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KAGECHIKA Hiroyuki  影近 弘之

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… Alternative Names

影近 弘之  カゲチカ ヒロユキ

KAHECHIKAK Hiroyuki  陰近 弘之

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Researcher Number 20177348
Other IDs
External Links
Affiliation (Current) 2025: 東京科学大学, 総合研究院, 教授
Affiliation (based on the past Project Information) *help 2023 – 2024: 東京医科歯科大学, 生体材料工学研究所, 教授
2012 – 2016: 東京医科歯科大学, 生体材料工学研究所, 教授
2012: 東京医科歯科大学, 疾患生命科学研究部, 教授
2011: 東京医科歯科大学, 大学院疾患生命科学研究部, 教授
2007 – 2011: Tokyo Medical and Dental University, SCHOOL OF BIOMEDICAL SCIENCE, PROFESSOR … More
2009: Tokyo Medical and Dental University, 疾患生命科学研究部, 教授
2007: 東京医科齢科大学, 大学院・疾患生命科学研究部, 教授
2006: Tokyo Med.Dent.Univ., School Biomed.Sci., Prof., 大学院疾患生命科学研究部, 教授
2006: 東京医科歯科大学, 疾患生命科学研究部, 教授
2005: 東京医科歯科大学, 大学院・疾患生命科学研究科, 教授
2004 – 2005: 東京医科歯科大学, 大学院・疾患生命科学研究部, 教授
2004: TOKYO MEDICAL AND DENTAL UNIVERCITY, SCHOLL OF BIOMEDICAL SCIENCE, PROFFECER, 教授
2004: 東京医科歯科大学, 大学院・疾患生命科学研究, 教授
1999 – 2004: 東京大学, 大学院・薬学系研究科, 助教授
2002: 東京大学, 大学院・薬学研究科, 助教授
1997 – 1998: University of Tokyo, Graduate School of Pharmaceutical Sciences, Research Associ, 大学院・薬学系研究科, 助手
1987 – 1996: 東京大学, 薬学部, 助手
1992: 東京大学, 薬部学, 助手 Less
Review Section/Research Field
Principal Investigator
医薬分子機能学 / Drug development chemistry / Biological Sciences / Living organism molecular science / Science and Engineering / Chemical pharmacy / Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related / Basic Section 47050:Environmental and natural pharmaceutical resources-related / Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related / Complex systems … More
Except Principal Investigator
… More 医薬分子機能学 / Endocrinology / Drug development chemistry / Medium-sized Section 47:Pharmaceutical sciences and related fields / Metabolomics / Chemical pharmacy / Complex systems / General pharmacology Less
Keywords
Principal Investigator
核内受容体 / レチノイド / RAR / アンタゴニスト / RXR / カルボラン / 不飽和脂肪酸 / 蛍光プローブ / ビタミンD / 分化誘導 … More / 結晶構造 / 芳香族ウレア / アミド結合 / レチノイン酸 / シス型優先性 / nuclear receptors / ビタミンK / 脂溶性ビタミン / 蛍光性リガンド / プロゲステロン / アンドロゲン / 遺伝子転写制御 / クマリン / LXR / アゴニスト / PPAR / トロポロン / シナジスト / レチノイドアンタゴニスト / レチノイドシナジスト / 芳香族グアニジン / 核酸認識分子 / 動的NMR / 構造展開 / non-genomic作用 / 遺伝子転写 / antidiabetes / synergist / carborane / floxane / tropolone / bioisoster / retinoids / 抗糖尿病〓 / 抗肥満 / 抗糖尿病 / 細胞分化 / アポトーシス / 白血病 / 転写因子 / 抗肥満・抗糖尿病 / フロキサン / バイオアイソスター / thyroid hormone / retinoid synergist / retinoid antagonist / retinoic acid / retinoid / チロイドホルモン / チアゾリジン / 構造活性相関 / N―メチルリシン / リシン / 酵素阻害剤 / 蛍光法 / スクリーニング / シプロヘプタジン / SET7/9 / 芳香族求核置換反応 / 検出法 / 阻害剤 / ヒストンメチル化酵素 / 抗腫瘍活性 / SXR / HepG2細胞 / K acid II / K acid I / メナキノン-4 / 抗炎症作用 / 細胞増殖 / 抗炎症効果 / 増殖抑制 / 癌細胞 / 酸化誘導体 / メナキノン / アダマンタン / ファーマコフォア / アンドロゲン受容体 / 蛍光センサー / ケイ素含有生理活性物質 / カルシウム濃度制御 / 高周期第14族元素 / 脂溶性ファーマコフォア / 脂質代謝 / ピロリジン / 生物学的等価性基 / アミド / スルフォンアミド / 生物学的等価性 / cis型二重結合 / 化合物ライブラリー / 疎水性ファーマコフォア / ケミカルバイオロジー / コンビナトリアル合成 / チアゾリジンジオン / 甲状腺ホルモン / AND型センサー / Riccardin C / seco-ステロイド骨格 / ビタミン D / 遺伝子発現 / ヘテロダイマー / IL-6 / 動脈硬化症 / KLF5 / バーチャルスクリーニング / ベンゾフロキサン / APL / カルボイン / オーファン受容体 / アラキドン酸 / モデリング / メラトニン / ホファン受容体 / ROR / DNAマイナーグルーブ結合性分子 / らせん分子 / シス型配座 / マイナーグルーブ / DNA結合分子 / 芳香族層状分子 / シス型 / 拡散認識分子 / 環状アミド / 層状分子 / 僧正分子 / 層状化合物 / 芳香族アミド … More
Except Principal Investigator
レチノイド / レチノイン酸 / アンタゴニスト / ビタミンA / retinoid / 分化 / 分化誘導 / 血管新生 / テレオシジン / レチノイドレセプタ- / retinoic acid receptor / PPAR / ステロイド / retinoic acid / 分子設計 / 核内受容体 / レセプター / 核内レセプター / 血管新生阻害 / 癌 / 白血病 / HL60 / endothelial cells / angiogenesis / all-trans retinoic acid / 動脈硬化 / レチノイン酸受容体 / 血管内皮細胞 / RXR / nuclear receptor / 一酸化窒素 / molecular design / differentiation / leukemia / レチノイドアンタゴニスト / ビタミンA酸 / 医薬品化学 / サリドマイド / RXRアンタゴニスト / 阻害剤 / 蛍光プローブ / リウマチ / アポトーシス / サイクリックADPリボース / ネオカルチノスタチン / 代謝拮抗剤 / 生体高分子 / チロキシン / 細胞分化 / TPA / レチノイドレセプター / 核レセプター / 構造活性相関 / Re80 / 癌治療 / 核レセプタ- / 転移 / 形態形成 / アンチセンスDNA / 遺伝子発現 / タンパク質ータンパク質相互作用阻害剤 / ファオルダマー / 大環状化合物 / らせん分子 / 環状構造 / らせん構造 / フォルダマー / 芳香族アミド / 受容体 / 血管内皮増殖因子 / phosphoinositide 3-kinase / endothelial NO synthase / nitric oxide(NO) / vascular endothelial cells / PI3キナーゼ / 内皮型一酸化窒素合成酵素 / RXR antagonist / adipocyte / diabetes / 生活習慣病 / PPARγ / 脂肪細胞 / 糖尿病 / thalidomide / bioprobe / enzyme inhibitor / antagonists / steroid hormone / structural development / 抗リウマチ活性 / 抗糖尿病活性 / シクロオキシゲナーゼ阻害剤 / エストロゲン / 抗アンドロゲン / シクロオキシゲナーゼ / ビタミンD_3 / 生物応答調節剤 / バチェラジン / チュブリン重合阻害剤 / 組胞分化誘導 / アンドロゲンアンタゴニスト / ビタミンDアンタゴニスト / プロテインキナーゼC / プロゲステロン / FXR / アンドロゲン / ビタミンD / Farnesoid X Receptor (FXR) / Liver X Receptor (LXR) / 核内受容体リガンド / 酵素阻害剤 / ステロイドホルモン / 構造展開 / steroid / teleocidin / protein kinase C / chemical synthesis / anti-HIV compound / tumor promoter / 核磁気共鳴スペクトル / 発癌プロモーター / 立体配座 / 有機合成化学 / プロテインキナーゼ / 化学合成 / 抗HIV化合物 / 発がんプロモーター / antagonist synergist / myeloma / tyroids / ベンゾラクタム / ジベンゾジアゼピン / フオルボール / 腫瘍悪性化 / チロイドリセプター / レチノイン酸レセプター / チロイド / retinoid receptor / cancer / retinoid antagonist / vitamin A / シリコン / がん / X線結晶解析 / 核中レセプター / 酸異性化 / リセプタータンパク / カルコンカルボン酸・分化 / テレフタル酸アリリド / 癌治療薬 / 生物学 / 生物物理 / 薬物動態学 / 代謝 / 全身循環 / 薬物動態 / 不整脈 / 心臓 / 生物物理学 / 生理学 / システム生物学 / 分子認識 / ホウ素クラスター / 疎水性相互作用 / アンドロゲン受容体 / エストロゲン受容体 / 医薬分子設計 / FREP / カベオラ / FRET / 核外作用 / 性ホルモン / ジヒドロピラン / ピロン / ジヒドロピロン / サポニン / 大豆 / ガン転移抑制作用 / 阻害活性 / MMP / DNAチップ / アロディニア / PGE_2 / リアノジン受容体 / 15R-TIC / リピドA / Cu-ATSM / ダントロレン誘導体 / 4'-チオリボヌクレオシド / 可視化プローブ / プロスグランジン / 34mCl / キナーゼ阻害剤 / 光親和性標識法 / MicroPET / プラナーポジトロンイメージング / 神経性疼痛 / Socius / ABCトランスポーター / non-RI光親和性標識法 / 3成分連結PG合成法 / シグナル解析 / 神経因性疼痛 / キナーゼ / 人工核酸 / 高速メチル化 / PET / タキソ-ル / ハリコンドリンB / 乾癖 / タキリ-ル / ハリコンンドリンB / フォルボール / ビタミンE / erb-A / フオルポール / ハービマイシンA / アンチセンスオリゴヌクレオチド / がん転移 / フィブロネクチン / G-蛋白質 / プリン / ras / 腫瘍血管新生 / 制癌剤 / HL-60細胞 / 制ガン剤 / レチノ安息香酸 / メソ-DNA / 計算化学 / 三重領 / 融解曲線 / エナンチオDNA / チロキシンレセプター / 鶏卵法検定 / 転移抑制 / 制がん剤 / 化学療法 / レチノイン酸レセプタ- / 対掌体 / DNA対掌体 / DNA / レチイン酸 / 分子進化 / Lーアラビノ-ス / レ-デオキシアデノシン / (dA)_6 / 三重鎖 / 核内レセプタ- / グルマコルケマイド / 発ガンプロモ-タ- / フオルポ-ルエステル / ビタンンA酸 / ビダミンA / 有機ゲルマニウム化合物 / 有機ケイ素化合物 / フォルボ-ルエステル / 発がんプロモ-タ- / 制がん Less
  • Research Projects

    (51 results)
  • Research Products

    (252 results)
  • Co-Researchers

    (67 People)
  •  Medicinal Chemsitry of Hydrophobic VItamins with Novel FunctionsPrincipal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2024 – 2026
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Review Section
      Basic Section 47010:Pharmaceutical chemistry and drug development sciences-related
      Basic Section 47050:Environmental and natural pharmaceutical resources-related
      Sections That Are Subject to Joint Review: Basic Section47010:Pharmaceutical chemistry and drug development sciences-related , Basic Section47050:Environmental and natural pharmaceutical resources-related
    • Research Institution
      Tokyo Medical and Dental University
  •  New molecular shapes from strained aromatic foldamer macrocycles and their application to development of PPI inhibitors

    • Principal Investigator
      棚谷 綾
    • Project Period (FY)
      2023 – 2026
    • Research Category
      Fund for the Promotion of Joint International Research (International Collaborative Research)
    • Review Section
      Medium-sized Section 47:Pharmaceutical sciences and related fields
    • Research Institution
      Ochanomizu University
  •  Development of novel detection method for histone methylation and HMT inhibitorsPrincipal Investigator

    • Principal Investigator
      Kagechika Hiroyuki
    • Project Period (FY)
      2014 – 2016
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Tokyo Medical and Dental University
  •  Development of novel vitamin K derivatives and elucidation of their biological functionsPrincipal Investigator

    • Principal Investigator
      KAGECHIKA Hiroyuki
    • Project Period (FY)
      2011 – 2013
    • Research Category
      Grant-in-Aid for Challenging Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Tokyo Medical and Dental University
  •  Establishment of Integrative Multi-level Systems Biology and its Applications

    • Principal Investigator
      KURACHI YOSHIHISA
    • Project Period (FY)
      2010 – 2015
    • Research Category
      Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
    • Review Section
      Complex systems
    • Research Institution
      Osaka University
  •  Development of specific modulators for nuclear receptors and elucidation of their functionsPrincipal Investigator

    • Principal Investigator
      KAGECHIKA Hiroyuki
    • Project Period (FY)
      2010 – 2014
    • Research Category
      Grant-in-Aid for Scientific Research on Innovative Areas (Research in a proposed research area)
    • Review Section
      Complex systems
    • Research Institution
      Tokyo Medical and Dental University
  •  Development of Receptor Regulators Utilizing Novel HydrophobicStructure and Its Application for Medicinal Drug Design

    • Principal Investigator
      ENDO Yasuyuki
    • Project Period (FY)
      2008 – 2012
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      Drug development chemistry
    • Research Institution
      Tohoku Pharmaceutical University
  •  Chemical biological approach for regulation of gene expressionPrincipal Investigator

    • Principal Investigator
      KAGECHIKA Hiroyuki
    • Project Period (FY)
      2007 – 2010
    • Research Category
      Grant-in-Aid for Scientific Research (A)
    • Research Field
      Living organism molecular science
    • Research Institution
      Tokyo Medical and Dental University
  •  核内受容体機能制御分子としての不飽和脂肪酸の医薬化学研究Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2007 – 2008
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Tokyo Medical and Dental University
  •  核内情報ネットワークの特異的制御分子に関する研究Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2006 – 2007
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Review Section
      Science and Engineering
    • Research Institution
      Tokyo Medical and Dental University
  •  創薬シーズとしての性ホルモン核外作用特異的リガンドのスクリーニング系の創製と応用

    • Principal Investigator
      古川 哲史
    • Project Period (FY)
      2006 – 2007
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      General pharmacology
    • Research Institution
      Tokyo Medical and Dental University
  •  EFFECTS OF ALL-TRANS RETINOIC ACID AND RETINOIDS ON ANGIOGENESIS

    • Principal Investigator
      SUGAWARA Akira
    • Project Period (FY)
      2006 – 2007
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Endocrinology
    • Research Institution
      Tohoku University
  •  核内情報伝達ネットワークを制御する脂溶性低分子化合物に関する研究Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2005 – 2006
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Review Section
      Science and Engineering
    • Research Institution
      Tokyo Medical and Dental University
  •  新規作用機構を有する脂肪細胞機能制御剤の創製研究Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2005 – 2006
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Living organism molecular science
    • Research Institution
      Tokyo Medical and Dental University
  •  MMP祖害活性を指標とした新規ガン転移抑制剤の開発

    • Principal Investigator
      杉本 昭子
    • Project Period (FY)
      2005 – 2006
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      Drug development chemistry
    • Research Institution
      Tokyo Medical and Dental University
  •  EFFECTS OF ATRA AND RETINOIDS ON ENDOTHELIAL FUNCTION

    • Principal Investigator
      SUGAWARA Akira
    • Project Period (FY)
      2004 – 2005
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Endocrinology
    • Research Institution
      TOHOKU UNIVERSITY
  •  核内レチノイド受容体を分子標的とした新規制癌剤の創製Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2002
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Review Section
      Biological Sciences
    • Research Institution
      The University of Tokyo
  •  Design and development of biological response modifiers

    • Principal Investigator
      HASHIMOTO Yuichi
    • Project Period (FY)
      2002 – 2006
    • Research Category
      Grant-in-Aid for Scientific Research (S)
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  Identification of RXR antagonists and characterization of potent stimulation of ST 13 preadipocyte differentiation

    • Principal Investigator
      SATO Mayumi
    • Project Period (FY)
      2002 – 2004
    • Research Category
      Grant-in-Aid for Scientific Research (C)
    • Research Field
      Metabolomics
    • Research Institution
      Tokyo Metropolitan Organization for Medical Research
  •  新規レチノイドの創製と癌治療への応用Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2001
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas (C)
    • Review Section
      Biological Sciences
    • Research Institution
      The University of Tokyo
  •  生物新機能と創薬をめざす生体内分子科学

    • Principal Investigator
      鈴木 正昭
    • Project Period (FY)
      2001 – 2005
    • Research Category
      Grant-in-Aid for Creative Scientific Research
    • Research Institution
      Gifu University
  •  Development of Novel Nuclear Receptor Regulators and Their Clinical UtilityPrincipal Investigator

    • Principal Investigator
      KAGECHIKA Hiroyuki
    • Project Period (FY)
      2001 – 2003
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  新規レチノイドの創製と癌治療への応用Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2000
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas (C)
    • Review Section
      Biological Sciences
    • Research Institution
      The University of Tokyo
  •  核内オーファン受容体RORのリガンド探索Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      2000 – 2001
    • Research Category
      Grant-in-Aid for Exploratory Research
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  アミド基の立体特性に基づく芳香族多層分子の構築と機能Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      1998 – 1999
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      Chemical pharmacy
    • Research Institution
      The University of Tokyo
  •  Development of Novel Nuclear Receptor ModulatorsPrincipal Investigator

    • Principal Investigator
      KAGECHIKA Hiroyuki
    • Project Period (FY)
      1998 – 2000
    • Research Category
      Grant-in-Aid for Scientific Research (B).
    • Research Field
      医薬分子機能学
    • Research Institution
      University of Tokyo
  •  生体高分子機能を修飾する抗がん化合物の合成と作用解析

    • Principal Investigator
      松田 彰
    • Project Period (FY)
      1996
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      Hokkaido University
  •  アミド結合の立体特性と生理活性物質構築への応用Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      1996
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  生体高分子機能を修飾する抗がん化合物の合成と作用解析

    • Principal Investigator
      松田 彰
    • Project Period (FY)
      1995
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      Hokkaido University
  •  レチノイドの化学・生物学・医学研究

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1995
    • Research Category
      Grant-in-Aid for Co-operative Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  アミド結合の立体物理化学と医薬化学への応用Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      1995
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      Chemical pharmacy
    • Research Institution
      The University of Tokyo
  •  Design, Synthesis and Biological Activity of Anti-HIV Compounds Derived from Teleocidins

    • Principal Investigator
      ENDO Yasuyuki
    • Project Period (FY)
      1995 – 1997
    • Research Category
      Grant-in-Aid for Scientific Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      University of Tokyo
  •  非細胞傷害性抗がん化合物の合成と作用解析

    • Principal Investigator
      松田 彰
    • Project Period (FY)
      1994
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      Hokkaido University
  •  核内情報伝達系の制御分子の合成と制がん作用機構

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1994 – 1995
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  アミド結合の立体特性の医薬化学への応用Principal Investigator

    • Principal Investigator
      影近 弘之
    • Project Period (FY)
      1994
    • Research Category
      Grant-in-Aid for Encouragement of Young Scientists (A)
    • Research Field
      医薬分子機能学
    • Research Institution
      The University of Tokyo
  •  臨床応用を目指すレチノイドの研究

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1993
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  非細胞傷害性抗がん化合物の合成と作用解析

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1993
    • Research Category
      Grant-in-Aid for Cancer Research
    • Research Institution
      The University of Tokyo
  •  Regulatory compound of nuclear receptor functions.

    • Principal Investigator
      SHUDO Koichi
    • Project Period (FY)
      1993 – 1995
    • Research Category
      Grant-in-Aid for Developmental Scientific Research (B)
    • Research Field
      医薬分子機能学
    • Research Institution
      University of Tokyo, Faculty of pharm.Sciences
  •  非細胞傷害性 抗がん化合物の合成と作用解析

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1992
    • Research Category
      Grant-in-Aid for Cancer Research
    • Research Institution
      The University of Tokyo
  •  核レセプター応答遺伝子の認識分子

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1992
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  核レセプタ-応答遺伝子の認識分子

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1991
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  臨床応用を目指すレチノイドの研究

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1991
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  ビタミンA酸および関連化合物による分化誘導とその機作

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1990
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  核内レセプタ-応答遺伝子の認識分子

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1990
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  臨床応用を目指す レチノイドの研究

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1990
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  Molecular design and synthesis of new retinoids

    • Principal Investigator
      SHUDO Koichi
    • Project Period (FY)
      1990 – 1992
    • Research Category
      Grant-in-Aid for Developmental Scientific Research (B)
    • Research Field
      Chemical pharmacy
    • Research Institution
      Univ. of Tokyo
  •  新しい作用機作をもつ抗がん剤の合成と特性

    • Principal Investigator
      SHUDO Koichi
    • Project Period (FY)
      1989
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  ビタミンA酸および関連化合物による分化誘導とその作用機作

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1989
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  新しい作用機作をもつ抗がん剤の合成と特性

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1988
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  ビタミンA酸および関連化合物による分化誘導とその作用機作

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1988
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo
  •  新しい作用機作をもつ抗がん剤の合成と特性

    • Principal Investigator
      首藤 紘一
    • Project Period (FY)
      1987
    • Research Category
      Grant-in-Aid for Scientific Research on Priority Areas
    • Research Institution
      The University of Tokyo

All 2024 2023 2016 2015 2014 2013 2012 2011 2010 2009 2008 2007 2006 2005 2004 2003 2002 Other

All Journal Article Presentation Book Patent

  • [Book] Expert Opinion(Thyromimetics : a review of recent reports and patents (2004-2009))2010

    • Author(s)
      Hirano, T., Kagechika, H.
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] フォルダマー、In超分子サイエンス&テクノロジー-基礎からイノベーションまで(国武豊喜監修)第3章、第1節、pp 467-4762009

    • Author(s)
      影近弘之
    • Total Pages
      10
    • Publisher
      NTS
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] Constructionof Coumarin Library for Development of Fluorescent Sensors, In' Combinatorialmethodologies for development of chemicaland biological sensors' Ed2009

    • Author(s)
      Hirano, T.; Kagechika, H.
    • Publisher
      Springer
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] Combinatorial methodologies for development of chemical and biological sensors(Ed. by Potyrailo, R. A. ; Mirsky, V. M., Construction of Coumarin Library for Development of Fluorescent Sensors, Chapter 18)2009

    • Author(s)
      Hirano, T., Kagechika, H.
    • Publisher
      Springer
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] フォルダマー、In超分子サイエンス & テクノロジー基礎からイノベーションまで(国武豊喜監修)第3章、第1節2009

    • Author(s)
      影近弘之、棚谷綾
    • Publisher
      NTS
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] Nuclear Receptor Drug Discovery in Gene Family Based MolecularDesign, Edited by Karen Lackey. Chapter 92008

    • Author(s)
      Hiroyuki Kagechika
    • Total Pages
      40
    • Publisher
      Wiley-Interscience
    • Data Source
      KAKENHI-PROJECT-19659022
  • [Book] Nuclear Receptor Drug Discovery in Gene Family Based Molecular Design, Edited by Karen Lackey. Chapter 92008

    • Author(s)
      Hiroyuki Kagechika
    • Total Pages
      40
    • Publisher
      Wiley-Interscience
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] NuclearReceptor Drug Discovery in Gene Family Based Molecular Design, Edited by KarenLackey2008

    • Author(s)
      Kagechika, H.; Tanatani, A.
    • Publisher
      Wiley-Interscience
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] Gene Family Based Molecular Design(Edited by Karen Lackey., Nuclear Receptor Drug Discovery, Chapter 9)2008

    • Author(s)
      Kagechika, H., Tanatani, A.
    • Publisher
      Wiley-Interscience
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Book] PPARs as Molecular targets for drug discovery2005

    • Author(s)
      KAGECHIKA H., Miyachi H
    • Total Pages
      7
    • Publisher
      日本臨床社
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Solvent-Dependent Conformational Switching of N-Methyl-N,N'- diarylsquaramide.2023

    • Author(s)
      Tanaka.; Takeda,F.; Kanda, M.; Kawahata,M.; Fujii,S.; Katagiri,K.; Masu, H.; Kagechika,H.; Tanatani, A.
    • Journal Title

      J. Org. Chem.

      Volume: 88 Issue: 17 Pages: 12289-12293

    • DOI

      10.1021/acs.joc.3c00918

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23KK0134, KAKENHI-PROJECT-23K06046
  • [Journal Article] Conformational Properties of Aromatic Amides Bearing Imidazole Ring and Acid-induced trans-cis Amide Switching.2023

    • Author(s)
      Takubo, C.; Kimura, S.; Ichinomiya, M.; Hayakawa, A.; Murata, M.; Urushibara, K.; Masu, H.; Katagiri, K.; Kawahata, M.; Kudo, M.; Azumaya, I.; Kagechika, H.; Tanatani, A.
    • Journal Title

      J. Org. Chem.

      Volume: 88 Issue: 24 Pages: 16707-16718

    • DOI

      10.1021/acs.joc.2c01295

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23KK0134
  • [Journal Article] Steric structure-activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9.2016

    • Author(s)
      Fujiwara T, Ohira K, Urushibara K, Ito A, Yoshida M, Kanai M, Tanatani A, Kagechika H, Hirano T.
    • Journal Title

      Bioorg. Med. Chem.

      Volume: 24 Issue: 18 Pages: 4318-4323

    • DOI

      10.1016/j.bmc.2016.07.024

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26221204, KAKENHI-PROJECT-26670052, KAKENHI-PROJECT-16K08318
  • [Journal Article] Identification of cyproheptadine as an inhibitor of SET domain containing lysine methyltransferase 7/9 (Set7/9) that regulates estrogen-dependent transcription.2016

    • Author(s)
      Takemoto Y, Ito A, Niwa H, Okamura M, Fujiwara T, Hirano T, Handa N, Umehara T, Sonoda T, Ogawa K, Tariq M, Nishino N, Dan S, Kagechika H, Yamori T, Yokoyama S, Yoshida M.
    • Journal Title

      J. Med. Chem.

      Volume: 59 Issue: 8 Pages: 3650-3660

    • DOI

      10.1021/acs.jmedchem.5b01732

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26221204, KAKENHI-PROJECT-16H05105, KAKENHI-PROJECT-26670052, KAKENHI-PROJECT-15K08019
  • [Journal Article] All trans-retinoic acid analogs promote cancer cell apoptosis through non-genomic Crabp1 mediating ERK1/2 phosphorylation2016

    • Author(s)
      Persaud, S. D.; Park, S. W.; Ishigami-Yuasa, M.; Koyano-Nakagawa, N.;, Kagechika, H.; Wei, L.-N.
    • Journal Title

      Sci. Rep

      Volume: 6 Issue: 1 Pages: 22396-22396

    • DOI

      10.1038/srep22396

    • Peer Reviewed / Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Journal Article] Structural development of canthin-5,6-dione moiety as a fluorescent dye and its application to novel fluorescent sensors.2016

    • Author(s)
      Yokoo, H.; Ohsaki, A.; Kagechika, H.; Hirano T.
    • Journal Title

      Tetrahedron

      Volume: 72 Issue: 39 Pages: 5872-5879

    • DOI

      10.1016/j.tet.2016.08.014

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-26670052, KAKENHI-PROJECT-15K08019, KAKENHI-PROJECT-16K01921
  • [Journal Article] Development of 1,3-diphenyladamantane derivatives as nonsteroidal progesterone receptor antagonists.2015

    • Author(s)
      Mori, S.; Takeuchi, Y.; Tanatani, A.; Kagechika, H.; Fujii, S.
    • Journal Title

      Bioorg. Med. Chem

      Volume: 23 Issue: 4 Pages: 803-809

    • DOI

      10.1016/j.bmc.2014.12.047

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-24590137, KAKENHI-PROJECT-25460146
  • [Journal Article] 6-Arylcoumarins: versatile scaffolds for fluorescent sensors2015

    • Author(s)
      Takuya Shiraishi, Hiroyuki Kagechika, Tomoya Hirano
    • Journal Title

      New Journal of Chemistry

      Volume: 39 Issue: 11 Pages: 8389-8396

    • DOI

      10.1039/c5nj01609f

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PROJECT-15K08019, KAKENHI-PROJECT-26670052
  • [Journal Article] A new cell-based assay to evaluate myogenesis in mouse myoblast C2C12 cells2015

    • Author(s)
      Kodaka, M.; Yang, Z.; Nakagawa, K.; Maruyama, J.; Xu, X.; Sarkar, A.; Ichimura, A.; Nasu, Y.; Ozawa, T.; Iwasa, H.; Ishigami-Yuasa, M.; Ito, S.; Kagechika, H.; Hata, Y.
    • Journal Title

      Exp. Cell. Res.

      Volume: 336 Issue: 2 Pages: 171-181

    • DOI

      10.1016/j.yexcr.2015.06.015

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-26670052, KAKENHI-PROJECT-26860185, KAKENHI-PROJECT-26293061, KAKENHI-PROJECT-26220805
  • [Journal Article] Design and synthesis of tetraol derivatives of 1,12-dicarba-closo-dodecaborane as non-secosteroidal vitamin D analogs.2014

    • Author(s)
      Fujii, S.; Kano, A.; Masuno, H.; Songkram, C.; Kawachi, E.; Hirano, T.; Tanatani, A.; Kagechika, H
    • Journal Title

      Bioorg. Med. Chem. Lett.

      Volume: 24 Issue: 18 Pages: 4515-4519

    • DOI

      10.1016/j.bmcl.2014.07.075

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-24590005, KAKENHI-PROJECT-24590137, KAKENHI-PROJECT-25460146
  • [Journal Article] Retinoic acid receptor signaling is required to maintain glucose-stimulated insulin secretion and β-cell mass.2014

    • Author(s)
      Brun, P.-J.; Grijalva, A.; Rausch, R.; Watson, E.; Yuen, J. J.; Das, B. C.; Shudo, K.; Kagechika, H.; Leibel, R. L.; Blaner, W. S.
    • Journal Title

      FASEB J

      Volume: 29 Issue: 2 Pages: 671-683

    • DOI

      10.1096/fj.14-256743

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Journal Article] Retinoic acid receptor-α up-regulates proopiomelanocortin gene expression in AtT20 corticotroph cells2014

    • Author(s)
      Uruno, A.; Saito-Hakoda, A.; Yokoyama, A.; Kogure, N.; Matsuda, K.; Parvin, R.; Shimizu, K.; Sato, I.; Kudo, M.; Yoshikawa, T.; Kagechika, H.; Iwasaki, Y.; Ito, S.; Sugawara, A.
    • Journal Title

      Endocr J

      Volume: 61 Issue: 11 Pages: 1105-1114

    • DOI

      10.1507/endocrj.EJ14-0115

    • NAID

      130004677954

    • ISSN
      0918-8959, 1348-4540
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-26460383
  • [Journal Article] Activation of liver X receptor suppresses the production of the IL-12 family of cytokines by blocking nuclear translocation of NF-kappa Bp502014

    • Author(s)
      Canavan, M.; McCarthy, C.; Ben Larbi, N.; Dowling, J. K.; Collins, L.; O'Sullivan, F.; Hurley, G.; Murphy, C.; Quinlan, A.; Moloney, G.; Darby, T.; MacSharry, J.; Kagechika, H.; Moynagh, P.; Melgar, S.; Loscher, C. E.
    • Journal Title

      Innate Immun.

      Volume: 20 Issue: 7 Pages: 675-687

    • DOI

      10.1177/1753425913501915

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Journal Article] Development of a novel fluorescent sensor to detect a specific range of pH2014

    • Author(s)
      Shiraishi, T.; Saito, T.; Kagechika, H.; Hirano, T.
    • Journal Title

      Tetrahedron Lett.

      Volume: 55 Issue: 50 Pages: 6784-6786

    • DOI

      10.1016/j.tetlet.2014.10.037

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-24590005, KAKENHI-PROJECT-26670052
  • [Journal Article] Design and synthesis of nonsteroidal progesterone receptor antagonists based on C,C’-diphenylcarborane scaffold as a hydrophobic pharmacophore.2014

    • Author(s)
      Fujii, S.; Yamada, A.; Nakano, E.; Takeuchi, Y.; Mori, S.; Masuno, H.; Kagechika, H.
    • Journal Title

      Eur. J. Med. Chem.

      Volume: 84 Pages: 264-277

    • DOI

      10.1016/j.ejmech.2014.07.034

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-25460146
  • [Journal Article] Screening with a Novel Cell-Based Assay for TAZ Activators Identifies a Compound That Enhances Myogenesis in C2C12 Cells and Facilitates Muscle Repair in a Muscle Injury Model.2014

    • Author(s)
      Yang, Z. Y.; Nakagawa, K.; Sarkar, A.; Maruyama, J.; Iwasa, H.; Bao, Y. J.; Ishigami-Yuasa, M.; Ito, S.; Kagechika, H.; Hata, S.; Nishina, H.; Abe, S.; Kitagawa, M.; Hata, Y.
    • Journal Title

      Mol. Cell. Biol.

      Volume: 34 Issue: 9 Pages: 1607-1621

    • DOI

      10.1128/mcb.01346-13

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23790325, KAKENHI-PLANNED-26114005, KAKENHI-PROJECT-26293012, KAKENHI-PROJECT-26293061, KAKENHI-PROJECT-26860185
  • [Journal Article] Synthesis and structure-activity relationship of p-carborane-based non-secosteroidal vitamin D analogs.2014

    • Author(s)
      Fujii, S.; Kano, A.; Songkram, C.; Masuno, H.; Tao da, Y.; Kawachi, E.; Hirano, T.; Tanatani, A.; Kagechika, H.
    • Journal Title

      Bioorg. Med. Chem.

      Volume: 22 Issue: 4 Pages: 1227-1235

    • DOI

      10.1016/j.bmc.2014.01.015

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-24590005, KAKENHI-PROJECT-24590137, KAKENHI-PROJECT-25460146
  • [Journal Article] Lipase-catalyzed asymmetric acylation of boron cluster-containing secondary alcohols.2014

    • Author(s)
      Mori, S.; Takagaki, R.; Fujii, S.; Matsumura, M.; Tanatani, A.; Kagechika, H.
    • Journal Title

      Tetrahedron Asymm.

      Volume: 25 Issue: 23 Pages: 1505-1512

    • DOI

      10.1016/j.tetasy.2014.10.009

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-24590137, KAKENHI-PROJECT-25460146, KAKENHI-PROJECT-26670052
  • [Journal Article] Structural development of p-carborane-based potent non-secosteroidal vitamin D analogs.2014

    • Author(s)
      Fujii, S.; Sekine, R.; Kano, A.; Masuno, H.; Songkram, C.; Kawachi, E.; Hirano, T.; Tanatani, A.; Kagechika, H.
    • Journal Title

      Bioorg. Med. Chem

      Volume: 22 Issue: 21 Pages: 5891-5901

    • DOI

      10.1016/j.bmc.2014.09.020

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-24590005, KAKENHI-PROJECT-24590137, KAKENHI-PROJECT-25460146
  • [Journal Article] Development of p-carborane-based nonsteroidal progesterone receptor antagonists.2014

    • Author(s)
      Fujii, S.; Nakano, E.; Yanagida, N.; Mori, S.; Masuno, H.; Kagechika, H.
    • Journal Title

      Bioorg. Med. Chem.

      Volume: 22 Issue: 19 Pages: 5329-5337

    • DOI

      10.1016/j.bmc.2014.07.049

    • Peer Reviewed / Acknowledgement Compliant
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-25460146
  • [Journal Article] Retinoid X receptor a attenuates host antiviral response by suppressing type I interferon.2014

    • Author(s)
      Ma, F.; Liu, S.-Y.; Razani, B.; Arora, N.; Li, B.; Kagechika, H.; Tontonoz, P.; Nunez, V.; Ricote, M.; Cheng, G.
    • Journal Title

      Nat. Commun

      Volume: 5 Issue: 1 Pages: 5494-5494

    • DOI

      10.1038/ncomms6494

    • Peer Reviewed / Open Access
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Journal Article] Synthesis and Structure–Activity Relationship Study of Triazine-Based Inhibitors of the DNA Binding of NF-κB2014

    • Author(s)
      Fujii, S.; Kobayashi, T.; Nakatsu, A.; Miyazawa, H.; Kagechika, H.
    • Journal Title

      Chemical and Pharmaceutical Bulletin

      Volume: 62 Issue: 7 Pages: 700-708

    • DOI

      10.1248/cpb.c14-00218

    • NAID

      130004053804

    • ISSN
      0009-2363, 1347-5223
    • Language
      English
    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-25460146
  • [Journal Article] The Retinoic Acid Receptor Agonist Am80 Increases Mucosal Inflammation in an IL-6 Dependent Manner During Trichuris muris Infection.2013

    • Author(s)
      Hurst, R. J. M.; De Caul, A.; Little, M. C.; Kagechika, H.; Else, K. J.
    • Journal Title

      J. Clin. Immunol.

      Volume: 33 Issue: 8 Pages: 1386-1394

    • DOI

      10.1007/s10875-013-9936-8

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Journal Article] Molecular mechanism of 9-cis-retinoic acid inhibition of adipogenesis in 3T3-L1 cells.2013

    • Author(s)
      Sagara, C.; Takahashi, K.; Kagechika, H.; Takahashi, N.
    • Journal Title

      Biochem. Biophys. Res. Commun.

      Volume: 433 Issue: 1 Pages: 102-107

    • DOI

      10.1016/j.bbrc.2013.02.057

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-22590074, KAKENHI-PROJECT-23659051
  • [Journal Article] Design and synthesis of 4-(4-benzoylaminophenoxy)phenol derivatives as androgen receptor antagonists.2013

    • Author(s)
      Yamada, A.; Fujii, S.; Mori, S.; Kagechika, H.
    • Journal Title

      ACS Med. Chem. Lett.

      Volume: 4 Issue: 10 Pages: 937-941

    • DOI

      10.1021/ml4001744

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-25460146
  • [Journal Article] Retinoid X Receptor Agonists Modulate Foxp3 + Regulatory T Cell and Th17 Cell Differentiation with Differential Dependence on Retinoic Acid Receptor Activation.2013

    • Author(s)
      Takeuchi, H.; Yokota-Nakatsuma, A.; Ohoka, Y.; Kagechika, H.; Kato, C.; Si-Young Song, S.-Y.; Iwata, M.
    • Journal Title

      J. Immunol.

      Volume: 191 Issue: 7 Pages: 3725-3733

    • DOI

      10.4049/jimmunol.1300032

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23390023, KAKENHI-PROJECT-23590317, KAKENHI-ORGANIZER-24111001, KAKENHI-PROJECT-24590106, KAKENHI-PUBLICLY-25111514, KAKENHI-PROJECT-25450190
  • [Journal Article] Structure-activity relationship study on benzoic acid part of diphenylamine-based retinoids2013

    • Author(s)
      Ohta, K.; Kawachi, E.; Shudo, K.; Kagechika, H
    • Journal Title

      Bioorg. Med. Chem. Lett

      Volume: 23 Issue: 1 Pages: 81-84

    • DOI

      10.1016/j.bmcl.2012.11.008

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-24790115, KAKENHI-PLANNED-22136013
  • [Journal Article] Chemical library screening for WNK signalling inhibitors using fluorescence correlation spectroscopy.2013

    • Author(s)
      Mori, T.; Kikuchi, E.; Watanabe, Y.; Fujii, S.; Ishigami-Yuasa, M.; Kagechika, H.; Sohara, E.; Rai, T.; Sasaki, S.; Uchida, S.
    • Journal Title

      Biochem. J.

      Volume: 455 Issue: 3 Pages: 339-345

    • DOI

      10.1042/bj20130597

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-22249032, KAKENHI-PROJECT-22390168, KAKENHI-PROJECT-24659412, KAKENHI-PROJECT-24790836, KAKENHI-PROJECT-25221306, KAKENHI-PROJECT-25460146, KAKENHI-PROJECT-25670406
  • [Journal Article] Increased Hydrophobicity and Estrogenic Activity of Simple Phenols with Silicon and Germanium- Containing Substituents2013

    • Author(s)
      Fujii, S.
    • Journal Title

      J. Med. Chem.

      Volume: 56 Issue: 1 Pages: 160-166

    • DOI

      10.1021/jm3013757

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128, KAKENHI-PLANNED-22136013
  • [Journal Article] Development of Androgen Recby Application of Ten-vertex p-Carborane as a Novel Hydrophobic Core Structure2012

    • Author(s)
      Shinya Fujii, Kiminori Ohta, Tokuhito Goto, Akifumi Oda, Hiroyuki Masuno, Ysuyuki Endo, Hiroyuki Kagechika
    • Journal Title

      Med. Chem. Commun

      Volume: 3 Issue: 6 Pages: 680-684

    • DOI

      10.1039/c2md00294a

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128, KAKENHI-PROJECT-23790137, KAKENHI-PROJECT-24790115, KAKENHI-PLANNED-22136013
  • [Journal Article] Retinoic acid receptor agonists regulate expression of ATP-binding cassette transporter G1 in macrophages2012

    • Author(s)
      Ayaori, M., 他15名
    • Journal Title

      Biochimica et Biophysica Acta-Molecular and Cell Biology of Lipids

      Volume: 1821 Issue: 4 Pages: 561-572

    • DOI

      10.1016/j.bbalip.2012.02.004

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-22310042, KAKENHI-PROJECT-22591003, KAKENHI-PROJECT-23659051, KAKENHI-PLANNED-22136013
  • [Journal Article] Retinoid X receptorgamma signaling accelerates CNSremyelination2011

    • Author(s)
      Huang, J. K.; Jarjour, A. A.; Nait-Oumesmar, B.; Kerninon, C.; Williams, A. Krezel, W.; Kagechika, H.; Bauer, J.; Zhao, C.; Baron-Van Evercooren, A.; Chambon, P.; ffrench-Constant, C.; Franklin, R. J. M.
    • Journal Title

      Nature Neurosci

      Volume: 14 Pages: 45-53

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Boron Cluster-based DevNon-Secosteroidal Vitamin D Receptor Ligands: Direct Observation of Hydrophobic Interaction between Protein Surface and Carborane2011

    • Author(s)
      Shinya Fujii, Hiroyuki Masuno, Yoshiyuki Taoda, Atsushi Kano, Angsuma Wongmayura, Makoto Nakabayashi, Nobutoshi Ito, Masato Shimizu, Emiko Kawachi, Tomoya Hirano, YasuyukiEndo, Aya Tanatani, Hiroyuki Kagechika
    • Journal Title

      J. Am. Chem. Soc

      Volume: 133 Issue: 51 Pages: 20933-20941

    • DOI

      10.1021/ja208797n

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390035, KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-22790106, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128
  • [Journal Article] Tributyltin chlorideinduces ABCA1 expression andapolipoprotein A-I-mediated cellularcholesterol efflux by activatingLXRalpha/RXR2011

    • Author(s)
      Cui, H.; Okuhira, K.; Ohoka, N.; Naito, M.; Kagechika, H.; Hirose, A, ; Nishimaki-Mogami, T.
    • Journal Title

      Biochem. Pharmacol

      Volume: 81 Pages: 819-824

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] p-Carborane Based AndrogenActive in LNCaP Cells with a Mutated Androgen Receptor2011

    • Author(s)
      Shinya Fujii, Ayumi Yamada, Keiko Tomita, Mao Nagano, Tokuhito Goto, Kiminori Ohta, Takashi Harayama, Yasuyuki Endo, Hiroyuki Kagechika
    • Journal Title

      Med. Chem. Commun

      Volume: 2 Issue: 9 Pages: 877-880

    • DOI

      10.1039/c1md00001b

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116, KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128
  • [Journal Article] Efficient and diversity-oriented total synthesis of Riccardin C and application to develop novel macrolactam derivatives2011

    • Author(s)
      Iwashita, M.
    • Journal Title

      Tetrahedron

      Volume: 67 Issue: 33 Pages: 6073-6082

    • DOI

      10.1016/j.tet.2011.06.018

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790128
  • [Journal Article] Diphenylamine-based Retinoid Anatagonists : Regulation of RAR and RXR Function Depending on the N-substituent2011

    • Author(s)
      Ohta, K.; Kawachi, E.; Fukasawa, H., Shudo, K.; Kagechika, H.
    • Journal Title

      Bioorg. Med. Chem

      Volume: 19 Issue: 8 Pages: 2501-2507

    • DOI

      10.1016/j.bmc.2011.03.026

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-21790116, KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-23659051
  • [Journal Article] 6-Arylcoumarins as novel nonsteroidal type progesterone antagonists : An example with receptor-binding-dependent fluorescence2011

    • Author(s)
      Sakai, H.
    • Journal Title

      J.Med.Chem.

      Volume: 54 Issue: 20 Pages: 7055-7065

    • DOI

      10.1021/jm2005404

    • Peer Reviewed
    • Data Source
      KAKENHI-PLANNED-22136013, KAKENHI-PROJECT-22790106, KAKENHI-PROJECT-23659051, KAKENHI-PROJECT-23790127, KAKENHI-PROJECT-23790128
  • [Journal Article] Efficient Induction of CCR9 onT Cells Requires Coactivation of RetinoicAcid Receptors and Retinoid X Receptors (RXRs): Exaggerated T Cell Homing to theIntestine by RXR Activation withOrganotins2010

    • Author(s)
      Takeuchi, H.; Yokota, A.; Ohoka, Y.; Kagechika, H.; kato, C.; Song, S.-Y.; Iwata, M.
    • Journal Title

      J. Immunol

      Volume: 185 Pages: 5289-5299

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Modulation of intramolecularheterodimer-induced fluorescencequenching of tricarbocyanine dye for thedevelopment of fluorescent sensors2010

    • Author(s)
      Hirano, T.; Akiyama, J.; Mori, S.; Kagechika, H.
    • Journal Title

      Org. Biomol. Chem

      Volume: 8 Pages: 5568-5575

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Inhibition of Mammary Carcinoma CellGrowth by RXR is Mediated by the Receptor's Oligomeric Switch2010

    • Author(s)
      Yasmin, R.; Kannan-Thulasiraman, P.; Kagechika, H.; Dawson, M. I.; Noy, N.
    • Journal Title

      J. Mol. Biol.

      Volume: 397 Pages: 1121-1131

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Retinoic Acid Induces Expression of theThyroid Hormone Transporter, Monocarboxylate Transporter 8(Mct8)2010

    • Author(s)
      Kogai, T.; Liu, Y.-Y.; Richter, L. L.; Mody, K.; Kagechika, H.; Bent, G. A.
    • Journal Title

      J. Biol. Chem

      Volume: 285 Pages: 27279-27288

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Design and Synthesis ofNovel Retinoid Synergists having aDibenzodiazepine Skeleton2010

    • Author(s)
      Ohta, K.; Kawachi, E.; Shudo, K.; Kagechika, H.
    • Journal Title

      Heterocycles

      Volume: 81 Pages: 2465-2470

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Developmentof novel bisubstrate-type inhibitors ofhistone methyltransferase SET7/92010

    • Author(s)
      Mori, S.; Iwase, K.; Iwanami, N.; Tanaka, Y.; Kagechika, H.; Hirano, T.
    • Journal Title

      Bioorg. Med. Chem

      Volume: 18 Pages: 8158-8168

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Activation of the PI3 Kinase Pathway By Retinoic Acid Mediates Sodium/Iodide Symporter Induction and Iodide Transport in MCF-7 Breast CancerCells2009

    • Author(s)
      Ohashi, E.; Kogai, T.; Kagechika, H.; Brent, G. A.
    • Journal Title

      Cancer Res

      Volume: 69 Pages: 3443-3450

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure2009

    • Author(s)
      Shinya Fujii, Kiminori Ohta, TokuhitoGoto, Hiroyuki Kagechika, Yasuyuki Endo
    • Journal Title

      Bioorg. Med. Chem

      Volume: 17 Issue: 1 Pages: 344-350

    • DOI

      10.1016/j.bmc.2008.10.060

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390035, KAKENHI-PROJECT-21790116
  • [Journal Article] Activation of Testicular Orphan Receptor 4 by Fatty Acids2009

    • Author(s)
      Tsai, N.-P., Huq, M., Gupta, P., Yamamoto, K., Kagechika, H., Wei, L.-N.
    • Journal Title

      Biochim.Biophys.Acta-Gene Regul.Mech. 1789

      Pages: 734-740

    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Acidicheterocycles as novel hydrophilicpharmacophore of androgen receptorligands with a carborane core structure. Bioorg2009

    • Author(s)
      Fujii, S.; Ohta, K.; Goto, T.; Kagechika, H.; Endo, Y.
    • Journal Title

      Med. Chem

      Volume: 17 Pages: 344-350

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Thetranscriotion factors Nur77 and retinoid X receptors participate in amphetamine-induced locomotor activities2009

    • Author(s)
      Bourhis, E.; Maheux, J.; Paquet, B.; Kagechika, H.; Shudo, K.; Rompre, P.; Rouillard, C.; Levesque, D.
    • Journal Title

      Psychopharmacol

      Volume: 202 Pages: 635-648

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] ApoC-III gene expression issharply increased during adipogenesis andis augmented by retinoid X receptor(RXR) agonists2009

    • Author(s)
      Takahashi, Y.; Inoue, J.; Kagechika, H.; Sato, R.
    • Journal Title

      FEBS Lett

      Volume: 583 Pages: 493-497

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Contribution of AP-1 interference induced by TAC-101 to tumor growth suppression in a hepatocellular carcinoma model2009

    • Author(s)
      Eshima, K., Fukaya S., Sugimoto, A., Mori, T., Yokoi, H., Yamamoto, Y., Sugiura, S., Honda, S., Masuko, N., Murakami, K., Yamasaki, Y., Kagechika, H.
    • Journal Title

      Tumor Biol. 30

      Pages: 1-7

    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure2009

    • Author(s)
      Fujii, S., Ohta, K., Goto, T., Kagechika, H., Endo, Y.
    • Journal Title

      Bioorg.Med.Chem. 17

      Pages: 344-350

    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Encapsulation of thesynthetic retinoids Am80 and LE540 intopolymeric micelles and the retinoids' rerease control2009

    • Author(s)
      Satoh, T.; Higuchi, Y.; Kawakami, S.; Hashida, M.; Kagechika, H.; Shudo, K.; Yokoyama, M.
    • Journal Title

      J. Controlled Release

      Volume: 136 Pages: 187-195

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Activation of Testicular Orphan Receptor4 by Fatty Acids2009

    • Author(s)
      Tsai, N.-P.; Huq, M.; Gupta, P.; Yamamoto, K.; Kagechika, H.; Wei, L.-N.
    • Journal Title

      Biochim. Biophys. Acta-Gene Regul. Mech

      Volume: 1789 Pages: 734-740

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Contribution of AP-1 interference induced by TAC-101 totumor growth suppression in ahepatocellular carcinoma model2009

    • Author(s)
      Eshima, K.; Fukaya S.; Sugimoto, A.; Mori, T.; Yokoi, H.; Yamamoto, Y.; Sugiura, S.; Honda, S.; Masuko, N.; Murakami, K.; Yamasaki, Y.; Kagechika, H.
    • Journal Title

      TumorBiol

      Volume: 30 Pages: 1-7

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Identification of an intermediate in the deboronation of ortho-carborane: an adduct of ortho-carborane with two nucleophiles on one boron atom2008

    • Author(s)
      Yoshiyuki Taoda, Takehiko Sawabe, Yasuyuki Endo, Kentaro Yamaguchi, Shinya Fujii, Hiroyuki Kagechika
    • Journal Title

      Chem. Commun

      Issue: 17 Pages: 2049-2051

    • DOI

      10.1039/b716079h

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-20390035
  • [Journal Article] The RXR agonists PA024 and HX630 have different abilities to activate LXR/RXR and to induce ABCA1 expression in macrophage cell line2008

    • Author(s)
      Nishimaki-Mogami, T., Tamehiro, N., Sato, Y., Okuhira, K., Sai, K., Kagechika, H., Shudo, K., Abe-Dohmae, S., Yokoyama, S., Ohno, Y., Inoue, K., Sawada, J.
    • Journal Title

      Biochem.Pharmacol. 76

      Pages: 1006-1013

    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Identification of An Intermediate in the Deboronation of or tho-Carborane : An Adduct of ortho-Carborane with Two Nucleophiles on One Boron Atom2008

    • Author(s)
      Taoda, Y.; Sawabe, T.; Endo, Y. Yamaguchi, K.; Fujii, S.; Kagechika, H.
    • Journal Title

      Chem. Commun

      Pages: 2049-2051

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] Effects of retinoic acids on the dendritic morphology of cultured hippocampal meurons2008

    • Author(s)
      Liu, Y.; Kagechika, H.; Ishikawa, J.; Hirano, H.; Matsukuma, S.; Tanaka, K.; Nakamura, S.
    • Journal Title

      J. Neurochem

      Volume: 106 Pages: 1104-1116

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] The RXRagonists PA024 and HX630 have different abilities to activate LXR/RXR and toinduce ABCA1 expression in macrophage cellline2008

    • Author(s)
      Nishimaki-Mogami, T.; Tamehiro, N.; Sato, Y.; Okuhira, K.; Sai, K.; Kagechika, H.; Shudo, K.; Abe-Dohmae, S.; Yokoyama, S.; Ohno, Y.; Inoue, K.; Sawada, J.
    • Journal Title

      Biochem. Pharmacol

      Volume: 76 Pages: 1006-1013

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] b-Cryptoxanthin, a novel natural RAR ligand, induces ATP-binding cassette transporters inmacrophages2007

    • Author(s)
      Matsumoto, A.; Mizukami, H.; Mizuno, S.; Umegaki, K.; Nishikawa, J.; Shudo, K.; Kagechika, H.; Inoue, M.
    • Journal Title

      Biochem. Pharmacol

      Volume: 74 Pages: 256-264

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] STAT5a/PPARg Pathway Regulates Involucrin Expression in Keratinocyte Differentiation2007

    • Author(s)
      Dai, X.; Sayama, K.; Shirakata, Y.; Hanakawa, Y.; Yamasaki, K.; Tokumaru, S.; Yang, L.; Wang, X.; Hirakawa, S.; Tohyama, M.; Yamauchi, T.; Kadowaki, T.; Kagechika, H.; Hashimoto, K.
    • Journal Title

      J. Invest. Dermatol

      Volume: 127 Pages: 1728-1735

    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Journal Article] All-trans retinoic acid induces in vitro angiogenesis viaretinoic acid receptor : possible involvement of endogenous vascular endothelial growth factor signaling.2007

    • Author(s)
      Saito A, Sugawara A, Uruno A, Kudo M, Kagechika H, Sato Y, Owada Y, Kondo H, Sato M, Kurabayashi M, Imaizumi M, Tsuchiya S, Ito S
    • Journal Title

      Endocrinology 148

      Pages: 1412-1423

    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] All-trans retinoic acid induces in vitro angiogenesis via retinoic acid receptor: possible involvement of endogenous vascular endothelial growth factor signaling.2007

    • Author(s)
      Saito A, Sugawara A, Uruno A, Kudo M, Kagechika H, Sato Y, Owada Y, Kondo H, Sato M, Kurabayashi M, Imaizumi M, Tsuchiya S, Ito S
    • Journal Title

      Endocrinology 148

      Pages: 1412-1423

    • Description
      「研究成果報告書概要(和文)」より
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] All-trans retinoic acid induces in vitro angiogenesis via retinoic acid receptor: possible involvement of endogenous vascular endothelial growth factor signaling2007

    • Author(s)
      Saito A, Sugawara A, Uruno A, Kudo M, Kagechika H, Sato Y, Owada Y, Kondo H, Sato M, Kurabayashi M, Imaizumi M, Tsuchiya S, Ito S.
    • Journal Title

      Endocrinology 148

      Pages: 1412-1423

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] 全トランス型レチノイン酸および合成レチノイドAm80の血管内皮細胞における遺伝子発現に及ぼす影響-マイクロアレイを用いた検討-。2006

    • Author(s)
      菅原 明, 斉藤明子, 宇留野晃, 今泉益栄, 工藤正孝, 影近弘之, 本郷道夫, 伊藤貞嘉
    • Journal Title

      血圧 13

      Pages: 250-252

    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] 全トランス型レチノイン酸および合成レチノイドAm80の血管内皮細胞における遺伝子発現に及ぼす影響-マイクロアレイを用いた検討-。2006

    • Author(s)
      菅原 明、斉藤明子、宇留野晃、今泉益栄、工藤正孝、影近弘之、本郷道夫、伊藤貞嘉
    • Journal Title

      血圧 13

      Pages: 250-252

    • Description
      「研究成果報告書概要(和文)」より
    • Peer Reviewed
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] Effects of ATRA and synthetic retinoid Am80 on endothelial gene expression-DNA microarray analyses2006

    • Author(s)
      Sugawara A, Saito A, Uruno A, Imaizumi M, Kudo M, Kagechika H, Hongo M, Ito S.
    • Journal Title

      Ketsuatsu 13

      Pages: 250-252

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Journal Article] Synthetic Retinoids : Recent Developments Concerning Structure and Clinical Utility2005

    • Author(s)
      Kagechika, H.
    • Journal Title

      J.Med.Chem. 48

      Pages: 5875-5883

    • Data Source
      KAKENHI-PROJECT-17035024
  • [Journal Article] Up-regulation of nitric oxide production in vascular endothelial cells by all-trans retinoic acid through the phosphoinositide 3-kinase/Akt pathway.2005

    • Author(s)
      Uruno A, Sugawara A, Kanatsuka H, Kagechika H, Saito A, Sato K, Kudo M, Takeuchi K, Ito S
    • Journal Title

      Circulation. 112

      Pages: 727-736

    • NAID

      120001182109

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-16590898
  • [Journal Article] PPARs as Molecular targets for drug discovery.2005

    • Author(s)
      KAGECHIKA H., Miyachi H.
    • Journal Title

      NIPPON RINSHO 63

      Pages: 549-555

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Synthetic Retinoids : Recent Developments Concerning Structure and Clinical Utility2005

    • Author(s)
      Kagechika, H.
    • Journal Title

      J.Med.Chem. 48

      Pages: 5875-5883

    • Data Source
      KAKENHI-PROJECT-17651120
  • [Journal Article] Nobel RXR antagonists enhance transactivaqtion of PPARγ and ST 13 preadipocyte differentiation.2004

    • Author(s)
      Sato M., A.Sugawara, N.Egawa, Y.Yajima, H.Kato, H.Kagechika
    • Journal Title

      12^<th> Internatinal Congress of Endocrinology

      Pages: 547-551

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Competitive RXR antagonists enhance transactivation of PPARγ and ST 13 preadipocyte differentiation 12^<th> International Congress of Endcrinology.2004

    • Author(s)
      MAYUMI SATO, AKIRA SUGAWARA, NAOTO EGAWA, YUKIKO YAJIMA, HIROYUKI KAGECHIKA.
    • Journal Title

      Portugal

      Pages: 831-904

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Novel retinoid X receptor (RXR) antagonists having a dicarba-closo-dodecaboane as a hydrophobic moiety.2004

    • Author(s)
      Ohta K, Iijima T, Kawachi E, Kagechika H, Endo Y.
    • Journal Title

      Bioorg Med Chem Lett 14

      Pages: 5913-5918

    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Nobel RXR antagonists enhance transactivaqtion of PPARγ and ST 13 Preadipocyte differentiation.2004

    • Author(s)
      Sato M., A.Sugawara, N.Egawa, Y.Yajima, H.Kato, H.Kagechika
    • Journal Title

      Internatinal Congress of Endocrinology

      Pages: 547-551

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Nobel RXR antagonists enhance transactivation of PPARg and ST 13 preadipocyte differentiation.2004

    • Author(s)
      Sato M, Sugawara A, Egawa N, Yajima Y, Kato H, Kagechika H
    • Journal Title

      12th Internatinal Congress of Endocrinology International Proceedings.

      Pages: 547-551

    • Data Source
      KAKENHI-PROJECT-16590898
  • [Journal Article] Design and synthesis of cyclic urea compounds : a pharmacological study for retinoidal activity.2004

    • Author(s)
      Kurihara M, Rouf AS, Kansui H, Kagechika H, Okuda H, Miyata N.
    • Journal Title

      Bioorg Med Chem Lett. 14(16)

      Pages: 4131-4134

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Design and synthesis of cyclic urea compounds : a pharmacological study for retinoidal activity2004

    • Author(s)
      Kurihara M, Rouf AS, Kansui H, Kagechika H, Okuda H, Miyata N.
    • Journal Title

      Bioorg Med Chem Lett 14

      Pages: 4131-4134

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Amide conformational switching induced by protonation of aromatic substituent..2003

    • Author(s)
      Yamasaki R, Tanatani A, Azumaya I, Saito S, Yamaguchi K, Kagechika H.
    • Journal Title

      Org Lett 5

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effect of synthetic retinoid, TAC-101, on experimental autoimmune disease.2003

    • Author(s)
      Miyagawa N, Homma T, Kagechika H, Shudo K, Nagai H.
    • Journal Title

      Pharmacology 7(1)

      Pages: 21-31

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Clinically potential subclasses of retinoid synergists revealed by gene expression profiling2003

    • Author(s)
      Ishida S, Shigemoto-Mogami Y, Kagechika H. et al.
    • Journal Title

      Mol Cancer Ther. 1

      Pages: 49-58

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Cyclooxygenase inhibitors derived from thalidomide.2003

    • Author(s)
      Suizu M, Muroya Y, Kakuta H, Kagechika H, Tanatani A, Nagasawa K, Hashimoto Y.
    • Journal Title

      Chem Pharm Bull (Tokyo) 9

      Pages: 1098-1102

    • NAID

      110003615465

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effects of retinoid ligands on RIP140 : molecular interaction with retinoid receptors and biological activity.2003

    • Author(s)
      Farooqui M, Franco PJ, Thompson J, Kagechika H, et al.
    • Journal Title

      Biochemistry 42

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Utility of boron clusters for drug design. Relation between estrogen receptor binding affinity and hydrophobicity of phenols bearing various types of carboranyl groups.2003

    • Author(s)
      Endo Y, Yamamoto K, Kagechika H.
    • Journal Title

      Bioorg Med Chem Lett. 13(22)

      Pages: 4089-4092

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effects of retinoid ligands on RIP 140 : molecular interaction with retinoid receptors and biological activity.2003

    • Author(s)
      Farooqui M, Franco PJ, Thompson J, Kagechika H, Chandraratna RA, Banaszak L, Wei LN.
    • Journal Title

      Biochemistry 42(4)

      Pages: 971-979

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Utility of boron clusters for drug design. Relation between estrogen receptor binding affinity and hydrophobicity of phenols bearing various types of carboranyl groups.2003

    • Author(s)
      Endo Y, Yamamoto K, Kagechika H.
    • Journal Title

      Bioorg Med Chem Lett 13

      Pages: 4089-4092

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Cyclooxygenase inhibitors derived from thalidomide.2003

    • Author(s)
      Suizu M, Muroya Y, Kakuta H, Kagechika H, Tanatani A, Nagasawa K, Hashimoto Y
    • Journal Title

      Chem Pharm Bull 9

      Pages: 1098-102

    • NAID

      110003615465

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Amide conformational switching induced by protonation of aromatic substituent.2003

    • Author(s)
      Yamasaki R, Tanatani A, Azumaya I, Saito S, Yamaguchi K, Kagechika H.
    • Journal Title

      Org Lett. 5(8)

      Pages: 1265-1267

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effect of synthetic retinoid, TAC-101, on experimental autoimmune disease.2003

    • Author(s)
      Miyagawa N, Homma T, Kagechika et al.
    • Journal Title

      Pharmacology. 7

      Pages: 21-31

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Clinically potential subclasses of retinoid synergists revealed by gene expression profiling.2003

    • Author(s)
      Ishida S, Shigemoto-Mogami Y, Kagechika H, Shudo K, Ozawa S, Sawada J, Ohno Y, Inoue K.
    • Journal Title

      Mol Cancer Ther. (1)

      Pages: 49-58

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Novel retinoid X receptor antagonists : specific inhibition of retinoid synergism in RXR-RAR heterodimer actions.2002

    • Author(s)
      Takahashi B, Ohta K, Kawachi E, Fukasawa H, Hashimoto Y, Kagechika H.
    • Journal Title

      J Med Chem. 45(16)

      Pages: 3327-3330

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effect of natural and synthetic retinoids on the proliferation and differentiation of three canine melanoma cell lines2002

    • Author(s)
      Ohashi E, Inoue K, Kagechika H, et al.
    • Journal Title

      J Vet Med Sci 64

    • NAID

      130000449408

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Novel synthetic retinoids and separation of the pleiotropic retinoidal activities.2002

    • Author(s)
      Kagechika H.
    • Journal Title

      Curr Med Chem. (5)

      Pages: 591-608

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Effect of natural and synthetic retinoids on the proliferation and differentiation of three canine melanoma cell lines.2002

    • Author(s)
      Ohashi E, Inoue K, Kagechika H, et al.
    • Journal Title

      J Vet Med Sci. 64(2)

      Pages: 169-172

    • NAID

      130000449408

    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Novel synthetic retinoids and separation of the pleiotropic retinoidal activities2002

    • Author(s)
      Kagechika H.
    • Journal Title

      Curr Med Chem 5

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Journal Article] Novel retinoid X receptor antagonists : specific inhibition of retinoid synergism in RXR-RAR heterodimer actions2002

    • Author(s)
      Takahashi B, Ohta K, Kawachi E, Fukasawa H, Hashimoto Y, Kagechika H.
    • Journal Title

      J Med Chem. 45

      Pages: 3327-3330

    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-14571118
  • [Patent] 新規アンドロゲン受容体アンタゴニスト2012

    • Inventor(s)
      影近弘之
    • Industrial Property Rights Holder
      影近弘之
    • Industrial Property Rights Type
      特許
    • Industrial Property Number
      2012-043959
    • Filing Date
      2012-02-29
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Patent] 新規アンドロゲン受容体アンタゴニスト2012

    • Inventor(s)
      影近弘之
    • Industrial Property Rights Holder
      東京医科歯科大学
    • Industrial Property Number
      2012-043959
    • Filing Date
      2012-02-29
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Patent] PRアンタゴニスト活性を有するクマリン誘導体2010

    • Inventor(s)
      棚谷綾、酒井悠、影近弘之、平野智也
    • Industrial Property Rights Holder
      お茶の水女子大学、東京医科歯科大学
    • Filing Date
      2010-02-26
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Patent] PRアンタゴニスト活性を有するクマリン誘導体2010

    • Inventor(s)
      棚谷綾, 酒井悠, 影近弘之, 平野智也
    • Industrial Property Rights Holder
      お茶の水女子大学、東京医科歯科大学
    • Industrial Property Number
      2010-043034
    • Filing Date
      2010-02-26
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Patent] レチノイドXレセプター機能調節剤2009

    • Inventor(s)
      影近弘之
    • Industrial Property Rights Holder
      東京医科歯科大学
    • Filing Date
      2009-03-03
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Patent] レチノイドXレセプター機能調節剤2009

    • Inventor(s)
      影近弘之
    • Industrial Property Rights Holder
      東京医科歯科大学
    • Industrial Property Number
      2009-004977
    • Filing Date
      2009-03-03
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] キラル側鎖をもつ芳香族スクアルアミドの立体構造解析2024

    • Author(s)
      久山和紗、片桐幸輔、川幡正俊、影近弘之、棚谷綾
    • Organizer
      日本化学会第104春季年会
    • Data Source
      KAKENHI-PROJECT-23KK0134
  • [Presentation] Dynamic Helical Property of Oligoamides with Imidazole Rings2023

    • Author(s)
      Aya Tanatani、Sakiko Kimura、Chiharu Takubo、Kosuke Katagiri、Masatoshi Kawahata、Hiroyuki Kagechika
    • Organizer
      Materials Research Meeting 2023 (MRM2023)
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-23KK0134
  • [Presentation] Development of Novel Fluorescent Sensors Based on Fluorescent Natural Compounds2016

    • Author(s)
      Hidetomo Yokoo, Tomoya Hirano, Ayumi Ohsaki, Hiroyuki Kagechika
    • Organizer
      252nd ACS National Meeting
    • Place of Presentation
      Philadelphia, USA
    • Year and Date
      2016-08-21
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Development of a facile method to detect the activity of histone methyltransferase based on SNAr reaction2016

    • Author(s)
      Yusuke Okazaki, Takashi Fujiwara, Asuka Takaguchi, Tomoya Hirano, Syuichi Mori, Hiroyuki Kagechika
    • Organizer
      International Chemical Biology Symposium 2016
    • Place of Presentation
      Madison, USA
    • Year and Date
      2016-10-24
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] SNAr反応を利用したヒストンメチル化酵素Set7/9の活性検出法の開発2016

    • Author(s)
      岡崎優祐、藤原敬士、平野智也、森修一、影近弘之
    • Organizer
      第60回日本薬学会関東支部会
    • Place of Presentation
      東京大学(東京都文京区)
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Suberene環部を修飾したCyproheptadine誘導体の合成とSet7/9に対する阻害活性評価2016

    • Author(s)
      平野道丈、平野智也、藤原敬士、大平香澄、伊藤昭博、吉田稔、影近弘之
    • Organizer
      日本薬学会第136年会
    • Place of Presentation
      パシフィコ横浜(横浜市)
    • Year and Date
      2016-03-26
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Structure-activity relationships of cyroheptadine as inhibitors of histone methyltransferase, Set7/92016

    • Author(s)
      Tomoya Hirano, Michitake Hirano, Takashi Fujiwara, Kasumi Ohira, Akihiro Ito, Minoru Yoshida, Hiroyuki Kagechika
    • Organizer
      International symposium for RIKEN epigenetics program
    • Place of Presentation
      理研中央研究所(和光市)
    • Year and Date
      2016-02-15
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Cyproheptadineを基にしたヒストンメチル化酵素Set7/9阻害剤の開発2016

    • Author(s)
      平野道丈、平野智也、藤原敬士、大平香澄、伊藤昭博、吉田稔、影近弘之
    • Organizer
      第60回日本薬学会関東支部会
    • Place of Presentation
      東京大学(東京都文京区)
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] ヒストンメチル化酵素Set7/9阻害剤の開発2015

    • Author(s)
      平野智也、藤原敬士、平野道丈、大平香澄、伊藤昭博、吉田稔、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第10回年会
    • Place of Presentation
      東北大学川内キャンパス(仙台市)
    • Year and Date
      2015-06-10
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Study for the development of inhibitors for Set7/92015

    • Author(s)
      Michitake Hirano, Tomoya Hirano, Takashi Fujiwara, Kasumi Ohira, Hiroyuki Kagechika, Akihiro Ito, Minoru Yoshida
    • Organizer
      3rd International retinoid meeting
    • Place of Presentation
      岐阜グランドホテル(岐阜市)
    • Year and Date
      2015-10-21
    • Int'l Joint Research
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] ヒストンメチル化酵素Set7/9阻害剤の開発2015

    • Author(s)
      平野道丈、平野智也、藤原敬士、大平香澄、伊藤昭博、吉田稔、影近弘之
    • Organizer
      第33回メディシナルケミストリーシンポジウム
    • Place of Presentation
      幕張国際研修センター(千葉市)
    • Year and Date
      2015-11-25
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] クマリン骨格を基盤とした新規アンドロゲン受容体アンタゴニストの創製2014

    • Author(s)
      古賀瞳、木下満里絵、藤井晋也、影近弘之、棚谷綾
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本大学(熊本)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 新規レチノイド及び関連物質の合成研究2014

    • Author(s)
      影近弘之
    • Organizer
      第345回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      京都
    • Year and Date
      2014-12-05
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] カルボランを基盤とした新規ビタミンD誘導体の創製2014

    • Author(s)
      八田健司、河内恵美子、増野弘幸、藤井晋也、影近弘之
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本大学(熊本)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] カルボランを基盤とした新規ビタミンD誘導体の創製2014

    • Author(s)
      八田健司, 河内恵美子, 増野弘幸, 藤井晋也, 影近弘之
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] クマリン骨格を基盤とした新規アンドロゲン受容体アンタゴニストの創製2014

    • Author(s)
      古賀瞳, 木下満里絵, 藤井晋也, 影近弘之, 棚谷綾
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] クマリン骨格を基盤とした新規アンドロゲン受容体アンタゴニストの創製2014

    • Author(s)
      古賀瞳、木下満里絵、藤井晋也、影近弘之、棚谷綾
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本大学(熊本)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] カルボランを基盤とした新規ビタミンD誘導体の創製2014

    • Author(s)
      八田健司、河内恵美子、増野弘幸、藤井晋也、影近弘之
    • Organizer
      日本薬学会第134年会
    • Place of Presentation
      熊本大学(熊本)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] アンドロゲン受容体アンタゴニスト活性を有する新規フェノキシフェノール誘導体の構造活性相関2013

    • Author(s)
      数井優子、山田歩、藤井晋也、影近弘之、棚谷綾
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      アステールプラザ(広島)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ビタミンK 酸化誘導体の系統的合成とその生理活性2013

    • Author(s)
      清水章貴, 藤井晋也, 影近弘之
    • Organizer
      日本薬学会第133年会
    • Place of Presentation
      横浜
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] アンドロゲン受容体アンタゴニスト活性を有する新規フェノキシフェノール誘導体の構造活性相関2013

    • Author(s)
      数井優子、山田歩、藤井晋也、影近弘之、棚谷綾
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      アステールプラザ(広島)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 疎水性球状分子を骨格とする新規プロゲステロン受容体アンタゴニストの創製2013

    • Author(s)
      森修一、竹内由起、中野英一、藤井晋也、棚谷綾、影近弘之
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      アステールプラザ(広島)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 球状疎水性ファーマコフォアを有する非セコステロイド型VDRリガンドの構造活性相関2013

    • Author(s)
      藤井晋也, Angsuma Wongmayura, 増野弘幸, 伊藤茂, 加納敦, 河内恵美子, 棚谷綾, 影近弘之
    • Organizer
      日本ビタミン学会第65回大会
    • Place of Presentation
      東京
    • Year and Date
      2013-05-17
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] クルクミンの構造要素を基盤とした新規アンドロゲン受容体アンタゴニストの創製2013

    • Author(s)
      藤井晋也, 山田歩, 森修一, 影近弘之
    • Organizer
      第24回日本レチノイド研究会学術集会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 新規ファーマコフォアの構築に基づくアンドロゲン受容体パ;ンアンタゴニストの創製2013

    • Author(s)
      藤井晋也、山田歩、森修一、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第8回年会
    • Place of Presentation
      東京医科歯科大学(東京)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 新規ファーマコフォアの構築に基づくアンドロゲン受容体パンアンタゴニストの創製2013

    • Author(s)
      藤井晋也, 山田歩, 森修一, 影近弘之
    • Organizer
      ケミカルバイオロジー学会第8回年会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] クルクミンの構造要素を基盤とした新規アンドロゲン受容体アンタゴニストの創製2013

    • Author(s)
      藤井晋也、山田歩、森修一、影近弘之
    • Organizer
      第24回日本レチノイド研究会学術集会
    • Place of Presentation
      星薬科大学(東京)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 球状疎水性ファーマコフォアを有する非セコステロイド型VDRリガンドの構造活性相関2013

    • Author(s)
      藤井晋也、Angsuma Wongmayura、増野弘幸、伊藤茂、加納敦、河内恵美子、棚谷綾、影近弘之
    • Organizer
      日本ビタミン学会第65回大会
    • Place of Presentation
      一橋講堂(東京)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Novel Estrogen Receptor Agonists Based on Silicon- and Germanium-Containing Hydrophobic Functionalities2013

    • Author(s)
      Masuno, H., Miyajima, Y., Fujii, S., Kagechika, H
    • Organizer
      The 2nd HD Physiology International Symposium on Multi-Level Systems Biology
    • Place of Presentation
      Tokyo
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 疎水性球状分子を骨格とする新規プロゲステロン受容体アンタゴニストの創製2013

    • Author(s)
      森修一, 竹内由起, 中野英一, 藤井晋也, 棚谷綾, 影近弘之
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      広島
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Novel Estrogen Receptor Agonists Based on Silicon- and Germanium-Containing Hydrophobic Functionalities2013

    • Author(s)
      Hiroyuki Masuno, Yu Miyajima, Shinya Fujii, Hiroyuki Kagechika
    • Organizer
      2nd HDP international symposium on Multi-Level Systems Biology
    • Place of Presentation
      MARUNOUCHI MY PLAZA HALL(東京)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 疎水性球状分子を骨格とする新規プロゲステロン受容体アンタゴニストの創製2013

    • Author(s)
      森修一、竹内由起、中野英一、藤井晋也、棚谷綾、影近弘之
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      アステールプラザ(広島)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 新規ファーマコフォアの構築に基づくアンドロゲン受容体パンアンタゴニストの創製2013

    • Author(s)
      藤井晋也、山田歩、森修一、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第8回年会
    • Place of Presentation
      東京医科歯科大学(東京)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of novel synthetic retinoids and their biological functions2013

    • Author(s)
      Hiroyuki Kagechika
    • Organizer
      1st International Retinoids Meeting 2013
    • Place of Presentation
      University of Calabria (Italy)
    • Invited
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ホウ素クラスターを基盤としたビタミンD の構造展開2013

    • Author(s)
      影近弘之,藤井晋也,増野弘幸
    • Organizer
      第341回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      奈良
    • Year and Date
      2013-12-06
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of novel synthetic retinoids and their biological functions2013

    • Author(s)
      Hiroyuki Kagechika
    • Organizer
      1st International Retinoids Meeting 2013
    • Place of Presentation
      University of Calabria (Italy)
    • Invited
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] 球状疎水性ファーマコフォアを有する非セコステロイド型VDRリガンドの構造活性相関2013

    • Author(s)
      藤井晋也、Angsuma Wongmayura、増野弘幸、伊藤茂、加納敦、河内恵美子、棚谷綾、影近弘之
    • Organizer
      日本ビタミン学会第65回大会
    • Place of Presentation
      一橋講堂(東京)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Development of Novel Estrogen Receptor Agonists Based on Silicon- and Germanium-Containing Hydrophobic Functionalities2013

    • Author(s)
      Hiroyuki Masuno, Yu Miyajima, Shinya Fujii, Hiroyuki Kagechika
    • Organizer
      2nd HDP international symposium on Multi-Level Systems Biology
    • Place of Presentation
      MARUNOUCHI MY PLAZA HALL(東京)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] クルクミンの構造要素を基盤とした新規アンドロゲン受容体アンタゴニストの創製2013

    • Author(s)
      藤井晋也、山田歩、森修一、影近弘之
    • Organizer
      第24回日本レチノイド研究会学術集会
    • Place of Presentation
      星薬科大学(東京)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] アンドロゲン受容体アンタゴニスト活性を有する新規フェノキシフェノール誘導体の構造活性相関2013

    • Author(s)
      数井優子, 山田歩, 藤井晋也, 影近弘之, 棚谷綾
    • Organizer
      第31回メディシナルケミストリーシンポジウム
    • Place of Presentation
      広島
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] D Development of novel synthetic retinoids and their biological functions2013

    • Author(s)
      Kagechika, H
    • Organizer
      1st International Retinoids Meeting 2013
    • Place of Presentation
      Italy
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Increased hydrophobicity and estrogenic activity of silicon- and germanium-containing phenols2013

    • Author(s)
      Shinya Fujii, Yu Miyajima, Hiroyuki Masuno, Hiroyuki Kagechika
    • Organizer
      14th Tetrahedron Symposium
    • Place of Presentation
      Vienna, Austria
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Increased hydrophobicity and estrogenic activity of silicon- and germanium-containing phenols2013

    • Author(s)
      Fujii, S., Miyajima, Y., Masuno, H., Kagechika, H
    • Organizer
      14th Tetrahedron Symposium
    • Place of Presentation
      Vienna, Austria
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Nuclear Receptor Ligands and Their CLinical Application2012

    • Author(s)
      Kagechika, H.
    • Organizer
      The 5th International Symp. for Future Technology Creating Better Human Health and Society(招待講演)
    • Place of Presentation
      岡山
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Various Functional Molecules Based on Hydrophobic and Fluorescent Scaffolds2012

    • Author(s)
      Hirano, T., Fujii, S., Mori, S., Tanatani, A., Kagechika, H
    • Organizer
      The 1st Official Conference of the International Chemical Biology Society (ICBS2012)
    • Place of Presentation
      Boston, USA
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] トリアルキルシリルおよびゲルミル基の性質と生理活性物質の疎水性構造への応用2012

    • Author(s)
      藤井晋也, 宮島友, 増野弘幸, 影近弘之
    • Organizer
      ケミカルバイオロジー学会第7回年会
    • Place of Presentation
      京都
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Nuclear Receptor Ligands and Their CLinical Application2012

    • Author(s)
      Kagechika, H
    • Organizer
      The 5th International Symposium for Future Technology Creating Better Human Health and Society
    • Place of Presentation
      Okayama
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Nuclear Receptor Ligands Based on Carborane as Hydrophobic Core Structure2012

    • Author(s)
      Fujii, S., Yamada, A., Ohta, K., Endo, Y., Kagechika, H
    • Organizer
      The 1st HD Physiology International Symposium: Integrative Multi-level Systems
    • Place of Presentation
      Tokyo
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Hydrophobic parameters, substituent constants and estrogenic activities of silyl- and germyl-containing phenols2012

    • Author(s)
      Fujii, S., Miyajima, Y., Masuno, H., Kagechika, H
    • Organizer
      Int Symp Med Chem
    • Place of Presentation
      Berlin
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of novel RXR ligands bearing tralkylsilyl or trialkylgermyl groups2012

    • Author(s)
      Masuno, H., Fujii, S., Kawach, E., Kagechika, H
    • Organizer
      The 1st HD Physiology International Symposium: Integrative Multi-level Systems
    • Place of Presentation
      Tokyo
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Design and Synthesis of Novel VDR Ligand having A Spherical Hydrophobic Structure2012

    • Author(s)
      Masuno, H., Fujii, S., Wongmayura, A., Ito, S., Kawachi, E., Tanatani, A., Kagechika, H
    • Organizer
      Vitamin D Workshop
    • Place of Presentation
      Houston, USA
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] クルクミンの構造要素を基盤とした新規AR アンタゴニストの創製2012

    • Author(s)
      山田歩, 藤井晋也, 影近弘之
    • Organizer
      日本薬学会第132年会
    • Place of Presentation
      札幌
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of novel carborane-based androgen receptor antagonists effective for mutated receptor2011

    • Author(s)
      Yamada, A., Fujii, S., Tomita, K., Nagano, M., Harayama, T., Ohta, K., Endo, Y., Kagechika, H
    • Organizer
      IME Boron XIV
    • Place of Presentation
      Niagara Falls, Canada
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] レチノイドX受容体の新規リガンドの創製2011

    • Author(s)
      影近弘之
    • Organizer
      第331回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      名古屋
    • Year and Date
      2011-07-08
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] レチノイドX受容体の新規リガンドの創製2011

    • Author(s)
      影近弘之
    • Organizer
      第331回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      名古屋
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Nuclear Receptor Ligands and Their CLinical Application2011

    • Author(s)
      Kagechika, H.
    • Organizer
      The 5th International Symp.for Future Technology Creating Better Human Health and Society
    • Place of Presentation
      岡山
    • Year and Date
      2011-03-15
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ケイ素およびゲルマニウムを持つレチノイドX 受容体(RXR)リガンドの開発2011

    • Author(s)
      増野弘幸, 藤井晋也, 前田満将, 前田貴志, 平野智也, 河内恵美子, 影近弘之
    • Organizer
      ビタミン学会第63回大会
    • Place of Presentation
      広島
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] レチノイドX 受容体の新規リガンドの創製2011

    • Author(s)
      影近弘之
    • Organizer
      第331回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      名古屋
    • Year and Date
      2011-07-08
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development and structural basis of novel non-secosteroidal VDR ligands based on hydrophobic carborane cage2011

    • Author(s)
      Fujii, S., Masuno, H., Nakabayashi, M., Hirano, T., Kawachi, E., Ito, N., Kagechika, H
    • Organizer
      IME Boron XIV
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Siliconand Germanium-containing Ligands for Nuclear Receptors2011

    • Author(s)
      Masuno, H., Fujii, S., Miyajima, Y., Kawachi, E., Kagechika, H
    • Organizer
      AIMECS11
    • Place of Presentation
      Tokyo
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Novel AR Antagonists Active in LNCaP Cells with Mutated Androgen Receptor2011

    • Author(s)
      Yamada, A., Fujii, S., Tomita, K., Nagano, M., Harayama, T., Ohta, K., Endo, Y., Kagechika, H
    • Organizer
      AIMECS11
    • Place of Presentation
      Tokyo
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] Development of Novel Synthetic Ligands for Nuclear Receptors2010

    • Author(s)
      Kagechika, H.
    • Organizer
      The 14th International Congress ofEndocrinology(ICE2010)
    • Place of Presentation
      Kyoto
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] カルボランを疎水性骨格とするビタミンD誘導体とその核内受容体結合様式2010

    • Author(s)
      影近弘之,藤井晋也,増野弘幸,平野智也,伊藤暢聡,伊倉貞吉,棚谷綾
    • Organizer
      第7回中性子捕獲療法学会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of NovelAndrogen Antagonists Based on Hydrophobic Boron Clusters2010

    • Author(s)
      Fujii, S., Yamada, A., Ohta, K., Endo, Y., Kagechika, H.
    • Organizer
      EFMC-ISMC2010 21^<st> International Symposium on MedicinalChemistry
    • Place of Presentation
      Brussels, Bergium
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] クマリン骨格を基盤とした蛍光センサーの効率的開発法の構築と、蛍光性プロゲステロン受容体リガンド開発への応用2010

    • Author(s)
      平野智也,酒井悠,白石拓也,森修一,藤井晋也,棚谷綾,影近弘之
    • Organizer
      第4回バイオ関連化学シンポジウム
    • Place of Presentation
      大阪
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Non-seco-Stroid-type Vitamin D Derivatives2010

    • Author(s)
      影近弘之
    • Organizer
      ICE2010 Official Satellite Symposium
    • Place of Presentation
      京都
    • Year and Date
      2010-03-31
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Synthetic Ligands for Nuclear Receptors2010

    • Author(s)
      Kagechika, H.
    • Organizer
      The 14^<th> International Congress of Endocrinology (ICE2010)
    • Place of Presentation
      京都
    • Year and Date
      2010-03-30
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 変異受容体にも有効な新規アンドロゲンアンタゴニストの創製2010

    • Author(s)
      山田 歩、冨田 景子、長野也 麻央、藤井晋、原山 尚、太田 公規、遠藤 泰之、影近弘之
    • Organizer
      日本薬学会第130年会
    • Place of Presentation
      岡山
    • Data Source
      KAKENHI-PROJECT-20390035
  • [Presentation] Development of Novel Nonsteroidal AndrogenReceptor Ligands Based on Hydrophobic BoronClusters2010

    • Author(s)
      Fujii, S., Ohta, K., Endo, Y., Kagechika, H.
    • Organizer
      ICE2010 Official Satellite Symposium-Nuclear Receptor and its Frontier-
    • Place of Presentation
      Kyoto
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] カルボランを疎水性骨格とする新規アンドロゲン受容体リガンドの創製2010

    • Author(s)
      藤井晋也,山田歩,太田公規,遠藤泰之,影近弘之
    • Organizer
      第7回中性子捕獲療法学会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] カルボランを疎水性骨格とするビタミンD誘導体とその核内受容体結合様式2010

    • Author(s)
      影近弘之
    • Organizer
      第7回中性子捕獲療法学会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ホウ素クラスターを疎水性骨格とする新規非セコステロイド型ビタミンD誘導体:受容体結合様式と構造展開2010

    • Author(s)
      藤井晋也,増野弘幸,垰田善之,加納敦,中林誠,伊藤暢聡,河内恵美子,清水正人,棚谷綾,平野智也,影近弘之
    • Organizer
      日本レチノイド研究会第21回学術集会
    • Place of Presentation
      高槻
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Synthetic Ligands for Nuclear Receptors2010

    • Author(s)
      影近弘之
    • Organizer
      The 14^<th> International Congress of Endocrinology
    • Place of Presentation
      京都
    • Year and Date
      2010-03-30
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 核内受容体を分子標的とした医薬化学研究-レチノイドを中心に2010

    • Author(s)
      影近弘之
    • Organizer
      Metabolic Syndrome Seminar
    • Place of Presentation
      岡山
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Non-seco-Stroid-type Vitamin DDerivatives2010

    • Author(s)
      Kagechika, H.
    • Organizer
      ICE2010 Official Satellite Symposium-Nuclear Receptor and its Frontier-
    • Place of Presentation
      Kyoto
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 変異ARを有するLNCaP細胞に対して有効な新規ARアンタゴニストの創製2010

    • Author(s)
      山田歩,富田景子,長野麻央,藤井晋也,原山尚,太田公規,遠藤泰之,影近弘之
    • Organizer
      ケミカルバイオロジー学会第5回年会
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] VDR活性をもつLCA誘導体の合成とVDR結合構造の解析2010

    • Author(s)
      増野弘幸,数井優子,伊倉貞吉,中林誠,伊藤暢聡,藤井晋也,河内恵美子,棚谷綾,影近弘之
    • Organizer
      ビタミン学会第62回大会
    • Place of Presentation
      岩手
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Nuclear Receptor Ligands for Cancer Therapy2009

    • Author(s)
      影近弘之
    • Organizer
      TMD-CMU International Symposium
    • Place of Presentation
      東京
    • Year and Date
      2009-10-14
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 変異ARに対して有効なカルボラン含有新規ARアンタゴニストの創製2009

    • Author(s)
      山田歩,富田景子,長野麻央,藤井晋也,原山尚,太田公規,遠藤泰之,影近弘之
    • Organizer
      第28回メディシナルケミストリーシンポジウム
    • Place of Presentation
      東京
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] ビタミンA新しい構造、機能、そして医薬へ2009

    • Author(s)
      影近弘之
    • Organizer
      第326回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      静岡
    • Year and Date
      2009-12-04
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of a novel "functional" fluorescent labeling reagents for variousligand molecules2009

    • Author(s)
      Hirano, T., Akiyama, J., Kagechika, H.
    • Organizer
      World Molecular ImagingCongress
    • Place of Presentation
      Montreal, Canada
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Crystal Structures of Non-secosteroidLigands Bound to Vitamin D NuclearReceptor2009

    • Author(s)
      Masuno, H., Fujii, S., Nakabayashi, M., Ikura, T., Ito, N., Shimizu, M., Kagechika, H.
    • Organizer
      14th Vitamin D Workshop
    • Place of Presentation
      Brugge, Belgium
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] ビタミンA 新しい構造、機能、そして医薬へ2009

    • Author(s)
      影近弘之
    • Organizer
      第326回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      静岡
    • Year and Date
      2009-12-04
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 10-vertex カルボランを用いたアンドロゲン受容体リガンドの創製2009

    • Author(s)
      藤井 晋也、太田 公規、遠藤 泰之、影近弘之
    • Organizer
      日本薬学会第129年会
    • Place of Presentation
      京都
    • Data Source
      KAKENHI-PROJECT-20390035
  • [Presentation] Development ofNovel Non-secosteroidal Vitamin DReceptor Ligands Based on Carborane as AHydrophobic Core Structure2009

    • Author(s)
      Fujii, S., Kano, A., Sekine, R., Kawachi, E., Masuno, H., Hirano, T., Tanatani, A., Kagechika, H.
    • Organizer
      14th Vitamin D Workshop
    • Place of Presentation
      Brugge, Belgium
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Non-secosteroidal Vitamin D Receptor Ligands Based on Carborane as A Hydrophobic Core Structure2009

    • Author(s)
      Fujii, A., Kano, A., Sekine, R., Kawachi, E., Masuno, H., Hirano, T., Tanatani, A., Kagechika, H.
    • Organizer
      14^<th> Vitamin D Workshop
    • Place of Presentation
      Brugge, Belgium
    • Year and Date
      2009-10-04
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] 新規非セコステロイド型VDRリガンドの構造展開と受容体結合様式の解析2009

    • Author(s)
      藤井晋也,加納敦,平野智也,河内恵美子,増野弘幸,棚谷綾,中林誠,伊倉貞吉,伊藤暢聡,清水正人,影近弘之
    • Organizer
      ビタミン学会第61回大会
    • Place of Presentation
      亀岡
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] カルボランを疎水性骨格とする新規非ステロイド型VDRリガンドの構造展開2009

    • Author(s)
      藤井晋也,加納敦,平野智也,河内恵美子,増野弘幸,棚谷綾,中林誠,伊倉貞吉,伊藤暢聡,清水正人,影近弘之
    • Organizer
      第35回反応と合成の進歩シンポジウム
    • Place of Presentation
      金沢
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Tricarbocyanine系蛍光物質の会合現象制御による蛍光センサーの開発2009

    • Author(s)
      平野智也,秋山淳,影近弘之
    • Organizer
      第24回生体機能関連化学シンポジウム
    • Place of Presentation
      福岡
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Novel synthetic RAR and RXR-selective agonists bearing aunique structure in the hydrophobic part2008

    • Author(s)
      Kagechika H, Muratake H, Amano Y, Noguchi M, Shudo K
    • Organizer
      FASEB meeting on Retinoid
    • Place of Presentation
      New Haven, USA
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Novel synthetic RAR- and RXR-selective agonists bearing a unique structure in the hydrophobic part2008

    • Author(s)
      Hiroyuki Kagechika
    • Organizer
      FASEB meeting on Retinoid
    • Place of Presentation
      New Haven, CT, USA
    • Year and Date
      2008-06-16
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Novel synthetic RAR- and RXR-selective agonists bearing a unique structure in the hydrophobic part2008

    • Author(s)
      Kagechika, H., Muratake, H., Amano, Y., Noguchi, M., Shudo. K.
    • Organizer
      FASEB meeting on Retinoid
    • Year and Date
      2008-06-15
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Novel non-seco-steroidal VDR ligands bearing a carborane as a hydrophobic pharmacophore2008

    • Author(s)
      Hiroyuki Kagechika
    • Organizer
      XIII IMEBORON
    • Place of Presentation
      Spain
    • Year and Date
      2008-09-21
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Novelnon-seco-steroidal VDR ligands bearing acarborane as a hydrophobic pharmacophore2008

    • Author(s)
      Kagechika H, Kano A, Fujii S, Hirano T, Kawachi E, Tanatani A
    • Organizer
      XIII IMEBORON
    • Place of Presentation
      Spain
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] カルボラン含有ビタミンD誘導体の創製とVDR結合様式2008

    • Author(s)
      影近弘之
    • Organizer
      第320回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      大阪
    • Year and Date
      2008-07-18
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] レチノイド : 活性ビタミンAの医薬展開2008

    • Author(s)
      影近弘之
    • Organizer
      第386回国際治療談話会例会
    • Place of Presentation
      東京
    • Year and Date
      2008-09-18
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Development of Novel Inhibitors of Histone Methyltransferase2008

    • Author(s)
      Hirano T, Hoshino K, Iwanami N, TanakaY, Kagechika H
    • Organizer
      236th ACS National Meeting
    • Place of Presentation
      Philadelphia, USA
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Utility of boron cluster for drug design:Design of androgen receptor/ estrogen receptor dual ligands bearing carborane for anti-prostate cancer drug2008

    • Author(s)
      Yasuyuki Endo , Tokuhito Goto, Kiminori Ohta, Shinya Fujii, Hiroyuki Kagechika
    • Organizer
      13th International Conferenceon Boron Chemistry
    • Place of Presentation
      Platja d'Aro, Spain
    • Data Source
      KAKENHI-PROJECT-20390035
  • [Presentation] Androgen receptor antagonists based on boron cluster as a hydrophobic core structure2008

    • Author(s)
      Shinya Fujii, Kiminori Ohta, Tokuhito Goto, Tomoharu Suzuki, Shigeru Ohta, Yuichi Hashimoto, Hiroyuki Kagechika, Yasuyuki Endo
    • Organizer
      13th International Conference on Boron Chemistry
    • Place of Presentation
      Platja d'Aro, Spain
    • Data Source
      KAKENHI-PROJECT-20390035
  • [Presentation] Synthetic Retinoids: Biological Functions and Clinical Utilities2007

    • Author(s)
      影近 弘之
    • Organizer
      第4回武田科学振興財団薬科学シンポジウム
    • Place of Presentation
      東京
    • Year and Date
      2007-12-03
    • Data Source
      KAKENHI-PROJECT-19659022
  • [Presentation] Mechanisms of ATRA-indiced angiogenesis: involvement of VEGF2007

    • Author(s)
      Saito A, Sugawara A, Uruno A, Kudo M, Kagechika H, Sato Y, Imaizumi M, Tsuchiya S, Ito S
    • Organizer
      18th Meeting of Japanese Society for Retinoid Research
    • Place of Presentation
      Tokyo
    • Year and Date
      2007-11-23
    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Presentation] Synthetic Retinoids: Biological Functions and Clinical Utilities2007

    • Author(s)
      影近 弘之
    • Organizer
      第4回武田科学振興財団薬科学シンポジウム
    • Place of Presentation
      東京
    • Year and Date
      2007-12-03
    • Data Source
      KAKENHI-PROJECT-19201044
  • [Presentation] Synthetic Retinoids: Biological Functions and Clinical Utilities2007

    • Author(s)
      影近 弘之
    • Organizer
      第4回武田科学振興財団薬科学シンポジウム
    • Place of Presentation
      東京
    • Year and Date
      2007-12-03
    • Data Source
      KAKENHI-PROJECT-18032026
  • [Presentation] 全トランス型レチノイン酸による血管新生促進機構の解明-レチノイン酸受容体及びVEGFシグナルの関与-2007

    • Author(s)
      斉藤明子、菅原 明、宇留野晃、工藤正孝、影近弘之、佐藤靖史、今泉益栄、土屋 滋、伊藤貞嘉
    • Organizer
      日本レチノイド研究会第18回学術集会
    • Place of Presentation
      東京
    • Year and Date
      2007-11-23
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Presentation] PPARαγデュアルリガンドによる血管新生の制御。2006

    • Author(s)
      佐藤眞友美、清水本武、宮地弘幸、影近弘之、菅原 明
    • Organizer
      第79回日本内分泌学会学術総会
    • Place of Presentation
      神戸
    • Description
      「研究成果報告書概要(和文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Presentation] Regulation of angiogenesis by PPARay dual ligand2006

    • Author(s)
      Sato M, Shimizu M, Miyaji H, Kagechika H, Sugawara A
    • Organizer
      79th Japan Endocrine Society Meeting
    • Place of Presentation
      Kobe
    • Description
      「研究成果報告書概要(欧文)」より
    • Data Source
      KAKENHI-PROJECT-18591015
  • [Presentation] Development of Fluorescent Sensors with its Functions Regulated by Chemical or Enzymatic Reaction

    • Author(s)
      Tomoya Hirano, Takuya Shiraishi, Toshiki Saito, Hiroyuki Kagechika
    • Organizer
      3rd International Chemical Biology Meeting
    • Place of Presentation
      San Fransisco, USA
    • Year and Date
      2014-11-17 – 2014-11-20
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Lipase-catalyzed asymmetric acylation of boron cluster-containing secondary alcohols

    • Author(s)
      Shuichi Mori, Ryohei Takagaki, Shinya Fujii, Mio Matsumura, Aya Tanatani, and Hiroyuki Kagechika
    • Organizer
      Active Enzyme Molecule 2014
    • Place of Presentation
      富山
    • Year and Date
      2014-12-17 – 2014-12-19
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 蛍光物質ライブラリーおよびその構築法を基にした多機能性蛍光センサー群の開発

    • Author(s)
      平野智也、白石拓也、齋藤俊樹、影近弘之
    • Organizer
      第8回バイオ関連化学シンポジウム
    • Place of Presentation
      岡山
    • Year and Date
      2014-09-11 – 2014-09-13
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] N-Aryl-N’-cyanoformamidineの立体構造解析

    • Author(s)
      デリホマル アニワル、伊藤茂、金井美紗衣、棚谷綾、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 蛍光物質ライブラリー構築を基にした蛍光センサー群の開発

    • Author(s)
      平野智也、白石拓也、齋藤俊樹、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第9回年会
    • Place of Presentation
      大阪
    • Year and Date
      2014-06-11 – 2014-06-13
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Development of Novel Synthetic Retinoids with Unique Hydrophobic Core Structure

    • Author(s)
      Hiroyuki Kagechika
    • Organizer
      FASEB 2nd International retinoid meeting
    • Place of Presentation
      Chicago, USA
    • Year and Date
      2014-06-01 – 2014-06-06
    • Invited
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ホウ素クラスターを基盤としたビタミンDの構造展開

    • Author(s)
      影近弘之、藤井晋也、増野弘幸
    • Organizer
      第341回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      奈良女子大学(奈良)
    • Data Source
      KAKENHI-PROJECT-23659051
  • [Presentation] アンドロゲン受容体アンタゴニスト活性を有する新規シラノール誘導体の創製

    • Author(s)
      山内夢人、藤井晋也、増野弘幸、河内恵美子、影近弘之
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ヒストンメチル化酵素活性評価系の開発研究

    • Author(s)
      藤原敬士、髙口明日香、森修一、平野智也、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] Lipase-catalyzed optical resolution and biological activity of boron-cluster-based progesterone receptor ligands

    • Author(s)
      Shuichi Mori, Ryohei Takagaki, Shinya Fujii, Mio Matsumura, Aya Tanatani, Hiroyuki Kagechika
    • Organizer
      3rd International Chemical Biology Meeting
    • Place of Presentation
      San Fransisco, USA
    • Year and Date
      2014-11-17 – 2014-11-20
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 高血圧治療薬開発を志向したWNKシグナル阻害剤の創薬

    • Author(s)
      鈴山帆乃佳、渡邊優子、森崇寧、菊池絵梨子、湯浅磨里、藤井晋也、内田信一、影近弘之
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] シラノール基を有する新規アンドロゲン受容体アンタゴニストの創製

    • Author(s)
      山内夢人、藤井晋也、河内恵美子、増野弘幸、影近弘之
    • Organizer
      日本レチノイド研究会第25回学術集会
    • Place of Presentation
      秋田
    • Year and Date
      2014-10-08 – 2014-10-09
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Hippoシグナル伝達系に関与する転写共役因子TAZの活性促進物質の探索

    • Author(s)
      デリホマル アニワル、伊藤茂、中川健太郎、楊沢宇、湯浅磨里、畑裕、影近弘之
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Investigation of regulatory compounds toward transcriptional co-activator TAZ

    • Author(s)
      Shigeru Ito, Kentaro Nakagawa, Zeyu Yang, Mari Yuasa, Yutaka Hata, Hiroyuki Kagechika
    • Organizer
      EMBO Conference Series: Chemical Biology 2014
    • Place of Presentation
      Heidelberg, Germany
    • Year and Date
      2014-08-20 – 2014-08-23
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 新規7-アミドクマリン誘導体のアンドロゲンアンタゴニスト活性

    • Author(s)
      古賀瞳、木下満里絵、藤井晋也、影近弘之、棚谷綾
    • Organizer
      日本レチノイド研究会第25回学術集会
    • Place of Presentation
      秋田
    • Year and Date
      2014-10-08 – 2014-10-09
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 特定の酵素により機能が制御されるカチオン蛍光センサーの開発

    • Author(s)
      白石拓也、平野智也、齊藤俊樹、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 転写共役因子 TAZ の活性を制御する化合物の探索

    • Author(s)
      伊藤茂、中川健太郎、楊沢宇、湯浅磨里、影近弘之、畑裕
    • Organizer
      日本ケミカルバイオロジー学会第9回年会
    • Place of Presentation
      大阪
    • Year and Date
      2014-06-11 – 2014-06-13
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Design and Synthesis of C,C’-Diphenylcarborane Derivatives as Novel Progesterone Receptor Antagonists

    • Author(s)
      Hiroyuki Kagechika, Eiichi Nakano, Ayumi Yamada, Yuki Takeuchi, Shuichi Mori, Hiroyuki Masuno, Shinya Fujii
    • Organizer
      IMEBoron XV
    • Place of Presentation
      Prague, Czech Republic
    • Year and Date
      2014-08-24 – 2014-08-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ヒストンメチル化酵素活性評価系の開発研究

    • Author(s)
      藤原敬士、髙口明日香、森修一、平野智也、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Development of Fluorescent Sensors with its Functions Regulated by Chemical or Enzymatic Reaction

    • Author(s)
      Tomoya Hirano, Takuya Shiraishi, Toshiki Saito, Hiroyuki Kagechika
    • Organizer
      3rd International Chemical Biology Meeting
    • Place of Presentation
      San Francisco, USA
    • Year and Date
      2014-11-17 – 2014-11-20
    • Data Source
      KAKENHI-PROJECT-26670052
  • [Presentation] クルクミン誘導体の構造展開による新規PRアンタゴニストの創製

    • Author(s)
      藤井晋也、山田歩、森修一、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第9回年会
    • Place of Presentation
      大阪
    • Year and Date
      2014-06-11 – 2014-06-13
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] クマリン骨格を基盤としたアンドロゲンアンタゴニストの創製研究

    • Author(s)
      古賀瞳、木下満里絵、藤井晋也、影近弘之、棚谷綾
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 合成レチノイドによるT細胞カルシウムイオン濃度上昇の阻害効果

    • Author(s)
      森修一、湯浅麻里、渡辺陽平、押田侑輝、影近弘之
    • Organizer
      日本レチノイド研究会第25回学術集会
    • Place of Presentation
      秋田
    • Year and Date
      2014-10-08 – 2014-10-09
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 蛍光物質ライブラリー構築を基にした蛍光センサー群の開発

    • Author(s)
      平野智也、白石拓也、齋藤俊樹、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第9回年会
    • Place of Presentation
      大阪
    • Year and Date
      2014-06-11 – 2014-06-13
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 新規ストア作動性カルシム流入阻害剤の探索と構造展開

    • Author(s)
      森修一、渡邉陽平、湯浅磨里、影近弘之
    • Organizer
      日本ケミカルバイオロジー学会第9回年会
    • Place of Presentation
      大阪
    • Year and Date
      2014-06-11 – 2014-06-13
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 蛍光物質ライブラリーおよびその構築法を基にした多機能性蛍光センサー群の開発

    • Author(s)
      平野智也、白石拓也、齋藤俊樹、影近弘之
    • Organizer
      第8回バイオ関連化学シンポジウム
    • Place of Presentation
      岡山
    • Year and Date
      2014-09-11 – 2014-09-13
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] カルボランを基盤とする非セコステロイド型VDRリガンドの疎水性部位の構造展開

    • Author(s)
      藤井晋也、八田健司、増野弘幸、河内恵美子、影近弘之
    • Organizer
      日本ビタミン学会第65回大会
    • Place of Presentation
      姫路
    • Year and Date
      2014-06-13 – 2014-06-14
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Novel Store-Operated Calcium Entry (SOCE) inhibitors having the retinoid-like structure

    • Author(s)
      Mari Ishigami-Yuasa, Shuichi Mori, Yohei Watanabe, Hiroyuki Kagechika
    • Organizer
      FASEB 2nd International retinoid meeting
    • Place of Presentation
      Chicago, USA
    • Year and Date
      2014-06-01 – 2014-06-06
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] カルボラン含有プロゲステロン受容体リガンドのリパーゼによる光学分割

    • Author(s)
      森修一、高垣亮平、藤井晋也、松村実生、棚谷綾、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 特定のpH領域を検出する蛍光センサー群の開発

    • Author(s)
      野地優希、平野智也、齋藤俊樹、白石拓也、影近弘之
    • Organizer
      日本薬学会第135年会
    • Place of Presentation
      神戸
    • Year and Date
      2015-03-26 – 2015-03-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] Synthesis and Characterization of Novel m-Ccarborane-Containing Porphyrinoid

    • Author(s)
      Shinya Fujii, Shotaro Iihama, Hiroyuki Kagechika
    • Organizer
      IMEBoron XV
    • Place of Presentation
      Prague, Czech Republic
    • Year and Date
      2014-08-24 – 2014-08-28
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] ホウ素クラスターを基盤としたビタミンDの構造展開

    • Author(s)
      影近弘之、藤井晋也、増野弘幸
    • Organizer
      第341回脂溶性ビタミン総合研究委員会
    • Place of Presentation
      奈良女子大学(奈良)
    • Data Source
      KAKENHI-PLANNED-22136013
  • [Presentation] 新規T細胞カルシウム濃度制御剤の創製」

    • Author(s)
      森修一、渡辺陽平、押田侑輝、湯浅磨里、影近弘之
    • Organizer
      第32回メディシナルケミストリーシンポジウム
    • Place of Presentation
      神戸
    • Year and Date
      2014-11-26 – 2014-11-28
    • Data Source
      KAKENHI-PLANNED-22136013
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