navenot J. M., Wang Z. X., Peiper S. C., Akamatsu M., Fujii N.
- Journal Title
  
  J. Med. Chem. 50
  
  Pages: 3222-3228
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Cyclic peptide analysis of the biologically active loop region in the laminin R3 chain LG4 module demonstrates the importance of peptide conformation on biological activity.2007
- Author(s)
  Kato Takagaki, K., Oishi, S., Nomizu, M.et al.
- Journal Title
  
  Biochemistry 46・7
  
  Pages: 1952-1960
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Structure-activity relationships of cyclic Peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone functionalities.2007
- Author(s)
  Ueda, S., Oishi, S., Fujii, N.et al.
- Journal Title
  
  J.Med.Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Gold-catalyzed hydroarylation of allenes : a highly regioselective carbon-carbon bond formation producing sixmembered rings.2007
- Author(s)
  Watanabe T., Oishi S., Fujii N., Ohno H.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 4821-4824
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the pTyr+1 position of Grb2 SH2 domain-binding tripeptides.2007
- Author(s)
  Kang, S.-U., Oishi, S., Burke, T.R., Jr.et al.
- Journal Title
  
  J.Med.Chem. 50・8
  
  Pages: 1978-1982
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] ケミカルバイオロジーを基盤とするペプチド創薬2007
- Author(s)
  大石真也, et. al.
- Journal Title
  
  遺伝子医学MOOK8ペプチドと創薬寒川賢治・南野直人編集
  
  Pages: 87-91
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides.2007
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Org. Lett. 9
  
  Pages: 3465-3468
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 272-278
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Direct Synthesis of 2-(Aminomethyl)indoles through Copper(I)-Catalyzed Domino Three-Component Coupling and Cyclization Reactions.2007
- Author(s)
  Ohno, H., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Angew.Chem.Int.Ed.Engl. 46・13
  
  Pages: 2295-2298
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene-and fluoroalkene-dipeptide isosteres.2007
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Biopolymers 88・2
  
  Pages: 272-278
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling2007
- Author(s)
  Watanabe T., Ueda S., Inuki S., Oishi S., Fujii N., Ohno H.
- Journal Title
  
  Chem. Commun.
  
  Pages: 4516-4518
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Structure-activity relationships of cyclic Peptide-based chemokine receptor CXCR4 antagonists : disclosing the importance of side-chain and backbone functionalities.2007
- Author(s)
  Ueda, S., Oishi, S., Fujii, N.et al.
- Journal Title
  
  J. Med. Chem. 50・2
  
  Pages: 192-198
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] A novel oxazolidine linker for the synthesis of peptide aldehydes.2007
- Author(s)
  Tanaka M., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Int. J. Pep. Res. Ther. 13
  
  Pages: 271-279
- NAID
  10020528946
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the pTyr+1 position of Grb2 SH2 domain-binding tripeptides.2007
- Author(s)
  Kang, S.-U., Oishi, S., Burke, T.R., Jr.et al.
- Journal Title
  
  J. Med. Chem. 50・8
  
  Pages: 1978-1982
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Cyclic peptide analysis of the biologically active loop region in the laminin R3 chain LG4 module demonstrates the importance of peptide conformation on biological activity.2007
- Author(s)
  Kato Takagaki, K., Oishi, S., Nomizu, M.et al.
- Journal Title
  
  Biochemistry 46・7
  
  Pages: 1952-1960
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis and biological evaluation of L-cysteine derivatives as mitotic kinesin Eg5 inhibitors.2007
- Author(s)
  Ogo N., Oishi S., Matsuno K., Sawada J., Fujii N., Asai A.
- Journal Title
  
  Bioorg. Med. Chem. Lett. 17
  
  Pages: 3921-3924
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] ペプチドをリードとした創薬2007
- Author(s)
  大石真也, et al.
- Journal Title
  
  蛋白質核酸酵素増刊ケミカルバイオロジー長野哲雄・長田裕之・菊地和也・上杉志成編集 52
  
  Pages: 1696-1701
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Application of tri-and tetrasubstituted alkene dipeptide mimetics toconformational studies of cyclic RGD peptides.2006
- Author(s)
  Oishi S., et al.
- Journal Title
  
  Tetrahedron 62
  
  Pages: 1416-1424
- Description
  「研究成果報告書概要(和文)」より
- Peer Reviewed
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita K., Niida A., Oishi S., Ohno H., Cluzeau J., Navenot J. M., Wang Z. X., Peiper S. C., Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. 14
  
  Pages: 7595-7603
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Bioorg. Med. Chem. 45・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utili-zing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations.2006
- Author(s)
  Niida, A., Oishi, S., Fujii, N.et al.
- Journal Title
  
  J. Org. Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.2006
- Author(s)
  Narumi T., Niida A., Tomita K., Oishi S., Otaka A., Ohno H., Fujii N.
- Journal Title
  
  Chem. Commun.
  
  Pages: 4720-4722
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Application of tri- and tetrasubstituted alkene dipeptide mimetics to conformational studies of cyclic RGD peptides2006
- Author(s)
  Oishi S., Miyamoto K., Niida A., Yamamoto M., Ajito K., Tamamura H., Otaka A., Kuroda Y., Asai A., Fujii N.
- Journal Title
  
  Tetrahedron 62
  
  Pages: 1416-1424
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Unequivocal synthesis of (Z)-alkene and (E)-fluoroalkene dipeptide isosteres to probe structural requirements of the peptide transporter PEPT1.2006
- Author(s)
  Niida A., Tomita K., Mizumoto M., Tanigaki H., Terada T., Oishi S., Otaka A., Inui K., Fujii N.
- Journal Title
  
  Org. Lett. 8
  
  Pages: 613-616
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Folliculin encoded by the BHD gene interacts with a novel binding protein, FNIPl, and AMPK, and is involved in AMPK and mTOR signaling.2006
- Author(s)
  Baba, M., Oishi, S., Zbar, B.et al.
- Journal Title
  
  Proc.Natl.Acad.Sci. 103・42
  
  Pages: 15552-15557
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Bioorg.Med.Chem. 45・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Synthesis of (Z)-alkene and (E)-fluoroalkenecontaining diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT2006
- Author(s)
  Niida A., Mizumoto M., Narumi T., Inokuchi E., Oishi S., Ohno H., Otaka A., Kitaura K., Fujii N.
- Journal Title
  
  J. Org. Chem. 71
  
  Pages: 4118-4129
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utili-zing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations.2006
- Author(s)
  Niida, A., Oishi, S., Fujii, N.et al.
- Journal Title
  
  J.Org.Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Application of tri- and tetrasubstituted alkene dipeptide mimetics to conformational studies of cyclic RGD peptides2006
- Author(s)
  Oishi, S. et al.
- Journal Title
  
  Tetrahedron 62・7
  
  Pages: 1416-1424
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Structure-activity relationship study on small peptidic GPR54 agonists.2006
- Author(s)
  Tomita, K., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Bioorg.Med.Chem. 45・22
  
  Pages: 7595-7603
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.2006
- Author(s)
  Narumi, T., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Chem. Commun. 45
  
  Pages: 4720-2722
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.2006
- Author(s)
  Narumi, T., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Chem.Commun. 45
  
  Pages: 4720-2722
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres.2006
- Author(s)
  Narumi, T., Oishi, S., Fujii, N.et al.
- Journal Title
  
  Chem.Commun. 45
  
  Pages: 4720-4722
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Folliculin encoded by the BHD gene interacts with a novel binding protein, FNIP1, and AMPK, and is involved in AMPK and mTOR signaling.2006
- Author(s)
  Baba, M., Oishi, S., Zbar, B.et al.
- Journal Title
  
  Proc.Natl.Acad.Sci. 103・42
  
  Pages: 15552-15557
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Folliculin encoded by the BHD gene interacts with a novel binding protein, FNIP1, and AMPK, and is involved in AMPK and mTOR signaling.2006
- Author(s)
  Baba, M., Oishi, S., Zbar, B.et al.
- Journal Title
  
  Proc. Natl. Acad. Sci. 103・42
  
  Pages: 15552-15557
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Design and synthesis of downsized metastin (45-54) analogs with maintenance of high GPR54 agonistic activity2006
- Author(s)
  Niida A., Wang Z., Tomita K, Oishi S., Tamamura H., Otaka A., Navenot J. M., Broach J. R., Peiper S. C., Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett. 16
  
  Pages: 134-137
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists.2006
- Author(s)
  Niida A., Tanigaki H., Inokuchi E., Sasaki Y., Oishi S., Ohno H., Tamamura H., Wang Z., Peiper S. C., Kitaura K., Otaka A., Fujii N.
- Journal Title
  
  J. Org. Chem. 71
  
  Pages: 3942-3951
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Synthesis of (Z)-alkene and (E)- fluoroalkene-containing diketopiperazine mimetics utili-zing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations.2006
- Author(s)
  Niida, A., Oishi, S., Fujii, N.et al.
- Journal Title
  
  J.Org.Chem. 71・11
  
  Pages: 4118-4129
- Data Source
  KAKENHI-PROJECT-18060020
[Journal Article] Ring-closing metathesis of C-terminal allylglycine residues with an N-terminal β-vinyl-substituted phosphotyrosyl mimetic as an approach to novel Grb2 SH2 domain-binding macrocycles2005
- Author(s)
  Oishi, S. et al.
- Journal Title
  
  ChemBioChem 6・4
  
  Pages: 668-674
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Evaluation of macrocyclic Grb2 SH2 domain-binding peptide mimetics prepared by ring-closing metathesis of C-terminal allylglycines with an N-terminal β-vinyl-substituted phosphotyrosyl mimetic2005
- Author(s)
  Oishi, S. et al.
- Journal Title
  
  Bioorg.Med.Chem. 13・7
  
  Pages: 2431-2438
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Design and synthesis of conformationally constrained Grb2 SH2 domain binding peptides employing y-methylphenylalanyl based phosphotyrosyl mimetics2005
- Author(s)
  Oishi, S. et al.
- Journal Title
  
  J.Med.Chem. 48・3
  
  Pages: 764-772
- Data Source
  KAKENHI-PROJECT-17790091
[Journal Article] Coiled-coil tag-probe system for quick labeling of membrane receptors in living cells.
- Author(s)
  Yano Y., Yano A., Oishi S., Sugimoto Y., Tsujimoto G., Fujii N., Matsuzaki K.
- Journal Title
  
  ACS Chem. Biol. (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Identification of novel nonpeptide CXCR4 antagonists by ligand-based design approach.
- Author(s)
  Ueda S., Kato M., Inuki S., Ohno H., Evans B., Wang Z., Peiper S. C., Izumi K., Kodama E., Matsuoka M., Nagasawa H., Oishi S., Fujii N.
- Journal Title
  
  Bioorg. Med. Chem. Lett. (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Novel screening systems for HIV-1 fusion mediated by two extra-virion heptad repeats of gp41.
- Author(s)
  Nishikawa H., Kodama E., Sakakibara A., Fukudome A., Izumi K., Oishi S., Fujii N., Matsuoka M.
- Journal Title
  
  Antivir. Res. (in press)
- NAID
  120002790066
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Structure-activity relationship of pyrazine-based CK2 inhibitors : synthesis and biological evaluation of 2,6-disubstituted pyrazine and 4,6-disubstituted pyrimidine derivatives.
- Author(s)
  Suzuki Y., Cluzeau J., Hara T., Hirasawa A.. Tsujimoto G., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Archiv. Pharm. (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Palladiumcatalysed biscyclisation of allenic bromoalkenes through zipper-mode cascade.
- Author(s)
  Okano A., Mizutani T., Oishi S., Tanaka T., Ohno H., Fujii N.
- Journal Title
  
  Chem. Commun. (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Journal Article] Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists.
- Author(s)
  Tomita K., Oishi S., Ohno H., Fujii N.
- Journal Title
  
  Biopolymers (in press)
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] 免疫原性低減型低分子抗体とその製造法2021
- Inventor(s)
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Holder
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Type
  特許
- Filing Date
  2021
- Overseas
- Data Source
  KAKENHI-PROJECT-18H02555
[Patent] 免疫原性低減型低分子抗体とその製造法2021
- Inventor(s)
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Holder
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Type
  特許
- Filing Date
  2021
- Overseas
- Data Source
  KAKENHI-PROJECT-20K21252
[Patent] 免疫原性低減型低分子抗体とその製造法2020
- Inventor(s)
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Holder
  野中元裕、大石真也、大野浩章、青木啓輔
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2020-105104
- Filing Date
  2020
- Data Source
  KAKENHI-PROJECT-18H02555
[Patent] 新規NK3受容体アゴニスト2014
- Inventor(s)
  藤井信孝、大野浩章、大石真也、三須良介、山田愛、山本昂輝、他
- Industrial Property Rights Holder
  国立大学法人京都大学、独立行政法人農業生物資源研究所
- Industrial Property Rights Type
  特許
- Filing Date
  2014-12-05
- Overseas
- Data Source
  KAKENHI-PROJECT-23689007
[Patent] Eg5阻害剤2014
- Inventor(s)
  藤井信孝、大野浩章、大石真也、竹内智起、浅井章良、澤田潤一
- Industrial Property Rights Holder
  京都大学、有限責任中間法人ファルマＩＰ
- Industrial Property Rights Type
  特許
- Filing Date
  2014-02-25
- Overseas
- Data Source
  KAKENHI-PROJECT-24659004
[Patent] 新規NK3受容体アゴニスト2013
- Inventor(s)
  藤井信孝、大石真也、他
- Industrial Property Rights Holder
  国立大学法人京都大学、独立行政法人農業生物資源研究所
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2013-253534
- Filing Date
  2013-12-06
- Data Source
  KAKENHI-PROJECT-23689007
[Patent] 新規NK3受容体アゴニスト2013
- Inventor(s)
  藤井信孝、大石真也、他
- Industrial Property Rights Holder
  国立大学法人京都大学、独立行政法人農業生物資源研究所
- Industrial Property Rights Type
  特許
- Filing Date
  2013-10-18
- Overseas
- Data Source
  KAKENHI-PROJECT-23689007
[Patent] Eg5阻害剤2013
- Inventor(s)
  藤井信孝、大野浩章、大石真也、竹内智起、浅井章良、澤田潤一
- Industrial Property Rights Holder
  京都大学、有限責任中間法人ファルマＩＰ
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2013-094147
- Filing Date
  2013-04-26
- Data Source
  KAKENHI-PROJECT-24659004
[Patent] 新規NK3受容体アゴニスト2012
- Inventor(s)
  藤井信孝、大野浩章、大石真也、野口太朗、三須良介
- Industrial Property Rights Holder
  藤井信孝、大野浩章、大石真也、野口太朗、三須良介
- Industrial Property Rights Type
  特許
- Industrial Property Number
  2012-231902
- Filing Date
  2012-10-19
- Data Source
  KAKENHI-PROJECT-23689007
[Patent] 酵母を用いた抗HIVペプチドの生産方法2010
- Inventor(s)
  大石真也, 他
- Industrial Property Rights Holder
  科学技術振興機構、月桂冠
- Industrial Property Number
  2010-046273
- Filing Date
  2010-03-03
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] 麹菌を用いた抗HIVペプチドの生産方法2010
- Inventor(s)
  大石真也, 他
- Industrial Property Rights Holder
  月桂冠、科学技術振興機構
- Industrial Property Number
  2010-030875
- Filing Date
  2010-02-16
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也、富田健嗣
- Industrial Property Rights Holder
  国立大学法人京都大学、武田薬品工業株式会社
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2015-02-27
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] Metastin derivative and use thereof2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2017-06-07
- Overseas
- Data Source
  KAKENHI-PROJECT-20057011
[Patent] METASTIN DERIVATIVE AND USE THEREOF2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2013-11-26
- Overseas
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] METASTIN DERIVATIVE AND USE THEREOF2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2013-11-26
- Overseas
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也、富田健嗣
- Industrial Property Rights Holder
  国立大学法人京都大学、武田薬品工業株式会社
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2015-02-27
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] Metastin derivative and use thereof2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2017-06-07
- Overseas
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] Eg5阻害剤2009
- Inventor(s)
  藤井信孝、大野浩章、大石真也, 他
- Industrial Property Rights Holder
  京都大学
- Filing Date
  2009-12-25
- Overseas
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也, 他
- Industrial Property Rights Holder
  京都大学
- Filing Date
  2009-04-28
- Overseas
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也, 他
- Industrial Property Rights Holder
  京都大学
- Filing Date
  2009-04-28
- Overseas
- Data Source
  KAKENHI-PROJECT-20057011
[Patent] Metastin derivative and use thereof2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2017-06-07
- Overseas
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] METASTIN DERIVATIVE AND USE THEREOF2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2013-11-26
- Overseas
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也、富田健嗣
- Industrial Property Rights Holder
  国立大学法人京都大学、武田薬品工業株式会社
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2015-02-27
- Data Source
  KAKENHI-PROJECT-20057011
[Patent] 修飾ペプチド及びその製造方法2009
- Inventor(s)
  藤井信孝、松岡雅雄、児玉栄一、大石真也、田中理紀、秦洋二、堤浩子、梶原一美、常盤礼
- Industrial Property Rights Holder
  科学技術振興機構、京都大学、月桂冠
- Industrial Property Number
  2009-164647
- Filing Date
  2009-07-13
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] METASTIN DERIVATIVE AND USE THEREOF2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2013-11-26
- Overseas
- Data Source
  KAKENHI-PROJECT-20057011
[Patent] Metastin derivative and use thereof2009
- Inventor(s)
  Nobutaka Fujii, Shinya Oishi, Kenji Tomita
- Industrial Property Rights Holder
  Kyoto University, Takeda Pharmaceutical Company
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2017-06-07
- Overseas
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] メタスチン誘導体およびその用途2009
- Inventor(s)
  藤井信孝、大石真也、富田健嗣
- Industrial Property Rights Holder
  国立大学法人京都大学、武田薬品工業株式会社
- Industrial Property Rights Type
  特許
- Filing Date
  2009-04-28
- Acquisition Date
  2015-02-27
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] 修飾ペプチド及びその製造方法2009
- Inventor(s)
  大石真也, 他
- Industrial Property Rights Holder
  科学技術振興機構、京都大学、月桂冠
- Industrial Property Number
  2009-164647
- Filing Date
  2009-07-13
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] Eg5阻害剤2008
- Inventor(s)
  藤井、大石, 他
- Industrial Property Rights Holder
  京都大学・ファルマIP
- Industrial Property Number
  2008-331963
- Filing Date
  2008-12-16
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] Eg5阻害剤2008
- Inventor(s)
  藤井、大石, 他
- Industrial Property Rights Holder
  京都大学・ファルマIP
- Industrial Property Number
  2008-331963
- Filing Date
  2008-12-26
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] メタスチン誘導体およびその用途2008
- Inventor(s)
  藤井、大石他
- Industrial Property Rights Holder
  京都大学・武田薬品工業
- Industrial Property Number
  2008-119235
- Filing Date
  2008-04-30
- Data Source
  KAKENHI-PROJECT-20057011
[Patent] メタスチン誘導体およびその用途2008
- Inventor(s)
  藤井信孝、大石真也、富田健嗣
- Industrial Property Rights Holder
  京都大学、武田薬品工業
- Industrial Property Number
  2008-119235
- Filing Date
  2008-04-30
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] メタスチン誘導体およびその用途2008
- Inventor(s)
  藤井、大石, 他
- Industrial Property Rights Holder
  泉都大学・武田薬品工業
- Industrial Property Number
  2008-000001
- Filing Date
  2008-04-30
- Data Source
  KAKENHI-PROJECT-20790098
[Patent] メタスチン誘導体およびその用途2008
- Inventor(s)
  藤井、大石, 他
- Industrial Property Rights Holder
  京都大学・武田薬品工業
- Industrial Property Number
  2008-119235
- Filing Date
  2008-04-30
- Data Source
  KAKENHI-PROJECT-20015021
[Patent] メタスチン誘導体およびその用途2008
- Inventor(s)
  藤井信孝, 大石真也, 富田健嗣
- Industrial Property Rights Holder
  国立大学法人京都大学
- Industrial Property Number
  2008-119235
- Filing Date
  2008-04-30
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] Eg5阻害剤および該化合物を含有してなる抗癌剤2007
- Inventor(s)
  浅井章良, 澤田潤一, 松野研司, 小郷尚久, 藤井信孝, 大石真也
- Industrial Property Rights Holder
  有限責任中間法人フアルマIP
- Industrial Property Number
  2007-069487
- Filing Date
  2007-03-16
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] 抗HIV剤2006
- Inventor(s)
  藤井信孝, 大石真也, 松岡雅雄, 児玉栄
- Industrial Property Rights Holder
  国立大学法人京都大学
- Industrial Property Number
  2006-290241
- Filing Date
  2006-10-25
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] GPR54アゴニスト活性を有する化合物2006
- Inventor(s)
  藤井信孝, 大石真也, 富田健嗣, 新居田歩
- Industrial Property Rights Holder
  国立大学法人京都大学
- Industrial Property Number
  2006-122305
- Filing Date
  2006-04-26
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Patent] N36結合ペプチドの製造方法2006
- Inventor(s)
  堤, 石田, 久田, 水本, 秦, 藤井, 松岡, 児玉, 大石
- Industrial Property Rights Holder
  月桂冠株式会
- Industrial Property Number
  2006-204827
- Filing Date
  2006-07-27
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] 鏡像タンパク質を活用した創薬研究2023
- Author(s)
  大石真也
- Organizer
  第12回有機「ものつくり」化学研究会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 創薬モダリティとしての応用を指向した鏡像モノボディの化学合成法の確立と応用2023
- Author(s)
  佐藤志乃, 岩本直也, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 野中元裕, 大石真也
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 創薬モダリティとしての応用を指向した鏡像モノボディの化学合成法の確立と応用2023
- Author(s)
  佐藤志乃, 岩本直也, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 野中元裕, 大石真也
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 免疫原性の低減を志向した鏡像VHH抗体の開発2023
- Author(s)
  青木啓輔, 野中元裕, 小田幸穂, 東克暁, 眞鍋麻彩子, 木村寛之, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡の中の中分子化合物からの医薬シーズの探索技術2023
- Author(s)
  大石真也
- Organizer
  日本薬学会第143年会
- Invited
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 鏡像タンパク質を活用した創薬研究2023
- Author(s)
  大石真也
- Organizer
  大阪大学蛋白質研究所セミナー：タンパク質に挑戦する化学
- Invited
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 鏡像タンパク質を活用した創薬研究2023
- Author(s)
  大石真也
- Organizer
  大阪大学蛋白質研究所セミナー：タンパク質に挑戦する化学
- Invited
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像タンパク質を活用した創薬研究2023
- Author(s)
  大石真也
- Organizer
  第12回有機「ものつくり」化学研究会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 免疫原性の低減を志向した鏡像VHH抗体の開発2023
- Author(s)
  青木啓輔, 野中元裕, 小田幸穂, 東克暁, 眞鍋麻彩子, 木村寛之, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 免疫チェックポイントを調節するタンパク質の化学合成研究2023
- Author(s)
  岩本直也, 佐々木順平, 青木啓輔, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第143年会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡の中の中分子化合物からの医薬シーズの探索技術2023
- Author(s)
  大石真也
- Organizer
  日本薬学会第143年会
- Invited
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Investigation of the immunogenicity of mirror-image single-domain antibody binding to vascular endothelial growth factor2022
- Author(s)
  Keisuke Aoki, Motohiro Nonaka, Sakiho Oda, Katsuaki Higashi, Asako Manabe, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第59回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] Synthesis and functional analysis of mirror-image monobody2022
- Author(s)
  Naoya Iwamoto, Yukino Sato, Asako Manabe, Shinsuke Inuki, Hiroaki Ohno, Motohiro Nonaka, Shinya Oishi
- Organizer
  第59回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像VHH抗体の免疫原性評価と免疫ライブラリーを用いた配列取得2022
- Author(s)
  眞鍋麻彩子, 前田佳夕, 青木啓輔, 薄井友輔, 髙橋里菜, 大野浩章, 森瀬譲二, 岡昌吾, 大石真也, 野中元裕
- Organizer
  第95回日本生化学会大会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 麻疹ウイルス膜融合阻害ペプチドの構造最適化研究2022
- Author(s)
  山口夕貴, 髙原葵, 青木啓輔, 中津亨, 平田和成, 鈴木聡志, 林宏典, 河治久実, 井貫晋輔, 大野浩章, 加藤博章, 村山和隆, 児玉栄一, 大石真也
- Organizer
  第39回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-21K19366
[Presentation] MCP-1に結合するミラーイメージ人工抗体の創製2022
- Author(s)
  三浦清楓, 近藤太志, 薄井友輔, 大石真也, 藤野公茂, 林剛介, 村上裕
- Organizer
  第16回バイオ関連化学シンポジウム
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] VEGF 結合活性を示す鏡像VHH 抗体の探索研究2022
- Author(s)
  青木啓輔, 野中元裕, 小田幸穂, 東克暁, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第39回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] メチル基にまつわる小さな話2022
- Author(s)
  大石真也
- Organizer
  第54回若手ペプチド夏の勉強会
- Invited
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] VEGF 結合活性を示す鏡像VHH 抗体の探索研究2022
- Author(s)
  青木啓輔, 野中元裕, 小田幸穂, 東克暁, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第39回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像VHH抗体の免疫原性評価と免疫ライブラリーを用いた配列取得2022
- Author(s)
  眞鍋麻彩子、前田佳夕、青木啓輔、薄井友輔、髙橋里菜、大野浩章、森瀬譲二、岡昌吾、大石真也、野中元裕
- Organizer
  第95回日本生化学会大会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 抗MCP-1人工抗体のミラーイメージ選択2022
- Author(s)
  三浦清楓, 近藤太志, 薄井友輔, 大石真也, 藤野公茂, 林剛介, 村上裕
- Organizer
  第12回CSJ化学フェスタ2022
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Synthesis and functional analysis of mirror-image monobody2022
- Author(s)
  Naoya Iwamoto, Yukino Sato, Asako Manabe, Shinsuke Inuki, Hiroaki Ohno, Motohiro Nonaka, Shinya Oishi
- Organizer
  第59回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] 血管内皮増殖因子VEGFに対して特異的に結合する鏡像VHH抗体の探索2022
- Author(s)
  青木啓輔, 野中元裕, 小田幸穂, 東克暁, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第54回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像モノボディの化学合成法の確立と機能評価2022
- Author(s)
  佐藤志乃, 岩本直也, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 野中元裕, 大石真也
- Organizer
  第39回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-22K19376
[Presentation] Investigation of the immunogenicity of mirror-image single-domain antibody binding to vascular endothelial growth factor2022
- Author(s)
  Keisuke Aoki, Motohiro Nonaka, Sakiho Oda, Katsuaki Higashi, Asako Manabe, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第59回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像モノボディの化学合成法の確立と機能評価2022
- Author(s)
  佐藤志乃, 岩本直也, 眞鍋麻彩子, 井貫晋輔, 大野浩章, 野中元裕, 大石真也
- Organizer
  第39回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Chemical protein synthesis for mirror-image screening2021
- Author(s)
  S. Oishi
- Organizer
  4th National Taiwan University School of Pharmacy Research Day and International Conference
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像タンパク質を活用した創薬研究2021
- Author(s)
  大石真也
- Organizer
  第94回日本生化学会大会：生理活性ペプチドと中分子創薬─新たな創薬ブレイクスルーを目指して
- Invited
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 溶解性向上タグを用いたTIGIT細胞外ドメインの化学合成研究2021
- Author(s)
  岩本直也, 佐々木順平, 青木啓輔, 薄井友輔, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第53回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Chemical protein synthesis for mirror-image screening2021
- Author(s)
  Shinya Oishi, Keitou Shu, Naoya Iwamoto, Takumi Ohara, Jumpei Sasaki, Keisuke Aoki, Yusuke Usui, Shinsuke Inuki, Hiroaki Ohno
- Organizer
  The 18th Akabori Conference
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Chemical protein synthesis for mirror-image screening2021
- Author(s)
  Shinya Oishi
- Organizer
  4th National Taiwan University School of Pharmacy Research Day and International Conference
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Chemical protein synthesis for mirror-image screening2021
- Author(s)
  S. Oishi
- Organizer
  The 18th Akabori Conference
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 溶解性向上タグを用いたTIGIT細胞外ドメインの化学合成研究2021
- Author(s)
  岩本直也, 佐々木順平, 青木啓輔, 薄井友輔, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第53回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] 鏡像VHH抗体の化学合成と免疫原性評価2020
- Author(s)
  青木啓輔、野中元裕、井貫晋輔、大野浩章、大石真也
- Organizer
  第70回日本薬学会関西支部大会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Investigation of the immunogenicity of mirror-image single-domain antibody2020
- Author(s)
  Keisuke Aoki, Motohiro Nonaka, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第57回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Coibamide Aの標的分子の同定と構造最適化への展開2020
- Author(s)
  大石真也
- Organizer
  第11回有機「ものつくり」研究会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 鏡像VHH抗体の化学合成と免疫原性評価2020
- Author(s)
  青木啓輔、野中元裕、井貫晋輔、大野浩章、大石真也
- Organizer
  第70回日本薬学会関西支部大会
- Data Source
  KAKENHI-PROJECT-20K21252
[Presentation] Synthesis of mirror-image protein of glutamate racemase2020
- Author(s)
  Takumi Ohara, Naoya Owamoto, Taro Noguchi, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  医薬系研究交流サロン
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Ｃ末端側からのNCLプロトコールを利用したTIGITタンパク質の合成研究2020
- Author(s)
  岩本直也、青木啓輔、佐々木順平、井貫晋輔、大野浩章、大石真也
- Organizer
  日本薬学会第140年会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Investigation of the immunogenicity of mirror-image single-domain antibody2020
- Author(s)
  Keisuke Aoki, Motohiro Nonaka, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第57回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 麻疹ウイルス膜融合阻害ペプチドの最小活性配列の同定と相互作用解析2019
- Author(s)
  高原葵、中津亨、平田和成、林宏典、河治久実、井貫晋輔、大野浩章、加藤博章、児玉栄一、大石真也
- Organizer
  第37回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Coibamide Aの固相合成法の改良と構造活性相関研究2019
- Author(s)
  喜多村隆志、川口晋作、井貫晋輔、大野浩章、大石真也
- Organizer
  第69回日本薬学会関西支部大会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 麻疹ウイルス膜融合阻害ペプチドの構造活性相関研究　―抗ウイルス活性に必要な最小配列の同定―2019
- Author(s)
  髙原葵、平田和成、林宏典、河治久実、井貫晋輔、大野浩章、児玉栄一、大石真也
- Organizer
  第69回日本薬学会関西支部大会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] XIAP BIR3ドメインの化学合成と鏡像スクリーニングへの応用2019
- Author(s)
  岩本直也, 周敬棠, 本田香織, 近藤恭光, 長田裕之, 井貫晋輔, 大野浩章, 藤井信孝, 大石真也
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Synthetic study on full-length hepatitis B virus core protein2019
- Author(s)
  Keisuke Aoki, Shugo Tsuda, Shinsuke Inuki, Hiroaki Ohno, Taku Yoshiya, Shinya Oishi
- Organizer
  第56回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 鏡像スクリーニングを指向したTIGITタンパク質の合成研究2019
- Author(s)
  青木啓輔, 佐々木順平, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第139年会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Synthesis of mirror-image protein of glutamate racemase2019
- Author(s)
  Takumi Ohara, Naoya Iwamoto, Taro Noguchi, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第12回有機触媒シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Synthetic study of TIGIT protein for mirror-image screening2019
- Author(s)
  Keisuke Aoki, Jumpei Sasaki, Naoya Iwamoto, Yusuke Usui, Shinsuke Inuki, Hiroaki Ohno and Shinya Oishi
- Organizer
  27th International Society of Heterocyclic Chemistry Congress
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Synthetic study on TIGIT protein for mirror-image screening2019
- Author(s)
  Naoya Iwamoto, Jumpei Sasaki, Keisuke Aoki, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  第56回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] カプシドタンパク質の化学合成と粒子形成の最適化2018
- Author(s)
  佐々木順平, 石場勲之, 津田修吾, 西尾秀喜, 片岡紀代, 渡士幸一, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] グルタミン酸ラセマーゼMurIの化学合成法の確立2018
- Author(s)
  大原拓己, 野口太朗, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Mirror-image Screening of Chiral Natural Products for SH2 Domain Inhibitors2018
- Author(s)
  Shinya Oishi, Taro Noguchi, Keitou Shu, Kaori Honda, Yasumitsu Kondoh, Hiroyuki Osada, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  10th International Peptide Symposium
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 鏡像スクリーニングを指向したTIGITタンパク質の合成研究2018
- Author(s)
  佐々木順平, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第68回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Synthetic Study of TIGIT Protein for Mirror-Image Screening2018
- Author(s)
  Jumpei Sasaki, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  10th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 鏡像レジデンスを活用した医薬品探索2018
- Author(s)
  大石真也
- Organizer
  日本化学会第98春季年会
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Pd触媒を用いたTHF環構築によるJaspine B 位置異性体の合成研究2018
- Author(s)
  宮川貴吏、本田真歩、中村真也、仲西功、井貫晋輔、大石真也、大野浩章
- Organizer
  日本薬学会第138年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Chemical Synthesis of Glutamate Racemase MurI by Native Chemical Ligation2018
- Author(s)
  Takumi Ohara, Taro Noguchi, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  10th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Screening Platform Using Synthetic Proteins for Access to Mirror-Image Library of Natural Products2018
- Author(s)
  Shinya Oishi
- Organizer
  The 17th Akabori Conference
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] グルタミン酸ラセマーゼMurIの化学合成法の確立2018
- Author(s)
  大原拓己, 野口太朗, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  第68回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 化合物アレイ技術を活用した医薬品探索─鏡の中の天然物からのものづくりに向けて─2018
- Author(s)
  大石真也
- Organizer
  日本化学会第98春季年会
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] グルタミン酸ラセマーゼMurIの化学合成法の確立2018
- Author(s)
  大原拓己, 野口太朗, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  「有機合成化学を起点とするものづくり戦略」最終シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] NK3受容体に作用する繁殖調整剤の創製研究2018
- Author(s)
  山本昂輝, 井貫晋輔, 大野浩章, 大石真也
- Organizer
  「有機合成化学を起点とするものづくり戦略」最終シンポジウム
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Structure Activity Relationship Study of the Helix-Inducible Motif in a Measles Virus Fusion Inhibitor2018
- Author(s)
  Aoi Takahara, Kumi Kawaji, Haruka Sekiguchi, Shinsuke Inuki, Hiroaki Ohno, Nobutaka Fujii, Eiichi Kodama, Shinya Oishi
- Organizer
  10th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] 新規KSP阻害薬のヒト乳癌細胞に対する効果2018
- Author(s)
  太田有紀、土屋聖子、武永美津子、新美純、渡邉大輝、大滝正訓、大石真也、藤井信孝、津川浩一郎、松本直樹
- Organizer
  第138年会日本薬学会
- Data Source
  KAKENHI-PROJECT-15K10074
[Presentation] Facile Fmoc-based Solid-Phase Synthesis of Coibamide2018
- Author(s)
  Takashi Kitamura, Shinsaku Kawaguchi, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi
- Organizer
  10th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-18H02555
[Presentation] Dictyodendrin類の多様性志向型全合成2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  第15回次世代を担う有機化学シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Total synthesis of dictyodendrins by the gold-catalyzed intermolecular cascade cyclization of conjugated diynes with pyrroles2017
- Author(s)
  Junpei Matsuoka, Yuka Matsuda, Yuiki Kawada, Shinya Oishi, Hiroaki Ohno
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 金触媒を用いた分子内連続環化反応を基盤としたAspidophylline Aの全合成研究2017
- Author(s)
  奥村怜司、大原礼子、熊谷洋、大石真也、大野浩章
- Organizer
  第59回天然有機化合物討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2017
- Author(s)
  関口遼、黒柳友子、小林由佳、藤井信孝、大野浩章、大石真也
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dictyodendrin類の網羅的全合成と誘導体の活性評価2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  第43回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 化学合成タンパク質・ペプチドを活用した医薬品探索技術2017
- Author(s)
  大石真也
- Organizer
  メディカルジャパン2017大阪研究成果企業化促進セミナー
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] CXCR7受容体選択的リガンドの構造活性相関研究2017
- Author(s)
  関口遼、黒柳友子、小林由佳、小林数也、赤路健一、藤井信孝、大野浩章、大石真也
- Organizer
  第35回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] キラルな天然物の有効活用を目指した医薬品探索技術2017
- Author(s)
  大石真也
- Organizer
  第7回関西バイオ創薬研究会
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 鏡像体タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2017
- Author(s)
  周敬棠、野口太朗、本田香織、近藤恭光、長田裕之、大野浩章、藤井信孝、大石真也
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Development of peptide macrocyclization protocol utilizing o-aminoanilide linker for flow chemistry2017
- Author(s)
  Takumi Ohara, Masato Kaneda, Tomo Saito, Hiroaki Ohno, Shinya Oishi
- Organizer
  第54回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of novel NK3 receptor antagonists with reduced environmental impact2017
- Author(s)
  Koki Yamamoto, Hiroaki Ohno, Nobutaka Fujii, Shinya Oishi
- Organizer
  254th ACS National Meeting
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 4-epi-Jaspine B位置異性体の合成と構造活性相関研究2017
- Author(s)
  宮川貴吏、本田真歩、小林由佳、中村真也、仲西功、藤井信孝、井貫晋輔、大石真也、大野浩章
- Organizer
  第34回有機合成化学セミナー
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dictyodendrin類の全合成研究2017
- Author(s)
  松岡純平、松田優佳、川田惟樹、大石真也、大野浩章
- Organizer
  日本薬学会第137回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Dbzリンカーを用いた環状ペプチドの合成研究2017
- Author(s)
  大原拓己、金田雅仁、齋藤知、大野浩章、大石真也
- Organizer
  第49回若手ペプチド夏の勉強会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 化学合成タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2016
- Author(s)
  周敬棠、大石真也、野口太朗、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第11回年会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Facile access to the mirror-image library of chiral natural product derivatives: identification of MDM2-p53 interaction inhibitor2016
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Strictamineの不斉形式全合成2016
- Author(s)
  熊谷洋、西山大亮、大石真也、藤井信孝、大野浩章
- Organizer
  第42回反応と合成の進歩シンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of a screening system for Grb2 SH2 domain inhibitors using synthetic proteins2016
- Author(s)
  Taro Noguchi, Hiroyuki Ishiba, Kaori Honda, Yasumitsu Kondoh, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii, Shinya Oishi
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 金触媒を用いたアスピドスペルマ型アルカロイド骨格構築法の開発--Aspidosprmidineの合成研究--2016
- Author(s)
  熊谷洋、大石真也、大野浩章
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Design of iron-chelating cyclic peptides2016
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  8th International Peptide Symposium
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of screening systems for c-Src SH2 domain inhibitors using synthetic proteins2016
- Author(s)
  Keitou Shu, Taro Noguchi, Nobutaka Fujii, Hiroaki Ohno, Shinya Oishi
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Design of Fe(II)-chelaing cyclic hexapeptide with bidentate pyridinyl-triazlole groups2016
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  第53回ペプチド討論会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] ヒト乳癌細胞に対する新規KSP(kinesin spindle protein)阻害薬の効果2016
- Author(s)
  太田有紀, 土屋聖子, 武永美津子, 角田智志, 大滝正訓, 新美純, 大石真也,　藤井信孝, 渡辺実, 武半優子, 飯利太朗, 松本直樹
- Organizer
  第37回日本臨床薬理学会
- Place of Presentation
  米子コンベンションセンター（鳥取県・米子市）
- Year and Date
  2016-12-01
- Data Source
  KAKENHI-PROJECT-15K10074
[Presentation] 長時間作用型PEG化NK3受容体作動薬の創製2016
- Author(s)
  桑井真司、大石真也、三須良介、大野浩章、山村崇、若林嘉浩、岡村裕昭、藤井信孝
- Organizer
  日本薬学会第136回年会
- Place of Presentation
  パシフィコ横浜（神奈川県横浜市）
- Year and Date
  2016-03-26
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 新規合成KSP(Kinesin spindle protein)阻害剤のヒト乳癌細胞に対する抗腫瘍効果に関する研究2016
- Author(s)
  土屋聖子, 太田有紀, 武永美津子, 大滝正訓, 新美純, 大石真也, 藤井信孝, 松本直樹, 津川浩一郎
- Organizer
  第24回日本乳癌学会学術総会
- Place of Presentation
  東京ビッグサイト（東京都・江東区）
- Year and Date
  2016-06-16
- Data Source
  KAKENHI-PROJECT-15K10074
[Presentation] Development of Novel CXCR7 Ligands: Selectivity Switch from CXCR4 Antagonists with Cyclic Pentapeptide Scaffold2016
- Author(s)
  Tomoko Kuroyanagi, Shinya Oishi, Tatsuhiko Kubo, Yuka Kobayashi, Haruka Sekiguchi, Ryosuke Misu, Hiroaki Ohno, Nicolas Montpas, Nikolaus Heveker, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Strictamineの全合成研究2016
- Author(s)
  西山大亮、大原礼子、熊谷洋、千葉浩亮、藤井信孝、大石真也、大野浩章
- Organizer
  第34回メディシナルケミストリーシンポジウム
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Gold-catalyzed construction of tetracyclic skeleton for aspidosperma alkaloid synthesis: Synthetic study on (±)-aspidospermidine2016
- Author(s)
  Hiroshi Kumagai, Shinya Oishi, Hiroaki Ohno
- Organizer
  ISONIS-10
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] MDM2タンパク質の化学合成と天然物の鏡像体化合物群からの医薬品探索への応用2016
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  第36回有機合成若手セミナー
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] ケモカイン受容体CXCR7 選択的リガンドの構造最適化研究2016
- Author(s)
  関口遼、大石真也、黒柳友子、小林由佳、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第11回年会
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Facile access to the mirror-image library of chiral natural product derivatives: identification of MDM2-p53 interaction inhibitor2016
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 創薬シーズ探索のためのものづくり：鏡の中の化合物へのアプローチ2016
- Author(s)
  大石真也
- Organizer
  日本化学会第96春季年会
- Place of Presentation
  同志社大学（京都府京田辺市）
- Year and Date
  2016-03-24
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Total synthesis of a novel cytotoxic depsipeptide from Okinawan marine cyanobacteria2016
- Author(s)
  Masato Kaneda, Shinya Oishi, Kosuke Sueyoshi, Toshiaki Teruya, Hiroaki Ohno and Nobutaka Fujii
- Organizer
  第8回武田振興財団薬科学シンポジウム
- Place of Presentation
  武田研修センター（大阪府吹田市）
- Year and Date
  2016-01-21
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 化学合成タンパク質を利用したc-Src SH2ドメイン阻害剤の探索法の開発2016
- Author(s)
  周敬棠、野口太朗、藤井信孝、大野浩章、大石真也
- Organizer
  第66回日本薬学会近畿支部総会・大会
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 天然物とその誘導体の鏡像体化合物群の活用を目指した新規スクリーニング法の開発2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学川内キャンパス（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Development of Novel CXCR7 Ligands by Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold2015
- Author(s)
  Shinya Oishi, Tomoko Kuroyanagi, Tatsuhiko Kubo, Nicolas Montpas, Yasushi Yoshikawa, Ryosuke Misu, Yuka Kobayashi, Hiroaki Ohno, Nikolaus Heveker, Toshio Furuya, and Nobutaka Fujii
- Organizer
  AIMECS2015
- Place of Presentation
  Jeju international convention center（韓国、済州島）
- Year and Date
  2015-10-18
- Invited / Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Identification of an MDM2-p53 interaction inhibitor from virtual mirror-image library of chiral natural product derivatives2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第52回ペプチド討論会
- Place of Presentation
  平塚市中央公民館（神奈川県平塚市）
- Year and Date
  2015-11-16
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Identification of a novel MDM2-p53 inhibitor using mirror-image-screening technology for chiral natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  SKO symposium
- Place of Presentation
  New Drug Development Center, Seoul University（韓国、ソウル）
- Year and Date
  2015-11-17
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2015
- Author(s)
  黒柳友子，大石真也，小林由佳，関口遼，三須良介，大野浩章，Montpas Nicolas，Heveker Nikolaus，藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] プロパルギル転位を伴う共役ジインの金触媒三連続環化反応を用いたカルバゾールの合成2015
- Author(s)
  田口将光、時水勇輔、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] キラル化合物の有効活用を目指した医薬品探索技術の開発2015
- Author(s)
  大石真也
- Organizer
  第21回ペプチドフォーラム
- Place of Presentation
  東京薬科大学千代田サテライトキャンパス（東京都千代田区）
- Year and Date
  2015-08-29
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 天然物とその誘導体の鏡像体化合物群の活用を目指した新規スクリーニング法の開発2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第10回年会
- Place of Presentation
  東北大学（宮城県仙台市）
- Year and Date
  2015-06-10
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] ケモカイン受容体CXCR7選択的リガンドの構造最適化研究2015
- Author(s)
  黒柳友子，大石真也，久保達彦，三須良介，小林由佳，大野浩章，Montpas Nicolas，Heveker Nikolaus，吉川寧，古谷利夫，藤井信孝
- Organizer
  第65回日本薬学会　近畿支部総会・大会
- Place of Presentation
  大阪大谷大学（大阪府羽曳野市）
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Novel screening approach for drug discovery from virtual mirror-image libaray of natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（米国、ホノルル市）
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] アポモルヒネによるMDM2-p53相互作用の阻害メカニズムの解明2015
- Author(s)
  石場勲之、大石真也、野口太朗、周敬棠、大野浩章、本田香織、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第65回日本薬学会近畿支部大会
- Place of Presentation
  大阪大谷大学（大阪府富田林市）
- Year and Date
  2015-10-17
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Identification of a novel MDM2-p53 inhibitor using mirror-image-screening technology for chiral natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  SKO symposium
- Place of Presentation
  ソウル国際大学（韓国、ソウル市）
- Year and Date
  2015-11-17
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 鏡像体タンパク質を利用した医薬品探索 ─鏡の中の化合物へのアプローチ─2015
- Author(s)
  大石真也
- Organizer
  創薬懇話会2015 in 徳島
- Place of Presentation
  グランドエクシブ鳴門ザ・ロッジ（徳島県鳴門市）
- Year and Date
  2015-07-01
- Invited
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] キラルな天然有機化合物の鏡像体群をリソースとしたMDM2-p53間相互作用阻害剤の探索2015
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] Investigation of inhibitory mechanism of apomorphine against MDM2-p53 interaction2015
- Author(s)
  Hiroyuki Ishiba, Shinya Oishi, Taro Noguchi, Keito Shu, Hiroaki Ohno, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  第52回ペプチド討論会
- Place of Presentation
  平塚市中央公民館（神奈川県平塚市）
- Year and Date
  2015-11-16
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] MDM2-p53タンパク質間相互作用に対するアポモルフィンの阻害メカニズムの解明2015
- Author(s)
  石場勲之、大石真也、野口太朗、周敬棠、大野浩章、藤井信孝
- Organizer
  創薬懇話会2015 in 徳島
- Place of Presentation
  グランドエクシブ鳴門ザ・ロッジ（徳島県鳴門市）
- Year and Date
  2015-07-01
- Data Source
  KAKENHI-PROJECT-15H04653
[Presentation] 環境調和型NK3受容体拮抗剤の創製研究2015
- Author(s)
  山本昂輝、大石真也、大野浩章、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] Novel screening approach for drug discovery from virtual mirror-image library of natural products2015
- Author(s)
  Taro Noguchi, Shinya Oishi, Kaori Honda, Yasumitsu Kondoh, Tamio Saito, Hiroaki Ohno, Hiroyuki Osada, Nobutaka Fujii
- Organizer
  Pacifichem 2015
- Place of Presentation
  Hilton Hawaiian Village（アメリカ、ホノルル）
- Year and Date
  2015-12-15
- Int'l Joint Research
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] PEG修飾による長時間作用型NK3受容体作動薬の創製2015
- Author(s)
  桑井真司、大石真也、三須良介、岡崎志穂、山本昂輝、大野浩章、山村崇、若林嘉浩、岡村裕昭、藤井信孝
- Organizer
  第33回メディシナルケミストリーシンポジウム
- Place of Presentation
  幕張国際研修センター（千葉県幕張市）
- Year and Date
  2015-11-25
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 共役ジインとピロールを用いた金触媒[4+2]型インドール合成と縮環骨格構築への展開2015
- Author(s)
  松田優佳、直江紗織、大石真也、藤井信孝、大野浩章
- Organizer
  第45回複素環化学討論会
- Place of Presentation
  早稲田大学（東京都新宿区）
- Year and Date
  2015-11-19
- Data Source
  KAKENHI-PROJECT-15H04654
[Presentation] 化合物アレイを用いた新規MDM2/MDMX-p53阻害剤探索法の開発2013
- Author(s)
  野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  日本薬学会第133年会
- Place of Presentation
  パシフィコ横浜（神奈川県）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] デフェリフェリクリシン誘導体の合成と構造機能相関研究への応用2013
- Author(s)
  小林由佳、大石真也、小林数也、大野浩章、堤浩子、秦洋二、藤井信孝
- Organizer
  日本薬学会第133年会
- Place of Presentation
  パシフィコ横浜（神奈川県）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] デフェリフェリクリシンの合成と新規キレート錯体の探索2012
- Author(s)
  小林由佳、小林数也、大石真也、堤浩子、秦洋二、大野浩章、藤井信孝
- Organizer
  第7回日本ケミカルバイオロジー学会年会
- Place of Presentation
  京都大学（京都府）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Structure-activity relationship study of neurokinin-3 receptor agonists2012
- Author(s)
  Noguchi T, Oishi S, Misu M, Ohno H, Yamamura T, Okamura H, Fujii N.
- Organizer
  第49回ペプチド討論会
- Place of Presentation
  鹿児島県民交流センター（鹿児島県）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] デフェリフェリクリシンの合成と新規金属キレート錯体の探索2012
- Author(s)
  小林由佳、小林数也、大石真也、大野浩章、堤浩子、秦洋二、藤井信孝
- Organizer
  第44回若手ペプチド夏の勉強会
- Place of Presentation
  ロッジ舞浜（大阪府）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Synthesis and investigation of novel metall complexes of deferriferrichrysin2012
- Author(s)
  小林由佳、小林数也、大石真也、堤浩子、秦洋二、大野浩章、藤井信孝
- Organizer
  第49回ペプチド討論会
- Place of Presentation
  鹿児島県民交流センター（鹿児島県）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Structure-activity relationship study of tachykinin peptides for develpment of novel neurokinin-3 receptor agonists2012
- Author(s)
  Misu R, Oishi S, Noguchi T, Yamada A, Ohno H, Yamamura T, Okamura H, Matsuda F, Ohkura S, Fujii N.
- Organizer
  2nd World Conference on Kisspeptin Signaling in the Brain
- Place of Presentation
  東京大学（東京都）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B) and their sphingosine kinase inhibitory activities2012
- Author(s)
  吉光佑二、宮垣潤、大石真也、藤井信孝、大野浩章
- Organizer
  ISMC2012
- Place of Presentation
  ベルリン（ドイツ）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究2012
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第42回複素環化学討論会
- Place of Presentation
  京都テルサ（京都府）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Development and application of fluorescent probes for monitoring CXCR4 receptor internalization2011
- Author(s)
  Oishi S, Masuda R, Tanahara N, Ohno H, Yano Y, Matsuzaki K, Hirasawa H, Tsujimoto G, Fujii N.
- Organizer
  Nature Chemical Biology Symposium 2011: Cancer Chemical Biology
- Place of Presentation
  Boston（United States of America）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Internalization of CXC chemokine receptor 4 (CXCR4) induced by polyphemusin II-derived antagonist peptides2011
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Nakase I, Futaki S, Fujii N.
- Organizer
  第48回ペプチド討論会
- Place of Presentation
  札幌コンベンションセンター（北海道）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] GPR54リガンドによるNPFF受容体の活性化2011
- Author(s)
  三須良介、大石真也、富田健嗣、説田章平、増田亮、大野浩章、難波陽介、家田菜穂子、井上直子、大蔵聡、上野山賀久、束村博子、前多敬一郎、平澤明、辻本豪三、藤井信孝
- Organizer
  第6回日本ケミカルバイオロジー学会年会
- Place of Presentation
  東京工業大学大岡山キャンパス（東京都）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] アルケン型及びアミジン型ジペプチドイソスターの合成とCXCR4拮抗剤の構造活性相関研究への応用2011
- Author(s)
  小林数也、大石真也、井ノ口恵利子、林亮子、富田健嗣、久保達彦、棚原憲子、大野浩章、藤井信孝、吉川寧、古谷利夫、志村和也、松岡雅雄
- Organizer
  第37回反応と合成の進歩シンポジウム
- Place of Presentation
  あわぎんホール（徳島県）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] アミジン型ペプチド結合等価体の合成と応用2011
- Author(s)
  井ノ口恵利子、山田愛、大石真也、久保達彦、大野浩章、保住健太郎、野水基義、志村和也、松岡雅雄、藤井信孝
- Organizer
  第6回日本ケミカルバイオロジー学会年会
- Place of Presentation
  東京工業大学大岡山キャンパス（東京都）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Synthesis and application of fluorescent SDF-1 derivatives2011
- Author(s)
  Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Structure-activity relationship study on a CXCR4 antagonist FC131 using alkene-type dipeptide isosteres2011
- Author(s)
  Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Naito N, Matsuoka M, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Potent CXCR4 antagonists containing amidine-type peptide bond isosteres2011
- Author(s)
  Kubo T, Inokuchi E, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  AIMECS11
- Place of Presentation
  京王プラザホテル（東京都）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Synthesis and biological evaluation of novel CXCR4 antagonists containing amidine-type peptide bond isosteres2011
- Author(s)
  Inokuchi E, Oishi S, Kubo T, Ohno H, Shimura K, Matsuoka M, Fujii N.
- Organizer
  22nd American Peptide Symposium
- Place of Presentation
  San Diego（United States of America）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Development of novel GPR54 agonists2010
- Author(s)
  Oishi S, et al.
- Organizer
  14th International Congress of Endocrinology, Satellite Symposi
- Place of Presentation
  京都
- Year and Date
  2010-03-30
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Development of novel GPR54 agonists2010
- Author(s)
  Oishi S, et al.
- Organizer
  14th International Congress of Endocrinology, Satellite Symposium
- Place of Presentation
  京都
- Year and Date
  2010-03-30
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 薬剤耐性株に有効な抗HIV活性ペプチドの創製と発現生産プロセスの開発2010
- Author(s)
  大石真也、梶原一美、田中理紀、大野浩章、藤井信孝
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-28
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 縮環インドール構造を有する新規Eg5阻害剤の開発2010
- Author(s)
  竹内智起、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本薬学会第130年会
- Place of Presentation
  岡山
- Year and Date
  2010-03-29
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Development of novel GPR54 agonists14th International Congress of Endocrinology2010
- Author(s)
  Shinya Oishi, Kenji Tomita, Hiroaki Ohno, Nobutaka Fujii.
- Organizer
  Satellite Symposium.
- Place of Presentation
  京都
- Year and Date
  2010-03-30
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  東京
- Year and Date
  2009-08-03
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-18
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Pd-Catalyzed Carbonylation of Amino Acid-Derived Allylic Carbonates2009
- Author(s)
  Inokuchi E, Oishi S, Ohno H, Fujii N, et al.
- Organizer
  8th Australian Peptide Conference
- Place of Presentation
  Queensland Australia
- Year and Date
  2009-10-12
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 固相上におけるペプチド鎖へのDTPAの新規標識法の開発2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ウイルスの変異に学ぶ抗HIV活性ペプチドのデザイン2009
- Author(s)
  大石真也
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-26
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Synthesis and Application of Novel Fluorescent-Labeled CXCR4 Antagonists2009
- Author(s)
  増田亮、大石真也, 他
- Organizer
  第10回文部科学省特定領域研究「がん」5領域若手研究者ワークショップ
- Place of Presentation
  蓼科
- Year and Date
  2009-09-02
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 有機銅-亜鉛複合試薬を用いたトリフルオロメチルアルケンジペプチドイソスターの新規合成法の開発2009
- Author(s)
  小林数也、大石真也, 他
- Organizer
  第35回反応と合成の進歩シンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-16
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Bioorganic Synthesis of End-Capped HIV-1 Fusion Inhibitory Peptides2009
- Author(s)
  Kajiwara K, Oishi S, et al.
- Organizer
  8th Australian Peptide Conference
- Place of Presentation
  Queensland Australia
- Year and Date
  2009-10-12
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] カルバゾール骨格を有する新規Eg5阻害剤のデザインと合成2009
- Author(s)
  渡部敏明、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-19
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 固相上におけるペプチド鎖へのDTPAの新規標識法の開発2009
- Author(s)
  増田亮、大石真也, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した新規化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 有機銅-亜鉛複合試薬を用いたトリフルオロメチルアルケンジペプチドイソスターの新規合成法の開発2009
- Author(s)
  小林数也、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第35回反応と合成の進歩シンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-16
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-18
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4に対する特異的ペプチドT140の蛍光標識プローブを用いた膀胱癌イメージング2009
- Author(s)
  西澤恒二、大石真也, 他
- Organizer
  第68回日本癌学会学術総会
- Place of Presentation
  横浜
- Year and Date
  2009-10-03
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 前立腺癌・膀胱癌に対するkinesin 5(Eg5)新規阻害剤の抗腫瘍効果2009
- Author(s)
  丁森泰、大石真也, 他
- Organizer
  第68回日本癌学会学術総会
- Place of Presentation
  横浜
- Year and Date
  2009-10-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した新規化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4に対する特異的ペプチドT140の蛍光標識プローブを用いた膀胱癌イメージング2009
- Author(s)
  西澤恒二、大石真也, 他
- Organizer
  第68回日本癌学会学術総会
- Place of Presentation
  横浜
- Year and Date
  2009-10-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Efficient Synthesis of Trifluoromethyl and Related Trisubstituted Alkene Dipeptide Isosteres by Pd-Catalyzed Carbonylation of Amino Acid-Derived Allylic Carbonates2009
- Author(s)
  Inokuchi E, Oishi S, et al.
- Organizer
  8th Australian Peptide Conference
- Place of Presentation
  Queensland Australia
- Year and Date
  2009-10-12
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第6回GPCR研究会
- Place of Presentation
  東京
- Year and Date
  2009-05-08
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  東京
- Year and Date
  2009-08-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ペプチドミメティクスの利用による新規GPR54アゴニストの創製2009
- Author(s)
  説田章平、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第6回GPCR研究会
- Place of Presentation
  東京
- Year and Date
  2009-05-08
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した新規化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也, 他
- Organizer
  第59回日本薬学会近畿支部総会
- Place of Presentation
  大阪
- Year and Date
  2009-10-24
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 抗HIV活性ペプチドSC35EKの生物有機化学的合成2009
- Author(s)
  梶原一美、大石真也, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  金沢
- Year and Date
  2009-11-05
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Synthesis and Application of Novel Fluorescent-Labeled CXCR4 Antagonists2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第10回文部科学省特定領域研究「がん」5領域若手研究者ワークショップ
- Place of Presentation
  蓼科
- Year and Date
  2009-09-02
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 固相上におけるペプチド鎖へのDTPAの新規標識法の開発2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  日本ケミカルバイオロジー研究会第4回年会
- Place of Presentation
  神戸
- Year and Date
  2009-05-18
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ケモカイン受容体CXCR4選択的蛍光プローブを活用した化合物評価系の構築2009
- Author(s)
  棚原憲子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第46回ペプチド討論会
- Place of Presentation
  北九州
- Year and Date
  2009-11-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Synthesis and Application of Novel Fluorescent-Labeled CXCR4 Antagonists2009
- Author(s)
  増田亮、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第10回文部科学省特定領域研究「がん」5領域若手研究者ワークショップ
- Place of Presentation
  蓼科
- Year and Date
  2009-09-02
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] アルケン型ジペプチドイソスターの合成とケモカイン受容体CXCR4拮抗剤の構造活性相関研究への応用2009
- Author(s)
  林亮子、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 縮環インドール構造を有する新規Eg5阻害剤の開発2009
- Author(s)
  竹内智起、大石真也、大野浩章、藤井信孝, 他
- Organizer
  第28回メディシナルケミストリーシンポジウム
- Place of Presentation
  東京
- Year and Date
  2009-11-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 環状ベプチドをリードとする非ペプチド性CXCR4拮抗剤の開発2008
- Author(s)
  大石真也, 他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 多様なジペフチドイゾースターの分岐的合成とGPR54アゴニストへの応用2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第27回メディシナルケミストリーシンポジウム
- Place of Presentation
  大阪
- Year and Date
  2008-11-26
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Development of novel non-peptide CXCR4 antagonists based on cyclic peptide structure2008
- Author(s)
  Oishi S., Katoh M., Ueda S., Inuki S., Ohno H., Barry Evans, Zi-xuan Wang, Stephen C. Peiper, Fujii N.
- Organizer
  3rd Annual Meeting of Japan Chemical Biology Society
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of Novel Pseudopeptide GPR54 Agonists with High Tolerance against MMP-Mediaed Digestion2008
- Author(s)
  Kenji Tomita, Shinya Oishi,Nobutaka Fujii, 他
- Organizer
  XXth International Symposium on Medicinal Chemistry
- Place of Presentation
  ウイーン
- Year and Date
  2008-09-01
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 新規ファルマコフォアを有するケモカインレセプターCXCR4アンタゴニストの構造活性相関研究2008
- Author(s)
  田中智博、大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-20
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] CXCR4 Antagonists : Relevance to Cancer Chemotherapy2008
- Author(s)
  Nobutaka Fujii, Shinya Oishi
- Organizer
  XXth International Symposium on Medicinal Chemistry
- Place of Presentation
  ウイーン
- Year and Date
  2008-09-03
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] マトリックスメタロプロテアーゼ耐性GPR54アゴニストの開発2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第45回ペプチド討論会
- Place of Presentation
  東京
- Year and Date
  2008-10-29
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Novel labeling protocol for cell-membrane proteins by tag-probe method-2008
- Author(s)
  Yano Y., Yano A., Oishi S., Sugimoto Y., Tsujimoto G., Fujii N., Matsuszaki K.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of fluorescent CXCR4 antagonist2008
- Author(s)
  Masuda R., Oishi S., Ueda S., Evans B., Peiper SC, Hirasawa A., Tsujimoto G., Ohno H., Fujii N.
- Organizer
  3rd Annual Meeting of Japan Chemical Biology Society
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也、藤井信孝、他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Design and synthesis of anti-HIV peptides having helix-inducible motifs2008
- Author(s)
  Watanabe K., Oishi S., Itoh S., Tanaka M., Hishikawa H., Watabe T., Izumi K., Sakagami Y., Kodama E., Matsuoka M., Ohno H., Fujii N.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] ジペプチドイソスターの分岐型合成による酵素耐性GPR54アゴニストの創出2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ペプチド結合とペプチドミメティクス2008
- Author(s)
  大石真也
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ペプチド・蛋白質化学を基盤とする新興・再興感染症治療薬の創製2008
- Author(s)
  大石真也
- Organizer
  第5回バイオメディカル研究会
- Place of Presentation
  大阪
- Year and Date
  2008-02-13
- Data Source
  KAKENHI-PROJECT-17790091
[Presentation] Model development for virtual screening of CYP-interactive compounds using CCA spatial model2008
- Author(s)
  Ogawa T., Minowa Y., Adachi T., Feng C, Niijima S., Oishi S., Fujii N., Okuno Y.
- Organizer
  5th Seminars on Biomedical Researches
- Place of Presentation
  Osaka
- Year and Date
  2008-02-13
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] X-ray crystal structure analysis of 6-helical bundle structure of T-20 (Fuzeon) -resistant HIV mutants2008
- Author(s)
  Watabe T., Oishi S., Nishikawa H., Watanabe K., Nakano H., Nakatsu T., Ohno H., Katoh H., Kodama E., Matsuoka M., Fujii N.
- Organizer
  88th Spring meeting of the chemical society of Japan
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] ジペプチドイソスターの分岐型合成による酵素耐性GPR54アゴニストの創出2008
- Author(s)
  富田健嗣、大石真也, 他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-04
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 多様なジペプチドイソスターの分岐的合成と応用2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第28回有機合成若手セミナー
- Place of Presentation
  大阪
- Year and Date
  2008-11-12
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4に対する蛍光標識リカンドの創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也、藤井信孝、他
- Organizer
  第45回ペプチド討論会
- Place of Presentation
  東京
- Year and Date
  2008-10-29
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 環状ペプチドをリードとする非ペプチド性CXCR4拮抗剤の開発2008
- Author(s)
  大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也、藤井信孝、他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Structure-activity relationship on CXCR4 antagonists having novel pharmacophores2008
- Author(s)
  Tanaka T., Tabe Y., Ohhashi N., Haseyama M., Tsutsumi H., Nomura W., Itoya K., Esaka R.,Oishi S., Fujji N., Wang Z., Peiper SC, Evans B., Tamamura H.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relathionship on pyrazine-based CK2 inhibitors2008
- Author(s)
  Suzuki Y., Cluzeau J., Oishi S., Ohno H., Fujii N., Hara T., Hirasawa A., Tsujimoto G.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Establishment of bioevaluation technology for drug discovery for GPCR -novel labeling protocol for cell-membrane proteins by tag-probe method-2008
- Author(s)
  Yano Y., Oishi S., Sugimoto Y., Tsujimoto G., Fujii N., Matsuzaki K.
- Organizer
  The 1st Symposium on Target Protein Research Program
- Place of Presentation
  Tokyo
- Year and Date
  2008-02-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也、藤井信孝、他
- Organizer
  第45回ペプチド討論会
- Place of Presentation
  東京
- Year and Date
  2008-10-29
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-04
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 多様なジペプチドイソスターの分岐的合成と応用2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第28回有機合成若手セミナー
- Place of Presentation
  大阪
- Year and Date
  2008-11-12
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 多様なジペプチドイソスターの分岐的合成とGPR54アゴニストへの応用2008
- Author(s)
  富田健嗣、大石真也, 他
- Organizer
  第27回メディシナルケミストリーシンポジウム
- Place of Presentation
  大阪
- Year and Date
  2008-11-26
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] CXCR4 Antagonists: Relevance to Cancer Chemotherapy2008
- Author(s)
  Nobutaka Fujii, Shinya Oishi
- Organizer
  XXth International Symposium on Medicinal Chemistry
- Place of Presentation
  ウイーン
- Year and Date
  2008-09-03
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也, 他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Contribution to chemical library by preparation of novel fragment compound -efficient synthesis of multi-substituted heterocycles having drug-like strucure-2008
- Author(s)
  Fujii N., Ohno H., Oishi S., Takemoto Y., Takasu K, Yasui Y., Tomioka K., Yamada K., Yamamoto Y.
- Organizer
  The 1st Symposium on Target Protein Research Program
- Place of Presentation
  Tokyo
- Year and Date
  2008-02-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也, 他
- Organizer
  第45回ペプチド討論会
- Place of Presentation
  東京
- Year and Date
  2008-10-29
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 環状ペプチドをリードとする非ペプチド性CXCR4拮抗剤の開発2008
- Author(s)
  大石真也, et al.
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of ergot alkaloids by paradium-catalyzed domino cyclizations of allenes2008
- Author(s)
  Inuki S., Oishi S., Fuji N., Ohno H.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of Z-alkene and E-fluoroalkene dipeptide isosteres as cis-amide bond equivalents2008
- Author(s)
  Tomita K, Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] ジペプチドイソスターの分岐型合成による酵素耐性GPR54アゴニストの創出2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第34回反応と合成の進歩シンポジウム
- Place of Presentation
  京都
- Year and Date
  2008-11-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] ペプチド結合とペプチドミメティクス2008
- Author(s)
  大石真也
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-03
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] ケモカイン受容体CXCR4に対する蛍光標識リガンドの創製と応用2008
- Author(s)
  増田亮、大石真也, 他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Synthesis of nitrogen heterocycles by palladium-catalyzed sp3 C-H activation.2008
- Author(s)
  Toshiaki Watanabe, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno
- Organizer
  The 9th Youngnam-Kinki Joint Symposium on Organometallic Chemistry
- Place of Presentation
  Kyoto
- Year and Date
  2008-01-25
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-04
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 環状ペプチドをリードとする非ペプチド性CXCR4拮抗剤の開発2008
- Author(s)
  大石真也、加藤学、上田聡、井貫晋輔、大野浩章、Barry Evans、Zi-xuan Wang、Stephen C.Peiper、藤井信孝
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 多様なジペプチドイソスターの分岐的合成と応用2008
- Author(s)
  富田健嗣、大石真也, 他
- Organizer
  第28回有機合成若手セミナー
- Place of Presentation
  大阪
- Year and Date
  2008-11-12
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] Development of screening system for anti-cancer lead compounds -for HIF-1-targeting agents -2008
- Author(s)
  Hattori A., Yagura T., Nishimura S., Oishi S., Fujii N., Kakeya H.
- Organizer
  The 1st Symposium on Target Protein Research Program
- Place of Presentation
  Tokyo
- Year and Date
  2008-02-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Selection of Chemicals for General Library2008
- Author(s)
  Yasuno K., Kojima H., Okabe T., Oishi S., Fujii N., Nagano T. Furuya T.
- Organizer
  The 1st Symposium on Target Protein Research Program
- Place of Presentation
  Tokyo
- Year and Date
  2008-02-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] CXCR4受容体アンタゴニストの蛍光標識体の創製と応用2008
- Author(s)
  増田亮、大石真也, 他
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-04
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] 多様なジペプチドイソスターの分岐的合成とGPR54アゴニストへの応用2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第27回メディシナルケミストリーシンポジウム
- Place of Presentation
  大阪
- Year and Date
  2008-11-26
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] 環状ペプチドをリードとする非ペプチド性CXCR4拮抗剤の開発2008
- Author(s)
  大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-19
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] 新規ファルマコフォアを有するケモカインレセプターCXCR4アンタゴニストの構造活性相関研究2008
- Author(s)
  田中智博、大石真也、藤井信孝、他
- Organizer
  日本ケミカルバイオロジー研究会第3回年会
- Place of Presentation
  東京
- Year and Date
  2008-05-20
- Data Source
  KAKENHI-PROJECT-20057011
[Presentation] Development of Novel Pseudopeptide GPR54 Agonists withHigh Tolerance against MMP-Mediaed Digestion2008
- Author(s)
  Kenji Tomita, Shinya Oishi, Nobutaka Fujii, 他
- Organizer
  XXth International Symposium on Medicinal Chemistry
- Place of Presentation
  ウイーン
- Year and Date
  2008-09-01
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Synthesis and application of fluorescent CXCR4 antagonist2008
- Author(s)
  Masuda R., Oishi S., Ueda S., Barry Evans, Stephen C. Peiper, Hirasawa A., Tsujimoto G., Ohno H., Fujii N.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective synthesis of trifluoromethylalkene dipeptide isosteres by nucliophilic CF3-introduction2008
- Author(s)
  Kobayashi K., Narumi T., Inokuchi E., Tomita K., Oishi S., Ohno H., Fujii N.
- Organizer
  The 128th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] ケモカイン受容体CXCR4に対する蛍光標識リガンドの創製と応用2008
- Author(s)
  増田亮、大石真也、藤井信孝、他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Structure-activity relathionship on pyrazine-based CK2 inhibitors2008
- Author(s)
  Suzuki Y., Jerome Cluzeau, Hara T., Hirasawa A., Tsujimoto G., Oishi S., Ohno H., Fujii N.
- Organizer
  3rd Annual Meeting of Japan Chemical Biology Society
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] ペプチド結合とペプチドミメティクス2008
- Author(s)
  大石真也
- Organizer
  第41回若手ペプチド夏の勉強会
- Place of Presentation
  京都
- Year and Date
  2008-08-03
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] マトリックスメタロプロテアーゼ耐性GPR54アゴニストの開発2008
- Author(s)
  富田健嗣、大石真也、藤井信孝、他
- Organizer
  第45回ペプチド討論会
- Place of Presentation
  東京
- Year and Date
  2008-10-29
- Data Source
  KAKENHI-PROJECT-20015021
[Presentation] Structure-activity relationship on CXCR4 antagonists having novel pharmacophores2008
- Author(s)
  Tanaka T., Nomura W., Tsutsumi H., Tabe Y., Ohhashi N., Itoya K., Oishi S., Fujii N., Evans B., Wang Z., Peiper SC, Tamamura H.
- Organizer
  3rd Annual Meeting of Japan Chemical Biology Society
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] 求核的CF3化反応による立体選択的トリフルオロメチルアルケン型ジペプチドイソスターの合成研究2008
- Author(s)
  小林数也、大石真也, 他
- Organizer
  第58回日本薬学会近畿支部総会
- Place of Presentation
  神戸
- Year and Date
  2008-10-25
- Data Source
  KAKENHI-PROJECT-20790098
[Presentation] ベプチド・蛋白質化学を基盤とする新興・再興感染症治療薬の創製2008
- Author(s)
  大石真也
- Organizer
  第5回バイオメディカル研究会
- Place of Presentation
  大阪
- Year and Date
  2008-02-13
- Data Source
  KAKENHI-PROJECT-18060020
[Presentation] Structure-activity relationship study on GPR54 agonist as novel anti-metastatic agent.2007
- Author(s)
  Tomita K., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  First JCA-AACR Special Joint Conference : The Latest Advances in Lung Cancer Research : From Basic Science to Therapeutics
- Place of Presentation
  Nagoya
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] From amino acids to peptide isosteres: Implication to genome-lead drug discovery.2007
- Author(s)
  Fujii N., Oishi S., Narumi T., Tomita K., Ohno H.
- Organizer
  2nd. World Congress of Pharmacy and Pharmaceutical Sciences
- Place of Presentation
  Beijing
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of fluorescent CXCR4 antagonist2007
- Author(s)
  Masuda R., Oishi S., Ueda S., Gotoh S., Ohno H., Evans B., Peiper SC, Hirasawa A., Tsujimoto G., Kodama E., Matsuoka M., Fujii N.
- Organizer
  44th Japanese Peptide Symposium
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] CXCR4 antagonists : Relevance to small cell lung cancer chemotherapy.2007
- Author(s)
  Fujii N., Oishi S., Ueda S.
- Organizer
  First JCA-AACR Special Joint Conference : The Latest Advances in Lung Cancer Research : From Basic Science to Therapeutics
- Place of Presentation
  Nagoya
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Anti-HIV activity of water-soluble analogue of C29, SC29EK2007
- Author(s)
  Naitoh T., Izumi K., Kodama E., Oishi S., Fujii N., Matsuoka M.
- Organizer
  21st Annual meeting of the Japan Society for AIDS research
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective synthesis of peptidomimetics based on acid-catalyzed ring-opening of □-aziridinyl-□, □-enoates.2007
- Author(s)
  Tamamura H., Tanaka T., Tsutsumi H., Nemoto K., Mizokami S., Ohashi N., Oishi S., Fujii N.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling2007
- Author(s)
  Watanabe T., Inuki S., Ueda S., Oishi S., Ohno H., Fujii N.
- Organizer
  6th AFMC International Medicinal Chemistry Symposium
- Place of Presentation
  Istanbul
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] From knowledge to controlling : implications of peptide-lead drug templates for genome-lead discovery.2007
- Author(s)
  Nobutaka Fujii, Hiroaki Ohno, Shinya Oishi
- Organizer
  RIKEN International Symposium on Chemical Biology
- Place of Presentation
  Hakone
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Design and synthesis of novel HIV fusion inhibitors2007
- Author(s)
  Shinya Oishi, et al.
- Organizer
  Virus Molecular Interactions : Therapeutic Targets
- Place of Presentation
  オックスフォード
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Construction of 2-(aminomethyl)indole motif by Cu-catalyzed multi-component reaction.2007
- Author(s)
  Ohta Y., Oishi S., Fujii N., Ohno H.
- Organizer
  234th ACS meeting & exposition
- Place of Presentation
  Boston
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Plasma concentration of metastins in pancreatic cancer patients2007
- Author(s)
  Katagiri F., Nagai K., Kida M., Tomita K., Oishi S., Takeyama M., Doi R., Fujii N.
- Organizer
  2nd annual meeding of Japan Chemical Biology Society
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of synthetic methodology for fused aromatic compounds by consecutive bond formations2007
- Author(s)
  Ohno H., Ohta Y., Oishi S., Fujii N., Iuchi M., Tanaka T.
- Organizer
  The 33rd Symposium on Progress in Organic Reactions in the Life Sciences
- Place of Presentation
  Nagasaki
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Pd-Catalyzed carbonylation of CF3-containing allylic carbonate : application to the synthesis of (Z)-trifluoromethylalkene dipeptide isosteres.2007
- Author(s)
  Inokuchi E., Narumi T., Tomita K., Niida A., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Organizer
  14th IUPAC Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
- Place of Presentation
  Nara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of a novel fusion inhibitor against T-20-resistant HIV-1.2007
- Author(s)
  Oishi S., Ito S., Nishikawa H., Tanaka M., Ohno H., Otaka A., Izumi K., Kodama E., Matsuoka M., Fujii N.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of fusion inhibitors against feline immunodeficiency virus (FIV)2007
- Author(s)
  Nishikawa H., Kodera Y., Tanaka M., Mizukoshi F., Tsujimoto H., Kodama E., Matsuoka M., Oishi S., Ohno H., Fujii N.
- Organizer
  2nd annual meeding of Japan Chemical Biology Society
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of trifluoroalkene dipeptide isosteres and the related compounds using paradium-catalyzed carbonylation2007
- Author(s)
  Inokuchi E., Narumi T., Niida A., Tomita K, Oishi S., Ohno H., Fujii N.
- Organizer
  27th Seminars on Organic Synthesis for Young Scientists
- Place of Presentation
  Kyoto
- Year and Date
  2007-11-15
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel FIV membrane fusion inhibitors.2007
- Author(s)
  Nishikawa H., Kodera Y., Oishi S., Tanaka M., Tochikura T., Kajiwara K., Ohno H., Mizukoshi F., Tsujimoto H., Kodama E., Matsuoka M., Fujii N.
- Organizer
  Virus Molecular Interactions : Therapeutic Targets
- Place of Presentation
  Oxford
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of ergot alkaloids by paradium-catalyzed domino cyclizations of allenes2007
- Author(s)
  Inuki S., Oishi S., Fuji N., Ohno H.
- Organizer
  The 57th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Osaka
- Year and Date
  2007-10-27
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and in vivo evaluation of 18F labeled fluorobenzoyl pentapeptide ([18F]TOM80) as a PET imaging agent for GPR54.2007
- Author(s)
  T. Fuchigami, N. Harada, H. Tsukada, M. Ogawa, H. Yamaguchi, H. Raku, K. Tomita, S. Ohishi, N. Fujii, Y. Magata
- Organizer
  Seventh Japan-China Joint Semiinar on Radiopharmaceutical Chemistry
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents.2007
- Author(s)
  Tomita K., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of trifluoroalkene dipeptide isosteres and the related compounds using paradium-catalyzed carbonylation2007
- Author(s)
  Inokuchi E., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  The 33rd Symposium on Progress in Organic Reactions in the Life Sciences
- Place of Presentation
  Nagasaki
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Design and synthesis of anti-HIV peptides having helix-inducible motifs2007
- Author(s)
  Watanabe K., Itoh S., Nishikawa H., Tanaka M., Oishi S., Ohno H., Izumi K., Kodama E., Matsuoka M., Fujii N.
- Organizer
  44th Japanese Peptide Symposium
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and structure-activity relationship on cystein derivatives having Eg5 inhibiory activity2007
- Author(s)
  Ogo N., Oishi S., Matsuno K., Sawada J., Fujii N., Asai A.
- Organizer
  The 26th Symposium on Medicinal Chemistry
- Place of Presentation
  Sagamihara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of fluoroalkenes of organometal-mediated C-F bond cleavage : application of stereoselective synthesis of multifunctionalized fluoroalkene dipeptide isosteres2007
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Organizer
  The 57th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Osaka
- Year and Date
  2007-10-27
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of carbazoles by palladium-catalyzed tandem N-arylation and oxidative C-H activation2007
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  Eighth Tetrahedron Symposium
- Place of Presentation
  Berlin
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of a novel fusion inhibitor against T-20-resistant HIV-12007
- Author(s)
  Shinya Oishi, et al.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  モントリオール
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel CXCR4 antagonist having an indole scaffold2007
- Author(s)
  Katoh M., Ueda S., Inuki S., Oishi S., Ohno H., Evans B., Wang Z., Peiper SC, Fujii N.
- Organizer
  The 26th Symposium on Medicinal Chemistry
- Place of Presentation
  Sagamihara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Prediction of drugcytochrome P450 interaction using chemical-biological correlation space model.2007
- Author(s)
  Teppei Ogawa, Yosuke Minowa, Tetsuya Adachi, Chunlai Fen, Satoshi Niijima, Shinya Oishi, Nobutaka Fujii, Yasushi Okuno
- Organizer
  Annual meeding of CBI society
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of fusion inhibitors based on resistant mutation against T-202007
- Author(s)
  Izumi K., Kodama E., Shimura K., Oishi S., Fujii N., Matsuoka M.
- Organizer
  21st Annual meeting of the Japan Society for AIDS research
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Palladium-catalyzed synthesis of carbazole by tandem N-arylation and C-H activation.2007
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 5th Symposium on Organic Chemistry - The Next Generation
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Design and synthesis of novel HIV fusion inhibitors.2007
- Author(s)
  〓inya Oishi
- Organizer
  Virus Molecular Interactions: Therapeutic Targets
- Place of Presentation
  Oxford
- Year and Date
  2007-09-17
- Data Source
  KAKENHI-PROJECT-17790091
[Presentation] Stereoselective synthesi of (Z)-trifluoromethylalkene dipeptide isosteres2007
- Author(s)
  Inokuchi E., Narumi T., Niida A., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Organizer
  The 127th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of a Novel Fusion Inhibitor against T-20-resistant HIV-1.2007
- Author(s)
  Oishi S.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Year and Date
  2007-06-29
- Data Source
  KAKENHI-PROJECT-17790091
[Presentation] Construction of 2-(aminomethyl)indole motif by Cu-catalyzed multi-component reaction.2007
- Author(s)
  Ohta Y., Oishi S., Fujii N., Ohno H.
- Organizer
  14th IUPAC Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
- Place of Presentation
  Nara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of (Z)-alkene and (E)-fluoroalkene dipeptide isosteres as cis amide equivalents2007
- Author(s)
  Tomita K., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  2nd annual meeding of Japan Chemical Biology Society
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Fluoroalkenes for peptidomimetics2007
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Kobayashi K., Oishi S., Ohno H., Fujii N.
- Organizer
  44th Japanese Peptide Symposium
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of Highly potent HIV fusion inhibitors2007
- Author(s)
  Tanaka M., Itoh S., Oishi S., Nishikawa H., Izumi K., Kodama E., MatsuokE M., Ohno H., Fujii N.
- Organizer
  2nd annual meeding of Japan Chemical Biology Society
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] HIV activity of T-20 derivatives2007
- Author(s)
  Shimane K., Izumi K., Kodama E., Oishi S., Fujii N., Matsuoka M.
- Organizer
  21st Annual meeting of the Japan Society for AIDS research
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of a Novel Fusion Inhibitor against T-20-resistant HIV-12007
- Author(s)
  Oishi S.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Year and Date
  2007-06-29
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of chemokine receptor CXCE4 antagonists using bio-mimetic strategy.2007
- Author(s)
  Tamamura H., Tanaka T., Tsutsumi H., Ohashi N., Hiramatsu K., Araki T., Ojida A., Hamachi I., Wang Z., Peiper SC, Trent JO., Ueda S., Oishi S., Fujii N.
- Organizer
  20th American Peptide Symposium
- Place of Presentation
  Montreal
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Palladium-catalyzed synthesis of carbazole by tandem N-arylation and C-H activation.2007
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 127th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of highly potent HIV fusion inhibitors by application of EK concept2007
- Author(s)
  Itoh S., Oishi S., Nishikawa H., Tanaka M., Watanabe K., Izumi K., Kodama E., Matsuoka M., Ohno H., Fujii N.
- Organizer
  The 127th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-affinity relationship study on fluorobenzoyl pentapeptides for GPR542007
- Author(s)
  Tomita K., Oishi S., Ohno H., Fujii N.
- Organizer
  The 127th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Propertie of intracellular fragment peptides of mouse prostaglandin E2 receptor mEP3b isoform.2007
- Author(s)
  Shinbo S., Yano Y., Oishi S., Fujii N., Sugimoto Y., Matsuzaki K.
- Organizer
  44th Japanese Peptide Symposium
- Place of Presentation
  Toyama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of GPR54 agonists as anti-metastasis agents.2007
- Author(s)
  Tomita K., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  The 8th workshop for cancer research for young scientists
- Place of Presentation
  Tateshina
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel CXCR4 antagonist having an indole scaffold2007
- Author(s)
  Katoh M., Ueda S., Inuki S., Oishi S., Ohno H., Fujii N.
- Organizer
  The 57th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Osaka
- Year and Date
  2007-10-27
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Unprecedented palladium- mediated carbon-fluorine bond cleavage : relevance to the synthesis of fluoroalkene dipeptidomimetics.2007
- Author(s)
  Narumi T., Inokuchi E., Tomita K, Oishi S., Ohno H., Fujii N.
- Organizer
  American Chemical Society 233rd National Meeting & Exposition
- Place of Presentation
  Chicago
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of ergot alkaloids by paradium-catalyzed domino cyclizations of allenes2007
- Author(s)
  Inuki S., Oishi S., Fuji N., Ohno H.
- Organizer
  27th Seminars on Organic Synthesis for Young Scientists
- Place of Presentation
  Kyoto
- Year and Date
  2007-11-15
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of synthetic method for trifluoromethylalkene dipeptide isosteres by paradium-catalyzed carbonylation2007
- Author(s)
  Inokuchi E., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  The 57th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Osaka
- Year and Date
  2007-10-27
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and applicatior of carbazoles by palladium-catalyzed tandem N-arylation and oxidative C-H activation.2007
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  14th IUPAC Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
- Place of Presentation
  Nara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Design and synthesis of novel HIV fusion inhibitors.2007
- Author(s)
  Oishi S., Ito S., Nishikawa H., Tanaka M., Ohno H., Otaka A., Izumi K., Kodama E., Matsuoka M., Fujii N.
- Organizer
  Virus Molecular Interactions : Therapeutic Targets
- Place of Presentation
  Oxford
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and application of Z-alkene and E-fluoroalkene dipeptide isosteres as cis-amide bond equivalents2007
- Author(s)
  Tomita K., Narumi T., Niida A., Oishi S., Ohno H., Fujii N.
- Organizer
  The 26th Symposium on Medicinal Chemistry
- Place of Presentation
  Sagamihara
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Design and synthesis of novel HIV fusion inhibitors2007
- Author(s)
  Shinya Oishi
- Organizer
  Virus Molecular Interactions: Therapeutic Targets
- Place of Presentation
  Oxford
- Year and Date
  2007-09-17
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres : Lys-Lys and Glu-Glu type FADIs.2007
- Author(s)
  Narumi T., Kodera Y., Tomita K., Inokuchi E., Oishi S., Ohno H., Fujii N.
- Organizer
  234th ACS meeting & exposition
- Place of Presentation
  Boston
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of cyclic pentapeptide- based CXCR4 antagonists for the treatment of CXCR4-mediated diseases.2007
- Author(s)
  Ueda S., Oishi S., Wang Z., Ohno H., Peiper SC, Fujii N.
- Organizer
  First JCA-AACR Special Joint Conference : The Latest Advances in Lung Cancer Research : From Basic Science to Therapeutics
- Place of Presentation
  Nagoya
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of fluoroalkenes by paradium-catalyzed C-F bond cleavage2006
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Oishi S., Ohno H., Fujii N.
- Organizer
  The 32th Symposium on Progress in Organic Reactions in the Life Sciences
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structureactivity relationship study on GPR54 agonists.2006
- Author(s)
  Tomita K., Niida A., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  ICOB-5 & ISCNP-25 IUPAC International Conference on Biodiversity and Natural Products
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship studies on cyclic peptide-based CXCK4 antagonists.2006
- Author(s)
  eda S., Oishi S., Wang Z., Araki T., Tamamura H., Ohno H., NakashimaH., Peiper SC, Fujii N.
- Organizer
  ICOB-5 & ISCNP-25 IUPAC International Conference on Biodiversity and Natural Products
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Discovery of novel low-molecular-weight GPR54 agonists.2006
- Author(s)
  Shinya Oishi, Kenji Tomita, Ayumu Niida, Miki Akamatsu, Toshihiko Masui, Ryuichiro Doi, Jean-Marc Navenot, Zixang Wang, Stephen C. Peiper, Nobutaka Fujii
- Organizer
  29th European Peptide Symposium
- Place of Presentation
  Gdansk
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Diastereoselective synthesis of (Z)-fluoroalkene dipeptide isosteres based on organocopper-mediated reduction/direct alkylation via transmetalation.2006
- Author(s)
  Tetsuo Narumi, Kenji Tomita, Ayumu Niida, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  29th European Peptide Symposium
- Place of Presentation
  Gdansk
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship studies on GPR54 agonists2006
- Author(s)
  Tomita K., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  The International Conference of 43rd Japanese Peptide Symposium and 4th Peptide Engineering Meeting
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of chemokine receptor CXCR4 antagonists having bivalent Zn-complex structure2006
- Author(s)
  Ogawa T., Tamamura H., Ojida A., Tsutsumi H., Masuno H., Nakajima H., Yamamoto N., Oishi S., Ohno H., Hamachi I., Fujii N.
- Organizer
  The 56th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Kyoto
- Year and Date
  2006-10-28
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesi of calbazoles by paradium-mediated tandem N-arylation and C-H activation2006
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 56th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Kyoto
- Year and Date
  2006-10-28
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of carbazoles by paradium-catalyzed tandem N-arylation and C-H activation2006
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 23rd Seminars on Organic Chemistry
- Place of Presentation
  Onuma
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] From amino acids to peptide isosteres : Implications to peptide-lead drug templates for genome-lead drug discovery.2006
- Author(s)
  Nobutaka Fujii, Shinya Oishi, Tetsuo Narumi, Kenji Tomita, Hiroaki Ohno
- Organizer
  232nd American Chemical Society National Meeting & Exposition
- Place of Presentation
  San Francisco
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Novel synthesis of fluoroalkene isosteres utilizing paradium-catalyzed cleavage of C-F bond activation2006
- Author(s)
  Narumi T., Niida A., Tomita K., Oishi S., Otaka A., Ohno H., Fujii N.
- Organizer
  The 126th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Sendai
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of synthetic methodology toward (Z)-fluoro- alkene dipeptide isosteres based on the concept of organometalic-mediated C-F bond cleavage.2006
- Author(s)
  Tetsuo Narumi, Kenji Tomita, Ayumu Niida, Yasuyo Kodera, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  ICOB-5 & ISCNP-25 IUPAC International Conference on Biodiversity and Natural Products
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] One-pot synthesis of carbazoles using paradium-catalyzed tandem N-arylation and C-H activation2006
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 7th Nagai Nagayoshi Memorial Symposium
- Place of Presentation
  Tokushima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] シスアミド等価型アルケンジベプチドイソスターの合成と応用2006
- Author(s)
  大石真也, et al.
- Organizer
  第32回反応と合成の進歩シンポジウム
- Place of Presentation
  広島
- Description
  「研究成果報告書概要(和文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Allylic hydrodefluorination under palladium catalysis for the synthesis of fluoroalkene dipeptide isosteres.2006
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Oishi S., Ohno H., Fujii H.
- Organizer
  The 10th International KYOTO Conference on New Aspects of Organic Chemistry
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of 2-(aminomethyl)indoles by organocopper-catalyzed three-component coupling2006
- Author(s)
  Ohta Y., Oishi S., Fujii N., Ohno H.
- Organizer
  The 56th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Kyoto
- Year and Date
  2006-10-28
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of highly potent HIV fusion inhibitors based on EK-concept2006
- Author(s)
  Itoh S., Oishi S., Nishikawa H., Tanaka M., Izumi K., Kodama E., Matsuoki M., Ohno H., Fujii N.
- Organizer
  The 25th Symposium on Medicinal Chemistry
- Place of Presentation
  Nagoya
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesi and application of cis-amide equivalent alkene dipeptide isosteres2006
- Author(s)
  Oishi S., Niida A., Narumi T., Tomita K., Inokuchi E., Ohno H., Kitaura K., Fujii N., Otaka A., Inui K.
- Organizer
  The 32th Symposium on Progress in Organic Reactions in the Life Sciences
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship study on novel CXCR4 antagonists having a cyclic scaffold2006
- Author(s)
  Watanabe T., Esaka R., Ogawa T., Ueda S., Tamamura H., Oishi S., Trent, JO., Wang, Z., Peiper, SC. Fujii N.
- Organizer
  The 126th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Sendai
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel antiviral agents against T-20 registant HIV2006
- Author(s)
  Itoh S., Oishi S., Nishikawa H., Tanaka M., Izumi K., Kodama E., Matsuoka M., Ohno H., Fujii N.
- Organizer
  The 56th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Kyoto
- Year and Date
  2006-10-28
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel CXCR4 antagonists having bivalent Zn-complexes2006
- Author(s)
  Ogawa T., Tamamura H., Ojida A., Tsutsumi H., Nakajima H., Oishi S., Ohno H., Hamachi I., Fujii N.
- Organizer
  The 25th Symposium on Medicinal Chemistry
- Place of Presentation
  Nagoya
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] A novel oxazolidine linker for the synthesis of peptide aldehydes.2006
- Author(s)
  Tanaka M., Oishi S., Ohno H., Fujii N.
- Organizer
  The International Conference of 43rd Japanese Peptide Symposium and 4th Peptide Engineering Meeting
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] New peptide design for HIV-1 fusion inhibitors against T-20resistant HIV-1 variants.2006
- Author(s)
  Nishikawa H., Kodama E., Ito S., Kajiwara K., Izumi K., Oishi S., Matsuoka M., Fujii N.
- Organizer
  The 3rd Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Place of Presentation
  Seoul
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Establishment anc clinical application of an enzyme immunoassay for metastin to determination of the human plasma levels.2006
- Author(s)
  Katagiri F., Tomita K., Oishi S., Takeyama M., Fujii N.
- Organizer
  The International Conference of 43rd Japanese Peptide Symposium and 4th Peptide Engineering Meeting
- Place of Presentation
  Yokohama
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of a novel photo-labile protecting group having 4(dimethylamino)phenacyl group and the application to peptide synthesis2006
- Author(s)
  Ueda S., Tomita K., Nomura M., Otaka A., Oishi S., Ohno H., Fujii N.
- Organizer
  1st Annual Meeting of Japan Chemical Biology Society
- Place of Presentation
  Tokyo
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] SAR and QSAR studies on N-terminal moieties of pentapeptide GPR54 agonists2006
- Author(s)
  Tomita K., Niida A., Harada T., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  The 126th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Sendai
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship studies on N-terminal acyl groups of pentapeptidic GPR54 agonists.2006
- Author(s)
  Tomita K., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  The 3rd Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists
- Place of Presentation
  Seoul
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Palladium-catalyzed synthesis of carbazole by tandem N-arylation and C-H activation.2006
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  The 10th International KYOTO Conference on New Aspects of Organic Chemistry
- Place of Presentation
  Kyoto
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of fluoroalkenes by paradium-catalyzed C-F bond cleavage2006
- Author(s)
  Narumi T., Tomita K., Inokuchi E., Oishi S., Ohno H., Fujii N.
- Organizer
  26th Seminar on Organic Synthesis for Young Scientists
- Place of Presentation
  Osaka
- Year and Date
  2006-12-14
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel photolabile protecting groups for carboxyl- and amino-groups2006
- Author(s)
  Ogawa T., Ueda S., Oishi S., Ohno H., Fujii N.
- Organizer
  33rd Seminars on Organic Reactions
- Place of Presentation
  Kyotanabe
- Year and Date
  2006-08-03
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective synthesis of (Z)-trifluoromethylalkene dipeptide isosteres and the application to bioactive peptides2006
- Author(s)
  Inokuchi E., Narumi T., Niida A., Tomita K., Oishi S., Ohno H., Fujii N.
- Organizer
  33rd Seminars on Organic Reactions
- Place of Presentation
  Kyotanabe
- Year and Date
  2006-08-03
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of novel photo-labile 4-(dimethylamino)phenacyl-type protecting groups for chemical biology2006
- Author(s)
  Ogawa T., Ueda S., Nomura M., Otaka A., Oishi S., Ohno H., Fujii N.
- Organizer
  Seminars on Biomedical Researches
- Place of Presentation
  Osaka
- Year and Date
  2006-09-12
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of 2-(aminomethyl)indoles by organocopper-mediated three-component coupling2006
- Author(s)
  Ohta Y., Oishi S., Fujii N., Ohno H.
- Organizer
  26th Seminar on Organic Synthesis for Young Scientists
- Place of Presentation
  Osaka
- Year and Date
  2006-12-14
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereselective synthesi of (Z)-trifluororhethyl alkene dipeptide isosteres and the application to bioactive peptides2006
- Author(s)
  Inokuchi E., Narumi T., Niida A., Tomita K., Oishi S., Ohno H., Fujii N.
- Organizer
  The 41th Seminars on Natural Products
- Place of Presentation
  Hokkaido
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of fluoroalkenes by organometal-mediated C-F bond cleavage : Application to highly functionalized fluoroalkene dipeptide isosteres2006
- Author(s)
  Narumi T., Tomita K., Niida A., Oishi S., Otaka A., Ohno H., Fujii N.
- Organizer
  The 4th Symposium on Organic Chemistry - The Next Generation -
- Place of Presentation
  Osaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship study on GPR54 agonists2006
- Author(s)
  Tomita K., Oishi S., Ohno H., Akamatsu M., Fujii N.
- Organizer
  The 34th Symposium on Structure-Activity Relationships
- Place of Presentation
  Niigata
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Development of anti-FIV agents having fusion inhibitory activiry2006
- Author(s)
  Kodera Y., Nishikawa H., Tanaka M., Mizukoshi F., Tsujimoto H., Kodama E., Matsuoka M., Oishi S., Ohno H., Fujii N.
- Organizer
  The 56th Kinki Regional Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Kyoto
- Year and Date
  2006-10-28
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Highly stereoselective synthesis of fluoroalkene isosteres and the application to bioactive peptides2006
- Author(s)
  Narumi T., Miyatani T., Niida A., Tomita K., Oishi S., Otaka H., Ohno H., Fujii N.
- Organizer
  The 126th Annual Meeting of the Pharmaceutical Society of Japan
- Place of Presentation
  Sendai
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Palladium-catalyzed synthesis of carbazole by tandem N-arylation and C-H activation.2006
- Author(s)
  Watanabe T., Ueda S., Oishi S., Fujii N., Ohno H.
- Organizer
  26th Seminar on Organic Synthesis for Young Scientists
- Place of Presentation
  Osaka
- Year and Date
  2006-12-14
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis of 2-(aminomethyl)indoles by organocopper-mediated three-component coupling2006
- Author(s)
  Ohta Y., Oishi S., Fujii N.. Ohno H.
- Organizer
  The 32th Symposium on Progress in Organic Reactions in the Life Sciences
- Place of Presentation
  Hiroshima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship studies on cyclic peptide-based CXCR4 antagonists : Side-chain and backbone modifications.2006
- Author(s)
  Satoshi Ueda, Shinya Oishi, Zixuan Wang, Hiroaki Ohno, Stephen C. Peiper, Nobutaka Fujii
- Organizer
  232nd American Chemical Society National Meeting & Exposition
- Place of Presentation
  San Francisco
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Solid-phase synthesis of peptide aldehydes using an oxazolidine linker2006
- Author(s)
  Tanaka M., Oishi S., Ohno H., Fujii N.
- Organizer
  The 7th Nagai Nagayoshi Memorial Symposium
- Place of Presentation
  Tokushima
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective of multi-functionalized fluoroalkene dipeptide isosteres2005
- Author(s)
  Narumi T., Niida A., Tomita K., Oishi S., Ohno H., Otaka H., Fujii N.
- Organizer
  Seminar on Organic Synthesis for Young Scientists
- Place of Presentation
  Kobe
- Year and Date
  2005-11-24
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres2005
- Author(s)
  Narumi T., Niida A., Tomita K., Oishi S., Otaka A., Ohno H., Fujii N.
- Organizer
  42th Japanese Peptide Symposium
- Place of Presentation
  Osaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and bioevaluation of peptidomimetics of CXCR4 antagonist FC1312005
- Author(s)
  Tamamura H., Hiramatsu K., Araki T., Ueda S., Oishi S., Esaka R., Zixuan Wang, Stephen C. Peoper, John 0. Trent, Nakajima H., Yamamoto N., Otaka A., Fujii N.
- Organizer
  42th Japanese Peptide Symposium
- Place of Presentation
  Osaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity study on small-molecule GPR54 agonists2005
- Author(s)
  Tomita K., Niida A., Oishi S., Ohno H., Otaka A., Fujii N.
- Organizer
  The 24th Symposium on Medicinal Chemistry
- Place of Presentation
  Oosaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Structure-activity relationship study on RW-amide-type hOT7T175 agonist2005
- Author(s)
  Tomita K., Niida A., Oishi S., Ohno H., Otaka A., Fujii N.
- Organizer
  42th Japanese Peptide Symposium
- Place of Presentation
  Osaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Stereoselective of multi-functionalized fluoroalkene dipeptide isosteres2005
- Author(s)
  Narumi T., Niida A., Tomita K, Oishi S., Ohno H., Otaka A., Fujii N.
- Organizer
  The 24th Symposium on Medicinal Chemistry
- Place of Presentation
  Oosaka
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Unequivocal synthesis of (Z)-alkene or (E)-fluoroalkene dipeptide isosteres via DKP mimetics to probe structural orrequirements of peptide transporter.2005
- Author(s)
  Niida A., Oishi S., Mizumoto M., Sasaki Y., Tomita K., Tamamura H., Otaka A., Terada T., Inui K. Fujii N.
- Organizer
  19th American Peptide Symposium
- Place of Presentation
  San Diego
- Description
  「研究成果報告書概要(欧文)」より
- Data Source
  KAKENHI-PROJECT-17209004
[Presentation] Synthesis and Functional Analysis of Deferriferrichrysin Derivatives
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Kazuya Kobayashi, Hiroaki Ohno, Hiroko Tsutsumi, Yoji Hata, Nobutaka Fujii
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] 新規ニューロキニン-3受容体アゴニストの創製研究
- Author(s)
  山本昂輝、大石真也、三須良介、野口太朗、大野浩章、山村崇、岡村裕昭、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学（大阪府豊中市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] キスペプチン受容体に対する蛍光プローブの創製研究
- Author(s)
  金田雅仁、大石真也、三須良介、大野浩章、藤井信孝
- Organizer
  日本薬学会第134年会
- Place of Presentation
  熊本大学黒髪キャンパス（熊本県熊本市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 化合物アレイを用いた新規mdm2/mdmx-p53阻害剤の探索法の開発とその応用
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第31回メディシナルケミストリーシンポジウム
- Place of Presentation
  アステールプラザ（広島県広島市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] ペプチダーゼ耐性を有する新規NK3受容体アゴニストの創製研究
- Author(s)
  三須良介、大石真也、山田愛、山本昂輝、野口太朗、大野浩章、山村崇、岡村裕昭、松田二子、大蔵聡、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学（大阪府豊中市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] NK3受容体リガンドの安定性評価と新規選択的アゴニストの創製
- Author(s)
  山田愛、三須良介、大石真也、大野浩章、松田二子、大蔵聡、藤井信孝
- Organizer
  第62回日本薬学会近畿支部大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、岩田顕、大槻和裕、丸山透、大石真也、大野浩章、藤井信孝
- Organizer
  日本ケミカルバイオロジー学会　第9回年会
- Place of Presentation
  大阪大学（大阪府豊中市）
- Year and Date
  2014-06-11 – 2014-06-13
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] ニューロキニン-3受容体アゴニストの構造活性相関研究
- Author(s)
  山本昂輝、三須良介、野口太朗、大野浩章、大石真也、山村崇、岡村裕昭、藤井信孝
- Organizer
  第11回GPCR研究会
- Place of Presentation
  日本科学未来館（東京都江東区）
- Year and Date
  2014-05-09 – 2014-05-10
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 生体機能の解明に向けたものづくり：生物活性環状ペプチドの設計と応用
- Author(s)
  大石真也
- Organizer
  第3回化学フェスタ
- Place of Presentation
  タワーホール船堀（東京都江戸川区）
- Invited
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Synthesis and functional characterization of fluorescent probes for GPR54
- Author(s)
  Masato Kaneda, Ryosuke Misu, Shinya Oishi, Hiroaki Ohno, and Nobutaka Fujii
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館（京都府京都市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 化合物アレイを用いた新規mdm2/mdmx-p53阻害剤の探索法の開発とその応用
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  第63回日本薬学会近畿支部大会
- Place of Presentation
  同志社女子大学（京都府京田辺市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Design and synthesis of fluorescent probes for GPR54
- Author(s)
  Masato Kaneda, Ryosuke Misu, Shinya Oishi, Hiroaki Ohno, and Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク（大阪府吹田市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] スフィンゴシンキナーゼ阻害活性を有するJaspine B誘導体の構造活性相関研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、岩田顕、大槻和裕、丸山透、中村真也、仲西功、大石真也、大野浩章、藤井信孝
- Organizer
  第32回メディシナルケミストリーシンポジウム
- Place of Presentation
  神戸国際会議場（兵庫県神戸市）
- Year and Date
  2014-11-26 – 2014-11-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] 新規ニューロキニン-3受容体アゴニストの創製研究
- Author(s)
  山本昂輝、大石真也、三須良介、野口太朗、大野浩章、山村崇、岡村裕昭、藤井信孝
- Organizer
  創薬懇話会2014 in 岐阜
- Place of Presentation
  ぎふ長良川温泉　ホテルパーク（岐阜県岐阜市）
- Year and Date
  2014-07-10 – 2014-07-11
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Development of Photoaffinity Probes for Characterization of the Receptor Binding Residues in Kisspeptins
- Author(s)
  Shinya Oishi, Shohei Setsuda, Ryosuke Misua Taro Noguchi, Masato Kaneda, Hiroaki Ohno, Barry Evans, Jean-Marc Navenot, Stephen C. Peiper, Nobutaka Fujii
- Organizer
  23rd American Peptide Symposium
- Place of Presentation
  ヒルトンワイコロアホテル（米国、コナ市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Synthesis of IB-01212 by Site-Selective N-Methylation of Peptide Bonds
- Author(s)
  ○Ryota Nabika, Shinya Oishi, Ryosuke Misu, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク（大阪府吹田市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Structure-activity Relationship Study of Tachykinin Peptides for Development of Novel Neurokinin-3 Receptor Selective Agonists
- Author(s)
  Ryosuke Misu, Shinya Oishi, Taro Noguchi, Ai Yamada, Hiroaki Ohno, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  23rd American Peptide Symposium
- Place of Presentation
  ヒルトンワイコロアホテル（米国、コナ市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Synthesis and Investigation of Ferrichrysin Derivatives
- Author(s)
  Yuka Kobayashi, Shinya Oishi, Kazuya Kobayashi, Hiroaki Ohno, Hiroko Tsutsumi, Yoji Hata, Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク（大阪府吹田市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] ウイルス変異に基づく抗HIV活性ペプチドのデザイン
- Author(s)
  大石真也
- Organizer
  生命分子機能研究会2013学術集会
- Place of Presentation
  長浜バイオ大学（滋賀県長浜市）
- Invited
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 鉄(II)イオン配位性ペプチドの設計と機能評価
- Author(s)
  小林由佳、大石真也、大野浩章、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  デザイン・クリエイティブセンター神戸（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Development of Novel Kinesin Spindle Protein (KSP) Inhibitors
- Author(s)
  Shinya Oishi
- Organizer
  The First Asian Conference for ''MONODUKURI'' Strategy by Synthetic Organic Chemistry
- Place of Presentation
  Southern Beach Hotel & Resort Okinawa（沖縄県糸満市）
- Invited
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] NK3受容体アゴニストの生体内安定性評価と新規誘導体の創製
- Author(s)
  三須良介、大石真也、山田愛、山本昂輝、野口太朗、大野浩章、山村崇、岡村裕昭、松田二子、大蔵聡、藤井信孝
- Organizer
  第11回GPCR研究会
- Place of Presentation
  日本科学未来館（東京都江東区）
- Year and Date
  2014-05-09 – 2014-05-10
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Kinesin Spindle Protein (KSP) Inhibitors with Diaryl Amine Scaffolds
- Author(s)
  Shinya Oishi, Tomoki Takeuchi, Hiroaki Ohno, Jun-ichi Sawada, Akira Asai, Nobuaka Fujii
- Organizer
  9th AFMC International Medicinal Chemistry Symposium
- Place of Presentation
  The Grand Hotel, Taipei（台湾、台北市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Optimization of neurokinin-3 receptor (NK3R)-selective agonists
- Author(s)
  Koki Yamamoto, Shinya Oishi, Ryosuke Misu, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Nobutaka Fujii
- Organizer
  第51回ペプチド討論会
- Place of Presentation
  徳島大学（徳島県徳島市）
- Year and Date
  2014-10-22 – 2014-10-24
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Jaspine Bおよびその誘導体の多様性指向型合成研究
- Author(s)
  宮垣潤、吉光佑二、大石真也、藤井信孝、大野浩章
- Organizer
  第62回日本薬学会近畿支部大会
- Place of Presentation
  武庫川女子大学（兵庫県）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Identification of Novel MDM2/MDMX-p53 interaction inhibitors by chemical array technology
- Author(s)
  ○野口太朗、大石真也、久保達彦、大野浩章、近藤恭光、斎藤臣雄、長田裕之、藤井信孝
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館（京都府京都市）
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Coibamide Aの合成研究
- Author(s)
  松田剛、並河亮太、大石真也、大野浩章、藤井信孝
- Organizer
  第63回日本薬学会近畿支部大会
- Place of Presentation
  同志社女子大学（京都府京田辺市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Characterization of the Receptor Binding Residues of Kisspeptins by Using Photoaffinity Probes
- Author(s)
  Ryosuke Misu, Shinya Oishi, Shohei Setsuda, Taro Noguchi, Masato Kaneda, Hiroaki Ohno, Barry Evans, Jean-Marc Navenot, Stephen C. Peiper, Nobutaka Fujii
- Organizer
  2nd Annual Conference ICBS2013
- Place of Presentation
  京都大学芝蘭会館（京都府京都市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 天然物の鏡像体化合物群の活用を目指した新規スクリーニング法の開発
- Author(s)
  野口太朗、大石真也、本田香織、近藤恭光、斎藤臣雄、大野浩章、長田裕之、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  デザイン・クリエイティブセンター神戸（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] クロスメタセシス反応を利用したスフインゴシンキナーゼ阻害剤の創製研究
- Author(s)
  本田真歩、宮垣潤、吉光佑二、大槻和裕、丸山透、中村真也、仲西功、大石真也、大野浩章、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  兵庫医療大学（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-24659046
[Presentation] Synthetic Studies on Coibamide A
- Author(s)
  Ryota Nabika, Shinya Oishi, Hiroaki Ohno, Nobutaka Fujii
- Organizer
  The First Asian Conference for ''MONODUKURI'' Strategy by Synthetic Organic Chemistry
- Place of Presentation
  Southern Beach Hotel & Resort Okinawa（沖縄県糸満市）
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] Evaluation of Biological Stability of Neurokinin-3 Receptor Agonists for the Development of Novel Biostable Analogs
- Author(s)
  Ryosuke Misu, Shinya Oishi, Taro Noguchi, Ai Yamada, Hiroaki Ohno, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  4th Asia-Pacific International Peptide Symposium
- Place of Presentation
  ホテル阪急エキスポパーク（大阪府吹田市）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 光アフィニティープローブを利用したキスペプチン類の受容体結合残基の同定
- Author(s)
  三須良介、大石真也、説田章平、野口太朗、金田雅仁、大野浩章、藤井信孝
- Organizer
  第8回ケミカルバイオロジー学会年会
- Place of Presentation
  東京医科歯科大学（東京都文京区）
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] ペプチド結合のN-メチル化反応を利用したIB-01212の合成研究
- Author(s)
  並河亮太、大石真也、三須良介、大野浩章、藤井信孝
- Organizer
  第40回反応と合成の進歩シンポジウム
- Place of Presentation
  東北大学　川内萩ホール（宮城県仙台市）
- Year and Date
  2014-11-10 – 2014-11-11
- Data Source
  KAKENHI-PROJECT-24659004
[Presentation] 新規ニューロキニン-3受容体アゴニストの創製と繁殖中枢制御への応用
- Author(s)
  山本昂輝、大石真也、三須良介、野口太朗、大野浩章、山村崇、岡村裕昭、藤井信孝
- Organizer
  日本薬学会第135年会
- Place of Presentation
  兵庫医療大学（兵庫県神戸市）
- Year and Date
  2015-03-26 – 2015-03-28
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] 縮環インドール類の新しい生物活性の探索：KSP阻害剤の創製
- Author(s)
  大石真也
- Organizer
  有機合成化学を起点とするものづくり戦略ミニシンポジウム
- Place of Presentation
  東京大学（東京都）
- Invited
- Data Source
  KAKENHI-PROJECT-23689007
[Presentation] Development of novel neurokinin-3 receptor selective agonists with resistance against proteolytic degradation
- Author(s)
  Ryosuke Misu, Shinya Oishi, Ai Yamada, Koki Yamamoto, Taro Noguchi, Hiroaki Ohno, Takashi Yamamura, Hiroaki Okamura, Fuko Matsuda, Satoshi Ohkura, Nobutaka Fujii
- Organizer
  第51回ペプチド討論会
- Place of Presentation
  徳島大学（徳島県徳島市）
- Year and Date
  2014-10-22 – 2014-10-24
- Data Source
  KAKENHI-PROJECT-23689007

1. FUJII Nobutaka (60109014)

# of Collaborated Projects: 9 results

# of Collaborated Products: 303 results
2. OHNO Hiroaki (30322192)

# of Collaborated Projects: 5 results

# of Collaborated Products: 103 results
3. 野中元裕 (70514173)

# of Collaborated Projects: 4 results

# of Collaborated Products: 17 results
4. HATTORI Akira (50300893)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
5. NISHIMURA Shinichi (30415260)

# of Collaborated Projects: 2 results

# of Collaborated Products: 0 results
6. UENOYAMA Yoshihisa (70324382)

# of Collaborated Projects: 2 results

# of Collaborated Products: 2 results
7. Kondo Yasumitsu (80333342)

# of Collaborated Projects: 2 results

# of Collaborated Products: 18 results
8. FUJIWARA Hiroshi (30252456)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
9. INOUE Hideshi (20184765)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
10. MARUYAMA Masato (00399445)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
11. ISHII Hirotaka (20445810)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
12. SUWA Makiko (30242241)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
13. MAGATA Yasuhiro (20209399)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
14. SAKAHARA Harumi (10187031)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
15. OGAWA Mikako (20344351)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
16. HIRANO Toru (30313951)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
17. TSUKADA Hideo (10393951)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
18. MASUTANI Hiroshi (50252523)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
19. ITOH Shinji (50362512)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
20. Saito Tamio (40260228)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
21. Kashiwada Yoshiki (30169429)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
22. Chihiro Tsukano (70524255)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
23. NAKANISHI Isao (10362576)

# of Collaborated Projects: 1 results

# of Collaborated Products: 2 results
24. Ohta Yuki (60387066)

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
25. 渡部毅 (00397788)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
26. 武永美津子 (10236490)

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
27. 大滝正訓 (20612683)

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
28. 束村博子 (00212051)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
29. 大蔵聡 (20263163)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
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# of Collaborated Projects: 1 results

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31. 羽田真悟 (40553441)

# of Collaborated Projects: 1 results

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32. 真方文絵 (50635208)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
33. 渡辺雄貴 (50781788)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
34. 中村翔 (50829223)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
35. 井上直子 (90377789)

# of Collaborated Projects: 1 results

# of Collaborated Products: 1 results
36. 児玉栄一 (50271151)

# of Collaborated Projects: 1 results

# of Collaborated Products: 2 results
37. 木村寛之 (50437240)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
38. 樋口隆弘 (30739850)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
39. 大黒多希子 (30767249)

# of Collaborated Projects: 1 results

# of Collaborated Products: 0 results
40. TSUCHIYA Seiko

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
41. NIIMI Jun

# of Collaborated Projects: 1 results

# of Collaborated Products: 4 results
42. KUWATA Takeo

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
43. 斉藤臣雄

# of Collaborated Projects: 0 results

# of Collaborated Products: 10 results
44. 前多敬一郎

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
45. 松下修三

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
46. 廣田毅

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results
47. 中瀬生彦

# of Collaborated Projects: 0 results

# of Collaborated Products: 1 results

Oishi Shinya 大石 真也

OISHI Shinya 大石 真也

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Development of Platform Technlogy for Therapeutic Applications of Mirror-image Functional ProteinsPrincipal Investigator

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Development of mirror-image antibody-like scaffolds and their applicationsPrincipal Investigator

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Development of Screening Platform for Mirror-image Antibody-like ScaffoldsPrincipal Investigator

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Development of Drug Discovery Technologies Using Mirror-image BiomoleculesPrincipal Investigator

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Develoment of a screening platform using mirror-image proteins and their application to drug discoveryPrincipal Investigator

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Oishi Shinya 大石真也

OISHI Shinya 大石真也