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Kunishima Munetaka  国嶋 崇隆

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… Alternative Names

KUNISHIMA Munetaka  国嶋 崇隆

国嶋 崇隆  クニシマ ムネタカ

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Researcher Number 10214975
Other IDs
External Links
Affiliation (Current) 2025: 神戸学院大学, 薬学部, 教授
Affiliation (based on the past Project Information) *help 2023 – 2025: 神戸学院大学, 薬学部, 教授
2008 – 2022: Kanazawa University, 薬学系, 教授
2007: Kobe Gakuin University, 薬学部, 教授
2006: 神戸学院大学, 薬学部, 助教授
2003 – 2004: 神戸学院大学, 薬学部, 助教授 … More
2002: 神戸学院大学, 薬学部, 講師
1998 – 1999: 神戸学院大学, 薬学部, 講師
1992: 神戸学院大学, 薬学部, 助手
1990: 神戸学院大学, 薬学部 Less
Review Section/Research Field
Principal Investigator
Chemical pharmacy / Chemical pharmacy / Medium-sized Section 47:Pharmaceutical sciences and related fields / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related / Basic Section 47050:Environmental and natural pharmaceutical resources-related
Except Principal Investigator
Basic Section 52040:Radiological sciences-related / Medium-sized Section 52:General internal medicine and related fields / Radiation science / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Tumor therapeutics / Risk sciences of radiation and chemicals / Medical pharmacy
Keywords
Principal Investigator
アミド / トリアジン / 脱水縮合 / 脱離基 / カルボカチオン / 脱水縮合剤 / 一分子求核置換反応 / アルキル化反応 / 含窒素複素環 / アルキル化剤 … More / 触媒反応 / トリアジノン / タンパク質 / 分子認識 / アリール化 / 対アニオン / 有機カチオン / 第4級アンモニウム / バイオコンジュゲーション / 抗体 / 求核置換反応 / 官能基変換 / 求核反応 / カルボカチオノイド / アルコール / SN1反応 / アルキル化 / カチオン安定化 / カチオン発生法 / トリアジン及び誘導体 / 一分子脱離反応 / 脱アミノ化剤 / リガンド / 反応剤 / アシル化剤 / 酸化剤 / 1,3,5-トリアジン / 親水性ゲル / エポキシ化剤 / 縮合剤 / 含窒素芳香族化合物 / bioorganic chemistry / dehydrocondensation / molecular recognistion / acyltransfer / amides / enzyme models / Host-Guest / クラウンエーテル / シクロデキストリン / ホストーゲスト / 超分子 / ホスト-ゲスト / 超分子化学 / 触媒的アミド化 / 人工酵素 / アシル基転移酵素 / 生物有機化学 / 脱水縮合反応 / アシル基転移 / 酵素モデル / ホストゲスト / 不斉アルキル化 / Carbocations / Asymmetric induction / 含窒素芳香環 / エステル / 電子欠乏性含窒素芳香環 / タンパク質検索 / タンパク質探索 / 標的タンパク質 / 標識化反応 / カリクサジン / カルボン酸 / オキサゾリン / 脂質 / ホスト化合物 / 標識化 / 脂質合成 / リポソーム / スフィンゴシン / セラミド / 膜融合 / アミド化反応 / 反応触媒 / 高分子化学 / モレキュラーインプリンティング … More
Except Principal Investigator
分子イメージング / 核医学 / セラノティクス / セラノスティクス / がん / SPECT / 放射性画像診断薬 / 個別化薬物療法 / 薬物代謝酵素活性 / 個体差要因 / 低分子化合物 / 阻害剤 / ヌクレオチド除去修復 / 胆汁排泄 / 核医学画像診断薬 / アミノ酸トランスポーター / 細胞内レドックス制御 / レドックス制御 / 画像診断薬 / トランスポーター / 治療標的 / がん細胞 / PET / SGLT / on water現象 / ミセル / ペプチド合成 / 水中合成 / 環境調和型合成 / がん関連アミノ酸トランスポーター / グルタミノリシス / 核医学画像診断法 / 汎用的基盤形成 / 薬効・副作用の個体差要因 / 薬物療法 / 代謝酵素活性測定 / 個別化適正使用 / cytochrome P450 / 核医学画像診断 / 代謝酵素活性 / 薬物代謝酵素 / 抗がん剤 / トランスポータ / 小動物イメージング / 個別化医療 / 薬物トランスポータ / 多剤耐性 / 個別化治療 / 増感作用 / シスプラチン / 抗癌剤 / 神経化学的評価 / 放射性診断薬 / 分子標的 / 治療効果判定 / 個体差 / 治療効果 / 遺伝子発現解析 / 精神神経疾患 / スクリーニング / 化合物ライブラリー / ケミカルバイオロジー / MRP2 / 薬物誘導性肝障害 / 可視化 / 副作用 / 薬物間相互作用 / 肝細胞 / 輸送体 Less
  • Research Projects

    (25 results)
  • Research Products

    (240 results)
  • Co-Researchers

    (33 People)
  •  カルボカチオノイド化学における学理の深化とその実践的展開Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      2025 – 2028
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
      Basic Section 47050:Environmental and natural pharmaceutical resources-related
      Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related
    • Research Institution
      Kobe Gakuin University
  •  Environmentally benign synthesis: development of a technique for the chemical synthesis of peptides in water using micelles as a reaction field.

    • Principal Investigator
      北條 恵子
    • Project Period (FY)
      2024 – 2026
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
    • Research Institution
      Kobe Gakuin University
  •  テトラアリールアンモニウムの合成法の開発Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      2023 – 2025
    • Research Category
      Grant-in-Aid for Challenging Research (Exploratory)
    • Review Section
      Medium-sized Section 47:Pharmaceutical sciences and related fields
    • Research Institution
      Kobe Gakuin University
  •  Development of Mitochondria-Targeted Theranostic Agents for Cancer-Specific Glutaminolysis

    • Principal Investigator
      小林 正和
    • Project Period (FY)
      2022 – 2024
    • Research Category
      Grant-in-Aid for Challenging Research (Exploratory)
    • Review Section
      Medium-sized Section 52:General internal medicine and related fields
    • Research Institution
      Kanazawa University
  •  細胞内レドックス制御を司るがん幹細胞治療の標的トランスポーター画像診断薬の開発

    • Principal Investigator
      川井 恵一
    • Project Period (FY)
      2022 – 2025
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Review Section
      Basic Section 52040:Radiological sciences-related
    • Research Institution
      Kanazawa University
  •  Establishment of methodology for controlling carbocations and its application to nucleophilic substitution reactionsPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2021 – 2023
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
    • Research Institution
      Kobe Gakuin University
      Kanazawa University
  •  Development of a highly selective bioconjugation method using protein interactionsPrincipal Investigator

    • Principal Investigator
      Kunishima Munetaka
    • Project Period (FY)
      2021 – 2022
    • Research Category
      Grant-in-Aid for Challenging Research (Exploratory)
    • Review Section
      Medium-sized Section 47:Pharmaceutical sciences and related fields
    • Research Institution
      Kanazawa University
  •  Development of theranostics probes targeting sodium-dependent glucose transporters

    • Principal Investigator
      小林 正和
    • Project Period (FY)
      2021 – 2024
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Review Section
      Basic Section 52040:Radiological sciences-related
    • Research Institution
      Kanazawa University
  •  Control of short-lived highly reactive carbocation species for drug discovery and life science applicationsPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2019 – 2020
    • Research Category
      Grant-in-Aid for Challenging Research (Exploratory)
    • Review Section
      Medium-sized Section 47:Pharmaceutical sciences and related fields
    • Research Institution
      Kanazawa University
  •  Establishment of Nuclear Medicine Diagnostic Method to Evaluate Drug Metabolizing Enzyme Activity for Personalized Pharmacotherapy Optimization

    • Principal Investigator
      Kawai Keiichi
    • Project Period (FY)
      2018 – 2020
    • Research Category
      Grant-in-Aid for Challenging Research (Exploratory)
    • Review Section
      Medium-sized Section 52:General internal medicine and related fields
    • Research Institution
      Kanazawa University
  •  Development of novel reagents taking the advantage of the electron deficient nitrogen-containing heterocyclesPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2017 – 2020
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kanazawa University
  •  Development of high accuracy multidrug resistance prediction method using SPECT imaging for individualized anticancer therapy

    • Principal Investigator
      KOBAYASHI Masato
    • Project Period (FY)
      2015 – 2017
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Radiation science
    • Research Institution
      Kanazawa University
  •  Development of novel pi-electron deficient nitrogen-containing heterocycles for dehydrocondensationsPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2014 – 2016
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kanazawa University
  •  Asymmetric induction by using carbocations as a reactive speciesPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2014 – 2015
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kanazawa University
  •  Application of chemical biology to a mechanistic study of human nucleotide excision repair

    • Principal Investigator
      MATSUNAGA Tsukasa
    • Project Period (FY)
      2013 – 2015
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Risk sciences of radiation and chemicals
    • Research Institution
      Kanazawa University
  •  Development of a molecular targeted radiolabeled diagnostic agent useful for personalized drug therapy of psychoneurotic diseases

    • Principal Investigator
      KAWAI Keiichi
    • Project Period (FY)
      2013 – 2016
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Radiation science
    • Research Institution
      Kanazawa University
  •  Analysis of a novel small-molecule compound inducing the degradation of a cisplatin resistance-related factor ERCC1

    • Principal Investigator
      MATSUNAGA Tsukasa
    • Project Period (FY)
      2013 – 2014
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Tumor therapeutics
    • Research Institution
      Kanazawa University
  •  Development of Efficient Sensing Method for Targeting Proteins Based on Dehydrocondensing ReactionsPrincipal Investigator

    • Principal Investigator
      KUNISHIMA MUNETAKA
    • Project Period (FY)
      2011 – 2013
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kanazawa University
  •  Application of Sandwich-cultured hepatocytes for analysis of drug-drug interaction on bile canalicular transporters

    • Principal Investigator
      TAMAI Ikumi
    • Project Period (FY)
      2011 – 2012
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Medical pharmacy
    • Research Institution
      Kanazawa University
  •  DEVELOPMENT OF REACTION FIEILDS FOR DEHYDROCONDENSATIONS TOWARD CREATION OF NEW TECHNOLOGIES ON THE BASIS OF TRIAZINE CHEMISTRYPrincipal Investigator

    • Principal Investigator
      KUNISHIMA Munetaka
    • Project Period (FY)
      2008 – 2010
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kanazawa University
  •  二本鎖脂質分子の膜内での化学合成によって誘起される膜の形態変化に関する研究Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      2006 – 2007
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kobe Gakuin University
  •  Development and application of artificial acyltransferase models based on host compoundsPrincipal Investigator

    • Principal Investigator
      KUNISHIMA Munetaka
    • Project Period (FY)
      2002 – 2004
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kobe Gakuin University
  •  新規な分子インプリンティング法を用いた反応触媒高分子の開発Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      1998 – 1999
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kobe Gakuin University
  •  2価希土類元素の特性を活用した分子内カルベン挿入反応の開発Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      1992
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kobe Gakuin University
  •  アルキリデンカルベンを活性種とする分子内環化反応の開発と医薬品合成への応用Principal Investigator

    • Principal Investigator
      国嶋 崇隆
    • Project Period (FY)
      1990
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Kobe Gakuin University

All 2024 2023 2022 2021 2020 2019 2018 2017 2016 2015 2014 2013 2012 2011 2010 2009 2008 2007 2006 2005 2004 2002 Other

All Journal Article Presentation Book Patent

  • [Book] 医療・診断をささえるペプチド化学-再生医療・DDS・診断への応用-2017

    • Author(s)
      北村正典、国嶋崇隆
    • Total Pages
      315
    • Publisher
      シーエムシー
    • ISBN
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Book] e-EROS (Encyclopedia of Reagents for Organic Synthesis) 4-(4,6-Dimethoxy-1,3,5-triazin-2-yl )-4-methylmorpholinium chloride2013

    • Author(s)
      M. Kitamura, M. Kunishima
    • Total Pages
      5
    • Publisher
      John Wiley & Sons, Ltd
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Book] e-EROS (Encyclopedia of Reagents for Organic Synthesis) 4-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride.2013

    • Author(s)
      Masanori Kitamura, Munetaka Kunishima
    • Total Pages
      5
    • Publisher
      John Wiley & Sons, Ltd
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Book] 化学フロンティア19創薬をめざす有機合成最前線, 宍戸宏造, 新藤充編策1章トリアジン誘導体を用いた脱水縮合反応2007

    • Author(s)
      国嶋 崇隆(分担執筆)
    • Publisher
      化学同人
    • Data Source
      KAKENHI-PROJECT-18659006
  • [Book] フルオラスケミストリー2005

    • Author(s)
      国嶋崇隆
    • Total Pages
      9
    • Publisher
      シーエムシー出版
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Book] 第5版 実験化学講座 16 有機化合物の合成IV 酸アミド,ラクタム2005

    • Author(s)
      国嶋崇隆
    • Total Pages
      55
    • Publisher
      丸善株式会社
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Book] 第5版実験化学講座第16巻,有機化合物の合成IV,1.7 酸アミドおよび酸イミド2005

    • Author(s)
      国嶋崇隆
    • Total Pages
      37
    • Publisher
      丸善
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Book] 第5版実験化学講座第16巻,有機化合物の合成IV,1.8 ラクタム2005

    • Author(s)
      国嶋崇隆
    • Total Pages
      20
    • Publisher
      丸善
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Carbocationoids, a concept for controlling highly reactive cationic species2024

    • Author(s)
      Fujita Hikaru、Shimada Daichi、Kudo Jotaro、Kosha Kazuyuki、Kakuyama Satoshi、Terasaki Hiromitsu、Kunishima Munetaka
    • Journal Title

      Communications Chemistry

      Volume: 7 Issue: 1

    • DOI

      10.1038/s42004-024-01139-w

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Journal Article] Hydrophobic‐Substrate‐Selective Dehydrative Condensations at the Emulsion Interface under Conditions where Competitive Reactions Proceed in the Bulk Aqueous Phase2023

    • Author(s)
      Matsumoto Takuya、Hirata Eri、Zhang Hanlin、Hioki Kazuhito、Kunishima Munetaka
    • Journal Title

      Asian Journal of Organic Chemistry

      Volume: 12 Issue: 1

    • DOI

      10.1002/ajoc.202200602

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-21K19331
  • [Journal Article] Epitope-Based Specific Antibody Modification2023

    • Author(s)
      Horie Saki、Mishiro Kenji、Nishino Mio、Domae Inori、Wakasugi Mitsuo、Matsunaga Tsukasa、Kunishima Munetaka
    • Journal Title

      ChemRxiv

      Volume: 2023

    • DOI

      10.26434/chemrxiv-2023-c0k4n

    • Open Access
    • Data Source
      KAKENHI-PROJECT-21K19331
  • [Journal Article] Nucleophilic substitution reactions of unbranched alkyl amines using triazine reagents2022

    • Author(s)
      Masanori Kitamura, Yuki Kitaoka, Hikaru Fujita, Munetaka Kunishima
    • Journal Title

      Tetrahedron Letters

      Volume: 93 Pages: 153692-153692

    • DOI

      10.1016/j.tetlet.2022.153692

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-21H02603
  • [Journal Article] Measurement of Hepatic CYP3A4 and 2D6 Activity Using Radioiodine-Labeled O-Desmethylvenlafaxine2022

    • Author(s)
      Mizutani Asuka、Kobayashi Masato、Aibe Riku、Muranaka Yuka、Nishi Kodai、Kitamura Masanori、Suzuki Chie、Nishii Ryuichi、Shikano Naoto、Magata Yasuhiro、Ishida Yasushi、Kunishima Munetaka、Kawai Keiichi
    • Journal Title

      International Journal of Molecular Sciences

      Volume: 23 Issue: 19 Pages: 11458-11458

    • DOI

      10.3390/ijms231911458

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-21K07503, KAKENHI-PROJECT-22K06517, KAKENHI-PROJECT-18K15554, KAKENHI-PROJECT-19K17194, KAKENHI-PROJECT-23K21423
  • [Journal Article] Synthesis and characterization of tetraphenylammonium salts2022

    • Author(s)
      Fujita Hikaru、Sasamoto Ozora、Kobayashi Shiori、Kitamura Masanori、Kunishima Munetaka
    • Journal Title

      Nature Communications

      Volume: 13 Issue: 1 Pages: 2537-2537

    • DOI

      10.1038/s41467-022-30282-y

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-22K06517, KAKENHI-PROJECT-21H02603
  • [Journal Article] Development of a triazinedione-based dehydrative condensing reagent containing 4-(dimethylamino)pyridine as an acyl transfer catalyst2021

    • Author(s)
      Jie Liu, Hikaru Fujita, Masanori Kitamura, Daichi Shimada, Munetaka Kunishima
    • Journal Title

      Organic & Biomolecular Chemistry

      Volume: 19 Issue: 21 Pages: 4712-4719

    • DOI

      10.1039/d1ob00450f

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-21H02603
  • [Journal Article] Development of a triazinedione-based dehydrative condensing reagent containing 4-(dimethylamino)pyridine as an acyl transfer catalyst2021

    • Author(s)
      Jie Liu, Hikaru Fujita, Masanori Kitamura, Daichi Shimada, Munetaka Kunishima
    • Journal Title

      Org. Biomol. Chem.

      Volume: 19

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] A versatile iodo(III)etherification of terminal ethynylsilanes using BF3-OiPr2 and alkyl benzyl ethers2021

    • Author(s)
      Matsumoto Takuya、Hagiyama Hiroshi、Kuribayashi Kanetsugu、Hioki Kazuhito、Fujita Hikaru、Ochiai Masahito、Kunishima Munetaka
    • Journal Title

      Organic & Biomolecular Chemistry

      Volume: 19 Issue: 17 Pages: 3825-3828

    • DOI

      10.1039/d1ob00479d

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Journal Article] <i>N</i>-Acyltriazinedione; a Novel Acylating Reagent Synthesized from a Triazinone-Type Condensing Reagent2021

    • Author(s)
      Yamada Kohei、Lee Jeongsu、Kota Mika、Karuo Yukiko、Kitamura Masanori、Kunishima Munetaka
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 69 Issue: 5 Pages: 498-502

    • DOI

      10.1248/cpb.c20-00952

    • NAID

      130008032816

    • ISSN
      0009-2363, 1347-5223
    • Year and Date
      2021-05-01
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06995, KAKENHI-PROJECT-17H03970, KAKENHI-PROJECT-19K06994
  • [Journal Article] Conjugation of 4-(dimethylamino)pyridine to primary amines in aqueous buffer solutions using an N-hydroxysuccinimide ester reagent2021

    • Author(s)
      Horie Saki、Fujita Hikaru、Yamashita Rina、Kunishima Munetaka
    • Journal Title

      Tetrahedron Letters

      Volume: 81 Pages: 153343-153343

    • DOI

      10.1016/j.tetlet.2021.153343

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-21K19331
  • [Journal Article] Trizaine-Based Dehydrative Condensation Reagents Bearing Carbon-Substituents2020

    • Author(s)
      2.Masanori Kitamura, Sayaka Komine, Kohei Yamada, Munetaka Kunishima
    • Journal Title

      Tetrahedron

      Volume: 76 Issue: 12 Pages: 130900-130900

    • DOI

      10.1016/j.tet.2019.130900

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06995, KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of Hydrophilic Polyacrylamide Gel-Based Condensing Reagents Comprised of Chlorotriazine2020

    • Author(s)
      Yamada Kohei、Hirozawa Shota、Xia Junqing、Kunishima Munetaka
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 68 Issue: 6 Pages: 534-537

    • DOI

      10.1248/cpb.c20-00074

    • NAID

      130007850055

    • ISSN
      0009-2363, 1347-5223
    • Year and Date
      2020-06-01
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06995, KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of Triazinone-Based Condensing Reagents for Amide Formation2019

    • Author(s)
      Kohei Yamada, Mika Kota, Kensuke Takahashi, Hikaru Fujita, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 84 Issue: 23 Pages: 15042-15051

    • DOI

      10.1021/acs.joc.9b01261

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-19K06995, KAKENHI-PROJECT-19K22489, KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of a Storable Triazinone-Based Reagent for O-p-Methoxybenzylation under Mild Heating Conditions2019

    • Author(s)
      Fujita Hikaru、Terasaki Hiromitsu、Kakuyama Satoshi、Hioki Kazuhito、Kunishima Munetaka
    • Journal Title

      Organic Letters

      Volume: 21 Issue: 9 Pages: 3093-3097

    • DOI

      10.1021/acs.orglett.9b00732

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] Preparation of Alkyl Ethers with Diallyltriazinedione‐Type Alkylating Agents (ATTACKs‐R) Under Acid Catalysis2019

    • Author(s)
      Hikaru Fujita, Rina Yamashita, Takanori Fujii, Kohei Yamada, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      European Journal of Organic Chemistry

      Volume: 2019 Issue: 27 Pages: 4436-4446

    • DOI

      10.1002/ejoc.201900607

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-19K06995, KAKENHI-PROJECT-19K22489, KAKENHI-PROJECT-17H03970
  • [Journal Article] Substitution of the Dimethylamino Group in Gramines and One-Pot Cyclization to Tetrahydro-β-carbolines Using a Triazine-Based Activating Agent2019

    • Author(s)
      Hikaru Fujita, Riho Nishikawa, Ozora Sasamoto, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 84 Issue: 13 Pages: 8380-8391

    • DOI

      10.1021/acs.joc.9b00039

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19K06994, KAKENHI-PROJECT-17H03970
  • [Journal Article] An Isolable and Bench-Stable Epoxidizing Reagent Based on Triazine: Triazox2018

    • Author(s)
      Yamada Kohei、Igarashi Yuki、Betsuyaku Tatsuki、Kitamura Masanori、Hirata Koki、Hioki Kazuhito、Kunishima Munetaka
    • Journal Title

      Organic Letters

      Volume: 20 Issue: 7 Pages: 2015-2019

    • DOI

      10.1021/acs.orglett.8b00560

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970, KAKENHI-PROJECT-16K08160, KAKENHI-PROJECT-16K08161
  • [Journal Article] Imido-substituted triazines as dehydrative condensing reagents for the chemoselective formation of amides in the presence of free hydroxy?groups2018

    • Author(s)
      Kitamura Masanori、Sasaki Suguru、Nishikawa Riho、Yamada Kohei、Kunishima Munetaka
    • Journal Title

      RSC Advances

      Volume: 8 Issue: 40 Pages: 22482-22489

    • DOI

      10.1039/c8ra03057j

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-17H03970, KAKENHI-PROJECT-16K08160, KAKENHI-PROJECT-16K08161
  • [Journal Article] Development of highly electron-deficient and less sterically-hindered phosphine ligands possessing 1,3,5-triazinyl groups2018

    • Author(s)
      Kazumi Abe, Masanori Kitamura, Hikaru Fujita, Munetaka Kunishima
    • Journal Title

      Molecular Catalysis

      Volume: 445 Pages: 87-93

    • DOI

      10.1016/j.mcat.2017.11.008

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-16K08161, KAKENHI-PROJECT-17H03970
  • [Journal Article] Triazine-Based Cationic Leaving Group: Synergistic Driving Forces for Rapid Formation of Carbocation Species2018

    • Author(s)
      Hikaru Fujita, Satoshi Kakuyama, Shuichi Fukuyoshi, Naoko Hayakawa, Akifumi Oda, Munetaka Kunishima
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 83 Issue: 8 Pages: 4568-4580

    • DOI

      10.1021/acs.joc.8b00331

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17K08257, KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of radioiodine labeled acetaminophen for specific, high-contrast imaging of malignant melanoma2018

    • Author(s)
      Wen Jing Zhu , Masato Kobayashi , Kohei Yamada , Kodai Nishi , Kotaro Takahashi , Asuka Mizutani , Ryuichi Nishii , Leo G. Flores II , Naoto Shikano , Munetaka Kunishima , Keiichi Kawai
    • Journal Title

      Nuclear Medicine and Biology

      Volume: 59 Pages: 16-21

    • DOI

      10.1016/j.nucmedbio.2017.12.008

    • Peer Reviewed / Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-16H05397, KAKENHI-PROJECT-15K09949, KAKENHI-PROJECT-18K19508
  • [Journal Article] Cooperation of the Neutral and the Cationic Leaving Group Pathways in Acid-Catalyzed O-Benzylation of TriBOT2018

    • Author(s)
      Fujita Hikaru、Hayakawa Naoko、Kunishima Munetaka
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 83 Issue: 17 Pages: 10684-10687

    • DOI

      10.1021/acs.joc.8b01505

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of Triazine-Based Benzylating Reagents Possessing <i>t</i>-Butyl Group on the Triazine Core: Thermally Controllable Reagents for the Initiation of Reaction2018

    • Author(s)
      Karuo Yukiko、Yamada Kohei、Kunishima Munetaka
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 66 Issue: 3 Pages: 303-308

    • DOI

      10.1248/cpb.c17-00897

    • NAID

      130006407119

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970, KAKENHI-PROJECT-16K08160
  • [Journal Article] Development of triazine-based esterifying reagents containing pyridines as a nucleophilic catalyst2018

    • Author(s)
      Yamada Kohei、Liu Jie、Kunishima Munetaka
    • Journal Title

      Organic & Biomolecular Chemistry

      Volume: 16 Issue: 35 Pages: 6569-6575

    • DOI

      10.1039/c8ob01660g

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] Study of <i>O</i>-Allylation Using Triazine-Based Reagents2017

    • Author(s)
      Kohei Yamada, Naoko Hayakawa, Hikaru Fujita, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 65 Issue: 1 Pages: 112-115

    • DOI

      10.1248/cpb.c16-00744

    • NAID

      130005187751

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-16K08161
  • [Journal Article] N,N’-Dimethylated Benzyloxytriazinedione: A Stable Solid Reagent for Acid-Catalyzed O-Benzylation2017

    • Author(s)
      Hikaru Fujita, Satoshi Kakuyama, Munetaka Kunishima
    • Journal Title

      Eur. J. Org. Chem.

      Volume: 2017 Issue: 4 Pages: 833-839

    • DOI

      10.1002/ejoc.201601387

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Journal Article] Development of a method for the synthesis of 2,4,5-trisubstituted oxazoles composed of carboxylic acid, amino acid, and boronic acid2017

    • Author(s)
      Yamada Kohei、Kamimura Naoto、Kunishima Munetaka
    • Journal Title

      Beilstein J. Org. Chem.

      Volume: 13 Pages: 1478-1485

    • DOI

      10.3762/bjoc.13.146

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] トリアジンの特性を活用した新規アルキル化剤2017

    • Author(s)
      国嶋崇隆,山田耕平,藤田光,北村正典
    • Journal Title

      有機合成化学協会誌

      Volume: 75 Pages: 1023-1034

    • NAID

      130006156694

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Journal Article] Development of Acid-Catalyzed Fluorous Benzylating Reagents Based on a Triazinedione Core2016

    • Author(s)
      Munetaka Kunishima, Ryohei Asao, Kohei Yamada, Masanori Kitamura, Hikaru Fujita
    • Journal Title

      J. Fluorine Chem

      Volume: 190 Pages: 68-74

    • DOI

      10.1016/j.jfluchem.2016.09.003

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-16K08161
  • [Journal Article] Development of a Triazine-based tert-Butylating Reagent, TriAT-tBu2016

    • Author(s)
      Kohei Yamada, Naoko Hayakawa, Hikaru Fujita, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      Eur. J. Org. Chem.

      Volume: 2016 Issue: 23 Pages: 4093-4098

    • DOI

      10.1002/ejoc.201600663

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-16K08161
  • [Journal Article] Hydroxy and Amino Group-Tolerant Synthesis of Six-Membered Cyclic Quaternary Ammonium Salts Using a Triazine-Based Reagent2016

    • Author(s)
      Masanori Kitamura, Seina Yamamura, Kohei Yamada, Munetaka Kunishima
    • Journal Title

      Asian J. Org. Chem.

      Volume: 5 Issue: 12 Pages: 1508-1517

    • DOI

      10.1002/ajoc.201600429

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-16K08161
  • [Journal Article] Potent triazine-based dehydrocondensing reagents substituted by an amido group2016

    • Author(s)
      Munetaka Kunishima, Daiki Kato, Nobu Kimura, Masanori Kitamura, Kohei Yamada, Kazuhito Hioki
    • Journal Title

      Beilstein J. Org. Chem.

      Volume: 12 Pages: 1897-1903

    • DOI

      10.3762/bjoc.12.179

    • Peer Reviewed / Acknowledgement Compliant / Open Access
    • Data Source
      KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-16K08161
  • [Journal Article] Mild Amide-Cleavage Reaction Mediated by Electrophilic Benzylation2016

    • Author(s)
      Kohei Yamada, Yukiko Karuo, Yuichi Tsukada, Munetaka Kunishima
    • Journal Title

      Chem. Eur. J.

      Volume: 22 Issue: 39 Pages: 14042-14047

    • DOI

      10.1002/chem.201603120

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Journal Article] Study of the Reactivities of Acid-Catalyzed O-Benzylating Reagents Based on Structural Isomers of 1,3,5-Triazine2015

    • Author(s)
      Hikaru Fujita, Naoko Hayakawa, and Munetaka Kunishima
    • Journal Title

      The Journal of Organic Chemistry

      Volume: 80 Issue: 21 Pages: 11200-11205

    • DOI

      10.1021/acs.joc.5b02059

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-13J07110, KAKENHI-PROJECT-26670001, KAKENHI-PROJECT-26293003
  • [Journal Article] O-Benzylation of Carboxylic Acids Using 2,4,6-Tris(benzyloxy)-1,3,5-triazine (TriBOT) under Acidic or Thermal Conditions2015

    • Author(s)
      Kohei Yamada, Saki Yoshida, Hikaru Fujita, Masanori Kitamura, and Munetaka Kunishima
    • Journal Title

      European Journal of Organic Chemistry

      Volume: 36 Issue: 36 Pages: 7997-8002

    • DOI

      10.1002/ejoc.201501172

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-13J07110, KAKENHI-PROJECT-25460012, KAKENHI-PROJECT-25460013, KAKENHI-PROJECT-26670001, KAKENHI-PROJECT-26293003
  • [Journal Article] Development of a New Benzylating Reagent Spontaneously Releasing Benzyl Cation Equivalents at Room Temperature2014

    • Author(s)
      Kohei Yamada, Yuichi Tsukada, Yukiko Karuo, Masanori Kitamura, Munetaka Kunishima
    • Journal Title

      Chem. Eur. J.

      Volume: 20 Issue: 38 Pages: 12274-12278

    • DOI

      10.1002/chem.201403158

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-25460013, KAKENHI-PROJECT-26293003, KAKENHI-PROJECT-26670001
  • [Journal Article] Synthesis of Pyrrolidinium Salts Using a Triazine-based Reagent under Mild Conditions2014

    • Author(s)
      Masanori Kitamura, Seina Yamamura, Hiroko Kobayashi, Mariko Yamamoto, Kayo Tada, Kazuhito Hioki, Kohei Yamada, Munetaka Kunishima
    • Journal Title

      Chem. Lett.

      Volume: 43 Issue: 10 Pages: 1593-1595

    • DOI

      10.1246/cl.140503

    • NAID

      130004427196

    • ISSN
      0366-7022, 1348-0715
    • Language
      English
    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-25460013, KAKENHI-PROJECT-26293003
  • [Journal Article] Specific Labeling of Streptavidin for Better Understanding of Ligand Modification in Modular Method for Affinity Labeling (MoAL)2014

    • Author(s)
      Munetaka Kunishima, Daiki Kato, Shuichi Nakanishi, Masanori Kitamura, Kohei Yamada, Keiji Terao, Tomoya Asano
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 62 Issue: 11 Pages: 1146-1150

    • DOI

      10.1248/cpb.c14-00468

    • NAID

      130004712907

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-25460013, KAKENHI-PROJECT-26293003
  • [Journal Article] Role of Linkers in Tertiary Amines That Mediate or Catalyze 1,3,5-Triazine-Based Amide-Forming Reactions2014

    • Author(s)
      M. Kitamura, F. Kawasaki, K. Ogawa, S. Nakanishi, H. Tanaka, K. Yamada, M. Kunishima
    • Journal Title

      J. Org. Chem

      Volume: 79 Issue: 8 Pages: 3709-3714

    • DOI

      10.1021/jo500376m

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004, KAKENHI-PROJECT-25460013, KAKENHI-PROJECT-26293003
  • [Journal Article] A new method using 2-chloro-4,6-dimethoxy-1,3,5-triazine for facile elimination of dimethylamino group in Eschenmoser’s methylenation for synthesis of a,b-unsaturated esters2013

    • Author(s)
      Kohei Yamada, Kazumasa Masaki, Yuri Hagimoto, Seina Kamiya, Munetaka Kunishima
    • Journal Title

      Tetrahedron Lett.

      Volume: 54 Issue: 13 Pages: 1758-1760

    • DOI

      10.1016/j.tetlet.2013.01.092

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004, KAKENHI-PROJECT-23790009
  • [Journal Article] Study of 1,3,5-Triazine-Based Catalytic Amide-Forming Reactions: Effect of Solvents and Basicity of Reactants2013

    • Author(s)
      Munetaka Kunishima, Masanori Kitamura, Hiroyuki Tanaka, Ichiro Nakakura, Takahiro Moriya, Kazuhito Hioki
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 61 Issue: 8 Pages: 882-886

    • DOI

      10.1248/cpb.c13-00368

    • NAID

      130003360818

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004, KAKENHI-PROJECT-25460013
  • [Journal Article] A Practical Method for p-Methoxybenzylation of Hydroxy Groups Using 2,4,6-Tris (p-methoxybenzyloxy)-1,3,5-triazine (TriBOT-PM)2013

    • Author(s)
      Kohei Yamada, Hikaru Fujita, Masanori Kitamura, Munetaka Kuni shima
    • Journal Title

      Synthesis

      Volume: 45 Issue: 21 Pages: 2989-2997

    • DOI

      10.1055/s-0033-1339713

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-13J07110, KAKENHI-PROJECT-23590004, KAKENHI-PROJECT-25460013
  • [Journal Article] Binding of Sulforhodamine B to Human Serum Albumin: A Spectroscopic Study.2013

    • Author(s)
      Kitamura M., Murakami K., Yamada K., Kawai K., Kunishima M.
    • Journal Title

      Dyes and Pigments.

      Volume: 99(3) Pages: 588-593

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-25293260
  • [Journal Article] Binding of sulforhodamine B to human serum albumin: A spectroscopic study2013

    • Author(s)
      Masanori Kitamura, Koji Murakami, Kohei Yamada, Keiichi Kawai, Munetaka Kunishima
    • Journal Title

      Dyes and Pigments

      Volume: 99 Issue: 3 Pages: 588-593

    • DOI

      10.1016/j.dyepig.2013.06.011

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Journal Article] A Novel Acid-Catalyzed O‐Benzylating Reagent with the Smallest Unit of Imidate Structure2012

    • Author(s)
      Kohei Yamada, Hikaru Fujita, Munetaka Kunishima
    • Journal Title

      Org. Lett.

      Volume: 14 Issue: 19 Pages: 5026-5029

    • DOI

      10.1021/ol302222p

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004, KAKENHI-PROJECT-23790009
  • [Journal Article] One-Pot Preparation of Oxazol-5(4<i>H</i>)-ones from Amino Acids in Aqueous Solvents2012

    • Author(s)
      H. Fujita, M. Kunishima
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 60 Issue: 7 Pages: 907-912

    • DOI

      10.1248/cpb.c12-00291

    • NAID

      130001852501

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Journal Article] Substrate-Selective Dehydrocondensation at an Interface of Micelles and Emulsions of Common Surfactants2012

    • Author(s)
      M. Kunishima, K. Kikuchi, Y. Kawai, K. Hioki
    • Journal Title

      Angew. Chem. Int. Ed

      Volume: 51 Issue: 9 Pages: 2080-2083

    • DOI

      10.1002/anie.201107706

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Journal Article] Study on 1,3,5-Triazine Chemistry in Dehydrocondensation: Gauche Effect on the Generation of Active Triazinylammonium Species2012

    • Author(s)
      Munetaka Kunishima, Takae Ujigawa, Yoshie Nagaoka, Chiho Kawachi, Kazuhito Hioki, Motoo Shiro
    • Journal Title

      Chem. Eur. J.

      Volume: 18 Issue: 49 Pages: 15856-15867

    • DOI

      10.1002/chem.201202236

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Journal Article] New approach to oligotriazoles using a cobalt complex of propargyl azides as a synthetic component2011

    • Author(s)
      Y.Tsukada, K.Yamada, M.Kunishima
    • Journal Title

      Tetrahedron Lett. Vol 52,印刷中

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Labeling study of avidin by modular method for affinity labeling (MoAL)2010

    • Author(s)
      S.Nakanishi, H.Tanaka, K.Hioki, K.Yamada, M.Kunishima
    • Journal Title

      Bioorg.Med.Chem.Lett. Vol.20

      Pages: 7050-7053

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Effects of stereochemistry and β-substituents on the rates of vinylic S_N2 reaction of hypervalent vinyl(phenyl)-λ3-iodanes with tetrabutylammonium halides2010

    • Author(s)
      K.Miyamoto, T.Okubo, M.Hirobe, M.Kunishima, M.Ochiai
    • Journal Title

      Tetrahedron Vol:66

      Pages: 5819-5826

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Convenient Modular Method for Affinity Labeling(MoAL Method)Based on a Catalytic Amidation2009

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Chem.Commun.

      Pages: 5597-5599

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] A Simple Practical Method for Synthesis of 4,6-Dimethoxy-1,3,5-triazin-2(1H)-one Using Dimethylamine-Functionalized Solid-Phase Reagent2009

    • Author(s)
      K.Hioki, K.Ohshima, Y.Sota, M.Tanaka, M.Kunishima
    • Journal Title

      Synthesis

      Pages: 542-544

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Synthesis of Aza-bridged Calix(4-methoxy)triazines toward Flattened p-Conjugated Macrocycles2009

    • Author(s)
      H.Tanaka, 1 A.Wada, M.Shiro, K.Hioki, D.Morisaki, M.Kunishima
    • Journal Title

      Heterocycles Vol.79

      Pages: 609-616

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Convenient Modular Method for Affinity Labeling (MoAL Method) Based on a Catalytic Amidation2009

    • Author(s)
      M.Kunishima, S.Nakanishi, J.Nishida, H.Tanaka, D.Morisaki, K.Hioki, H.Nomoto
    • Journal Title

      Chem. Commun.

      Pages: 5597-5599

    • NAID

      120002165223

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Convenient One-Pot Synthesis of 2-Oxazolines from Carboxylic Acids2008

    • Author(s)
      K.Hioki, Y.Takechi, N.Kimura, H.Tanaka, M.Kunishima
    • Journal Title

      Chem.Pharm.Bull. Vol.56

      Pages: 1735-1737

    • NAID

      110007004709

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] 反応場の特性を基盤とする反応制御と実用的試薬の開発研究2008

    • Author(s)
      国嶋崇隆
    • Journal Title

      薬誌 Vol.128

      Pages: 425-438

    • NAID

      110006646597

    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Direct Preparation of Primary Amides by Reaction of Carboxylic Acids and Ammonia in Alcohols Using DMT-MM2008

    • Author(s)
      T.Mizuhara, K.Hioki, M.Yamada, H.Sasaki, D.Morisaki, M.Kunishima
    • Journal Title

      Chem Lett. Vol.37

      Pages: 1190-1191

    • NAID

      10024397464

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Antitumor Studies-Part 2 : Structure-Activity Relationship Study for Flavin Analogs Including Investigations on Their in vitro Antitumor Assay and Docking Simulation into Protein Tyrosine Kinase.2008

    • Author(s)
      H.I.Ali, K.Tomita, E.Akaho, M.Kunishima, Y.Kawashima, T.Yamagishi, H.Ikeya, T.Nagamatsu
    • Journal Title

      Eur.J.Med.Chem. Vol.43

      Pages: 1376-1389

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] 反応場の特性を基盤とする反応制御と実用的試薬の開発研究2008

    • Author(s)
      国嶋 崇隆
    • Journal Title

      薬学雑 3(印刷中)

    • NAID

      110006646597

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-18659006
  • [Journal Article] 機能拡張性を備えた実用的なポリマー型脱水縮合剤の開発2008

    • Author(s)
      国嶋崇隆
    • Journal Title

      薬学研究の進歩 Vol.24

      Pages: 29-35

    • Data Source
      KAKENHI-PROJECT-20390007
  • [Journal Article] Primary-Amine-Specific Lactamization of ω-Amino Acids by an Artificial Cyclotransferase Based on [18]Crown-62006

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Angew.Chem.Int.Ed. 45-8

      Pages: 1252-1255

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Primary-Amine-Specific Lactamization of ω-Amino Acids by an Artificial Cyclotransferase Based on 〔18〕Crown-62006

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Angew. Chem. Int. Ed. 45,8

      Pages: 1252-1255

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Spontaneous Membrane Fusion Induced by Chemical Formation of Ceramides in a Lipid Bilayer2006

    • Author(s)
      M.Kunishima et al.
    • Journal Title

      J. Am. Chem. Soc. 128

      Pages: 14452-14452

    • Data Source
      KAKENHI-PROJECT-18659006
  • [Journal Article] Unusual Rate Enhancement of Bimolecular Dehydrocondensation Forming Amides at the Interface of Micelles of Fatty Acid Salt2005

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Angew. Chem. Int. Ed. 44,44

      Pages: 7254-7257

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Development of Novel Polymer-type Dehydrocondensing Reagents Comprised of Chlorotriazines2005

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Chem.Commun. 21

      Pages: 2698-2700

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Development of Novel Polymer-type Dehydrocondensing Reagents Comprised of Chlorotriazines2005

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Chem. Commun. 21

      Pages: 2698-2700

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] メディアとしての水の特性を利用したアミド化反応2005

    • Author(s)
      国嶋崇隆
    • Journal Title

      ファルマシア 44,7

      Pages: 654-658

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Unusual Rate Enhancement of Bimolecular Dehydrocondensation Forming Amides at the Interface of Micelles of Fatty Acid Salt2005

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Angew.Chem.Int.Ed. 44-44

      Pages: 7254-7257

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] 新規トリアジン型脱水縮合剤の合成と用途開発2004

    • Author(s)
      国嶋崇隆
    • Journal Title

      和光純報 72

      Pages: 8-8

    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Substrate-Specific Amidation of Carboxylic Acids in a Liquid-Liquid Two-Phase System Using Cyclodextrins As an Inverse Phase Transfer Catalyst2004

    • Author(s)
      M.Kunishima, Y.Watanabe, K.Terao, S.Tani
    • Journal Title

      Eur.J.Org.Chem.

      Pages: 4535-4535

    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Substrate-Specific Amidation of Carboxylic Acids in a Liquid-Liquid Two-Phase System Using Cyclodextrins As an Inverse Phase Transfer Catalyst2004

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Eur. J. Org. Chem 22

      Pages: 4535-4540

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Substrate-Specific Amidation of Carboxylic Acids in a Liquid-Liquid Two-Phase System Using Cyclodextrins As an Inverse Phase Transfer Catalyst2004

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Eur J.Org.Chem. 22

      Pages: 4535-4540

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Development of a Simple System for Dehydrocondensation Using Solid-Phase Adsorption of a Water-Soluble Dehydrocondensing Reagent (DMT-MM)2004

    • Author(s)
      Y.Watanabe, T.Fuji, K.Hioki, S.Tani, M.Kunishima
    • Journal Title

      Chem.Pharm.Bull. 52

      Pages: 1223-1223

    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Approach to Green Chemistry of DMT-MM : Recovery and Recycle of Coproduct to Chloromethane-Free DMT-MM2002

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Tetrahedron Lett. 43-18

      Pages: 3323-3326

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Journal Article] Approach to Green Chemistry of DMT-MM : Recovery and Recycle of Coproduct to Chloromethane-Free DMT-MM2002

    • Author(s)
      Munetaka Kunishima
    • Journal Title

      Tetrahedron Lett., 43,18

      Pages: 3323-3326

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] SGLT機能画像診断薬2023

    • Inventor(s)
      小林正和,川井恵一,國嶋崇隆,他4名
    • Industrial Property Rights Holder
      小林正和,川井恵一,國嶋崇隆,他4名
    • Industrial Property Rights Type
      特許
    • Filing Date
      2023
    • Data Source
      KAKENHI-PROJECT-23K21423
  • [Patent] xCT機能活性阻害剤2023

    • Inventor(s)
      川井恵一,国嶋崇隆,玉井郁巳,小林正和,松本拓也 他3名
    • Industrial Property Rights Holder
      川井恵一,国嶋崇隆,玉井郁巳,小林正和,松本拓也 他3名
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2023-028079
    • Filing Date
      2023
    • Data Source
      KAKENHI-PROJECT-23K24277
  • [Patent] トリアジンジオン化合物2020

    • Inventor(s)
      國嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人 金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2020-118568
    • Filing Date
      2020
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Patent] トリアジノン化合物2016

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2016-034845
    • Filing Date
      2016-02-25
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] 酸化剤2016

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2016-210433
    • Filing Date
      2016-10-27
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] トリアジン含有ポリマー、その製造方法、及びその脱水縮合剤としての用途2016

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2016-034723
    • Filing Date
      2016-02-25
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] トリアジンジオン化合物2015

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-208908
    • Filing Date
      2015-10-23
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Patent] トリアジン化合物2015

    • Inventor(s)
      国嶋 崇隆
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-037118
    • Filing Date
      2015-02-26
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Patent] トリアジン化合物2015

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-037118
    • Filing Date
      2015-02-26
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] 脱水縮合剤2015

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-016112
    • Filing Date
      2015-01-29
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] 脱水縮合剤2015

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-016113
    • Filing Date
      2015-01-29
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] トリアジンジオン化合物2015

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2015-208908
    • Filing Date
      2015-10-23
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Patent] N型糖タンパク質の製造方法2013

    • Inventor(s)
      國嶋崇隆、山田耕平
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2013-026997
    • Filing Date
      2013-02-14
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] N型糖タンパク質の製造方法2013

    • Inventor(s)
      国嶋崇隆、山田耕平
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2013-026997
    • Filing Date
      2013-02-14
    • Overseas
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] 薬物と高分子化合物相互作用確認 用試薬及び相互作用の検査2012

    • Inventor(s)
      国嶋崇隆、山 田耕平、木野徹平
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2012-027242
    • Filing Date
      2012-02-10
    • Overseas
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] 分子イメージングにより代謝機能を測定するための検査薬2012

    • Inventor(s)
      川井恵一、玉井郁巳、国嶋崇隆太、中西猛夫、小林正和
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Number
      2012-044231
    • Filing Date
      2012-02-29
    • Data Source
      KAKENHI-PROJECT-23659076
  • [Patent] 不斉脱水縮合剤2012

    • Inventor(s)
      国嶋崇隆,北村正典,山田耕平,正木一将
    • Industrial Property Rights Holder
      国立大学法人金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2012-227249
    • Filing Date
      2012-10-12
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] 10.薬物と高分子化合物相互作用確認用試薬及び相互作用の検査2012

    • Inventor(s)
      国嶋崇隆、山田耕平、木野徹平
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Number
      2012-027242
    • Filing Date
      2012
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] 不斉脱水縮合剤2012

    • Inventor(s)
      国嶋崇隆、北村正典、山 田耕平、 正木一将
    • Industrial Property Rights Holder
      金沢大学
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2012-227249
    • Filing Date
      2012-10-12
    • Overseas
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Patent] 脱水縮合反応により相転移を生じ得る分子集合体およびその相転移方法2005

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      JST
    • Industrial Property Number
      2005-021241
    • Filing Date
      2005-01-28
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 脱水縮合反応により相転移を生じ得る分子集合体およびその相転移方法2005

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      JST
    • Filing Date
      2005-12-12
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 水界面への集積性を有する脱水縮合剤2005

    • Inventor(s)
      国嶋 崇隆
    • Industrial Property Rights Holder
      科学技術振興機構
    • Filing Date
      2005-01-31
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 水界面への集積性を有する脱水縮合剤2005

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      JST
    • Filing Date
      2005-01-31
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 塩化シアヌル誘導体,その製造法およびその使用2004

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      TLOひょうご
    • Industrial Property Number
      2004-032253
    • Filing Date
      2004-02-09
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 1,3,5-トリアジン環を環構成要素として含むシクロファン型化合物、その製造方法、中間体及びその利用2004

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      JST
    • Industrial Property Number
      2004-032598
    • Filing Date
      2004-02-09
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Patent] 水界面への集積性を有する脱水縮合剤2004

    • Inventor(s)
      国嶋崇隆
    • Industrial Property Rights Holder
      JST
    • Industrial Property Number
      2004-033284
    • Filing Date
      2004-02-10
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14572025
  • [Presentation] SN1反応の高活性中間体を取り出す新規方法論:カルボカチオノイド2024

    • Author(s)
      島田大地, 藤田光, 高社和行, 工藤丈太郎, 国嶋崇隆
    • Organizer
      日本薬学会第144年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] gem-ジヨードニオアルケンのヨードニオ基置換反応の開発検討2024

    • Author(s)
      村谷大輝, 松本拓也, 小林礼奈, 栗林兼続, 藤田光, 三代憲司, 国嶋 崇隆
    • Organizer
      日本薬学会第144年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] gem-ジヨードニオアルケン類β位トリフルオロメタンスルホニルオキシ基置換反応の開発検討2024

    • Author(s)
      小川幸己, 松本拓也, 熊田侑戯, 村谷大輝, 栗林兼続, 藤田光, 三代憲司, 国嶋崇隆
    • Organizer
      日本薬学会第144年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] オルト位にケイ素置換基を有するトリフェニルアミンの合成2024

    • Author(s)
      佐藤友里杏, 藤田光, 小林栞, 国嶋崇隆
    • Organizer
      日本薬学会第144年会
    • Data Source
      KAKENHI-PROJECT-23K18180
  • [Presentation] 新たな高求電子性活性種カルボカチオノイドの構造及び反応性の解析2023

    • Author(s)
      高社和行, 藤田光, 島田大地, 工藤丈太郎, 国嶋崇隆
    • Organizer
      2023年度有機合成化学北陸セミナー
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 縮環構造を持たないテトラアリールアンモニウムの合成及び基本的性質の解明2023

    • Author(s)
      笹本大空、藤田光、小林栞、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第143年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 抗体の新規化学修飾法の開発2023

    • Author(s)
      堀江彩紀,三代憲司,西野未桜,堂前いのり,若杉光生,松永司,国嶋崇隆
    • Organizer
      日本薬学会第143年会
    • Data Source
      KAKENHI-PROJECT-21K19331
  • [Presentation] アルコキシ基交換を利用したトリアジンジオン型酸触媒アルキル化剤の合成2023

    • Author(s)
      八木谷知美、藤田光、国嶋崇隆
    • Organizer
      日本薬学会第143年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 分子間反応によるO-アルキル化を利用したエポキシドの開環反応2023

    • Author(s)
      松井孝憲, 藤田光, 国嶋崇隆
    • Organizer
      第52回複素環化学討論会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 高いアルキル化能を有する新規活性種カルボカチオノイドのNMR解析2023

    • Author(s)
      高社和行, 藤田光, 島田大地, 工藤丈太郎, 国嶋崇隆
    • Organizer
      第40回メディシナルケミストリーシンポジウム
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] カルボカチオノイド:不安定カチオン種を制御する新規方法論2023

    • Author(s)
      島田大地, 藤田光, 高社和行, 工藤丈太郎, 国嶋崇隆
    • Organizer
      2023年度有機合成化学北陸セミナー,
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] Synthesis of gem-diiodonio-alkenes2023

    • Author(s)
      松本拓也, 栗林兼続, 熊田侑戯, 藤田光, 三代憲司, 国嶋崇隆
    • Organizer
      第26回 ヨウ素学会シンポジウム
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] フェノキシ基の置換を利用するトリアジンジオン化合物の誘導体化法の開発2023

    • Author(s)
      島田大地、藤田光、工藤丈太郎、脊戸里々佳、国嶋崇隆
    • Organizer
      日本薬学会第143年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 未踏分子テトラフェニルアンモニウム塩の合成2022

    • Author(s)
      笹本大空、藤田光、小林栞、北村正典、国嶋崇隆
    • Organizer
      第20回次世代を担う有機化学シンポジウム
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] β-トリフリルオキシ-α,α-ビス(フェニルヨードニオ)エチレン類の合成:三つの強力な電子求引性置換基を有するエチレンユニットの開発2022

    • Author(s)
      栗林兼続、松本拓也、国嶋崇隆
    • Organizer
      第25回ヨウ素学会シンポジウム
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] トリアジンジオン型酸触媒パラメトキシベンジル化剤を用いたカルバマートとアミドのN-保護反応2022

    • Author(s)
      藤田 光、小林 栞、脊戸 里々佳、国嶋 崇隆
    • Organizer
      日本薬学会第142年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] トリアジンジオン型アルキル化剤を用いた酸触媒ベンジル化反応におけるトリアジニウム中間体の形成2022

    • Author(s)
      島田 大地、藤田 光、角山 哲史、国嶋 崇隆
    • Organizer
      日本薬学会第142年会
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] カチオン特性の制御と活用を指向する有機化学2022

    • Author(s)
      国嶋崇隆
    • Organizer
      岐阜薬科大学大学院薬学研究科特別講義、JST・SPRING事業講演会、日本プロセス化学会出前講義
    • Invited
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 炭素及び窒素カチオンを機軸とする有機化学2022

    • Author(s)
      国嶋崇隆
    • Organizer
      有機合成化学協会九州・山口支部 第34会若手研究者のためのセミナー
    • Invited
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] トリアジン型酸化剤Triazoxを用いた芳香族カルボン酸からカルバマートへの変換反応の開発2022

    • Author(s)
      藤田光、加藤利幸、国嶋崇隆
    • Organizer
      創薬懇話会2022 in 名古屋
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] カチオンを基盤とする有機化学2022

    • Author(s)
      国嶋崇隆
    • Organizer
      京都大学薬学研究科特別講演会
    • Invited
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] ヘテロ原子間結合を含有しない新規ウロニウム型脱水縮合剤の開発2022

    • Author(s)
      水島岳、藤田光、国嶋崇隆
    • Organizer
      第39回メディシナルケミストリーシンポジウム
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] Estimation of hepatic CYP3A4 and 2D6 activity by imaging with radioiodine-labeled O-Desmethylvenlafaxine2022

    • Author(s)
      Mizutani A, Kobayashi M, Muranaka Y, Nishi K, Suzuki C, Nishii R, Shikano N, Magata Y, Ishida Y, Kunishima M, Kawai K
    • Organizer
      13th World Federation of Nuclear Medicine and Biology
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-23K21423
  • [Presentation] 含窒素複素環を脱離基とするカルボカチオンの可逆的発生法の開発2021

    • Author(s)
      北岡 佑紀,藤田 光,工藤 丈太郎,寺崎 博満,角山 哲史,国嶋 崇隆
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-19K22489
  • [Presentation] 簡便に合成できる新規トリアジン型エポキシ化剤の開発2021

    • Author(s)
      加藤 利幸,別役 樹,藤田 光,国嶋 崇隆
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] Chemoselective alkoxylation in the synthesis of β-λ3-iodanyl-β-silyl enol ethers using BF3-OiPr2 and alkyl benzyl ethers2021

    • Author(s)
      Takuya Matsumoto, Hiroshi Hagiyama, Kanetsugu Kuribayashi, Kazuhito Hioki, Hikaru Fujita, Masahito Ochiai, Munetaka Kunishima
    • Organizer
      AFMC International Medicinal Chemistry Symposium 2021
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] Conjugation of an aminopyridine-based nucleophilic catalyst to aliphatic primary amines in aqueous media using an N-hydroxysuccinimide ester reagent2021

    • Author(s)
      Saki Horie, Hikaru Fujita, Rina Yamashita, Munetaka Kunishima
    • Organizer
      The 2021 International Chemical Congress of Pacific Basin Societies
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-21K19331
  • [Presentation] Para-methoxybenzyl protection of secondary amides under acidic conditions2021

    • Author(s)
      Hikaru Fujita, Ririka Seto, Munetaka Kunishima
    • Organizer
      The 2021 International Chemical Congress of Pacific Basin Societies
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] ピリジン型求核触媒を内包した新規脱水縮合剤の開発2021

    • Author(s)
      藤田 光、劉 杰、島田 大地、北村 正典、国嶋 崇隆
    • Organizer
      創薬懇話会2021 in 京都
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] Synthesis of triphenylamines bearing three adjacent substituents on the phenyl groups2021

    • Author(s)
      Ozora Sasamoto, Hikaru Fujita, Munetaka Kunishima
    • Organizer
      The 2021 International Chemical Congress of Pacific Basin Societies
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-21H02603
  • [Presentation] 含窒素複素環を脱離基とするカルボカチオンの可逆的発生法の開発2021

    • Author(s)
      北岡 佑紀,藤田 光,工藤 丈太郎,寺崎 博満,角山 哲史,国嶋 崇隆
    • Organizer
      日本薬学会第141年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 含窒素複素環化合物を用いたカルボカチオンの安定化及び反応性の制御2020

    • Author(s)
      工藤 丈太郎,藤田 光,寺崎 博,角山 哲史,国嶋 崇隆
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 含窒素複素環化合物を用いたカルボカチオンの安定化及び反応性の制御2020

    • Author(s)
      工藤 丈太郎,藤田 光,寺崎 博,角山 哲史,国嶋 崇隆
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-19K22489
  • [Presentation] トリアジンジオン型アルキル化剤を用いたアミドの酸触媒N-パラメトキシベンジル化反応の開発2020

    • Author(s)
      脊戸 里々佳,藤田 光,国嶋 崇隆
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンジオン型アシル化剤の反応性に関する研究2020

    • Author(s)
      李 政洙、軽尾 有紀子、古田 美佳、山田 耕平、北村 正典、国嶋 崇隆
    • Organizer
      日本薬学会第140年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 薬物代謝酵素CYP2D6の活性定量を目的とした新規放射性画像診断薬の開発2019

    • Author(s)
      水谷明日香,高須啓彰,小林正和,西 弘大,北村正典,国嶋宗隆,西井龍一,鈴木千恵,間賀田泰寛,川井恵一
    • Organizer
      第15回小動物インビボイメージング研究会
    • Data Source
      KAKENHI-PROJECT-18K19508
  • [Presentation] Triazine-Based Dehydrative Condensing Reagents Bearing Carbon-Substituents2019

    • Author(s)
      Masanori Kitamura, Sayaka Komine, Kohei Yamada and Munetaka Kunishima
    • Organizer
      27th International Society of Heterocyclic Chemistry Congress
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 含窒素芳香環の特性を活用したアルキル化剤の開発2019

    • Author(s)
      国嶋崇隆
    • Organizer
      フルオラス科学研究会 第12回シンポジウム
    • Invited
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] Stable Triazinone-Based Reagent for O-p-Methoxybenzylation under Mild Heating Conditions2019

    • Author(s)
      Hikaru Fujita, Hiromitsu Terasaki, Satoshi Kakuyama, Kazuhito Hioki, and Munetaka Kunishima
    • Organizer
      The 4th International Symposium on Process Chemistry (ISPC 2019)
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンジオン骨格を基盤としたアルキル化剤の置換基効果2019

    • Author(s)
      藤井崇徳, 山下莉奈, 藤田光, 角山哲史, 山田耕平, 北村正典, 国嶋崇隆
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] アミノ基を脱離基とした温和なアルキル化反応の開発2019

    • Author(s)
      北岡 佑紀,北村 正典,藤田 光,国嶋 崇隆
    • Organizer
      日本薬学会第139年会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] クロロトリアジンによるインドールアルカロイドの変換反応:テトラヒドロ-β-カルボリン誘導体の簡便合成法の開発2019

    • Author(s)
      藤田光,西川理穂,笹本大空,北村正典,国嶋崇隆
    • Organizer
      第37回メディシナルケミストリーシンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 光レドックス触媒によるトリアジニルアンモニウム塩のC-N結合開裂反応の開発2019

    • Author(s)
      小林葉月、山田耕平、国嶋崇隆
    • Organizer
      第45回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンジオン骨格を基盤とした種々アルキル化剤の開発2018

    • Author(s)
      山下莉奈,藤井崇徳,藤田光,山田耕平,北村正典,国嶋崇隆
    • Organizer
      第36回メディシナルケミストリーシンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンを基盤とした単離可能なエポキシ化剤Triazoxの開発2018

    • Author(s)
      別役樹,五十嵐佑貴,山田耕平,北村正典,平田紘基,日置和人,国嶋崇隆
    • Organizer
      日本プロセス化学会 2018 ウィンターシンポジウム
    • Invited
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 光増感触媒を用いたイナミンの生成及びそれを利用した光活性化型脱水縮合反応の開発2018

    • Author(s)
      木村 武史, 三代 憲司, 国嶋 崇隆
    • Organizer
      日本薬学会北陸支部第130回例会
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 親水性ポリアクリルアミドゲルを担体とする脱水縮合剤の開発2018

    • Author(s)
      廣澤翔太,夏俊卿,山田耕平,国嶋崇隆
    • Organizer
      第44回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンを基盤とした単離可能なエポキシ化剤Triazoxの開発2018

    • Author(s)
      別役樹,五十嵐佑貴,山田耕平,北村正典,平田紘基,日置和人,国嶋崇隆
    • Organizer
      日本プロセス化学会 2018 サマーシンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジンジオンを基盤とする新規アシル化剤の開発2017

    • Author(s)
      古田美佳、軽尾友紀子、 李政洙、山田耕平、北村正典、国嶋 崇隆
    • Organizer
      日本薬学会第137年会
    • Place of Presentation
      仙台国際センター、仙台
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] カルボン酸、アミノ酸、ボロン酸からなる多様性志向型三置換オキサゾール合成法の開発2017

    • Author(s)
      山田耕平,上村直人,国嶋崇隆
    • Organizer
      第35回メディシナルケミストリーシンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 新規トリアジン型酸化剤の開発と反応2017

    • Author(s)
      五十嵐佑貴、別役樹、山田耕平、国嶋崇隆
    • Organizer
      日本薬学会第137年会
    • Place of Presentation
      仙台国際センター、仙台
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 実用的な酸触媒アルキル化剤の開発2017

    • Author(s)
      角山哲史、藤田光、寺﨑博満、山田耕平、国嶋崇隆
    • Organizer
      日本プロセス化学会 2017 サマーシンポジウム
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] トリアジニルピリジニウム塩を用いたエステル化反応の開発2017

    • Author(s)
      劉杰、山田耕平、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第137年会
    • Place of Presentation
      仙台国際センター、仙台
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 求核触媒を内包した新規エステル化剤の開発2017

    • Author(s)
      劉杰、山田耕平、北村正典、国嶋崇隆
    • Organizer
      第43回反応と合成の進歩シンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] 酸触媒ジアルキルトリアジンジオン型フルオラスベンジル化剤の開発2017

    • Author(s)
      山田 耕平,藤井 崇徳,山下 莉奈,国嶋 崇隆
    • Organizer
      フルオラス科学研究会第10回シンポジウム
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] Development of Electron-Poor Phosphine Ligands Having 1,3,5-Triazinyl Groups2017

    • Author(s)
      Kazumi Abe, Masanori Kitamura, Hikaru Fujita, Munetaka Kunishima, Faculty of Pharmaceutical Sciences, Kanazawa University, Kanazawa, Japan
    • Organizer
      26th International Society of Heterocyclic Chemistry
    • Data Source
      KAKENHI-PROJECT-17H03970
  • [Presentation] カルボン酸・アミノ酸・アリールボロン酸からなる三置換オキサゾールの短工程合成法の開発2016

    • Author(s)
      上村直人、山田耕平、藤田光、国嶋崇隆
    • Organizer
      第46回複素環化学討論会
    • Place of Presentation
      歌劇座、金沢
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] サイトⅠ特異的な薬物タンパク結合を検出する蛍光標識化アルブミンの開発2016

    • Author(s)
      瀧澤祐美佳, 山田耕平, 国嶋崇隆
    • Organizer
      日本薬学会第136年会
    • Place of Presentation
      パシフィコ横浜、横浜
    • Year and Date
      2016-03-28
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of HSA Sensor for Detection of Site II Drug Binding.2016

    • Author(s)
      Kunishima M.
    • Organizer
      Asian Chemical Biology Initiative (ACBI) 2016 Jakarta Meeting
    • Place of Presentation
      Jakarta, Indonesia
    • Year and Date
      2016-01-30
    • Invited / Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of triazine-type dehydrocondensing reagents having an amido group2016

    • Author(s)
      Daiki Kato, Nobu Kimura, Kohei Yamada, Masanori Kitamura, Munetaka Kunishima
    • Organizer
      XXVII European Colloquium on Heterocyclic Chemistry (ECHC 2016)
    • Place of Presentation
      Beurs van berlage, Amsterdam, Netherlands
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 塩化トリアジンを用いた六員環状第四級アンモニウム塩合成法の開発2016

    • Author(s)
      北村正典、山村聖奈、山田耕平、国嶋崇隆
    • Organizer
      第34回メディシナルケミストリーシンポジウム
    • Place of Presentation
      つくば国際会議場、つくば
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] アミド基を置換基に有するトリアジニルアンモニウム型脱水縮合剤の開発2016

    • Author(s)
      古田美佳, 山田耕平, 藤田光, 国嶋崇隆
    • Organizer
      日本薬学会第136年会
    • Place of Presentation
      パシフィコ横浜、横浜
    • Year and Date
      2016-03-29
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 新規トリアジノン型脱水縮合剤の開発2016

    • Author(s)
      古田美佳、高橋 健輔、山田耕平、藤田光、国嶋崇隆
    • Organizer
      第46回複素環化学討論会
    • Place of Presentation
      歌劇座、金沢
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 互変異性化を駆動力とした新規トリアジン型酸化剤の開発2016

    • Author(s)
      五十嵐佑貴、山田耕平、平田紘基、国嶋崇隆
    • Organizer
      日本薬学会北陸支部第128回例会
    • Place of Presentation
      北陸大学、金沢
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] ポリアクリルアミドを担体とする親水性固定化脱水縮合剤の開発2016

    • Author(s)
      夏俊卿, 山田耕平, 国嶋崇隆
    • Organizer
      日本薬学会第136年会
    • Place of Presentation
      パシフィコ横浜、横浜
    • Year and Date
      2016-03-28
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] アミノトリアジンを脱離基とするベンジル化剤の開発:置換基効果に基づく分解反応の制御2015

    • Author(s)
      軽尾友紀子、小峰彩、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-26
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of a method for the synthesis of trisubstituted oxazoles by Suzuki-Miyaura Coupling2015

    • Author(s)
      Yamada K, Kamimura N, Fujita H, Kunishima M.
    • Organizer
      the 18th IUPAC International Symposium on Organometallic Chemistry Directed Towards Organic Synthesis
    • Place of Presentation
      Barcelona, Spain
    • Year and Date
      2015-06-29
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of acid-catalyzed alkylating reagents based on triazine chemistry2015

    • Author(s)
      Hayakawa N, Yamada K, Fujita H, Kitamura M, Yoshimura K, Kunishima M.
    • Organizer
      The 3rd International Symposium on Process Chemistry
    • Place of Presentation
      Kyoto International Conference Center, Kyoto, Japan
    • Year and Date
      2015-07-15
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] トリアジン骨格を基盤とする酸触媒tert-ブチル化剤の開発2015

    • Author(s)
      早川奈緒子、山田耕平、藤田光、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-26
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] π電子欠乏性新規トリアジン型脱水縮合剤の開発2015

    • Author(s)
      木村円、矢内秀、山田耕平、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-26
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] カルボン酸・アミノ酸・アリールボロン酸からなる三置換オキサゾール合成法の開発2015

    • Author(s)
      上村直人、山田耕平、藤田光、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-28
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Quick and mild methods for cleavage of amide-bonds by using a triazine-based benzylating reagent2015

    • Author(s)
      Karuo Y, Yamada K, Kunishima M.
    • Organizer
      2015 International Chemical Congress of Pacific Basin Societies
    • Place of Presentation
      Honolulu, Hawaii, USA
    • Year and Date
      2015-12-16
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Study of the reactivity of benzyloxytriazine derivatives (BOTs) for acid catalyzed O-benzylation2015

    • Author(s)
      Fujita H, Kunishima M.
    • Organizer
      2015 International Chemical Congress of Pacific Basin Societies
    • Place of Presentation
      Honolulu, Hawaii, USA
    • Year and Date
      2015-12-16
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] 電子的効果の軽微な置換基を有するトリアジン型縮合剤の反応性に関する研究学会等名2015

    • Author(s)
      小峰彩、北村正典、岡田有加里、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-28
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] トリアジン骨格を基盤とする酸触媒tert-ブチル化剤の開発2015

    • Author(s)
      早川奈緒子、山田耕平、藤田光、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-26
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] トリアジン型酸触媒ベンジル化剤のジプロトン化機構によるO-ベンジル化反応2015

    • Author(s)
      藤田光, 国嶋崇隆
    • Organizer
      第41回反応と合成の進歩シンポジウム
    • Place of Presentation
      近畿大学、大阪
    • Year and Date
      2015-10-27
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] 薬物タンパク結合を検出する蛍光標識化アルブミンの開発2015

    • Author(s)
      巻口真穂, 木野徹平, 山田耕平, 浅野智哉, 国嶋崇隆
    • Organizer
      日本薬学会北陸支部第127回例会
    • Place of Presentation
      富山大学、富山
    • Year and Date
      2015-11-15
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 電子欠乏性トリアジニルホスフィン配位子の開発2015

    • Author(s)
      安倍一実、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、クリエイティブセンター神戸
    • Year and Date
      2015-03-27
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Quick and mild methods for cleavage of amide-bonds by using a triazine-based benzylating reagent2015

    • Author(s)
      Karuo Y, Yamada K, Kunishima M.
    • Organizer
      2015 International Chemical Congress of Pacific Basin Societies
    • Place of Presentation
      Honolulu, Hawaii, USA
    • Year and Date
      2015-12-16
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] アミノトリアジンを脱離基とするベンジル化剤の開発:置換基効果に基づく分解反応の制御2015

    • Author(s)
      軽尾友紀子、小峰彩、北村正典、国嶋崇隆
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸、神戸学院大学
    • Year and Date
      2015-03-26
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] Study of the reactivity of benzyloxytriazine derivatives (BOTs) for acid catalyzed O-benzylation2015

    • Author(s)
      Fujita H, Kunishima M.
    • Organizer
      2015 International Chemical Congress of Pacific Basin Societies
    • Place of Presentation
      Honolulu, Hawaii, USA
    • Year and Date
      2015-12-16
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 新規酸触媒トリアジノン型ベンジル化剤の開発2015

    • Author(s)
      角山哲史, 藤田光, 北村正典, 山田耕平, 国嶋崇隆
    • Organizer
      第45回複素環化学討論会
    • Place of Presentation
      早稲田大学、東京
    • Year and Date
      2015-11-20
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of acid-catalyzed alkylating reagents based on triazine chemistry2015

    • Author(s)
      Hayakawa N, Yamada K, Fujita H, Kitamura M, Yoshimura K, Kunishima M.
    • Organizer
      The 3rd International Symposium on Process Chemistry
    • Place of Presentation
      Kyoto International Conference Center, Kyoto, Japan
    • Year and Date
      2015-07-15
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] イメージングによる肝臓の薬物代謝酵素CYP活性測定を可能にするヨウ素標識診断薬の開発2015

    • Author(s)
      水谷明日香,髙橋浩太郎,外間つづみ,小林正和,北村正典,国嶋宗隆,川井恵一,福地一樹.
    • Organizer
      第55回日本核医学会学術総会
    • Place of Presentation
      ハイアットリージェンシー東京(東京都千代田区)
    • Year and Date
      2015-11-05
    • Data Source
      KAKENHI-PROJECT-15K09949
  • [Presentation] 新規酸触媒トリアジノン型ベンジル化剤の開発2015

    • Author(s)
      角山哲史, 藤田光, 北村正典, 山田耕平, 国嶋崇隆
    • Organizer
      第45回複素環化学討論会
    • Place of Presentation
      早稲田大学、東京
    • Year and Date
      2015-11-20
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] Effect of carbon substituents on the reactivity of triazine-based dehydrocondensing reagents2015

    • Author(s)
      Komine S, Kitamura M, Kunishima M.
    • Organizer
      2015 International Chemical Congress of Pacific Basin Societies
    • Place of Presentation
      Honolulu, Hawaii, USA
    • Year and Date
      2015-12-16
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 酸触媒ベンジル化剤TriBOTを用いた低環境負荷型エステル化反応の開発2014

    • Author(s)
      山田耕平、吉田紗季、吉村和真、藤田光、北村正典、河合伸高、国嶋崇隆
    • Organizer
      日本プロセス化学会 2014 サマーシンポジウム
    • Place of Presentation
      東京、タワーホール船堀
    • Year and Date
      2014-08-01
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 未知の薬物標的タンパク質の探索を志向した親和標識化法2014

    • Author(s)
      加藤大輝, 北村正典, 山田耕平, 浅野智哉, 国嶋崇隆
    • Organizer
      創薬懇話会 2014 in 岐阜
    • Place of Presentation
      岐阜、岐阜長良川温泉 ホテルパーク
    • Year and Date
      2014-07-09
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] トリアジニルアミンを脱離基とした分子内閉環反応によるピロリジニウム塩の合成2014

    • Author(s)
      山村聖奈,北村正典,小林比呂子,山本真理子,多田佳世,日置和人,山田耕平,国嶋崇隆
    • Organizer
      第40回反応と合成の進歩シンポジウム
    • Place of Presentation
      仙台、東北大学 川内萩ホール
    • Year and Date
      2014-11-11
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 電子欠乏性アミノトリアジンを脱離基としたベンジル化剤の開発2014

    • Author(s)
      軽尾友紀子, 塚田裕以智, 山田耕平, 北村正典, 国嶋崇隆
    • Organizer
      第44回複素環化学討論会
    • Place of Presentation
      北海道、札幌市民ホール
    • Year and Date
      2014-09-11
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] 電子欠乏性アミノトリアジンを脱離基としたベンジル化剤の開発2014

    • Author(s)
      軽尾友紀子, 塚田裕以智, 山田耕平, 北村正典, 国嶋崇隆
    • Organizer
      第44回複素環化学討論会
    • Place of Presentation
      北海道、札幌市民ホール
    • Year and Date
      2014-09-11
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] Development of a new benzylating reagent which releases benzyl cation-like species at room temperature2014

    • Author(s)
      Kohei Yamada, Yukiko Karuo, Yuichi Tsukada, Masanori Kitamura, Munetaka Kunishima
    • Organizer
      14th Tetrahedron Symposium Asia Edition
    • Place of Presentation
      Singapore、Singapore EXPO Convention and Exhibition Centre
    • Year and Date
      2014-10-30
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] ベンジルカチオン種の求電子付加に基づくアミド結合開裂反応の開発2014

    • Author(s)
      軽尾友紀子,山田耕平,北村正典,国嶋崇隆
    • Organizer
      創薬懇話会 2014 in 岐阜
    • Place of Presentation
      岐阜、岐阜長良川温泉 ホテルパーク
    • Year and Date
      2014-07-09
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] Development of a new benzylating reagent which releases benzyl cation-like species at room temperature2014

    • Author(s)
      Kohei Yamada, Yukiko Karuo, Yuichi Tsukada, Masanori Kitamura, Munetaka Kunishima
    • Organizer
      14th Tetrahedron Symposium Asia Edition
    • Place of Presentation
      Singapore、Singapore EXPO Convention and Exhibition Centre
    • Year and Date
      2014-10-30
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] 酸触媒ベンジル化剤TriBOTを用いた低環境負荷型エステル化反応の開発2014

    • Author(s)
      山田耕平、吉田紗季、吉村和真、藤田光、北村正典、河合伸高、国嶋崇隆
    • Organizer
      日本プロセス化学会 2014 サマーシンポジウム
    • Place of Presentation
      東京、タワーホール船堀
    • Year and Date
      2014-08-01
    • Data Source
      KAKENHI-PROJECT-26670001
  • [Presentation] 脱水縮合反応を基盤とするタンパク質修飾法(MoAL法)におけるプローブ設計とその評価2014

    • Author(s)
      加藤大輝,山田耕平,北村正典,浅野 智哉,国嶋崇隆
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本大学(熊本県)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] ベンジルカチオン種の求電子付加に基づくアミド結合開裂反応の開発2014

    • Author(s)
      軽尾友紀子,山田耕平,北村正典,国嶋崇隆
    • Organizer
      創薬懇話会 2014 in 岐阜
    • Place of Presentation
      岐阜、岐阜長良川温泉 ホテルパーク
    • Year and Date
      2014-07-09
    • Data Source
      KAKENHI-PROJECT-26293003
  • [Presentation] イミダートの最小単位のみで構成される酸触媒アリールメチル化剤の開発2013

    • Author(s)
      山田耕平、藤田光、国嶋崇隆
    • Organizer
      日本プロセス化学会 2013 サマーシンポジウム
    • Place of Presentation
      つくば国際会議場(茨城県)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] カルボキシ基を標的とする生体分子の化学修飾2013

    • Author(s)
      国嶋崇隆
    • Organizer
      Endo-M研究会
    • Place of Presentation
      金沢勤労者プラザ(石川県)
    • Year and Date
      2013-05-17
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] A new acid-catalyzed benzylating reagent with the smallest unit of imidate structure: TriBOT2013

    • Author(s)
      Hikaru Fujita, Kohei Yamada, Munetaka Kunishima
    • Organizer
      14th Tetrahedron Symposium
    • Place of Presentation
      Hilton Vienna(Vienna, Austria)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 古い化合物の新しい化学~1,3,5-トリアジンを基軸とする反応の開拓~2013

    • Author(s)
      国嶋崇隆
    • Organizer
      化学千一夜2013 「明日の化学への夢を語ろう」
    • Place of Presentation
      参天製薬㈱能登工場(石川県)
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] カルボキシ基を標的とする 生体分子の化学修飾2013

    • Author(s)
      国嶋崇隆
    • Organizer
      Endo-M 研究会
    • Place of Presentation
      金沢勤労者プラザ(石川県)
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] ベンジルイミダートを経由するアミド結合切断反応の開発2013

    • Author(s)
      軽尾友紀子,山田耕平,北村正典,国嶋崇隆
    • Organizer
      第39回反応と合成の進歩シンポジウム
    • Place of Presentation
      九州大学医学部百年講堂(福岡県)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 酸触媒トリアジン型パラメトキシベンジル化剤 (TriBOT-PM) の開発2013

    • Author(s)
      藤田光、山田耕平、北村正典、国嶋崇隆
    • Organizer
      第43回複素環化学討論会
    • Place of Presentation
      長良川国際会議場(岐阜県)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 古い化合物の新しい化学〜1,3,5-トリアジンを基軸とする反応の開拓〜2013

    • Author(s)
      国嶋崇隆
    • Organizer
      化学千一夜2013「明日の化学への夢を語ろう」
    • Place of Presentation
      参天製薬㈱能登工場(石川県)
    • Year and Date
      2013-06-07
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] トリアジンの特性を利用した新反応剤の開発2012

    • Author(s)
      国嶋崇隆
    • Organizer
      日本プロセス化学会2012サマーシンポジウム
    • Place of Presentation
      京都テルサ(京都府)
    • Year and Date
      2012-07-19
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 脱水縮合反応を利用したシクロオキシゲナーゼの特異的標識化反応2011

    • Author(s)
      国嶋崇隆
    • Organizer
      第37回反応と合成の進歩シンポジウム
    • Place of Presentation
      あわぎんホール(徳島県)
    • Year and Date
      2011-11-07
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 脱水縮合反応を利用したシクロオキシゲナーゼの特異的標識化反応2011

    • Author(s)
      国嶋崇隆,鶴崎亮,中西修一,辻慎也,山田耕平
    • Organizer
      第37回反応と合成の進歩シンポジウム
    • Place of Presentation
      あわぎんホール(徳島)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] Specific Labeling of Avidin and Streptavidin by Modular Method for Affinity Labeling2011

    • Author(s)
      S. Nakanishi, K. Yamada, M. Kunishima
    • Organizer
      8th AFMC International Medicinal Chemistry Symposium
    • Place of Presentation
      京王プラザホテル(東京)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] カルボキシル基を標的とする生体分子の有機化学2011

    • Author(s)
      国嶋崇隆
    • Organizer
      日本薬学会 九州支部主催 特別講演会(招待講演)
    • Place of Presentation
      長崎大学(長崎)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] Labeling Study of Cyclooxygenase-1 (COX-1) by Modular Method for Affinity Labeling (MoAL)2011

    • Author(s)
      M. Kunishima, R. Tsurusaki, K. Yamada, S. Tsuji, S. Nakanishi
    • Organizer
      8th AFMC International Medicinal Chemistry Symposium
    • Place of Presentation
      京王プラザホテル(東京)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] カルボキシル基を標的とする生体分子の有機化学2011

    • Author(s)
      国嶋崇隆
    • Organizer
      日本薬学会九州支部主催特別講演会
    • Place of Presentation
      長崎大学(長崎県)
    • Year and Date
      2011-06-06
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] An Efficient Dehydrocondensing Reaction Accelerated at a Micellar Interface2010

    • Author(s)
      国嶋崇隆
    • Organizer
      環太平洋化学会 (PacifiChem 2010)
    • Place of Presentation
      ハワイコンベンションセンター(USA)
    • Year and Date
      2010-12-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] Convenient modular method for specific labeling of targeting proteins by catalytic amidation: MoAL Method2010

    • Author(s)
      Munetaka Kunishima
    • Organizer
      環太平洋化学会(PacifiChem2010)
    • Place of Presentation
      ハワイコンベンションセンター(U.S.A.)
    • Year and Date
      2010-12-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] Convenient modular method for specific labeling of targeting proteins by catalytic amidation : MoAL Method2010

    • Author(s)
      国嶋崇隆
    • Organizer
      環太平洋化学会 (PacifiChem 2010)
    • Place of Presentation
      ハワイコンベンションセンター(USA)
    • Year and Date
      2010-12-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] An Eflicient Dehydrocondensing Reaction Accelerated at a Micellar Interface2010

    • Author(s)
      Munetaka Kunishima
    • Organizer
      環太平洋化学会(PacifiChem2010)
    • Place of Presentation
      ハワイコンベンションセンター(U.S.A.) 招待講演
    • Year and Date
      2010-12-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] 触媒的脱水縮合反応を基盤とするモジュール式アフィニティーラベル化法(MoAL 法)の開発2009

    • Author(s)
      国嶋崇隆
    • Organizer
      日本ケミカルバイオロジー学会第4回年会
    • Place of Presentation
      神戸市産業振興センター(兵庫県)
    • Year and Date
      2009-05-19
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] 触媒的脱水縮合反応を基盤とするモジュール式アフィニティーラベル化法(MoAL法)の開発2009

    • Author(s)
      国嶋崇隆
    • Organizer
      日本ケミカルバイオロジー学会第4回年会
    • Place of Presentation
      神戸市産業振興センター(兵庫)
    • Year and Date
      2009-05-19
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] トリアジン型脱水縮合剤の開発と応用2009

    • Author(s)
      国嶋崇隆
    • Organizer
      平成21年度前期有機合成化学講習会
    • Place of Presentation
      長井記念ホール(東京都)
    • Year and Date
      2009-06-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] トリアジン型脱水縮合剤の開発と応用2009

    • Author(s)
      国嶋崇隆
    • Organizer
      平成21年度前期有機合成化学講習会
    • Place of Presentation
      長井記念ホール(東京)
    • Year and Date
      2009-06-17
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] 生体分子を標的とする特異的アミド化反応2008

    • Author(s)
      国嶋 崇隆
    • Organizer
      日本薬学会第128年会
    • Place of Presentation
      横浜
    • Year and Date
      2008-03-27
    • Data Source
      KAKENHI-PROJECT-18659006
  • [Presentation] 酸アミド結合の効率的な形成を目指した新技術の開拓 -トリアジン型縮合剤の開発と応川-2008

    • Author(s)
      国嶋崇隆
    • Organizer
      名城大学大学院総合学術研究科グリーンバイオビジネス創製プロジェクト平成20年度第4回プロジェクトセミナー
    • Place of Presentation
      名城大学
    • Year and Date
      2008-11-29
    • Data Source
      KAKENHI-PROJECT-20390007
  • [Presentation] 界面を反応場とする脱水縮合反応2007

    • Author(s)
      国嶋 崇隆
    • Organizer
      平成19年度第1回粉体接合研究会
    • Place of Presentation
      神戸
    • Year and Date
      2007-06-27
    • Data Source
      KAKENHI-PROJECT-18659006
  • [Presentation] トリアジンの特性を利用した新反応剤の開発

    • Author(s)
      国嶋崇隆,鶴崎亮,中西修一,辻慎也,山田耕平
    • Organizer
      日本プロセス化学会 2012 サマーシンポジウム
    • Place of Presentation
      京都テルサ(京都府)
    • Invited
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] プロトン性溶媒中でのエナンチオ選択的アミド化触媒の開発.

    • Author(s)
      正木一将、北村正典、国嶋崇隆
    • Organizer
      第38回反応と合成の進歩シンポジウム
    • Place of Presentation
      タワーホール船堀(東京都)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] Synthesis and Evaluation of Iodinated Cyclopropanecarboxylic Acid {3-[6-(Phenylamino)- pyrimidin-4-ylamino]-phenyl}-amides as EGFR-TK Imaging Agents.

    • Author(s)
      Yoshimoto M., Kimura S., Yamada K., Hirata M., Ohmomo Y., Kunishima M., Kawai K., Fujii H.
    • Organizer
      20th International Symposium on Radiopharmaceutical Sciences
    • Place of Presentation
      Jeju International Convention Center (Korea)
    • Data Source
      KAKENHI-PROJECT-25293260
  • [Presentation] Preparation of Hydrogel Particles by a in situ Generated Condensing Agent

    • Author(s)
      K. Iwahara, K. Hioki, M. Kitamura, K. Yamada, H. Ichikawa, M. Kunishima
    • Organizer
      IKCOC12
    • Place of Presentation
      リーガロイヤルホテル京都(京都府)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 血清アルブミンに対する薬物の結合を簡便に検出するセンサーの開発

    • Author(s)
      木野 徹平, 山田 耕平, 浅野 智哉, 国嶋 崇隆
    • Organizer
      日本薬学会第133年会
    • Place of Presentation
      パフィシコ横浜(神奈川県)
    • Data Source
      KAKENHI-PROJECT-23590004
  • [Presentation] 究極的に簡素化されたイミダート等価構造を持つ新規ベンジル化剤:TriBOT

    • Author(s)
      藤田光、山田耕平、国嶋崇隆
    • Organizer
      第38回反応と合成の進歩シンポジウム
    • Place of Presentation
      タワーホール船堀(東京都)
    • Data Source
      KAKENHI-PROJECT-23590004
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  • 2.  TAMAI Ikumi (20155237)
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    # of Collaborated Projects: 3 results
    # of Collaborated Products: 1 results
  • 13.  HOJO Keiko (20289028)
    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
  • 14.  INOBE Manabu (10312414)
    # of Collaborated Projects: 2 results
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    # of Collaborated Projects: 2 results
    # of Collaborated Products: 0 results
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    # of Collaborated Projects: 2 results
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    # of Collaborated Projects: 2 results
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  • 18.  松本 拓也 (40800214)
    # of Collaborated Projects: 2 results
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  • 19.  TANAKA Hiroyuki (40378873)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 5 results
  • 20.  MORISAKI Daiki (30462740)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 3 results
  • 21.  NAKANISHI Takeo (30541742)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 22.  GOTO Kyoko (50180245)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
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    # of Collaborated Projects: 1 results
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  • 24.  ENDO Yoshio (30211783)
    # of Collaborated Projects: 1 results
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  • 25.  OKAZAWA Hidehiko (50360813)
    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
  • 26.  SHIKANO Naoto (80295435)
    # of Collaborated Projects: 1 results
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    # of Collaborated Projects: 1 results
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    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
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    # of Collaborated Projects: 1 results
    # of Collaborated Products: 0 results
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    # of Collaborated Projects: 1 results
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